DrugMapper


Display Options: Drug type Therapeutic Area Route of administration Mechanism of Action Indication Status		Total: 1496


Small molecule Approved OTHER ORAL Bacterial Infections Bacterial dihydropteroate synthase inhibitor


Small molecule Approved OTHER INJECTION; ORAL; RECTAL Urinary Bladder Neoplasms; Altitude Sickness; Hypertension, Pulmonary; Premature Birth; Heart Arrest; Acute Kidney Injury; Headache; Asthma; Lung Diseases, Obstructive Adenosine receptor antagonist


Small molecule Approved OTHER INJECTION; ORAL Depressive Disorder; Carcinoma, Non-Small-Cell Lung; Depressive Disorder, Major; Hypertension, Pulmonary; Leukemia, Myeloid, Acute; Prostatic Neoplasms; Altitude Sickness; Apnea; Kidney Diseases; Leukemia; Pseudohypoparathyroidism; Renal Insufficiency, Chronic; Virus Diseases; Pulmonary Disease, Chronic Obstructive; Respiratory Insufficiency; Asthma; Bronchitis, Chronic; Lung Diseases, Obstructive Adenosine receptor antagonist

Small molecule

Approved

OTHER

INJECTION; ORAL

Depressive Disorder; Carcinoma, Non-Small-Cell Lung; Depressive Disorder, Major; Hypertension, Pulmonary; Leukemia, Myeloid, Acute; Prostatic Neoplasms; Altitude Sickness; Apnea; Kidney Diseases; Leukemia; Pseudohypoparathyroidism; Renal Insufficiency, Chronic; Virus Diseases; Pulmonary Disease, Chronic Obstructive; Respiratory Insufficiency; Asthma; Bronchitis, Chronic; Lung Diseases, Obstructive

Adenosine receptor antagonist


Small molecule Approved OTHER ORAL Osteomyelitis; Burns; Toxoplasmosis, Cerebral; Chorioretinitis; Toxoplasmosis, Congenital; Bacterial Infections Bacterial dihydropteroate synthase inhibitor


Small molecule Approved OTHER ORAL Diabetes, Gestational; Mood Disorders; Psoriasis; Alopecia Areata; Colitis, Ulcerative; Colorectal Neoplasms; Inflammatory Bowel Diseases; Lung Neoplasms; Neoplasms; Osteogenesis Imperfecta; Penile Induration; Premature Birth; Sarcopenia; Anemia, Sickle Cell; Blood Coagulation Disorders; Crohn Disease; Death, Sudden, Cardiac; Diabetes Mellitus; Diabetic Neuropathies; Disseminated Intravascular Coagulation; Endometrial Neoplasms; Giant Cell Tumor of Bone; Giant Cell Tumors; Heart Failure; Hepatitis C; HIV Infections; Hyperparathyroidism, Primary; Insulin Resistance; Latent Autoimmune Diabetes in Adults; Lupus Erythematosus, Cutaneous; Malnutrition; Migraine Disorders; Optic Neuritis; Prostatic Neoplasms; Restless Legs Syndrome; Uterine Cervical Neoplasms; Alzheimer Disease; Asthma; Bone Diseases, Metabolic; Breast Neoplasms; Burns; Colonic Neoplasms; Diabetes Mellitus, Type 1; Diabetes Mellitus, Type 2; Familial Hypophosphatemic Rickets; Femoral Neck Fractures; Fractures, Bone; Hepatitis C, Chronic; Hip Fractures; Hyperprolactinemia; Hypocalcemia; Leukemia; Lipid Metabolism Disorders; Lymphoma; Lymphoma, Non-Hodgkin; Melanoma; Menopause; Multiple Sclerosis; Myocardial Ischemia; Non-alcoholic Fatty Liver Disease; Obesity; Osteitis Deformans; Osteoarthritis, Knee; Osteoporosis; Osteoporosis, Postmenopausal; Pain; Polycystic Ovary Syndrome; Pregnancy; Prostatic Neoplasms, Castration-Resistant; Renal Insufficiency, Chronic; Severe Acute Respiratory Syndrome; Tuberculosis; Tuberculosis, Pulmonary; Vitamin D Deficiency; Hypoparathyroidism; Hypophosphatemia, Familial; Rickets, Hypophosphatemic Vitamin D receptor agonist

Small molecule

Approved

OTHER

ORAL

Diabetes, Gestational; Mood Disorders; Psoriasis; Alopecia Areata; Colitis, Ulcerative; Colorectal Neoplasms; Inflammatory Bowel Diseases; Lung Neoplasms; Neoplasms; Osteogenesis Imperfecta; Penile Induration; Premature Birth; Sarcopenia; Anemia, Sickle Cell; Blood Coagulation Disorders; Crohn Disease; Death, Sudden, Cardiac; Diabetes Mellitus; Diabetic Neuropathies; Disseminated Intravascular Coagulation; Endometrial Neoplasms; Giant Cell Tumor of Bone; Giant Cell Tumors; Heart Failure; Hepatitis C; HIV Infections; Hyperparathyroidism, Primary; Insulin Resistance; Latent Autoimmune Diabetes in Adults; Lupus Erythematosus, Cutaneous; Malnutrition; Migraine Disorders; Optic Neuritis; Prostatic Neoplasms; Restless Legs Syndrome; Uterine Cervical Neoplasms; Alzheimer Disease; Asthma; Bone Diseases, Metabolic; Breast Neoplasms; Burns; Colonic Neoplasms; Diabetes Mellitus, Type 1; Diabetes Mellitus, Type 2; Familial Hypophosphatemic Rickets; Femoral Neck Fractures; Fractures, Bone; Hepatitis C, Chronic; Hip Fractures; Hyperprolactinemia; Hypocalcemia; Leukemia; Lipid Metabolism Disorders; Lymphoma; Lymphoma, Non-Hodgkin; Melanoma; Menopause; Multiple Sclerosis; Myocardial Ischemia; Non-alcoholic Fatty Liver Disease; Obesity; Osteitis Deformans; Osteoarthritis, Knee; Osteoporosis; Osteoporosis, Postmenopausal; Pain; Polycystic Ovary Syndrome; Pregnancy; Prostatic Neoplasms, Castration-Resistant; Renal Insufficiency, Chronic; Severe Acute Respiratory Syndrome; Tuberculosis; Tuberculosis, Pulmonary; Vitamin D Deficiency; Hypoparathyroidism; Hypophosphatemia, Familial; Rickets, Hypophosphatemic

Vitamin D receptor agonist


Small molecule Approved CANCER; MUSCULOSKELETAL; OTHER; PREGNANCY AND GYNECOLOGY INJECTION; ORAL; TOPICAL; VAGINAL Reperfusion Injury; Brain Injuries; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Shock; Urinary Bladder, Overactive; Alzheimer Disease; Angina, Unstable; Anorexia Nervosa; Bone Diseases, Metabolic; Colonic Neoplasms; Coronary Disease; Diabetes Mellitus; Endometrial Hyperplasia; Endometrial Neoplasms; Hot Flashes; Hypercholesterolemia; Hypertension; Lupus Erythematosus, Systemic; Memory Disorders; Myocardial Infarction; Myocardial Ischemia; Stroke; Thrombosis; Turner Syndrome; Atrophic Vaginitis; Atrophy; Breast Neoplasms; Dyspareunia; Hypogonadism; Menopause; Osteoporosis; Osteoporosis, Postmenopausal; Primary Ovarian Insufficiency Estrogen receptor agonist

Small molecule

Approved

CANCER; MUSCULOSKELETAL; OTHER; PREGNANCY AND GYNECOLOGY

INJECTION; ORAL; TOPICAL; VAGINAL

Reperfusion Injury; Brain Injuries; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Shock; Urinary Bladder, Overactive; Alzheimer Disease; Angina, Unstable; Anorexia Nervosa; Bone Diseases, Metabolic; Colonic Neoplasms; Coronary Disease; Diabetes Mellitus; Endometrial Hyperplasia; Endometrial Neoplasms; Hot Flashes; Hypercholesterolemia; Hypertension; Lupus Erythematosus, Systemic; Memory Disorders; Myocardial Infarction; Myocardial Ischemia; Stroke; Thrombosis; Turner Syndrome; Atrophic Vaginitis; Atrophy; Breast Neoplasms; Dyspareunia; Hypogonadism; Menopause; Osteoporosis; Osteoporosis, Postmenopausal; Primary Ovarian Insufficiency

Estrogen receptor agonist


Small molecule Approved OTHER ORAL Digestive System Diseases Unknown


Small molecule Approved OTHER ORAL Thrombosis Vitamin k epoxide reductase complex subunit 1 isoform 1 inhibitor


Small molecule Approved OTHER TOPICAL Osteomyelitis; Amyotrophic Lateral Sclerosis; Eye Infections; Leishmaniasis; Trypanosomiasis DNA inhibitor


Small molecule Approved OTHER ORAL Epilepsy Sodium channel alpha subunit blocker


Small molecule Approved OTHER INJECTION Unknown Heavy metals chelating agent


Small molecule Approved OTHER INJECTION; ORAL Hemorrhage Dopamine D1 receptor antagonist


Small molecule Approved OTHER ORAL Epilepsy Voltage-gated T-type calcium channel blocker


Small molecule Approved OTHER ORAL Graves Ophthalmopathy; Thyrotoxicosis; Hyperthyroidism; Thyroid Diseases Thyroid peroxidase inhibitor


Small molecule Approved OTHER INJECTION; ORAL Osteomyelitis; Carcinoma, Squamous Cell; Neoplasms; Stomach Neoplasms; Bacteremia; Infections; Pharyngitis; Pneumococcal Infections; Pneumonia; Tonsillitis Bacterial penicillin-binding protein inhibitor


Small molecule Approved OTHER VAGINAL Unknown Estrogen receptor alpha agonist


Small molecule Approved OTHER ORAL Unknown Histamine H1 receptor antagonist


Small molecule Approved OTHER INJECTION Osteomyelitis; Bacterial Infections; Sepsis; Infections Unknown


Protein Approved OTHER FOR RX COMPOUNDING; INJECTION; OPHTHALMIC; TOPICAL Osteomyelitis; Paranasal Sinus Diseases; Arrhythmias, Cardiac; Bacterial Infections; Burns; Infections; Pneumonia C55-isoprenyl pyrophosphate inhibitor


Small molecule Approved DENTISTRY; NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER BUCCAL; ORAL; RECTAL; TOPICAL Attention Deficit Disorder with Hyperactivity; Complex Regional Pain Syndromes; Humeral Fractures; Morton Neuroma; Parathyroid Neoplasms; Skin Neoplasms; Spinal Fractures; Tinnitus; Brain Neoplasms; Carcinoma, Squamous Cell; Glioblastoma; Glycogen Storage Disease Type II; Hypertension, Pulmonary; Keratosis, Actinic; Lung Neoplasms; Neuroma; Premature Birth; Thromboembolism; Anus Diseases; Anxiety; Carcinoma; Cocaine-Related Disorders; Cognitive Dysfunction; Cystitis, Interstitial; Diabetic Neuropathies; Dysmenorrhea; Heart Diseases; Infertility; Irritable Bowel Syndrome; Leiomyoma; Macular Degeneration; Myofascial Pain Syndromes; Neoplasms; Osteoarthritis, Knee; Renal Colic; Rib Fractures; Scleroderma, Localized; Severe Acute Respiratory Syndrome; Shoulder Impingement Syndrome; Shoulder Pain; Skin Diseases; Temporomandibular Joint Disorders; Trigeminal Neuralgia; Urinary Incontinence; Urinary Tract Infections; Breast Neoplasms; Carpal Tunnel Syndrome; Chronic Pain; Colorectal Neoplasms; Common Cold; Cough; Dysuria; Fibromyalgia; Headache; Heart Arrest; Hemorrhage; Ileus; Low Back Pain; Migraine Disorders; Muscular Diseases; Nutrition Disorders; Obesity; Obesity, Morbid; Osteoporosis, Postmenopausal; Paget Disease, Extramammary; Parathyroid Diseases; Periarthritis; Peripheral Nervous System Diseases; Pharyngitis; Pre-Eclampsia; Pregnancy; Pulpitis; Scoliosis; Shock, Septic; Sinusitis; Stomatitis; Stroke; Tennis Elbow; Urinary Bladder, Overactive; Uterine Cervical Dysplasia; Wounds and Injuries; Arrhythmias, Cardiac; Arthritis; Back Pain; Burns; Bursitis; Hemorrhoids; Inflammation; Insect Bites and Stings; Muscle Cramp; Myalgia; Neuralgia; Neuralgia, Postherpetic; Osteoarthritis; Pain; Premature Ejaculation; Pruritus; Rectal Diseases; Sprains and Strains; Sunburn; Tendinopathy; Urethritis Sodium channel alpha subunit blocker

Small molecule

Approved

DENTISTRY; NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER

BUCCAL; ORAL; RECTAL; TOPICAL

Attention Deficit Disorder with Hyperactivity; Complex Regional Pain Syndromes; Humeral Fractures; Morton Neuroma; Parathyroid Neoplasms; Skin Neoplasms; Spinal Fractures; Tinnitus; Brain Neoplasms; Carcinoma, Squamous Cell; Glioblastoma; Glycogen Storage Disease Type II; Hypertension, Pulmonary; Keratosis, Actinic; Lung Neoplasms; Neuroma; Premature Birth; Thromboembolism; Anus Diseases; Anxiety; Carcinoma; Cocaine-Related Disorders; Cognitive Dysfunction; Cystitis, Interstitial; Diabetic Neuropathies; Dysmenorrhea; Heart Diseases; Infertility; Irritable Bowel Syndrome; Leiomyoma; Macular Degeneration; Myofascial Pain Syndromes; Neoplasms; Osteoarthritis, Knee; Renal Colic; Rib Fractures; Scleroderma, Localized; Severe Acute Respiratory Syndrome; Shoulder Impingement Syndrome; Shoulder Pain; Skin Diseases; Temporomandibular Joint Disorders; Trigeminal Neuralgia; Urinary Incontinence; Urinary Tract Infections; Breast Neoplasms; Carpal Tunnel Syndrome; Chronic Pain; Colorectal Neoplasms; Common Cold; Cough; Dysuria; Fibromyalgia; Headache; Heart Arrest; Hemorrhage; Ileus; Low Back Pain; Migraine Disorders; Muscular Diseases; Nutrition Disorders; Obesity; Obesity, Morbid; Osteoporosis, Postmenopausal; Paget Disease, Extramammary; Parathyroid Diseases; Periarthritis; Peripheral Nervous System Diseases; Pharyngitis; Pre-Eclampsia; Pregnancy; Pulpitis; Scoliosis; Shock, Septic; Sinusitis; Stomatitis; Stroke; Tennis Elbow; Urinary Bladder, Overactive; Uterine Cervical Dysplasia; Wounds and Injuries; Arrhythmias, Cardiac; Arthritis; Back Pain; Burns; Bursitis; Hemorrhoids; Inflammation; Insect Bites and Stings; Muscle Cramp; Myalgia; Neuralgia; Neuralgia, Postherpetic; Osteoarthritis; Pain; Premature Ejaculation; Pruritus; Rectal Diseases; Sprains and Strains; Sunburn; Tendinopathy; Urethritis

Sodium channel alpha subunit blocker


Small molecule Approved OTHER ORAL Infections; Rhinitis, Allergic, Seasonal; Postoperative Nausea and Vomiting Histamine H1 receptor antagonist


Small molecule Approved OTHER ORAL Epilepsy Voltage-gated T-type calcium channel blocker


Small molecule Approved OTHER TOPICAL Unknown Bacterial enoyl-[acyl-carrier-protein] reductase inhibitor


Small molecule Approved OTHER TOPICAL Scabies Unknown


Small molecule Approved OTHER ORAL Dermatomyositis; Glioblastoma; Graves Ophthalmopathy; Hyperthyroidism; Thyroid Diseases Thyroid peroxidase inhibitor

Small molecule

Approved

OTHER

ORAL

Adenocarcinoma of Lung; Adenomyosis; Fatigue; Fractures, Bone; Peripheral Vascular Diseases; Sleep Initiation and Maintenance Disorders; Anemia, Sickle Cell; Digestive System Diseases; Head and Neck Neoplasms; Herpes Simplex; Hypertriglyceridemia; Inflammation; Leukoplakia, Oral; Neuralgia, Postherpetic; Ulcer; Acute Lung Injury; Adenoma; Barrett Esophagus; Blood Coagulation Disorders; Carotid Stenosis; Depressive Disorder, Major; Depressive Disorder, Treatment-Resistant; Disseminated Intravascular Coagulation; Duodenal Ulcer; Endometrial Neoplasms; Glioblastoma; Heart Diseases; HIV Infections; Hypercholesterolemia; Hypertension, Pulmonary; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Lupus Erythematosus, Systemic; Melanoma; Metabolic Syndrome; Nasopharyngeal Neoplasms; Neoplasms; Ovarian Neoplasms; Periodontitis; Placental Insufficiency; Pneumonia; Pneumonia, Viral; Pregnancy; Prostatic Neoplasms; Pulmonary Disease, Chronic Obstructive; Rectal Neoplasms; Respiratory Distress Syndrome; Respiratory Insufficiency; Sepsis; Tension-Type Headache; Tobacco Use Disorder; Tuberculosis; Uterine Cervical Neoplasms; Venous Thrombosis; Vitamin D Deficiency; Abortion, Habitual; Acute Chest Syndrome; Acute Coronary Syndrome; Adenomatous Polyposis Coli; Angina, Stable; Aortic Valve Stenosis; Asthma; Atherosclerosis; Atrial Fibrillation; Bipolar Disorder; Blindness; Brain Infarction; Breast Neoplasms; Carcinoma, Hepatocellular; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Cardiomyopathy, Hypertrophic; Cardiovascular Diseases; Cataract; Cerebral Infarction; Cerebrovascular Disorders; Colitis, Ulcerative; Colonic Neoplasms; Colorectal Neoplasms; Colorectal Neoplasms, Hereditary Nonpolyposis; Diabetes Mellitus; Diabetes Mellitus, Type 2; Diabetic Retinopathy; Esophageal Neoplasms; Fetal Growth Retardation; Gastrointestinal Hemorrhage; Heart Failure; Hemorrhage; Hypertension; Infertility; Intracranial Aneurysm; Intracranial Arteriosclerosis; Ischemia; Ischemic Attack, Transient; Ischemic Stroke; Lipid Metabolism Disorders; Low Back Pain; Macular Degeneration; Meningitis; Mucocutaneous Lymph Node Syndrome; Multiple Myeloma; Myocardial Ischemia; Non-ST Elevated Myocardial Infarction; Osteoarthritis; Osteonecrosis; Peptic Ulcer; Peripheral Arterial Disease; Pharyngitis; Polycythemia Vera; Pre-Eclampsia; Prostatic Neoplasms, Castration-Resistant; Psychotic Disorders; Renal Insufficiency, Chronic; Retinal Artery Occlusion; Retinal Vein Occlusion; Rheumatic Heart Disease; Schizophrenia; Severe Acute Respiratory Syndrome; ST Elevation Myocardial Infarction; Stomach Neoplasms; Stomach Ulcer; Thrombocythemia, Essential; Thrombophilia; Varicose Ulcer; Vascular Diseases; Venous Thromboembolism; Wounds and Injuries; Arthritis; Back Pain; Common Cold; Coronary Artery Disease; Coronary Disease; Dysmenorrhea; Fever; Headache; Migraine Disorders; Muscle Cramp; Myalgia; Myocardial Infarction; Pain; Spasm; Stroke; Thrombosis; Toothache

Cyclooxygenase inhibitor

Protein

Approved

OTHER

INJECTION

Optic Neuritis; Polycystic Ovary Syndrome; Vitreoretinopathy, Proliferative; Glomerulonephritis; Glomerulonephritis, Membranous; Renal Insufficiency, Chronic; Amyotrophic Lateral Sclerosis; Dermatomyositis; Diabetic Nephropathies; Epilepsy; Migraine Disorders; Multiple Sclerosis, Chronic Progressive; Sarcoidosis; Scleritis; Uveitis; Arthritis, Rheumatoid; Multiple Sclerosis; Multiple Sclerosis, Relapsing-Remitting; Nephrotic Syndrome; Neuroblastoma; Multiple Sclerosis; Spasms, Infantile

Melanocortin receptor 2 agonist


Small molecule Approved OTHER INJECTION; OPHTHALMIC; ORAL; OTIC; TOPICAL Osteomyelitis; Acne Vulgaris; Bacterial Infections; Eye Infections Bacterial 70S ribosome inhibitor


Small molecule Approved OTHER INJECTION; ORAL Sunburn; Rhinitis, Allergic, Seasonal; Cough; Sinusitis Histamine H1 receptor antagonist


Small molecule Approved OTHER ORAL Osteomyelitis; Colitis, Ulcerative; Crohn Disease; Tuberculosis Dihydrofolate reductase inhibitor


Small molecule Approved DIABETES DRUGS & ENDOCRINOLOGY; OTHER; RHEUMATOLOGY ORAL Osteomyelitis; Glioblastoma; Hypertension, Pulmonary; Intestinal Obstruction; Nausea; Cholangitis, Sclerosing; Peripheral Nervous System Diseases; Spondylitis, Ankylosing; Arthritis, Psoriatic; Arthritis, Juvenile; Arthritis, Rheumatoid; Colitis, Ulcerative Arachidonate 5-lipoxygenase inhibitor


Small molecule Approved OTHER INJECTION; ORAL Lung Diseases, Obstructive Phosphodiesterase 3A inhibitor


Small molecule Approved OTHER ORAL Unknown Histamine H2 receptor antagonist


Small molecule Approved OTHER ORAL Unknown Unknown


Small molecule Approved OTHER ORAL Epilepsy Sodium channel alpha subunit blocker