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Total: 6532
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
TRANSDERMAL
Alzheimer Disease; Fibromyalgia; Stroke; Substance-Related Disorders; Parkinson Disease; Restless Legs Syndrome
D2-like dopamine receptor agonist
Small molecule
Approved
CARDIOVASCULAR; OTHER; RESPIRATORY
ORAL
Anemia, Sickle Cell; Altitude Sickness; Asthma; Hypoplastic Left Heart Syndrome; Severe Acute Respiratory Syndrome; Idiopathic Pulmonary Fibrosis; Vascular Diseases; Familial Primary Pulmonary Hypertension; Hypertension; Hypertension, Pulmonary; Pulmonary Arterial Hypertension
Endothelin receptor, ET-A/ET-B antagonist
Small molecule
Approved
Unknown
Unknown
Hypertension; Stroke
Renin inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Breast Neoplasms; Bronchiolitis Obliterans Syndrome; Chordoma; Colonic Neoplasms; Huntington Disease; Cerebellar Ataxia; Glioma; Graft vs Host Disease; Hypertension, Pulmonary; Leukemia, Myeloid, Acute; Melanoma; Neuroma, Acoustic; Paraganglioma; Parkinson Disease; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Synovitis, Pigmented Villonodular; Alzheimer Disease; Gastrointestinal Stromal Tumors; Leukemia; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid; Neoplasms; Sarcoma
Unknown
Small molecule
Approved
Unknown
Unknown
Colorectal Neoplasms; Diabetic Nephropathies; Asthma; Dermatitis; Eczema; Rhinitis; Rhinitis, Allergic, Perennial; Rhinitis, Allergic, Seasonal; Rhinitis, Vasomotor; Urticaria; Hypersensitivity
Unknown
Small molecule
Approved
IMMUNE SYSTEM; OTHER
ORAL
Hypertriglyceridemia; AIDS Dementia Complex; Arthritis, Rheumatoid; Cognitive Dysfunction; Graft vs Host Disease; Hematologic Neoplasms; Hodgkin Disease; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Myelodysplastic Syndromes; Sarcoma, Kaposi; Severe Acute Respiratory Syndrome; Stroke; Acquired Immunodeficiency Syndrome; Infections; HIV Infections; Virus Diseases
C-C chemokine receptor type 5 antagonist
Small molecule
Approved
OTHER
ORAL
Head and Neck Neoplasms; Hepatitis C; Leukemia, Biphenotypic, Acute; Paraparesis, Tropical Spastic; HTLV-I Infections; Liver Cirrhosis, Biliary; Multiple Sclerosis, Relapsing-Remitting; Acquired Immunodeficiency Syndrome; HIV Infections; Infections; Virus Diseases
Unknown
Small molecule
Approved
UROLOGY AND KIDNEY
INTRAVENOUS
Adenocarcinoma; Astrocytoma; Brain Neoplasms; Breast Neoplasms, Male; Carcinoma; Colonic Neoplasms; Colorectal Neoplasms; Diffuse Intrinsic Pontine Glioma; Genital Neoplasms, Female; Glioma; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Lung Neoplasms; Oligodendroglioma; Paraganglioma; Peritoneal Neoplasms; Prostatic Neoplasms; Urethral Neoplasms; Uterine Cervical Neoplasms; Adenoma; Arthritis, Rheumatoid; Carcinoid Tumor; Carcinoma, Endometrioid; Carcinoma, Hepatocellular; Carcinoma, Islet Cell; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Central Nervous System Neoplasms; Endometrial Neoplasms; Fallopian Tube Neoplasms; Ganglioneuroblastoma; Glioblastoma; Gliosarcoma; Hodgkin Disease; Insulinoma; Ischemia; Kidney Neoplasms; Leukemia; Leukemia, Myeloid, Acute; Liver Neoplasms; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Non-Hodgkin; Melanoma; Multiple Myeloma; Multiple Sclerosis, Relapsing-Remitting; Myelodysplastic Syndromes; Neuroblastoma; Osteosarcoma; Ovarian Neoplasms; Pancreatic Neoplasms; Peripheral Arterial Disease; Prostatic Neoplasms, Castration-Resistant; Retroviridae Infections; Rhabdomyosarcoma; Sarcoma; Small Cell Lung Carcinoma; Somatostatinoma; Thyroid Neoplasms; Urinary Bladder Neoplasms; Breast Neoplasms; Hepatoblastoma; Lymphoma; Neoplasm Metastasis; Rhabdomyosarcoma, Alveolar; Rhabdomyosarcoma, Embryonal; Carcinoma, Renal Cell; Lymphoma, Mantle-Cell; Neoplasms
FK506-binding protein 1A inhibitor
Small molecule
Approved
OTHER
INTRAVENOUS
Astrocytoma; Gliosarcoma; Head and Neck Neoplasms; Bile Duct Neoplasms; Breast Neoplasms, Male; Burkitt Lymphoma; Carcinoma, Non-Small-Cell Lung; Carcinoma, Renal Cell; Carcinoma, Verrucous; Cholangiocarcinoma; Colorectal Neoplasms; Gallbladder Neoplasms; Hypopharyngeal Neoplasms; Leukemia; Liver Neoplasms; Lung Neoplasms; Lymphoma; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Large-Cell, Anaplastic; Lymphoma, Mantle-Cell; Melanoma; Oropharyngeal Neoplasms; Ovarian Neoplasms; Pancreatic Neoplasms; Peritoneal Neoplasms; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Retroviridae Infections; Sarcoma; Squamous Cell Carcinoma of Head and Neck; Stomach Neoplasms; Tongue Neoplasms; Urethral Neoplasms; Urinary Bladder Neoplasms; Endometrial Neoplasms; Breast Neoplasms; Neoplasms
Tubulin inhibitor
Small molecule
Approved
Unknown
ORAL
Carcinoma, Renal Cell; Endometrial Neoplasms; Prostatic Neoplasms, Castration-Resistant; Renal Insufficiency, Chronic; Thyroid Neoplasms; Urinary Bladder Neoplasms; Adenocarcinoma; Bile Duct Neoplasms; Brain Neoplasms; Carcinoma, Ductal; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Colorectal Neoplasms; Esophageal Neoplasms; Gallbladder Neoplasms; Melanoma; Ovarian Neoplasms; Pancreatic Neoplasms; Paraganglioma; Peritoneal Neoplasms; Pituitary Neoplasms; Stomach Neoplasms; Uterine Cervical Neoplasms; Brain Diseases; Breast Neoplasms; Head and Neck Neoplasms; Neoplasms; Sarcoma
Unknown
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
ORAL
Carcinoma, Non-Small-Cell Lung; Head and Neck Neoplasms; Esophageal Neoplasms; Glioma; Multiple Sclerosis; Neoplasms; Schizophrenia; Sleep Initiation and Maintenance Disorders; Stroke; Brain Injuries; Depressive Disorder; Disorders of Excessive Somnolence; Fatigue; Obesity; Sleep Apnea Syndromes; Attention Deficit Disorder with Hyperactivity; Narcolepsy; Sleep Apnea, Obstructive; Sleep Wake Disorders
Dopamine transporter inhibitor
Small molecule
Approved
IMMUNE SYSTEM; OTHER; UROLOGY AND KIDNEY
INTRAVENOUS
Meningitis; Appendicitis; Cholecystitis; Pancreatitis; Peritonitis; Pneumonia; Pneumonia, Ventilator-Associated; Bacterial Infections; Intraabdominal Infections; Pyelonephritis; Urinary Tract Infections
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
Unknown
Unknown
Staphylococcal Infections; Infections; Impetigo; Staphylococcal Skin Infections
70S ribosome inhibitor
Small molecule
Approved
Unknown
Unknown
Breast Neoplasms; Neoplasms; Ovarian Neoplasms; Parkinson Disease; Scleroderma, Systemic; Leukemia, Myelogenous, Chronic, BCR-ABL Positive
Bcr/Abl fusion protein inhibitor
Small molecule
Approved
Unknown
Unknown
Amphetamine-Related Disorders; Cocaine-Related Disorders; Multiple Sclerosis; Substance-Related Disorders; Bipolar Disorder; Depressive Disorder; Feeding and Eating Disorders; Attention Deficit Disorder with Hyperactivity
Unknown
Small molecule
Approved
Unknown
Unknown
Heart Failure; Hypertension; Radiodermatitis; Alzheimer Disease; Autistic Disorder; Enteritis; Hypertension, Portal; Kidney Failure, Chronic; Lesch-Nyhan Syndrome; Liver Cirrhosis; Phenylketonurias; Pulmonary Disease, Chronic Obstructive
Unknown
Small molecule
Approved
OTHER; UROLOGY AND KIDNEY
ORAL
Urinary Incontinence; Urinary Bladder, Overactive; Urinary Incontinence, Urge
Muscarinic acetylcholine receptor M2 antagonist
Small molecule
Approved
Unknown
Unknown
Autonomic Dysreflexia; Urinary Incontinence, Stress; Urinary Bladder, Neurogenic; Urinary Bladder, Overactive; Polyuria; Urinary Incontinence
Unknown
Small molecule
Approved
Unknown
Unknown
Neoplasms
Diagnostic agent
Small molecule
Approved
CANCER
SUBCUTANEOUS
beta-Thalassemia; Blood Platelet Disorders; Diabetes Mellitus, Type 1; Diabetic Foot; End Stage Liver Disease; Glioblastoma; Graft vs Host Disease; Kidney Diseases; Leukemia; Leukemia, Biphenotypic, Acute; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Myeloid, Acute; Lymphoma, Follicular; Lymphoma, Mantle-Cell; Myelodysplastic Syndromes; Neutropenia; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Sarcoma; Syndrome; Thalassemia; Anemia, Sickle Cell; Fanconi Anemia; Gliosarcoma; Granulomatous Disease, Chronic; Head and Neck Neoplasms; Hematologic Neoplasms; Hodgkin Disease; Lymphoma, Large B-Cell, Diffuse; Lymphoma, T-Cell; Lymphopenia; Pancreatic Neoplasms; Scleroderma, Systemic; Hematopoietic Stem Cell Transplantation; Lymphoma; Lymphoma, Non-Hodgkin; Multiple Myeloma; Neoplasms
C-X-C chemokine receptor type 4 partial agonist
Small molecule
Approved
OTHER
ORAL
Fibromyalgia; Hepatitis C, Chronic; Depressive Disorder; Depressive Disorder, Major
Norepinephrine transporter inhibitor
Small molecule
Approved
CARDIOVASCULAR; OTHER
INTRAVENOUS
Vascular Diseases; Scoliosis; Hypertension; Hypertension, Malignant; Stroke; Cardiovascular Diseases
Voltage-gated L-type calcium channel blocker
Small molecule
Approved
Unknown
Unknown
Amnesia; Colorectal Neoplasms; Depressive Disorder; Inflammation; Neural Tube Defects; Obesity, Morbid; Premature Birth; Psychomotor Agitation; Renal Insufficiency; Renal Insufficiency, Chronic; Coronary Disease; Depressive Disorder, Treatment-Resistant; Hypotension; Leukemia; Migraine Disorders; Neoplasms; Postoperative Nausea and Vomiting; Pulmonary Disease, Chronic Obstructive; Tonsillitis; Wounds and Injuries; Atrial Fibrillation; Back Pain; Brain Injuries; Delirium; Genital Neoplasms, Male; Heart Diseases; Hypertension; Liver Cirrhosis; Obesity; Pain; Pruritus; Reperfusion Injury; Respiratory Distress Syndrome; Respiratory Insufficiency; Severe Acute Respiratory Syndrome; Status Epilepticus; Stroke; Subarachnoid Hemorrhage
Unknown
Small molecule
Approved
MUSCULOSKELETAL; OTHER
ORAL
Tourette Syndrome; Movement Disorders; Chorea; Huntington Disease
Synaptic vesicular amine transporter inhibitor
Small molecule
Approved
Unknown
Unknown
Arthritis; Back Pain; Bursitis; Contusions; Muscle Cramp; Myalgia; Pain; Sprains and Strains; Tendinopathy; Wounds and Injuries
Unknown
Small molecule
Approved
Unknown
IV (INFUSION)
Leukemia, Biphenotypic, Acute; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Leukemia, Plasma Cell; Lymphoma, B-Cell; Myelodysplastic Syndromes; Prostatic Neoplasms; Amyloidosis, Familial; Anemia, Hemolytic, Autoimmune; Breast Neoplasms; Hematologic Neoplasms; Leukemia; Leukemia, Hairy Cell; Lymphoma, T-Cell, Peripheral; Ovarian Neoplasms; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Small Cell Lung Carcinoma; Waldenstrom Macroglobulinemia; Hodgkin Disease; Immunoblastic Lymphadenopathy; Leukemia, Lymphocytic, Chronic, B-Cell; Lymphoma; Lymphoma, B-Cell, Marginal Zone; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Lymphoma, Non-Hodgkin; Multiple Myeloma; Neoplasms
Unknown
Small molecule
Approved
OTHER
INTRAVENOUS
Cardiovascular Diseases; Myocardial Perfusion Imaging
Adenosine A2a receptor agonist
Small molecule
Approved
CARDIOVASCULAR; OTHER
ORAL
Coronary Disease; Hypercholesterolemia; Hyperlipidemia, Familial Combined; Lipid Metabolism Disorders; Cardiovascular Diseases
Peroxisome proliferator-activated receptor alpha agonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
ORAL
Back Pain; Chronic Pain; Diabetic Neuropathies; Hallux Valgus; Joint Diseases; Low Back Pain; Neoplasms; Neuralgia; Osteoarthritis; Osteoarthritis, Hip; Osteoarthritis, Knee; Pain
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Fallopian Tube Neoplasms; Ileus; Ovarian Neoplasms; Peritoneal Neoplasms; Urinary Bladder Neoplasms; Constipation
Mu opioid receptor antagonist
Small molecule
Approved
Unknown
Unknown
Intestinal Obstruction; Kidney Diseases; Liver Diseases; Opioid-Related Disorders; Gastroparesis; Pancreatitis; Constipation; Enteral Nutrition; Ileus
Unknown
Small molecule
Approved
Unknown
Unknown
Colonic Polyps
Unknown