| Synonyms: | |
| Status: | Approved (1968) |
| Entry Type: | Small molecule |
| Molecule Category: | UNKNOWN |
| ATC: | R02AB30 |
| UNII: | 5IE62321P4 |
Pharmacology
| Action | Mechanism of Action | Reference |
|---|---|---|
| INHIBITOR | Cell membrane inhibitor |
| Targets | EC50(nM) | IC50(nM) | Kd(nM) | Ki(nM) | Inhibition(%) | |
|---|---|---|---|---|---|---|
|
Enzyme
Cytochrome P450
Cytochrome P450 family 5
Cytochrome P450 family 5A
Cytochrome P450 5A1
|
- | 774 | - | - | - | |
|
Enzyme
Kinase
Protein Kinase
TK protein kinase group
Tyrosine protein kinase Src family
|
- | 1094 | - | - | - | |
|
Membrane receptor
Family A G protein-coupled receptor
Peptide receptor (family A GPCR)
Short peptide receptor (family A GPCR)
Endothelin receptor
|
- | 2983 | - | 1835 | - | |
|
Membrane receptor
Family A G protein-coupled receptor
Peptide receptor (family A GPCR)
Short peptide receptor (family A GPCR)
Melanocortin receptor
|
- | 2013 | - | 1888 | - | |
|
Membrane receptor
Family A G protein-coupled receptor
Peptide receptor (family A GPCR)
Short peptide receptor (family A GPCR)
Neurokinin receptor
|
- | 4564 | - | 1521 | - |
Indications
| Mesh Heading | Maximum Phase | Mesh ID | Reference |
|---|---|---|---|
| Hordeolum | 3 | D006726 | ClinicalTrials |
Cross References
| Resources | Reference |
|---|---|
| ChEMBL | CHEMBL1201469 |
| FDA SRS | 5IE62321P4 |
CONTENTS