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Total: 50
Small molecule
Approved
DENTISTRY; NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
BUCCAL; ORAL; RECTAL; TOPICAL
Abortion, Spontaneous; Attention Deficit Disorder with Hyperactivity; Brain Neoplasms; Carcinoma, Squamous Cell; Cicatrix; Complex Regional Pain Syndromes; Glioblastoma; Glycogen Storage Disease Type II; Hypertension, Pulmonary; Keratosis, Actinic; Lung Neoplasms; Morton Neuroma; Neoplasms, Cystic, Mucinous, and Serous; Neuroma; Parathyroid Neoplasms; Premature Birth; Radius Fractures; Skin Neoplasms; Spinal Fractures; Thromboembolism; Tinnitus; Anus Diseases; Anxiety; Cancer Pain; Carcinoma; Cocaine-Related Disorders; Cognitive Dysfunction; Cystitis, Interstitial; Diabetic Neuropathies; Dysmenorrhea; Dysphonia; Geographic Atrophy; Heart Diseases; Humeral Fractures; Infertility; Irritable Bowel Syndrome; Leiomyoma; Myofascial Pain Syndromes; Neoplasms; Renal Colic; Rib Fractures; Scleroderma, Localized; Severe Acute Respiratory Syndrome; Shoulder Impingement Syndrome; Shoulder Pain; Skin Diseases; Temporomandibular Joint Disorders; Trigeminal Neuralgia; Urinary Incontinence; Urinary Tract Infections; Analgesia; Breast Neoplasms; Carpal Tunnel Syndrome; Chronic Pain; Colorectal Neoplasms; Common Cold; Cough; Dysuria; Fibromyalgia; Fractures, Bone; Headache; Heart Arrest; Hemorrhage; Ileus; Low Back Pain; Migraine Disorders; Muscular Diseases; Nutrition Disorders; Obesity; Obesity, Morbid; Osteoarthritis, Knee; Osteoporosis, Postmenopausal; Paget Disease, Extramammary; Parathyroid Diseases; Periarthritis; Peripheral Nervous System Diseases; Pharyngitis; Pre-Eclampsia; Pregnancy; Pulpitis; Scoliosis; Shock, Septic; Sinusitis; Stomatitis; Stroke; Tennis Elbow; Urinary Bladder Neoplasms; Urinary Bladder, Overactive; Uterine Cervical Dysplasia; Wounds and Injuries; Arrhythmias, Cardiac; Arthritis; Back Pain; Burns; Bursitis; Hemorrhoids; Inflammation; Insect Bites and Stings; Muscle Cramp; Myalgia; Neuralgia; Neuralgia, Postherpetic; Osteoarthritis; Pain; Premature Ejaculation; Pruritus; Rectal Diseases; Sprains and Strains; Sunburn; Tendinopathy; Urethritis
Sodium channel alpha subunit blocker
Small molecule
Approved
CANCER; NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
BUCCAL; SUBLINGUAL; TRANSDERMAL
Burns; Opioid-Related Disorders; Respiratory Distress Syndrome; Brain Injuries; Breast Neoplasms; Delirium; Fractures, Bone; Hypospadias; Hypotension; Irritable Bowel Syndrome; Pregnancy; Pulpitis; Scoliosis; Subarachnoid Hemorrhage; Abscess; Adenoma; Aortic Coarctation; Diabetic Neuropathies; Liver Diseases; Low Back Pain; Lung Diseases; Migraine Disorders; Neoplasm Metastasis; Obesity; Obesity, Morbid; Osteoarthritis; Pancreatic Neoplasms; Renal Insufficiency, Chronic; Respiratory Insufficiency; Severe Acute Respiratory Syndrome; Sleep Apnea, Obstructive; Stomach Neoplasms; Acute Pain; Cancer Pain; Chronic Pain; Neoplasms; Pain
Mu opioid receptor agonist
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER; PEDIATRICS
INTRAVENOUS; ORAL
Hepatitis B, Chronic; Parkinson Disease; Severe Acute Respiratory Syndrome; Cocaine-Related Disorders; Epilepsy, Reflex; HIV Infections; Nausea; Substance-Related Disorders; Anxiety; Dementia; Depressive Disorder; Schizophrenia; Bipolar Disorder; Epilepsies, Partial; Epilepsy; Glossopharyngeal Nerve Diseases; Seizures; Trigeminal Neuralgia
Sodium channel alpha subunit blocker
Small molecule
Approved
EMERGENCY MEDICINE; NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
INJECTION
Aortic Coarctation; Brain Neoplasms; Hernia, Ventral; HIV Infections; Lung Diseases; Neuralgia; Obesity, Morbid; Prostatic Neoplasms, Castration-Resistant; Sarcoma; Sinusitis; Stress Disorders, Post-Traumatic; Subarachnoid Hemorrhage; Vasospasm, Intracranial; Abdominal Pain; Appendicitis; Atrial Fibrillation; Blepharoptosis; Blood Coagulation Disorders; Cleft Palate; Complex Regional Pain Syndromes; Dupuytren Contracture; Fasciitis, Plantar; Femoral Neck Fractures; Headache; Hemorrhage; Hernia, Umbilical; Hip Fractures; Hypospadias; Hypotension; Lacrimal Apparatus Diseases; Low Back Pain; Mucositis; Musculoskeletal Diseases; Osteoarthritis, Hip; Pregnancy; Pulpitis; Rib Fractures; Shoulder Pain; Spinal Stenosis; Analgesia; Ankle Fractures; Breast Neoplasms; Breech Presentation; Carcinoma, Non-Small-Cell Lung; Chronic Pain; Cough; Fractures, Bone; Genital Neoplasms, Female; Hallux Valgus; Hemorrhoids; Hernia, Inguinal; Ileus; Liver Diseases; Lung Neoplasms; Migraine Disorders; Neoplasms; Osteoarthritis; Osteoarthritis, Knee; Pancreatic Neoplasms; Pancreatitis, Chronic; Peritoneal Neoplasms; Postoperative Nausea and Vomiting; Radiculopathy; Radius Fractures; Rotator Cuff Injuries; Toothache; Urethral Stricture; Wounds and Injuries; Acute Pain; Hernia; Pain
Sodium channel protein type IV alpha subunit blocker
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
ORAL
Burning Mouth Syndrome; Neuralgia; Marijuana Abuse; REM Sleep Behavior Disorder; Anxiety; Dementia; Depressive Disorder; Epilepsia Partialis Continua; Epilepsy, Tonic-Clonic; Pain; Schizophrenia; Status Epilepticus; Epilepsy; Panic Disorder; Seizures
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
ORAL
Astrocytoma; Brain Injuries; Burkitt Lymphoma; Carcinoma, Non-Small-Cell Lung; Central Nervous System Neoplasms; Colorectal Neoplasms; Epilepsies, Partial; Lung Neoplasms; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Medulloblastoma; Melanoma; Nasopharyngeal Carcinoma; Neoplasms; Ovarian Neoplasms; Paraganglioma; Sarcoma; Shock; Urinary Bladder Neoplasms; Wounds and Injuries; Alopecia; Brain Neoplasms; Breast Neoplasms; Carcinoma, Squamous Cell; Ependymoma; Glioblastoma; Glioma; Head and Neck Neoplasms; HIV Infections; Leukemia; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Lymphoma; Myelodysplastic Syndromes; Neuralgia; Pancreatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Retinitis Pigmentosa; Small Cell Lung Carcinoma; Supranuclear Palsy, Progressive; Thyroid Neoplasms; Uveal Melanoma; Alcoholism; Alzheimer Disease; Anxiety; Autistic Disorder; Dementia; Depressive Disorder; Migraine Disorders; Muscular Atrophy, Spinal; Paraparesis, Tropical Spastic; Psychomotor Agitation; Schizophrenia; Status Epilepticus; Bipolar Disorder; Epilepsy; Epilepsy, Absence; Epilepsy, Complex Partial; Mitochondrial Diseases; Seizures
Succinate semialdehyde dehydrogenase inhibitor
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM
INTRAMUSCULAR
Anorexia Nervosa; Bulimia; Bulimia Nervosa; Child Development Disorders, Pervasive; Dermatitis, Atopic; Melanoma; Mental Disorders; Psoriasis; Schizophrenia; Smoking Cessation; Alcohol Drinking; Alcohol-Related Disorders; Back Pain; Breast Neoplasms; Colitis, Ulcerative; Coronavirus Infections; Crohn Disease; Cystitis, Interstitial; Depressive Disorder, Major; Diabetic Neuropathies; Dry Eye Syndromes; Fatigue; Fibromyalgia; Low Back Pain; Marijuana Abuse; Migraine Disorders; Obsessive-Compulsive Disorder; Post-Acute COVID-19 Syndrome; Respiratory Distress Syndrome; Severe Acute Respiratory Syndrome; Trichotillomania; Amphetamine-Related Disorders; Borderline Personality Disorder; Chronic Pain; Cocaine-Related Disorders; Depressive Disorder; Endometriosis; Gambling; Heroin Dependence; HIV Infections; Multiple Sclerosis; Obesity; Opioid-Related Disorders; Pain; Stress Disorders, Post-Traumatic; Substance-Related Disorders; Tobacco Use Disorder; Alcoholism
Opioid receptors; mu/kappa/delta antagonist
Small molecule
Approved
IMMUNE SYSTEM; NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER; PEDIATRICS
ORAL
Alopecia; Child Development Disorders, Pervasive; Glioblastoma; Premature Birth; Psychotic Disorders; Abortion, Spontaneous; Anemia, Sickle Cell; Breast Neoplasms; HIV Infections; Hyperemesis Gravidarum; Intervertebral Disc Displacement; Low Back Pain; Marijuana Abuse; Mucositis; Multiple Sclerosis; Neoplasms; Paget Disease, Extramammary; Peripheral Nervous System Diseases; Postoperative Complications; Prostatic Neoplasms, Castration-Resistant; Rotator Cuff Injuries; Sleep Wake Disorders; Substance-Related Disorders; Substance Withdrawal Syndrome; Tinnitus; Tobacco Use Disorder; Urinary Bladder Neoplasms; Wounds and Injuries; Alcohol Drinking; Alcoholism; Anxiety; Azoospermia; Brain Injuries; Carpal Tunnel Syndrome; Chronic Pain; Cystitis, Interstitial; Delirium; Dementia; Depressive Disorder; Diabetic Neuropathies; Dyspepsia; Epilepsies, Partial; Fibromyalgia; Head and Neck Neoplasms; Herpes Zoster; Hot Flashes; Intervertebral Disc Degeneration; Liver Cirrhosis; Lung Diseases; Neuralgia; Opioid-Related Disorders; Oropharyngeal Neoplasms; Pain; Pelvic Organ Prolapse; Postoperative Nausea and Vomiting; Pruritus; Schizophrenia; Scoliosis; Sleep Initiation and Maintenance Disorders; Tremor; Vomiting; Epilepsy; Neuralgia, Postherpetic; Restless Legs Syndrome; Seizures
Voltage-gated calcium channel modulator
Protein
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
SUBCUTANEOUS
Cardiomyopathies; Coronavirus Infections; Severe Acute Respiratory Syndrome; HIV Infections; Multiple Sclerosis, Relapsing-Remitting; Multiple Sclerosis; Neoplasms
Interferon alpha/beta receptor agonist
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
ORAL
Fasting; HIV Infections; Lecithin Cholesterol Acyltransferase Deficiency; Mental Disorders; Alcoholism; Cocaine-Related Disorders; Cognitive Dysfunction; Multiple Sclerosis, Chronic Progressive; Multiple Sclerosis, Relapsing-Remitting; Neuralgia, Postherpetic; Neurofibromatosis 1; Opioid-Related Disorders; Substance-Related Disorders; Anxiety; Dementia; Epilepsy, Absence; Feeding and Eating Disorders; Mood Disorders; Obesity; Pain; Peripheral Nervous System Diseases; Schizophrenia; Bipolar Disorder; Depressive Disorder; Epilepsies, Partial; Epilepsy; Epilepsy, Tonic-Clonic; Lennox Gastaut Syndrome; Seizures
Sodium channel alpha subunit blocker
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
ORAL
Breast Neoplasms; Neoplasms; Schizophrenia; Stress Disorders, Post-Traumatic; Alzheimer Disease; Atrial Fibrillation; Bipolar Disorder; Cerebellar Ataxia; Child Development Disorders, Pervasive; Depressive Disorder; Depressive Disorder, Major; Melanoma; Multiple Sclerosis; Multiple Sclerosis, Chronic Progressive; Muscular Atrophy, Spinal; Obsessive-Compulsive Disorder; Peripheral Nervous System Diseases; Spinal Cord Injuries; Huntington Disease; Multiple System Atrophy; Spinal Cord Diseases; Spinocerebellar Ataxias; Supranuclear Palsy, Progressive; Amyotrophic Lateral Sclerosis
Sodium channel alpha subunit blocker
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER; PEDIATRICS
ORAL
Bulimia Nervosa; Cognitive Dysfunction; Feeding and Eating Disorders; Hernias, Diaphragmatic, Congenital; HIV Infections; Liver Diseases; Alcohol Drinking; Amphetamine-Related Disorders; Brain Ischemia; Deafness; Diabetes Mellitus; Hearing Loss, Sudden; Marijuana Abuse; Multiple Sclerosis; Parkinson Disease; Sciatica; Stress Disorders, Post-Traumatic; Alcoholism; Anxiety; Bipolar Disorder; Bulimia; Cocaine-Related Disorders; Dementia; Depressive Disorder; Diabetes Mellitus, Type 2; Epilepsies, Partial; Epilepsy, Tonic-Clonic; Essential Tremor; Gambling; Headache; Hyperlipidemias; Hypertension; Hypertriglyceridemia; Metabolic Syndrome; Mood Disorders; Obesity; Obsessive-Compulsive Disorder; Pain; Prader-Willi Syndrome; Schizophrenia; Smoking Cessation; Tobacco Use Disorder; Tourette Syndrome; Epilepsy; Lennox Gastaut Syndrome; Migraine Disorders; Seizures
Carbonic anhydrase II inhibitor
Small molecule
Approved
GASTROINTESTINAL; NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
INJECTION; INTRAVENOUS
Gram-Negative Bacterial Infections; Osteomyelitis; Pancreatitis; Respiratory Insufficiency; Appendicitis; Communicable Diseases; Hematologic Neoplasms; Tuberculosis; Tuberculosis, Pulmonary; Enterobacteriaceae Infections; Lung Diseases; Mental Disorders; Neonatal Sepsis; Pneumonia; Pneumonia, Bacterial; Pneumonia, Ventilator-Associated; Pyelonephritis; Sepsis; Shock, Septic; Urinary Bladder Neoplasms; Bacteremia; Bacterial Infections; Infections; Intraabdominal Infections; Meningitis; Meningitis, Bacterial; Urinary Tract Infections
Bacterial penicillin-binding protein inhibitor
Protein
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
UNKNOWN
Stroke; Alzheimer Disease; Asthma; Colitis, Ulcerative; Crohn Disease; Multiple Organ Failure; Polyradiculoneuropathy, Chronic Inflammatory Demyelinating; Pulmonary Disease, Chronic Obstructive; Hepatitis C; Influenza, Human; Multiple Sclerosis, Relapsing-Remitting; Pneumonia; Respiratory Distress Syndrome; Severe Acute Respiratory Syndrome; Multiple Sclerosis; Neoplasms
Interferon alpha/beta receptor agonist
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
NASAL; ORAL
Migraine Disorders
Serotonin 1b (5-HT1b) receptor agonist
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
ORAL
Amyloid Neuropathies, Familial; Cocaine-Related Disorders; Executive Function; Neuroblastoma; Alcoholism; Brain Injuries; Gambling; Obsessive-Compulsive Disorder; Pick Disease of the Brain; Schizophrenia; Tobacco Use Disorder; Liver Failure; Parkinson Disease
Catechol O-methyltransferase inhibitor
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
INTRAVENOUS; ORAL
Aphasia; Canavan Disease; Essential Tremor; Lymphoma, Follicular; Stroke; Alzheimer Disease; Anemia, Sickle Cell; Bipolar Disorder; Brain Neoplasms; Cocaine-Related Disorders; Cognitive Dysfunction; Dyskinesia, Drug-Induced; Epilepsy, Absence; Epilepsy, Reflex; Glioblastoma; Leukemia, Myeloid, Acute; Neuralgia, Postherpetic; Neuroblastoma; Obsessive-Compulsive Disorder; Opioid-Related Disorders; Paraganglioma; Parkinson Disease; Polyneuropathies; Psychotic Disorders; Restless Legs Syndrome; Stress Disorders, Post-Traumatic; Torticollis; Alcoholism; Anxiety; Dementia; Depressive Disorder; Epilepsies, Partial; Movement Disorders; Panic Disorder; Schizophrenia; Status Epilepticus; Subarachnoid Hemorrhage; Substance Withdrawal Syndrome; Epilepsy; Epilepsy, Tonic-Clonic; Seizures
Synaptic vesicle glycoprotein 2A modulator
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
ORAL
Amphetamine-Related Disorders; Epilepsy; Gastrointestinal Stromal Tumors; Obesity; Cocaine-Related Disorders; Parkinson Disease
Catechol O-methyltransferase inhibitor
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER; PREGNANCY AND GYNECOLOGY
ORAL; VAGINAL
Atrophy; Menopause
Estrogen receptor agonist
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
ORAL
Sleep Wake Disorders; Anxiety; Dementia; Depressive Disorder; Schizophrenia; Sleep Initiation and Maintenance Disorders
GABA A receptor alpha-1/beta-1/gamma-2 positive allosteric modulator
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
TRANSDERMAL
Amphetamine-Related Disorders; Central Nervous System Diseases; Cocaine-Related Disorders; Down Syndrome; Substance-Related Disorders; Anxiety; Brain Injuries; Cognitive Dysfunction; Delirium; Dementia, Vascular; Depressive Disorder; Neurobehavioral Manifestations; Schizophrenia; Supranuclear Palsy, Progressive; Alzheimer Disease; Dementia; Parkinson Disease
Cholinesterases; ACHE & BCHE inhibitor
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
ORAL
Cocaine-Related Disorders; Hearing Loss, Noise-Induced; Tobacco Use Disorder; Essential Tremor; Hearing Loss; Obesity; Parkinson Disease; Alcoholism; Epilepsy, Complex Partial; Feeding and Eating Disorders; Migraine Disorders; Psychotic Disorders; Schizophrenia; Smoking Cessation; Weight Gain; Epilepsies, Partial; Epilepsy; Seizures
Sodium channel alpha subunit blocker
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER; PEDIATRICS
ORAL
Neoplasms; Multiple Sclerosis; Aggression; Anxiety; Dementia; Depressive Disorder; Epilepsies, Partial; Neuralgia; Psychomotor Agitation; Schizophrenia; Epilepsy; Seizures
Sodium channel alpha subunit blocker
Antibody
Approved
CANCER; NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
INJECTION; INTRAVENOUS
Anemia; Arthritis, Rheumatoid; Epidermolysis Bullosa; Fallopian Tube Neoplasms; Fanconi Anemia; Kidney Diseases; Leukemia, Prolymphocytic, T-Cell; Lymphohistiocytosis, Hemophagocytic; Lymphoma, Follicular; Lymphoma, Non-Hodgkin; Multiple Myeloma; Neoplasms, Neuroepithelial; Neuroblastoma; Ovarian Neoplasms; Peritoneal Neoplasms; Renal Insufficiency; Vasculitis; Anemia, Aplastic; Anemia, Hemolytic, Autoimmune; beta-Thalassemia; Crohn Disease; Diabetes Mellitus, Type 1; Graft vs Host Disease; Granulomatous Disease, Chronic; Hematologic Neoplasms; Hemoglobinopathies; Histiocytosis; Hodgkin Disease; Immune System Diseases; Kidney Failure, Chronic; Kidney Neoplasms; Leukemia, Biphenotypic, Acute; Leukemia, Erythroblastic, Acute; Leukemia, Large Granular Lymphocytic; Leukemia, Lymphoid; Leukemia, Prolymphocytic; Liver Diseases; Lymphoma, Large B-Cell, Diffuse; Mycosis Fungoides; Myeloproliferative Disorders; Myositis, Inclusion Body; Neoplasms; Osteopetrosis; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Purpura, Thrombocytopenic, Idiopathic; Severe Combined Immunodeficiency; Sezary Syndrome; Thalassemia; Waldenstrom Macroglobulinemia; Anemia, Sickle Cell; Granuloma, Lethal Midline; Immunoblastic Lymphadenopathy; Leukemia; Leukemia, Myeloid, Acute; Lymphoma; Lymphoma, T-Cell, Peripheral; Multiple Sclerosis, Relapsing-Remitting; Myelodysplastic Syndromes; Leukemia, Lymphocytic, Chronic, B-Cell; Multiple Sclerosis
CAMPATH-1 antigen inhibitor
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER; RESPIRATORY
ORAL
Astrocytoma; Depressive Disorder, Major; Glioblastoma; Head and Neck Neoplasms; Heart Failure; Muscular Dystrophies; Neoplasms; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Cushing Syndrome; Dementia, Vascular; Diabetes Mellitus, Type 2; Eisenmenger Complex; Essential Hypertension; Gastroparesis; Hypertension; Multiple Myeloma; Obesity; Pancreatic Neoplasms; Priapism; Scleroderma, Systemic; Sexual Dysfunction, Physiological; Stroke; Glucose Intolerance; Heart Defects, Congenital; Insulin Resistance; Lung Diseases, Interstitial; Muscular Dystrophy, Duchenne; Premature Ejaculation; Raynaud Disease; Transposition of Great Vessels; Erectile Dysfunction; Hypertension, Pulmonary; Prostatic Hyperplasia; Pulmonary Arterial Hypertension
Phosphodiesterase 5A inhibitor
Small molecule
Approved
EMERGENCY MEDICINE; MUSCULOSKELETAL; NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
ORAL
Carcinoma, Squamous Cell; Cough; Essential Tremor; Marijuana Abuse; Oropharyngeal Neoplasms; Pregnancy; Refractive Errors; Tobacco Use Disorder; Alcoholism; Complex Regional Pain Syndromes; Dental Anxiety; Diabetes Mellitus; Dry Eye Syndromes; Irritable Bowel Syndrome; Nausea; Pancreatitis, Chronic; Pruritus; Urinary Bladder, Overactive; Anxiety; Breast Neoplasms; Burning Mouth Syndrome; Chronic Pain; Dementia; Depressive Disorder; Diabetic Neuropathies; Epilepsies, Partial; Epilepsy, Complex Partial; Epilepsy, Tonic-Clonic; Fractures, Bone; Headache; Herpes Zoster; Intervertebral Disc Degeneration; Migraine Disorders; Mononeuropathies; Muscle Cramp; Neuralgia, Postherpetic; Neurotic Disorders; Opioid-Related Disorders; Osteoarthritis; Pain; Peripheral Nervous System Diseases; Prostatitis; Radiculopathy; Restless Legs Syndrome; Schizophrenia; Sleep Initiation and Maintenance Disorders; Anxiety Disorders; Epilepsy; Fibromyalgia; Neuralgia; Seizures; Spinal Cord Injuries
Voltage-gated calcium channel modulator
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
ORAL
Marijuana Abuse; Anxiety Disorders; Sleep Apnea, Obstructive; Sleep Initiation and Maintenance Disorders
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
ORAL
Marijuana Abuse; Burns; Migraine with Aura; Migraine without Aura; Pulmonary Disease, Chronic Obstructive; Severe Acute Respiratory Syndrome; Sleep Apnea, Obstructive; Substance-Related Disorders; Tobacco Use Disorder; Bipolar Disorder; Depressive Disorder; Sleep Wake Disorders; Sleep Initiation and Maintenance Disorders
Melatonin receptor agonist
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER; PEDIATRICS
ORAL
Neuralgia; Epilepsy; Dementia; Depressive Disorder; Epilepsia Partialis Continua; Low Back Pain; Pain; Schizophrenia; Anxiety; Lennox Gastaut Syndrome; Seizures
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
ORAL
Obsessive-Compulsive Disorder; Anxiety; Autistic Disorder; Bipolar Disorder; Dementia; Depressive Disorder; Mood Disorders; Psychotic Disorders; Schizophrenia
Dopamine D2 receptor antagonist
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
TRANSDERMAL
Alzheimer Disease; Fibromyalgia; Stroke; Substance-Related Disorders; Parkinson Disease; Restless Legs Syndrome
D2-like dopamine receptor agonist
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
ORAL
Carcinoma, Non-Small-Cell Lung; Head and Neck Neoplasms; Esophageal Neoplasms; Glioma; Multiple Sclerosis; Neoplasms; Schizophrenia; Sleep Initiation and Maintenance Disorders; Stroke; Brain Injuries; Depressive Disorder; Disorders of Excessive Somnolence; Fatigue; Obesity; Sleep Apnea Syndromes; Attention Deficit Disorder with Hyperactivity; Narcolepsy; Sleep Apnea, Obstructive; Sleep Wake Disorders
Dopamine transporter inhibitor
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER; PEDIATRICS
ORAL
Pain; Epilepsy; Lennox Gastaut Syndrome; Seizures
Sodium channel alpha subunit blocker
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM
TOPICAL
Amyotrophic Lateral Sclerosis; Brain Injuries; Cough; Migraine Disorders; Pruritus; Stroke; Cardiovascular Diseases; Facial Pain; HIV Infections; Hypertension, Pulmonary; Morton Neuroma; Myofascial Pain Syndromes; Nausea; Neuralgia, Postherpetic; Neuroma; Tennis Elbow; Vomiting; Angina, Stable; Breast Neoplasms; Common Cold; Diabetic Neuropathies; Head and Neck Neoplasms; Herpes Zoster; Osteoarthritis, Knee; Peripheral Nervous System Diseases; Arthralgia; Arthritis; Back Pain; Bursitis; Contusions; Muscle Cramp; Myalgia; Neuralgia; Osteoarthritis; Pain; Sprains and Strains; Tendinopathy
Vanilloid receptor opener
Enzyme
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
INTRAVENOUS
Gaucher Disease
Glucocerebroside hydrolytic enzyme