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Total: 61
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER; RHEUMATOLOGY
ORAL
Glioblastoma; Hypertension, Pulmonary; Intestinal Obstruction; Leukemia, Myeloid, Acute; Nausea; Osteomyelitis; Paraganglioma; Cholangitis, Sclerosing; Peripheral Nervous System Diseases; Premature Birth; Spondylitis, Ankylosing; Arthritis, Psoriatic; Arthritis, Juvenile; Arthritis, Rheumatoid; Colitis, Ulcerative
Arachidonate 5-lipoxygenase inhibitor
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY
ORAL
Alzheimer Disease; Depression; Depressive Disorder; Depressive Disorder, Major
Monoamine oxidase inhibitor
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Diabetes Mellitus; Lecithin Cholesterol Acyltransferase Deficiency; Metabolic Syndrome; Photosensitivity Disorders; Diabetic Nephropathies; Kidney Diseases; Atherosclerosis; Coronary Disease; Death, Sudden, Cardiac; Diabetes Mellitus, Type 2; Essential Hypertension; Hypercholesterolemia; Kidney Calculi; Polycystic Kidney, Autosomal Dominant; Pre-Eclampsia; Angina Pectoris; Cardiovascular Diseases; Edema; Glomerulonephritis; Heart Failure; Hypertension; Kidney Failure, Chronic; Liver Cirrhosis; Myocardial Infarction; Nephrotic Syndrome; Toxemia
Thiazide-sensitive sodium-chloride cotransporter inhibitor
Small molecule
Approved
CARDIOVASCULAR; DIABETES DRUGS & ENDOCRINOLOGY; OTHER
BUCCAL; IMPLANTATION; INJECTION; NASAL; TRANSDERMAL
Aging; Cerebral Arterial Diseases; Dyspareunia; Insulin Resistance; Kallmann Syndrome; Pain; Penile Induration; Polycystic Ovary Syndrome; Acquired Immunodeficiency Syndrome; Anorexia Nervosa; Carcinoma, Intraductal, Noninfiltrating; Dwarfism; Heart Failure; Hereditary Breast and Ovarian Cancer Syndrome; Multiple Sclerosis; Muscle Weakness; Obesity; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Sarcopenia; Spinal Cord Injuries; Testicular Neoplasms; Coronary Disease; Disorders of Sex Development; Erectile Dysfunction; Hip Fractures; Infertility; Kidney Failure, Chronic; Menopause; Metabolic Syndrome; Hypogonadism; Klinefelter Syndrome; Neoplasms; Orchitis; Sexual Dysfunctions, Psychological
Androgen Receptor agonist
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER
INJECTION; INTRAMUSCULAR; SUBCUTANEOUS
Pregnancy; Premature Birth
Progesterone receptor agonist
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; MUSCULOSKELETAL; OTHER; PREGNANCY AND GYNECOLOGY; RHEUMATOLOGY
ORAL; TOPICAL; TRANSDERMAL; VAGINAL
Blood Coagulation Disorders; Cerebral Arterial Diseases; Diabetes Mellitus; Diabetes Mellitus, Type 1; Diabetes Mellitus, Type 2; Polycystic Ovary Syndrome; Aging; Alzheimer Disease; Atherosclerosis; Bulimia Nervosa; Carcinoid Tumor; Depression, Postpartum; Depressive Disorder; Dry Eye Syndromes; Hereditary Breast and Ovarian Cancer Syndrome; HIV Infections; Migraine Disorders; Prostatic Neoplasms; Psychotic Disorders; Schizophrenia; Severe Acute Respiratory Syndrome; Triple Negative Breast Neoplasms; Urinary Tract Infections; Amenorrhea; Anorexia Nervosa; Bone Diseases, Metabolic; Coronary Disease; Dysmenorrhea; Endometriosis; Heart Diseases; Hot Flashes; Infertility; Multiple Sclerosis; Myocardial Ischemia; Non-alcoholic Fatty Liver Disease; Obesity; Pain; Prostatic Neoplasms, Castration-Resistant; Sexual Dysfunction, Physiological; Stress Disorders, Post-Traumatic; Turner Syndrome; Atrophic Vaginitis; Atrophy; Breast Neoplasms; Dyspareunia; Hypogonadism; Menopause; Osteoporosis; Osteoporosis, Postmenopausal; Primary Ovarian Insufficiency
Estrogen receptor alpha agonist
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER; PREGNANCY AND GYNECOLOGY
INJECTION; INTRAUTERINE; ORAL; VAGINAL
Amphetamine-Related Disorders; Gliosarcoma; Anorexia Nervosa; Bulimia Nervosa; Cocaine-Related Disorders; Depression, Postpartum; Depressive Disorder; Endometrial Neoplasms; HIV Infections; Marijuana Abuse; Orthostatic Intolerance; Placenta Previa; Polycystic Ovary Syndrome; Pre-Eclampsia; Severe Acute Respiratory Syndrome; Tobacco Use Disorder; Uterine Cervical Dysplasia; Vulvar Lichen Sclerosus; Alzheimer Disease; Angina, Unstable; Bone Diseases; Bone Diseases, Metabolic; Brain Injuries; Breast Neoplasms; Cardiovascular Diseases; Coronary Disease; Diabetes Mellitus; Epilepsy; Hypercholesterolemia; Hypertension; Infertility; Infertility, Female; Leiomyoma; Memory Disorders; Menopause; Myocardial Ischemia; Osteoporosis; Ovarian Hyperstimulation Syndrome; Ovarian Neoplasms; Pregnancy; Premature Birth; Thrombosis; Amenorrhea; Endometrial Hyperplasia; Uterine Hemorrhage
Progesterone receptor agonist
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER
INJECTION; INTRACRANIAL
Hereditary Breast and Ovarian Cancer Syndrome; Leukemia, Plasma Cell; Lymphoma, T-Cell, Cutaneous; Mycosis Fungoides; Neuroblastoma; Sezary Syndrome; Brain Neoplasms; Colorectal Neoplasms; Gliosarcoma; Graft vs Host Disease; Hematologic Diseases; Leukemia, Lymphocytic, Chronic, B-Cell; Lymphoma, T-Cell, Peripheral; Melanoma; Multiple Sclerosis, Relapsing-Remitting; Myasthenia Gravis; Neoplasms, Plasma Cell; Neuromyelitis Optica; Opsoclonus-Myoclonus Syndrome; Ovarian Neoplasms; Polyradiculoneuropathy, Chronic Inflammatory Demyelinating; Prostatic Neoplasms, Castration-Resistant; Sarcoma; Stiff-Person Syndrome; Breast Neoplasms; Central Nervous System Neoplasms; Leukemia; Lymphoma; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Oligodendroglioma; Paraganglioma; Astrocytoma; Ependymoma; Glioblastoma; Glioma; Hodgkin Disease; Lymphoma, Non-Hodgkin; Medulloblastoma; Multiple Myeloma; Neoplasms
DNA inhibitor
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; MUSCULOSKELETAL; OTHER
ORAL
Atrophy; Breast Neoplasms; Hypogonadism; Menopause; Primary Ovarian Insufficiency
Estrogen receptor agonist
Small molecule
Approved
CARDIOVASCULAR; DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Diabetes Mellitus, Type 2; Glioblastoma; Hypertension, Pulmonary; Neoplasms; Primary Myelofibrosis; Heart Diseases; Pneumonia; Diabetes Mellitus, Type 1; Essential Hypertension; Severe Acute Respiratory Syndrome; Cardiovascular Diseases; Collagen Diseases; Diabetic Nephropathies; Diabetic Retinopathy; Heart Failure; Hypertension; Myocardial Infarction; Renal Insufficiency; Ventricular Dysfunction, Left
Angiotensin-converting enzyme inhibitor
Small molecule
Approved
CARDIOVASCULAR; DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Depressive Disorder; Depressive Disorder, Major; Cardiovascular Diseases
Beta-1 adrenergic receptor partial agonist
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; HEMATOLOGY; OTHER
ORAL
Angina, Stable; Ischemic Stroke; Spinal Cord Injuries; Brain Injuries; Diabetes Mellitus, Type 1; Stroke; Diabetes, Gestational; Diabetes Mellitus; Diabetes Mellitus, Type 2
Sulfonylurea receptor 1, Kir6.2 blocker
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Pancreatic Neoplasms; Atherosclerosis; Renal Insufficiency, Chronic; Diabetes Mellitus; Diabetes Mellitus, Type 2
Sulfonylurea receptor 1, Kir6.2 blocker
Protein
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER; PEDIATRICS
INJECTION
Unknown
Growth hormone-releasing hormone receptor agonist
Protein
Approved
DIABETES DRUGS & ENDOCRINOLOGY; HEMATOLOGY; OTHER
UNKNOWN
Adenocarcinoma; Anemia, Refractory, with Excess of Blasts; Carcinoma, Pancreatic Ductal; Hepatitis B, Chronic; Leukemia, Plasma Cell; Liver Neoplasms; Neoplasm Metastasis; Parkinson Disease; Periodontitis; Sepsis; Alzheimer Disease; Biliary Tract Neoplasms; Brain Neoplasms; Breast Neoplasms, Male; Carcinoma, Endometrioid; Carcinoma, Intraductal, Noninfiltrating; Carcinoma, Non-Small-Cell Lung; Carcinoma, Renal Cell; Carcinoma, Squamous Cell; Central Nervous System Neoplasms; Colorectal Neoplasms; Cystadenoma, Serous; Down Syndrome; Esophageal Neoplasms; Fallopian Tube Neoplasms; Gallbladder Neoplasms; Glioblastoma; Gliosarcoma; Hematologic Neoplasms; HIV Infections; Hodgkin Disease; Inflammatory Breast Neoplasms; Kidney Diseases; Kidney Neoplasms; Leishmaniasis, Cutaneous; Leukemia, Lymphocytic, Chronic, B-Cell; Lung Neoplasms; Lymphoma, Follicular; Myelodysplastic-Myeloproliferative Diseases; Myeloproliferative Disorders; Neoplasms, Plasma Cell; Osteosarcoma; Ovarian Neoplasms; Peritoneal Neoplasms; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Pulmonary Alveolar Proteinosis; Severe Acute Respiratory Syndrome; Squamous Cell Carcinoma of Head and Neck; Stomach Neoplasms; Triple Negative Breast Neoplasms; Breast Neoplasms; Crohn Disease; Cytomegalovirus Retinitis; Ganglioneuroblastoma; Infections; Leukemia; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Lymphoma; Lymphoma, Non-Hodgkin; Melanoma; Multiple Myeloma; Myelodysplastic Syndromes; Neuroblastoma; Pancreatic Neoplasms; Rhabdomyosarcoma; Sarcoma; Urinary Bladder Neoplasms; Uveal Melanoma; Leukemia, Myeloid, Acute; Neoplasms
Granulocyte-macrophage colony-stimulating factor receptor agonist
Protein
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER; PEDIATRICS
INJECTION; SUBCUTANEOUS
Prostatic Neoplasms
Gonadotropin-releasing hormone receptor agonist
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; MUSCULOSKELETAL; OTHER; RHEUMATOLOGY
ORAL
Lecithin Cholesterol Acyltransferase Deficiency; Carcinoma, Hepatocellular; Pancreatic Neoplasms; Colorectal Neoplasms; Muscular Diseases; Pain; Sprains and Strains; Acute Pain; Arthritis, Juvenile; Arthritis, Rheumatoid; Osteoarthritis; Rheumatic Diseases
Cyclooxygenase-2 inhibitor
Small molecule
Approved
DERMATOLOGY; DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Hyperplasia; Hypogonadism; Acne Vulgaris; Carcinoma, Non-Small-Cell Lung; Prostatic Neoplasms, Castration-Resistant; Retinal Diseases; Alopecia; Prostatic Hyperplasia; Prostatic Neoplasms
Steroid 5-alpha-reductase 2 inhibitor
Small molecule
Approved
CARDIOVASCULAR; DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Cholangitis, Sclerosing; Alcoholism; Burns; Diabetic Nephropathies; HIV Infections; Huntington Disease; Inflammatory Bowel Diseases; Metabolic Syndrome; Multiple Myeloma; Non-alcoholic Fatty Liver Disease; Obesity; Atherosclerosis; Coronary Disease; Diabetic Retinopathy; Hyperlipidemia, Familial Combined; Hyperlipidemias; Hyperlipoproteinemias; Hyperlipoproteinemia Type III; Hypertension; Hypertriglyceridemia; Lipid Metabolism Disorders; Lipodystrophy; Liver Cirrhosis, Biliary; Metabolic Diseases; Cardiovascular Diseases; Diabetes Mellitus; Diabetes Mellitus, Type 2; Dyslipidemias; Hypercholesterolemia; Hypothyroidism
Peroxisome proliferator-activated receptor alpha agonist
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER; PEDIATRICS
ORAL
Acidosis, Lactic; Acquired Immunodeficiency Syndrome; AIDS-Associated Nephropathy; AIDS Dementia Complex; HIV Infections; Virus Diseases
Human immunodeficiency virus type 1 reverse transcriptase inhibitor
Small molecule
Approved
DERMATOLOGY; DIABETES DRUGS & ENDOCRINOLOGY; OTHER; UROLOGY AND KIDNEY
INJECTION; ORAL; TOPICAL
Hematologic Neoplasms; Anemia, Aplastic; Anemia, Sickle Cell; Graft vs Host Disease; Lichen Planus, Oral; Thalassemia; Conjunctivitis, Allergic; Keratoconjunctivitis; Delayed Graft Function; Dermatitis, Atopic; Eczema; Immune System Diseases; Kidney Transplantation; Liver Transplantation
FK506-binding protein 1A inhibitor
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Hypotension, Orthostatic; Nesidioblastosis; Obesity; Aging; Kidney Neoplasms; Non-alcoholic Fatty Liver Disease; Atherosclerosis; Coronary Disease; Diabetes, Gestational; Hypercholesterolemia; Hypertension; Metabolic Diseases; Metabolic Syndrome; Diabetes Mellitus; Diabetes Mellitus, Type 2
Maltase-glucoamylase inhibitor
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Atherosclerosis; Coronary Disease; Hypercholesterolemia; Hypertension; Diabetes Mellitus; Diabetes Mellitus, Type 2
Sulfonylurea receptor 1, Kir6.2 blocker
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER
INJECTION
Chordoma; Fanconi Anemia; Kidney Neoplasms; Leukemia, Myeloid, Acute; Liver Neoplasms; Mesothelioma; Myeloproliferative Disorders; Neoplasms; Neoplasms, Germ Cell and Embryonal; Neoplasms, Plasma Cell; Neuroblastoma; Retinoblastoma; Breast Neoplasms; Central Nervous System Neoplasms; Colorectal Neoplasms; Endometrial Neoplasms; Fallopian Tube Neoplasms; Hodgkin Disease; Leukemia; Lymphoma; Lymphoma, Non-Hodgkin; Myelodysplastic Syndromes; Peritoneal Neoplasms; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Rectal Neoplasms; Sarcoma; Urinary Bladder Neoplasms; Uterine Cervical Neoplasms; Carcinoma; Hepatoblastoma; Lung Neoplasms; Multiple Myeloma; Peripheral Nervous System Diseases; Trigeminal Neuralgia; Head and Neck Neoplasms; Ovarian Neoplasms; Xerostomia
Reactive metabolite scavenging agent
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; IMMUNE SYSTEM; OTHER
ORAL
Alzheimer Disease; Glioma; Colorectal Neoplasms; Lymphoma; Lymphoma, Non-Hodgkin; Paraparesis, Tropical Spastic; Sarcoma, Kaposi; Small Cell Lung Carcinoma; Acquired Immunodeficiency Syndrome; AIDS-Associated Nephropathy; Carcinoma, Hepatocellular; Diarrhea; Liver Cirrhosis; Tuberculosis; Autoimmune Diseases; Hepatitis; Hepatitis B; Hepatitis B, Chronic; HIV Infections; Infections; Inflammation; Virus Diseases
DNA inhibitor
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Breast Neoplasms; Obesity; Substance-Related Disorders; Cocaine-Related Disorders; Endometriosis; Infertility; Paget Disease, Extramammary; Pituitary ACTH Hypersecretion; Polycystic Ovary Syndrome; Diabetes Mellitus; Ovarian Hyperstimulation Syndrome; Restless Legs Syndrome; Parkinson Disease; Pituitary Neoplasms
Dopamine D2 receptor agonist
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Cardiovascular Diseases; Heart Failure; Hypertension; Myocardial Infarction; Ventricular Dysfunction, Left
Angiotensin-converting enzyme inhibitor
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Postoperative Nausea and Vomiting; Sleep Apnea, Obstructive; Stomach Diseases; Alcoholism; Amphetamine-Related Disorders; Anorexia; Anorexia Nervosa; Cachexia; Cocaine-Related Disorders; Fibromyalgia; Paraganglioma; Substance-Related Disorders; Weight Loss; Anxiety; Child Development Disorders, Pervasive; Dementia; Heroin Dependence; Nausea; Schizophrenia; Depressive Disorder; Depressive Disorder, Major; Sleep Initiation and Maintenance Disorders
Adrenergic receptor alpha-2 antagonist
Small molecule
Approved
CARDIOVASCULAR; DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Acute Coronary Syndrome; Aortic Valve Insufficiency; Cardiomyopathy, Hypertrophic; Diabetic Nephropathies; Nephritis, Hereditary; Peripheral Arterial Disease; Renal Insufficiency, Chronic; Atherosclerosis; Atrial Fibrillation; Chagas Cardiomyopathy; Coronary Disease; Diabetes Mellitus, Type 2; Essential Hypertension; Hypercholesterolemia; Hypertension, Pulmonary; Kidney Diseases; Lipid Metabolism Disorders; Metabolic Syndrome; Non-ST Elevated Myocardial Infarction; Severe Acute Respiratory Syndrome; ST Elevation Myocardial Infarction; Cardiovascular Diseases; Diabetes Mellitus; Heart Failure; Hypertension; Myocardial Infarction; Stroke; Ventricular Dysfunction, Left
Type-1 angiotensin II receptor antagonist
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Diabetes Mellitus, Type 1; Diabetes Mellitus; Diabetes Mellitus, Type 2
Lysosomal alpha-glucosidase inhibitor
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Anemia, Sickle Cell; Arthritis, Rheumatoid; Gastrointestinal Stromal Tumors; Malaria; Mitochondrial Diseases; Neoplasms; Parkinson Disease; Prostatic Neoplasms, Castration-Resistant; Atherosclerosis; Coronary Disease; Cystic Fibrosis; Hypercholesterolemia; Hypertension; Diabetes Mellitus; Diabetes Mellitus, Type 2
Sulfonylurea receptor 1, Kir6.2 blocker
Antibody
Approved
DIABETES DRUGS & ENDOCRINOLOGY; IMMUNE SYSTEM; OTHER
SINGLE-USE
DiGeorge Syndrome; Kidney Tubular Necrosis, Acute; Leukemia, Myeloid, Acute; Multiple Myeloma; Neoplasms; Uremia; Amyotrophic Lateral Sclerosis; Colitis, Ulcerative; Glioblastoma; Glomerulosclerosis, Focal Segmental; Granuloma, Lethal Midline; Hodgkin Disease; Kidney Diseases; Renal Insufficiency, Chronic; Uveitis; Diabetes Mellitus, Type 1; Emphysema; Graft vs Host Disease; Infections; Reperfusion Injury; Delayed Graft Function; Immune System Diseases; Kidney Transplantation
Interleukin-2 receptor inhibitor
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER; UROLOGY AND KIDNEY
INJECTION; INTRAVENOUS; ORAL
Breast Neoplasms; Multiple Myeloma; Neoplasms; Neoplasms, Plasma Cell; Pancreatitis, Chronic; Carcinoma, Pancreatic Ductal; Diabetes Mellitus, Type 2; Diabetic Nephropathies; Hypocalcemia; Pancreatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Albuminuria; Glomerulonephritis, IGA; Hyperparathyroidism; Hypertrophy, Left Ventricular; Kidney Diseases; Proteinuria; Hyperparathyroidism, Secondary; Parathyroid Diseases; Renal Insufficiency, Chronic
Vitamin D receptor agonist
Small molecule
Approved
CARDIOVASCULAR; DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Cardiovascular Diseases; Brain Injuries; Pain; Severe Acute Respiratory Syndrome; Atherosclerosis; Breast Neoplasms; Coronary Disease; Diabetes Mellitus, Type 1; Diabetes Mellitus, Type 2; Essential Hypertension; Hypercholesterolemia; Hypertension, Renovascular; Proteinuria; Renal Artery Obstruction; Angina Pectoris; Diabetes Mellitus; Heart Failure; Hypertension; Myocardial Infarction; Stroke
Type-1 angiotensin II receptor antagonist
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER; RHEUMATOLOGY
ORAL
Breast Diseases; Breast Neoplasms; Bronchiolitis Obliterans Syndrome; Hemosiderosis; HIV Infections; Melanoma; Neoplasms; IgA Vasculitis; Lupus Erythematosus, Systemic; Lymphoproliferative Disorders; Multiple Myeloma; Pemphigoid, Bullous; Prostatic Neoplasms, Castration-Resistant; Sjogren's Syndrome; Smoldering Multiple Myeloma; Uveitis; Central Nervous System Neoplasms; Lupus Nephritis; Myasthenia Gravis; Polymyalgia Rheumatica; Severe Acute Respiratory Syndrome; Arthritis, Psoriatic; Arthritis, Rheumatoid
Dihydroorotate dehydrogenase inhibitor