Pharmacology

Action Mechanism of Action Reference
INHIBITOR DNA topoisomerase I inhibitor
Primary Target
tumor associated calcium signal transducer 2

Indications

Mesh Heading Maximum Phase Mesh ID Reference
Neoplasms 4 D009369 ClinicalTrials
Endometrial Neoplasms 3 D016889 ClinicalTrials
Endometrial Neoplasms 3 D016889 ClinicalTrials
Carcinoma, Non-Small-Cell Lung 3 D002289 ClinicalTrials
Urogenital Neoplasms 3 D014565 ClinicalTrials
Urinary Bladder Neoplasms 2 D001749 ClinicalTrials
Glioblastoma 2 D005909 ClinicalTrials
Prostatic Neoplasms, Castration-Resistant 2 D064129 ClinicalTrials
Uterine Cervical Neoplasms 2 D002583 ClinicalTrials
Urinary Bladder Neoplasms 2 D001749 ClinicalTrials
Urinary Bladder Neoplasms 2 D001749 ClinicalTrials
Klatskin Tumor 2 D018285 ClinicalTrials
Thyroid Neoplasms 2 D013964 ClinicalTrials
Lung Neoplasms 2 D008175 ClinicalTrials
Mesothelioma 2 D008654 ClinicalTrials
Ovarian Neoplasms 2 D010051 ClinicalTrials
Brain Diseases 2 D001927 ClinicalTrials
Esophageal Neoplasms 2 D004938 ClinicalTrials
Thymoma 2 D013945 ClinicalTrials
Thymoma 2 D013945 ClinicalTrials
Stomach Neoplasms 1 D013274 ClinicalTrials
Meningeal Carcinomatosis 1 D055756 ClinicalTrials
Small Cell Lung Carcinoma 1 D055752 ClinicalTrials

Cross References

Resources Reference
CAS NUMBER 1491917-83-9
ChEMBL CHEMBL3545262
FDA SRS M9BYU8XDQ6
Guide to Pharmacology 8253
PubChem 91668186