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Total: 31
Small molecule
Approved
CANCER; MUSCULOSKELETAL; OTHER; PREGNANCY AND GYNECOLOGY
INJECTION; ORAL; TOPICAL; VAGINAL
Memory; Reperfusion Injury; Brain Injuries; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Shock; Urinary Bladder, Overactive; Alzheimer Disease; Angina, Unstable; Anorexia Nervosa; Bone Diseases; Bone Diseases, Metabolic; Cardiovascular Diseases; Colonic Neoplasms; Coronary Disease; Cystitis, Interstitial; Diabetes Mellitus; Endometrial Neoplasms; Heart Diseases; Hot Flashes; Hypercholesterolemia; Hypertension; Lupus Erythematosus, Systemic; Memory Disorders; Myocardial Infarction; Myocardial Ischemia; Stroke; Thrombosis; Turner Syndrome; Atrophic Vaginitis; Atrophy; Breast Neoplasms; Dyspareunia; Hypogonadism; Menopause; Osteoporosis; Osteoporosis, Postmenopausal; Primary Ovarian Insufficiency
Estrogen receptor agonist
Small molecule
Approved
DERMATOLOGY; IMMUNE SYSTEM; OTHER; PREGNANCY AND GYNECOLOGY
INJECTION; ORAL; TOPICAL; VAGINAL
Central Serous Chorioretinopathy; Cholangitis, Sclerosing; Osteomyelitis; Periapical Periodontitis; Pouchitis; Prostatic Neoplasms, Castration-Resistant; Appendicitis; Brain Diseases; Carcinoma, Non-Small-Cell Lung; Clostridium Infections; Colitis, Ulcerative; Giardiasis; Leukemia, Lymphocytic, Chronic, B-Cell; Lichen Planus, Oral; Malnutrition; Pancreatic Neoplasms; Periodontal Diseases; Pilonidal Sinus; Rectal Neoplasms; Tuberculosis; Tuberculosis, Multidrug-Resistant; Uterine Cervical Neoplasms; Abscess; Blepharitis; Candidiasis; Colorectal Neoplasms; Crohn Disease; Diarrhea; Enterocolitis, Pseudomembranous; Fecal Incontinence; Gingivitis; Helicobacter Infections; Hemorrhoids; Hidradenitis Suppurativa; HIV Infections; Lymphoma, Non-Hodgkin; Mycoses; Pain; Pelvic Inflammatory Disease; Periodontitis; Skin Diseases; Trichomonas Vaginitis; Vaginal Discharge; Vaginitis; Amebiasis; Bacterial Infections; Duodenal Ulcer; Infections; Intraabdominal Infections; Pneumonia; Rosacea; Sepsis; Trichomonas Infections; Uterine Cervicitis; Vaginosis, Bacterial
DNA inhibitor
Small molecule
Approved
IMMUNE SYSTEM; PREGNANCY AND GYNECOLOGY
BUCCAL; INJECTION
Intertrigo; Stomatitis; HIV Infections; Otomycosis; Infections; Mycoses; Pruritus; Tinea; Tinea Pedis
Cytochrome P450 51 inhibitor
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; MUSCULOSKELETAL; OTHER; PREGNANCY AND GYNECOLOGY; RHEUMATOLOGY
ORAL; TOPICAL; TRANSDERMAL; VAGINAL
Blood Coagulation Disorders; Cerebral Arterial Diseases; Diabetes Mellitus; Diabetes Mellitus, Type 1; Diabetes Mellitus, Type 2; Polycystic Ovary Syndrome; Aging; Alzheimer Disease; Atherosclerosis; Bulimia Nervosa; Carcinoid Tumor; Depression, Postpartum; Depressive Disorder; Dry Eye Syndromes; Hereditary Breast and Ovarian Cancer Syndrome; HIV Infections; Migraine Disorders; Prostatic Neoplasms; Psychotic Disorders; Schizophrenia; Severe Acute Respiratory Syndrome; Triple Negative Breast Neoplasms; Urinary Tract Infections; Amenorrhea; Anorexia Nervosa; Bone Diseases, Metabolic; Coronary Disease; Dysmenorrhea; Endometriosis; Heart Diseases; Hot Flashes; Infertility; Multiple Sclerosis; Myocardial Ischemia; Non-alcoholic Fatty Liver Disease; Obesity; Pain; Prostatic Neoplasms, Castration-Resistant; Sexual Dysfunction, Physiological; Stress Disorders, Post-Traumatic; Turner Syndrome; Atrophic Vaginitis; Atrophy; Breast Neoplasms; Dyspareunia; Hypogonadism; Menopause; Osteoporosis; Osteoporosis, Postmenopausal; Primary Ovarian Insufficiency
Estrogen receptor alpha agonist
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER; PREGNANCY AND GYNECOLOGY
INJECTION; INTRAUTERINE; ORAL; VAGINAL
Amphetamine-Related Disorders; Gliosarcoma; Anorexia Nervosa; Bulimia Nervosa; Cocaine-Related Disorders; Depression, Postpartum; Depressive Disorder; Endometrial Neoplasms; HIV Infections; Marijuana Abuse; Orthostatic Intolerance; Placenta Previa; Polycystic Ovary Syndrome; Pre-Eclampsia; Severe Acute Respiratory Syndrome; Tobacco Use Disorder; Uterine Cervical Dysplasia; Vulvar Lichen Sclerosus; Alzheimer Disease; Angina, Unstable; Bone Diseases; Bone Diseases, Metabolic; Brain Injuries; Breast Neoplasms; Cardiovascular Diseases; Coronary Disease; Diabetes Mellitus; Epilepsy; Hypercholesterolemia; Hypertension; Infertility; Infertility, Female; Leiomyoma; Memory Disorders; Menopause; Myocardial Ischemia; Osteoporosis; Ovarian Hyperstimulation Syndrome; Ovarian Neoplasms; Pregnancy; Premature Birth; Thrombosis; Amenorrhea; Endometrial Hyperplasia; Uterine Hemorrhage
Progesterone receptor agonist
Protein
Approved
MUSCULOSKELETAL; OTHER; PREGNANCY AND GYNECOLOGY
INJECTION; NASAL
Bone Diseases, Metabolic; Menopause; Osteoporosis; Bone Resorption; Hypercalcemia; Osteitis Deformans; Osteoporosis, Postmenopausal; Parathyroid Diseases
Calcitonin receptor agonist
Small molecule
Approved
OTHER; PREGNANCY AND GYNECOLOGY
IMPLANTATION; INTRAUTERINE; ORAL
Diabetes Mellitus; Diabetes Mellitus, Type 2; Hepatitis B, Chronic; Hepatitis C, Chronic; Leukemia, Lymphocytic, Chronic, B-Cell; Neoplasms; Non-alcoholic Fatty Liver Disease; Adenomyosis; Endometrial Neoplasms; HIV Infections; Ovarian Neoplasms; Pain; Pregnancy; Anorexia Nervosa; Bone Diseases, Metabolic; Dysmenorrhea; Endometriosis; Hemorrhage; Migraine Disorders; Menorrhagia
Progesterone receptor agonist
Small molecule
Approved
OTHER; PREGNANCY AND GYNECOLOGY
VAGINAL
Candidiasis, Vulvovaginal; Vaginitis; Vulvovaginitis
Cytochrome P450 51 inhibitor
Small molecule
Approved
OTHER; PREGNANCY AND GYNECOLOGY
INJECTION; INTRAVENOUS; ORAL
Back Pain; Hypotension; Liver Cirrhosis; Skin Neoplasms; Spinal Cord Neoplasms; Cerebral Hemorrhage; Epistaxis; Intervertebral Disc Degeneration; Osteoarthritis, Knee; Shock, Septic; Subarachnoid Hemorrhage; Urinary Bladder Neoplasms; Anemia; Angioedemas, Hereditary; Aortic Aneurysm, Abdominal; Astrocytoma; Blood Coagulation Disorders; Bone Neoplasms; Brain Injuries; Brain Neoplasms; Burns; Coronary Disease; Femoral Neck Fractures; Fractures, Bone; Gastrointestinal Hemorrhage; Genital Neoplasms, Female; Head and Neck Neoplasms; Hematologic Neoplasms; Hematoma; Hematoma, Subdural, Intracranial; Hemoptysis; Hip Fractures; Ileus; Inflammation; Joint Diseases; Leiomyoma; Melanoma; Melanosis; Meningioma; Nasal Polyps; Neoplasms; Osteoarthritis; Pain; Paraganglioma; Pelvic Organ Prolapse; Placenta Accreta; Placenta Previa; Postpartum Hemorrhage; Prostatic Neoplasms, Castration-Resistant; Scoliosis; Sepsis; Severe Acute Respiratory Syndrome; Shock; Shoulder Impingement Syndrome; Telangiectasia, Hereditary Hemorrhagic; Thrombocytopenia; von Willebrand Diseases; Wounds and Injuries; Hemophilia A; Hemorrhage; Menorrhagia
Plasminogen inhibitor
Small molecule
Approved
ENT; EYE; OTHER; PEDIATRICS; PREGNANCY AND GYNECOLOGY
INJECTION; OPHTHALMIC; ORAL; OTIC
Hearing Loss; Osteomyelitis; Conjunctivitis, Bacterial; Diabetic Foot; Glaucoma; Glaucoma, Open-Angle; Ocular Hypertension; Otitis Media; Pelvic Inflammatory Disease; Urinary Tract Infections; Acne Vulgaris; Bacterial Infections; Bronchitis, Chronic; Corneal Ulcer; Eye Infections; Infections; Otitis Externa
Bacterial DNA gyrase inhibitor
Small molecule
Approved
CANCER; OTHER; PREGNANCY AND GYNECOLOGY
INJECTION; INTRAVENOUS
Breast Neoplasms, Male; Carcinoma, Endometrioid; Carcinoma, Renal Cell; Colonic Neoplasms; Cystadenoma, Serous; Digestive System Diseases; Lymphoma; Multiple Myeloma; Myelodysplastic Syndromes; Myeloproliferative Disorders; Nausea; Neoplasms, Plasma Cell; Sarcoma, Synovial; Vaginal Neoplasms; Vulvar Neoplasms; Biliary Tract Neoplasms; Carcinoma, Hepatocellular; Carcinoma, Intraductal, Noninfiltrating; Carcinoma, Large Cell; Carcinoma, Neuroendocrine; Carcinoma, Ovarian Epithelial; Carcinoma, Transitional Cell; Colorectal Neoplasms; Gastrointestinal Stromal Tumors; Hereditary Breast and Ovarian Cancer Syndrome; Leiomyosarcoma; Leukemia; Liver Neoplasms; Mediastinal Neoplasms; Melanoma; Osteosarcoma; Pancreatic Neoplasms; Penile Neoplasms; Retroviridae Infections; Salivary Gland Neoplasms; Sarcoma, Ewing; Small Cell Lung Carcinoma; Testicular Neoplasms; Thyroid Carcinoma, Anaplastic; Tonsillar Neoplasms; Triple Negative Breast Neoplasms; Urethral Neoplasms; Uterine Neoplasms; Adenocarcinoma of Lung; Anorexia; Cachexia; Carcinoma; Carcinoma, Squamous Cell; Endometrial Neoplasms; Esophageal Neoplasms; Fallopian Tube Neoplasms; Fatigue; Genital Neoplasms, Male; Hypersensitivity; Hypopharyngeal Neoplasms; Inflammatory Breast Neoplasms; Kidney Neoplasms; Laryngeal Neoplasms; Lung Neoplasms; Mouth Neoplasms; Nasopharyngeal Carcinoma; Nasopharyngeal Neoplasms; Neoplasm Metastasis; Neutropenia; Oropharyngeal Neoplasms; Ovarian Neoplasms; Paranasal Sinus Neoplasms; Peritoneal Neoplasms; Pharyngeal Neoplasms; Prostatic Neoplasms, Castration-Resistant; Sarcoma; Squamous Cell Carcinoma of Head and Neck; Urinary Bladder Neoplasms; Urogenital Neoplasms; Uterine Cervical Neoplasms; Adenocarcinoma; Breast Neoplasms; Carcinoma, Non-Small-Cell Lung; Head and Neck Neoplasms; Neoplasms; Prostatic Neoplasms; Stomach Neoplasms
Tubulin inhibitor
Small molecule
Approved
OTHER; PREGNANCY AND GYNECOLOGY
ORAL
Brain Neoplasms; Carcinoma, Endometrioid; Carcinoma, Non-Small-Cell Lung; Leiomyoma; Lymphoma, Non-Hodgkin; Mesothelioma; Pregnancy, Ectopic; Adenomyosis; Anovulation; Carcinoma; Carcinoma, Lobular; Dwarfism; Endometriosis; Fallopian Tube Neoplasms; Hemangiosarcoma; Hermanski-Pudlak Syndrome; Infertility, Male; Inflammatory Breast Neoplasms; Leiomyosarcoma; Liver Neoplasms; Lymphangioleiomyomatosis; Peritoneal Neoplasms; Triple Negative Breast Neoplasms; Uterine Cervical Neoplasms; Uterine Neoplasms; Abortion, Spontaneous; Azoospermia; Carcinoma, Intraductal, Noninfiltrating; Endometrial Neoplasms; Follicular Cyst; Hereditary Breast and Ovarian Cancer Syndrome; Hypogonadism; Infertility; Menopause; Neoplasm Metastasis; Osteoporosis; Ovarian Hyperstimulation Syndrome; Ovarian Neoplasms; Polycystic Ovary Syndrome; Pregnancy; Breast Neoplasms; Neoplasms
Cytochrome P450 19A1 inhibitor
Small molecule
Approved
OTHER; PREGNANCY AND GYNECOLOGY
ORAL
Prostatic Neoplasms, Castration-Resistant; Sleep Apnea, Obstructive; Alzheimer Disease; HIV Infections; Neuralgia; Albuminuria; Diabetes Mellitus, Type 2; Diabetic Nephropathies; Essential Hypertension; Heart Diseases; Kidney Diseases; Kidney Failure, Chronic; Lipid Metabolism Disorders; Polycystic Kidney Diseases; Severe Acute Respiratory Syndrome; Cardiovascular Diseases; Diabetes Mellitus; Hypertension; Myocardial Infarction; Stroke
Type-1 angiotensin II receptor antagonist
Antibody
Approved
PREGNANCY AND GYNECOLOGY
INTRAVENOUS
Adenocarcinoma, Follicular; Adrenal Cortex Neoplasms; Anus Neoplasms; Appendiceal Neoplasms; Breast Diseases; Carcinoid Tumor; Carcinoma, Ovarian Epithelial; Carcinoma, Renal Cell; Ependymoma; Fallopian Tube Neoplasms; Hodgkin Disease; Insulinoma; Lymphoma, Non-Hodgkin; Lymphoma, T-Cell, Cutaneous; Mycosis Fungoides; Oropharyngeal Neoplasms; Parathyroid Neoplasms; Pericardial Effusion; Peritoneal Neoplasms; Pleural Effusion; Skin Diseases; Somatostatinoma; Testicular Neoplasms; Thyroid Neoplasms; Uterine Cervical Neoplasms; Vaginal Neoplasms; Vulvar Neoplasms; Adenocarcinoma; Bile Duct Neoplasms; Carcinoma; Carcinoma, Ductal; Carcinoma, Non-Small-Cell Lung; Cholangiocarcinoma; Colonic Neoplasms; Digestive System Neoplasms; Endometrial Neoplasms; Gallbladder Neoplasms; Head and Neck Neoplasms; Hemangiosarcoma; Hematologic Neoplasms; Leukemia; Leukemia, Myeloid, Acute; Lung Neoplasms; Neoplasm Metastasis; Osteosarcoma; Ovarian Neoplasms; Pancreatic Neoplasms; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Salivary Gland Neoplasms; Sarcoma; Squamous Cell Carcinoma of Head and Neck; Triple Negative Breast Neoplasms; Urethral Neoplasms; Urinary Bladder Neoplasms; Urogenital Neoplasms; Biliary Tract Neoplasms; Brain Diseases; Breast Neoplasms, Male; Carcinoma, Intraductal, Noninfiltrating; Colorectal Neoplasms; Esophageal Neoplasms; Inflammatory Breast Neoplasms; Breast Neoplasms; Neoplasms; Stomach Neoplasms
Receptor protein-tyrosine kinase erbB-2 inhibitor
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER; PREGNANCY AND GYNECOLOGY
ORAL; VAGINAL
Atrophy; Menopause
Estrogen receptor agonist
Protein
Approved
OTHER; PREGNANCY AND GYNECOLOGY
INJECTION
Arthritis, Rheumatoid; Endometriosis; Infertility; Ovarian Hyperstimulation Syndrome; Prostatic Hyperplasia
Unknown
Small molecule
Approved
OTHER; PREGNANCY AND GYNECOLOGY
ORAL
Osteoarthritis, Knee; Pancreatitis; Pain; Pharyngitis; Arthritis, Rheumatoid; Dysmenorrhea; Osteoarthritis; Rheumatic Diseases
Cyclooxygenase-2 inhibitor
Antibody
Approved
MUSCULOSKELETAL; PREGNANCY AND GYNECOLOGY
SUBCUTANEOUS
Crohn Disease; Kidney Diseases; Ovarian Neoplasms; Aortic Valve Stenosis; Carcinoma, Non-Small-Cell Lung; Colorectal Neoplasms; Fibrous Dysplasia of Bone; Gout; Histiocytosis, Langerhans-Cell; Hypersensitivity; Infertility, Male; Inflammatory Breast Neoplasms; Melanoma; Multiple Myeloma; Neoplasms; Osteoarthritis, Hip; Osteolysis; Osteosarcoma; Thyroid Neoplasms; Anorexia Nervosa; Arthritis, Rheumatoid; Bone Diseases, Metabolic; Carcinoma; Carcinoma, Renal Cell; Diabetes Mellitus; Fractures, Bone; Lung Neoplasms; Osteogenesis Imperfecta; Prostatic Neoplasms, Castration-Resistant; Bone Diseases; Bone Resorption; Breast Neoplasms; Giant Cell Tumor of Bone; Giant Cell Tumors; Hypercalcemia; Neoplasm Metastasis; Neoplasms, Bone Tissue; Osteoporosis; Osteoporosis, Postmenopausal
Tumor necrosis factor ligand superfamily member 11 inhibitor
Small molecule
Approved
PREGNANCY AND GYNECOLOGY
ORAL
Adenomyosis; Breast Neoplasms; Charcot-Marie-Tooth Disease; Depressive Disorder; Menopause; Premenstrual Syndrome; Hemorrhage; Contraception, Postcoital; Leiomyoma
Progesterone receptor modulator
Antibody
Approved
PREGNANCY AND GYNECOLOGY
SINGLE-USE
Breast Diseases; Breast Neoplasms, Male; Colonic Neoplasms; Rectal Neoplasms; Carcinoma, Neuroendocrine; Carcinoma, Non-Small-Cell Lung; Colorectal Neoplasms; Fallopian Tube Neoplasms; Hemangiosarcoma; Hematologic Neoplasms; Neoplasm Metastasis; Pancreatic Neoplasms; Peritoneal Neoplasms; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Esophageal Neoplasms; Inflammatory Breast Neoplasms; Ovarian Neoplasms; Stomach Neoplasms; Breast Neoplasms; Neoplasms
Receptor protein-tyrosine kinase erbB-2 inhibitor
Small molecule
Approved
PREGNANCY AND GYNECOLOGY
ORAL
Paget Disease, Extramammary; Atrophic Vaginitis; Atrophy; Dyspareunia; Menopause
Estrogen receptor modulator
Combination
Approved
OTHER; PREGNANCY AND GYNECOLOGY
ORAL; ORAL-21; ORAL-28
Unknown
Unknown
Combination
Approved
OTHER; PREGNANCY AND GYNECOLOGY
ORAL; ORAL-21; ORAL-28
Unknown
Unknown
Combination
Approved
PREGNANCY AND GYNECOLOGY
ORAL
Unknown
Unknown
Combination
Approved
OTHER; PREGNANCY AND GYNECOLOGY
ORAL
Unknown
Unknown
Combination
Approved
OTHER; PREGNANCY AND GYNECOLOGY
ORAL; ORAL-28
Unknown
Unknown
Combination
Approved
DIABETES DRUGS & ENDOCRINOLOGY; MUSCULOSKELETAL; OTHER; PREGNANCY AND GYNECOLOGY
ORAL-28
Unknown
Unknown
Combination
Approved
PREGNANCY AND GYNECOLOGY
VAGINAL
Unknown
Unknown
Combination
Approved
PREGNANCY AND GYNECOLOGY
ORAL
Unknown
Unknown
Combination
Approved
MUSCULOSKELETAL; OTHER; PREGNANCY AND GYNECOLOGY
ORAL; ORAL-21; ORAL-28
Unknown
Unknown
Small molecule
Approved
OTHER; PREGNANCY AND GYNECOLOGY
INJECTION
Unknown
Unknown