DrugMapper


Display Options: Drug type Therapeutic Area Route of administration Mechanism of Action Indication Status		Total: 1496


Small molecule Approved OTHER ORAL Bacterial Infections Bacterial dihydropteroate synthase inhibitor


Small molecule Approved OTHER INJECTION; ORAL; RECTAL Altitude Sickness; Hypertension, Pulmonary; Premature Birth; Urinary Bladder Neoplasms; Heart Arrest; Acute Kidney Injury; Headache; Asthma; Lung Diseases, Obstructive Adenosine receptor antagonist


Small molecule Approved OTHER INJECTION; ORAL Carcinoma, Non-Small-Cell Lung; Depressive Disorder; Depressive Disorder, Major; Hypertension, Pulmonary; Leukemia, Myeloid, Acute; Lung Neoplasms; Prostatic Neoplasms; Altitude Sickness; Apnea; Hernias, Diaphragmatic, Congenital; Kidney Diseases; Leukemia; Pseudohypoparathyroidism; Renal Insufficiency, Chronic; Severe Acute Respiratory Syndrome; Virus Diseases; Pulmonary Disease, Chronic Obstructive; Respiratory Insufficiency; Asthma; Bronchitis, Chronic; Lung Diseases, Obstructive Adenosine receptor antagonist

Small molecule

Approved

OTHER

INJECTION; ORAL

Carcinoma, Non-Small-Cell Lung; Depressive Disorder; Depressive Disorder, Major; Hypertension, Pulmonary; Leukemia, Myeloid, Acute; Lung Neoplasms; Prostatic Neoplasms; Altitude Sickness; Apnea; Hernias, Diaphragmatic, Congenital; Kidney Diseases; Leukemia; Pseudohypoparathyroidism; Renal Insufficiency, Chronic; Severe Acute Respiratory Syndrome; Virus Diseases; Pulmonary Disease, Chronic Obstructive; Respiratory Insufficiency; Asthma; Bronchitis, Chronic; Lung Diseases, Obstructive

Adenosine receptor antagonist


Small molecule Approved OTHER ORAL Osteomyelitis; Burns; Toxoplasmosis, Cerebral; Chorioretinitis; Toxoplasmosis, Congenital; Bacterial Infections; Malaria Bacterial dihydropteroate synthase inhibitor


Small molecule Approved OTHER ORAL Alopecia Areata; Bone Diseases, Metabolic; Colitis, Ulcerative; Colorectal Neoplasms; Diabetes, Gestational; Diabetes Mellitus, Type 2; Infertility; Inflammatory Bowel Diseases; Lung Neoplasms; Mood Disorders; Neoplasms; Penile Induration; Premature Birth; Sarcopenia; Anemia, Sickle Cell; Blood Coagulation Disorders; Crohn Disease; Death, Sudden, Cardiac; Diabetes Mellitus; Diabetic Neuropathies; Disseminated Intravascular Coagulation; Endometrial Neoplasms; Heart Failure; Hepatitis C; HIV Infections; Insulin Resistance; Latent Autoimmune Diabetes in Adults; Lupus Erythematosus, Cutaneous; Malnutrition; Migraine Disorders; Neuralgia; Optic Neuritis; Osteogenesis Imperfecta; Polycystic Ovary Syndrome; Prostatic Neoplasms; Restless Legs Syndrome; Spinal Cord Injuries; Uterine Cervical Neoplasms; Alzheimer Disease; Asthma; Breast Neoplasms; Burns; Cardiovascular Diseases; Cluster Headache; Colonic Neoplasms; Coronary Disease; Diabetes Mellitus, Type 1; Femoral Neck Fractures; Hepatitis C, Chronic; Hip Fractures; Hypocalcemia; Leukemia; Lipid Metabolism Disorders; Lymphoma; Lymphoma, Non-Hodgkin; Melanoma; Menopause; Multiple Sclerosis; Myocardial Ischemia; Neonatal Sepsis; Non-alcoholic Fatty Liver Disease; Obesity; Osteoarthritis, Knee; Osteoporosis; Osteoporosis, Postmenopausal; Pain; Pregnancy; Prostatic Neoplasms, Castration-Resistant; Renal Insufficiency, Chronic; Severe Acute Respiratory Syndrome; Tuberculosis; Tuberculosis, Pulmonary; Vitamin D Deficiency; Hypoparathyroidism; Hypophosphatemia, Familial; Rickets, Hypophosphatemic Vitamin D receptor agonist

Small molecule

Approved

OTHER

ORAL

Alopecia Areata; Bone Diseases, Metabolic; Colitis, Ulcerative; Colorectal Neoplasms; Diabetes, Gestational; Diabetes Mellitus, Type 2; Infertility; Inflammatory Bowel Diseases; Lung Neoplasms; Mood Disorders; Neoplasms; Penile Induration; Premature Birth; Sarcopenia; Anemia, Sickle Cell; Blood Coagulation Disorders; Crohn Disease; Death, Sudden, Cardiac; Diabetes Mellitus; Diabetic Neuropathies; Disseminated Intravascular Coagulation; Endometrial Neoplasms; Heart Failure; Hepatitis C; HIV Infections; Insulin Resistance; Latent Autoimmune Diabetes in Adults; Lupus Erythematosus, Cutaneous; Malnutrition; Migraine Disorders; Neuralgia; Optic Neuritis; Osteogenesis Imperfecta; Polycystic Ovary Syndrome; Prostatic Neoplasms; Restless Legs Syndrome; Spinal Cord Injuries; Uterine Cervical Neoplasms; Alzheimer Disease; Asthma; Breast Neoplasms; Burns; Cardiovascular Diseases; Cluster Headache; Colonic Neoplasms; Coronary Disease; Diabetes Mellitus, Type 1; Femoral Neck Fractures; Hepatitis C, Chronic; Hip Fractures; Hypocalcemia; Leukemia; Lipid Metabolism Disorders; Lymphoma; Lymphoma, Non-Hodgkin; Melanoma; Menopause; Multiple Sclerosis; Myocardial Ischemia; Neonatal Sepsis; Non-alcoholic Fatty Liver Disease; Obesity; Osteoarthritis, Knee; Osteoporosis; Osteoporosis, Postmenopausal; Pain; Pregnancy; Prostatic Neoplasms, Castration-Resistant; Renal Insufficiency, Chronic; Severe Acute Respiratory Syndrome; Tuberculosis; Tuberculosis, Pulmonary; Vitamin D Deficiency; Hypoparathyroidism; Hypophosphatemia, Familial; Rickets, Hypophosphatemic

Vitamin D receptor agonist


Small molecule Approved CANCER; MUSCULOSKELETAL; OTHER; PREGNANCY AND GYNECOLOGY INJECTION; ORAL; TOPICAL; VAGINAL Memory; Reperfusion Injury; Brain Injuries; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Shock; Urinary Bladder, Overactive; Alzheimer Disease; Angina, Unstable; Anorexia Nervosa; Bone Diseases; Bone Diseases, Metabolic; Cardiovascular Diseases; Colonic Neoplasms; Coronary Disease; Cystitis, Interstitial; Diabetes Mellitus; Endometrial Neoplasms; Heart Diseases; Hot Flashes; Hypercholesterolemia; Hypertension; Lupus Erythematosus, Systemic; Memory Disorders; Myocardial Infarction; Myocardial Ischemia; Stroke; Thrombosis; Turner Syndrome; Atrophic Vaginitis; Atrophy; Breast Neoplasms; Dyspareunia; Hypogonadism; Menopause; Osteoporosis; Osteoporosis, Postmenopausal; Primary Ovarian Insufficiency Estrogen receptor agonist

Small molecule

Approved

CANCER; MUSCULOSKELETAL; OTHER; PREGNANCY AND GYNECOLOGY

INJECTION; ORAL; TOPICAL; VAGINAL

Memory; Reperfusion Injury; Brain Injuries; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Shock; Urinary Bladder, Overactive; Alzheimer Disease; Angina, Unstable; Anorexia Nervosa; Bone Diseases; Bone Diseases, Metabolic; Cardiovascular Diseases; Colonic Neoplasms; Coronary Disease; Cystitis, Interstitial; Diabetes Mellitus; Endometrial Neoplasms; Heart Diseases; Hot Flashes; Hypercholesterolemia; Hypertension; Lupus Erythematosus, Systemic; Memory Disorders; Myocardial Infarction; Myocardial Ischemia; Stroke; Thrombosis; Turner Syndrome; Atrophic Vaginitis; Atrophy; Breast Neoplasms; Dyspareunia; Hypogonadism; Menopause; Osteoporosis; Osteoporosis, Postmenopausal; Primary Ovarian Insufficiency

Estrogen receptor agonist


Small molecule Approved OTHER ORAL Digestive System Diseases Unknown


Small molecule Approved OTHER ORAL Thrombosis Vitamin k epoxide reductase complex subunit 1 isoform 1 inhibitor


Small molecule Approved OTHER TOPICAL Osteomyelitis; Amyotrophic Lateral Sclerosis; Eye Infections; Leishmaniasis; Trypanosomiasis DNA inhibitor


Small molecule Approved OTHER ORAL Epilepsy Sodium channel alpha subunit blocker


Small molecule Approved OTHER INJECTION Unknown Heavy metals chelating agent


Small molecule Approved OTHER INJECTION; ORAL Hemorrhage Dopamine D1 receptor antagonist


Small molecule Approved OTHER ORAL Epilepsy Voltage-gated T-type calcium channel blocker


Small molecule Approved OTHER ORAL Ischemic Stroke; Graves Disease; Graves Ophthalmopathy; Thyrotoxicosis; Hyperthyroidism; Thyroid Diseases Thyroid peroxidase inhibitor


Small molecule Approved OTHER INJECTION; ORAL Carcinoma, Squamous Cell; Neoplasms; Osteomyelitis; Stomach Neoplasms; Syphilis; Bacteremia; Infections; Pneumonia Bacterial penicillin-binding protein inhibitor


Small molecule Approved OTHER VAGINAL Unknown Estrogen receptor alpha agonist


Small molecule Approved OTHER ORAL Unknown Histamine H1 receptor antagonist


Small molecule Approved OTHER INJECTION Osteomyelitis; Bacterial Infections; Sepsis; Infections Unknown


Protein Approved OTHER FOR RX COMPOUNDING; INJECTION; OPHTHALMIC; TOPICAL Osteomyelitis; Paranasal Sinus Diseases; Arrhythmias, Cardiac; Bacterial Infections; Burns; Eye Infections; Infections; Pneumonia C55-isoprenyl pyrophosphate inhibitor


Small molecule Approved DENTISTRY; NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER BUCCAL; ORAL; RECTAL; TOPICAL Abortion, Spontaneous; Attention Deficit Disorder with Hyperactivity; Brain Neoplasms; Carcinoma, Squamous Cell; Cicatrix; Complex Regional Pain Syndromes; Glioblastoma; Glycogen Storage Disease Type II; Hypertension, Pulmonary; Keratosis, Actinic; Lung Neoplasms; Morton Neuroma; Neoplasms, Cystic, Mucinous, and Serous; Neuroma; Parathyroid Neoplasms; Premature Birth; Radius Fractures; Skin Neoplasms; Spinal Fractures; Thromboembolism; Tinnitus; Anus Diseases; Anxiety; Cancer Pain; Carcinoma; Cocaine-Related Disorders; Cognitive Dysfunction; Cystitis, Interstitial; Diabetic Neuropathies; Dysmenorrhea; Dysphonia; Geographic Atrophy; Heart Diseases; Humeral Fractures; Infertility; Irritable Bowel Syndrome; Leiomyoma; Myofascial Pain Syndromes; Neoplasms; Renal Colic; Rib Fractures; Scleroderma, Localized; Severe Acute Respiratory Syndrome; Shoulder Impingement Syndrome; Shoulder Pain; Skin Diseases; Temporomandibular Joint Disorders; Trigeminal Neuralgia; Urinary Incontinence; Urinary Tract Infections; Analgesia; Breast Neoplasms; Carpal Tunnel Syndrome; Chronic Pain; Colorectal Neoplasms; Common Cold; Cough; Dysuria; Fibromyalgia; Fractures, Bone; Headache; Heart Arrest; Hemorrhage; Ileus; Low Back Pain; Migraine Disorders; Muscular Diseases; Nutrition Disorders; Obesity; Obesity, Morbid; Osteoarthritis, Knee; Osteoporosis, Postmenopausal; Paget Disease, Extramammary; Parathyroid Diseases; Periarthritis; Peripheral Nervous System Diseases; Pharyngitis; Pre-Eclampsia; Pregnancy; Pulpitis; Scoliosis; Shock, Septic; Sinusitis; Stomatitis; Stroke; Tennis Elbow; Urinary Bladder Neoplasms; Urinary Bladder, Overactive; Uterine Cervical Dysplasia; Wounds and Injuries; Arrhythmias, Cardiac; Arthritis; Back Pain; Burns; Bursitis; Hemorrhoids; Inflammation; Insect Bites and Stings; Muscle Cramp; Myalgia; Neuralgia; Neuralgia, Postherpetic; Osteoarthritis; Pain; Premature Ejaculation; Pruritus; Rectal Diseases; Sprains and Strains; Sunburn; Tendinopathy; Urethritis Sodium channel alpha subunit blocker

Small molecule

Approved

DENTISTRY; NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER

BUCCAL; ORAL; RECTAL; TOPICAL

Abortion, Spontaneous; Attention Deficit Disorder with Hyperactivity; Brain Neoplasms; Carcinoma, Squamous Cell; Cicatrix; Complex Regional Pain Syndromes; Glioblastoma; Glycogen Storage Disease Type II; Hypertension, Pulmonary; Keratosis, Actinic; Lung Neoplasms; Morton Neuroma; Neoplasms, Cystic, Mucinous, and Serous; Neuroma; Parathyroid Neoplasms; Premature Birth; Radius Fractures; Skin Neoplasms; Spinal Fractures; Thromboembolism; Tinnitus; Anus Diseases; Anxiety; Cancer Pain; Carcinoma; Cocaine-Related Disorders; Cognitive Dysfunction; Cystitis, Interstitial; Diabetic Neuropathies; Dysmenorrhea; Dysphonia; Geographic Atrophy; Heart Diseases; Humeral Fractures; Infertility; Irritable Bowel Syndrome; Leiomyoma; Myofascial Pain Syndromes; Neoplasms; Renal Colic; Rib Fractures; Scleroderma, Localized; Severe Acute Respiratory Syndrome; Shoulder Impingement Syndrome; Shoulder Pain; Skin Diseases; Temporomandibular Joint Disorders; Trigeminal Neuralgia; Urinary Incontinence; Urinary Tract Infections; Analgesia; Breast Neoplasms; Carpal Tunnel Syndrome; Chronic Pain; Colorectal Neoplasms; Common Cold; Cough; Dysuria; Fibromyalgia; Fractures, Bone; Headache; Heart Arrest; Hemorrhage; Ileus; Low Back Pain; Migraine Disorders; Muscular Diseases; Nutrition Disorders; Obesity; Obesity, Morbid; Osteoarthritis, Knee; Osteoporosis, Postmenopausal; Paget Disease, Extramammary; Parathyroid Diseases; Periarthritis; Peripheral Nervous System Diseases; Pharyngitis; Pre-Eclampsia; Pregnancy; Pulpitis; Scoliosis; Shock, Septic; Sinusitis; Stomatitis; Stroke; Tennis Elbow; Urinary Bladder Neoplasms; Urinary Bladder, Overactive; Uterine Cervical Dysplasia; Wounds and Injuries; Arrhythmias, Cardiac; Arthritis; Back Pain; Burns; Bursitis; Hemorrhoids; Inflammation; Insect Bites and Stings; Muscle Cramp; Myalgia; Neuralgia; Neuralgia, Postherpetic; Osteoarthritis; Pain; Premature Ejaculation; Pruritus; Rectal Diseases; Sprains and Strains; Sunburn; Tendinopathy; Urethritis

Sodium channel alpha subunit blocker


Small molecule Approved OTHER ORAL Infections; Rhinitis, Allergic, Seasonal; Postoperative Nausea and Vomiting Histamine H1 receptor antagonist


Small molecule Approved OTHER ORAL Epilepsy Voltage-gated T-type calcium channel blocker


Small molecule Approved OTHER TOPICAL Unknown Bacterial enoyl-[acyl-carrier-protein] reductase inhibitor


Small molecule Approved OTHER TOPICAL Scabies Unknown


Small molecule Approved OTHER ORAL Gliosarcoma; Dermatomyositis; Glioblastoma; Graves Disease; Polymyositis; Graves Ophthalmopathy; Hyperthyroidism; Thyroid Diseases Thyroid peroxidase inhibitor

Small molecule

Approved

OTHER

ORAL

Adenocarcinoma of Lung; Adenomyosis; Aging; Anemia, Sickle Cell; Digestive System Diseases; Fatigue; Fractures, Bone; Head and Neck Neoplasms; Herpes Simplex; Hypertriglyceridemia; Inflammation; Leukemia, Hairy Cell; Leukoplakia, Oral; Liver Diseases, Alcoholic; Neuralgia, Postherpetic; Peripheral Vascular Diseases; Sleep Initiation and Maintenance Disorders; Ulcer; Acute Lung Injury; Adenoma; Barrett Esophagus; Blood Coagulation Disorders; Carotid Stenosis; Depressive Disorder; Depressive Disorder, Major; Depressive Disorder, Treatment-Resistant; Disseminated Intravascular Coagulation; Duodenal Ulcer; Endometrial Neoplasms; Glioblastoma; HIV Infections; Hypercholesterolemia; Hypertension, Pulmonary; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Lupus Erythematosus, Systemic; Melanoma; Metabolic Syndrome; Mouth Neoplasms; Nasopharyngeal Carcinoma; Neoplasms; Ovarian Neoplasms; Pancreatic Neoplasms; Periodontitis; Placental Insufficiency; Pneumonia, Viral; Pregnancy; Prostatic Neoplasms; Purpura, Thrombocytopenic, Idiopathic; Purpura, Thrombotic Thrombocytopenic; Rectal Neoplasms; Respiratory Distress Syndrome; Respiratory Insufficiency; Respiratory Tract Diseases; Sepsis; Tension-Type Headache; Tobacco Use Disorder; Tuberculosis; Uterine Cervical Neoplasms; Venous Thrombosis; Vitamin D Deficiency; Abortion, Habitual; Acute Chest Syndrome; Acute Coronary Syndrome; Adenomatous Polyposis Coli; Angina, Stable; Aortic Valve Stenosis; Asthma; Asthma, Aspirin-Induced; Atherosclerosis; Atrial Fibrillation; Bipolar Disorder; Blindness; Brain Infarction; Breast Neoplasms; Carcinoma, Hepatocellular; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Cardiomyopathy, Hypertrophic; Cardiovascular Diseases; Cataract; Cerebral Infarction; Cerebrovascular Disorders; Colitis, Ulcerative; Colonic Neoplasms; Colorectal Neoplasms; Colorectal Neoplasms, Hereditary Nonpolyposis; Diabetes Mellitus; Diabetes Mellitus, Type 2; Diabetic Retinopathy; Esophageal Neoplasms; Fetal Growth Retardation; Gastrointestinal Hemorrhage; Heart Diseases; Heart Failure; Hemorrhage; Hip Fractures; Hypertension; Infertility; Influenza, Human; Intracranial Aneurysm; Intracranial Arteriosclerosis; Ischemia; Ischemic Attack, Transient; Ischemic Stroke; Lipid Metabolism Disorders; Low Back Pain; Macular Degeneration; Meningitis; Mucocutaneous Lymph Node Syndrome; Multiple Myeloma; Multiple Sclerosis; Myocardial Ischemia; Non-ST Elevated Myocardial Infarction; Osteoarthritis; Osteonecrosis; Peptic Ulcer; Peripheral Arterial Disease; Pharyngitis; Pneumonia; Polycythemia Vera; Pre-Eclampsia; Prostatic Neoplasms, Castration-Resistant; Psychotic Disorders; Pulmonary Disease, Chronic Obstructive; Renal Insufficiency, Chronic; Retinal Artery Occlusion; Retinal Vein Occlusion; Rheumatic Heart Disease; Schizophrenia; Severe Acute Respiratory Syndrome; ST Elevation Myocardial Infarction; Stomach Neoplasms; Stomach Ulcer; Thrombocythemia, Essential; Thrombophilia; Varicose Ulcer; Vascular Diseases; Venous Thromboembolism; Wounds and Injuries; Arthritis; Back Pain; Common Cold; Coronary Artery Disease; Dysmenorrhea; Fever; Headache; Migraine Disorders; Muscle Cramp; Myalgia; Myocardial Infarction; Pain; Spasm; Stroke; Thrombosis; Toothache

Cyclooxygenase inhibitor

Protein

Approved

OTHER

INJECTION

Glomerulonephritis; Glomerulonephritis, Membranous; Optic Neuritis; Polycystic Ovary Syndrome; Renal Insufficiency, Chronic; Vitreoretinopathy, Proliferative; Amyotrophic Lateral Sclerosis; Dermatomyositis; Diabetic Nephropathies; Epilepsy; Migraine Disorders; Multiple Sclerosis, Chronic Progressive; Sarcoidosis; Scleritis; Uveitis; Arthritis, Rheumatoid; Glomerulosclerosis, Focal Segmental; Kidney Diseases; Multiple Sclerosis, Relapsing-Remitting; Nephrotic Syndrome; Multiple Sclerosis; Spasms, Infantile

Melanocortin receptor 2 agonist


Small molecule Approved OTHER INJECTION; OPHTHALMIC; ORAL; OTIC; TOPICAL Osteomyelitis; Acne Vulgaris; Bacterial Infections; Eye Infections Bacterial 70S ribosome inhibitor


Small molecule Approved OTHER INJECTION; ORAL Sunburn; Back Pain; Common Cold; Cough; Fever; Headache; Hypersensitivity; Nasal Obstruction; Pain; Pharyngitis; Rhinitis, Allergic, Seasonal; Sinusitis Histamine H1 receptor antagonist


Small molecule Approved OTHER ORAL Osteomyelitis; Colitis, Ulcerative; Crohn Disease; Tuberculosis, Pulmonary; Tuberculosis Dihydrofolate reductase inhibitor

Small molecule

Approved

DIABETES DRUGS & ENDOCRINOLOGY; OTHER; RHEUMATOLOGY

ORAL

Glioblastoma; Hypertension, Pulmonary; Intestinal Obstruction; Leukemia, Myeloid, Acute; Nausea; Osteomyelitis; Paraganglioma; Cholangitis, Sclerosing; Peripheral Nervous System Diseases; Premature Birth; Spondylitis, Ankylosing; Arthritis, Psoriatic; Arthritis, Juvenile; Arthritis, Rheumatoid; Colitis, Ulcerative

Arachidonate 5-lipoxygenase inhibitor


Small molecule Approved OTHER INJECTION; ORAL Lung Diseases, Obstructive Phosphodiesterase 3A inhibitor


Small molecule Approved OTHER ORAL Unknown Histamine H2 receptor antagonist


Small molecule Approved OTHER ORAL Unknown Unknown


Small molecule Approved OTHER ORAL Epilepsy Sodium channel alpha subunit blocker