DrugMapper


Display Options: Drug type Therapeutic Area Route of administration Mechanism of Action Indication Status		Total: 6532


Small molecule Approved Unknown Unknown Unknown Unknown


Small molecule Approved Unknown Unknown Osteoporosis; Idiopathic Pulmonary Fibrosis; Essential Hypertension; Stroke; Hypertension; Marfan Syndrome; Severe Acute Respiratory Syndrome; Cardiovascular Diseases Unknown


Small molecule Approved Unknown Unknown Colonic Neoplasms; Breast Neoplasms; Chordoma; Huntington Disease; Alzheimer Disease; Cerebellar Ataxia; Giant Cell Tumors; Glioma; Graft vs Host Disease; Hypertension, Pulmonary; Leukemia, Myeloid, Acute; Melanoma; Neurilemmoma; Parkinson Disease; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Synovitis, Pigmented Villonodular; Gastrointestinal Stromal Tumors; Leukemia; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid; Sarcoma; Neoplasms Unknown

Small molecule

Approved

Unknown

Colonic Neoplasms; Breast Neoplasms; Chordoma; Huntington Disease; Alzheimer Disease; Cerebellar Ataxia; Giant Cell Tumors; Glioma; Graft vs Host Disease; Hypertension, Pulmonary; Leukemia, Myeloid, Acute; Melanoma; Neurilemmoma; Parkinson Disease; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Synovitis, Pigmented Villonodular; Gastrointestinal Stromal Tumors; Leukemia; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid; Sarcoma; Neoplasms

Unknown


Small molecule Approved UROLOGY AND KIDNEY INTRAVENOUS Adenocarcinoma; Astrocytoma; Brain Neoplasms; Breast Neoplasms, Male; Carcinoma; Colonic Neoplasms; Colorectal Neoplasms; Diffuse Intrinsic Pontine Glioma; Genital Neoplasms, Female; Glioma; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Lung Neoplasms; Oligodendroglioma; Peritoneal Neoplasms; Prostatic Neoplasms; Urethral Neoplasms; Uterine Cervical Neoplasms; Adenoma; Arthritis, Rheumatoid; Carcinoma, Endometrioid; Carcinoma, Hepatocellular; Carcinoma, Islet Cell; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Central Nervous System Neoplasms; Endometrial Neoplasms; Fallopian Tube Neoplasms; Ganglioneuroblastoma; Glioblastoma; Gliosarcoma; Hodgkin Disease; Insulinoma; Ischemia; Kidney Neoplasms; Leukemia; Leukemia, Myeloid, Acute; Liver Neoplasms; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Non-Hodgkin; Melanoma; Multiple Myeloma; Multiple Sclerosis, Relapsing-Remitting; Myelodysplastic Syndromes; Neuroblastoma; Osteosarcoma; Ovarian Neoplasms; Peripheral Arterial Disease; Prostatic Neoplasms, Castration-Resistant; Retroviridae Infections; Sarcoma; Small Cell Lung Carcinoma; Somatostatinoma; Thyroid Neoplasms; Urinary Bladder Neoplasms; Breast Neoplasms; Hepatoblastoma; Lymphoma; Lymphoma, Mantle-Cell; Neoplasm Metastasis; Rhabdomyosarcoma, Alveolar; Rhabdomyosarcoma, Embryonal; Carcinoma, Renal Cell; Neoplasms FK506-binding protein 1A inhibitor

Small molecule

Approved

UROLOGY AND KIDNEY

INTRAVENOUS

Adenocarcinoma; Astrocytoma; Brain Neoplasms; Breast Neoplasms, Male; Carcinoma; Colonic Neoplasms; Colorectal Neoplasms; Diffuse Intrinsic Pontine Glioma; Genital Neoplasms, Female; Glioma; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Lung Neoplasms; Oligodendroglioma; Peritoneal Neoplasms; Prostatic Neoplasms; Urethral Neoplasms; Uterine Cervical Neoplasms; Adenoma; Arthritis, Rheumatoid; Carcinoma, Endometrioid; Carcinoma, Hepatocellular; Carcinoma, Islet Cell; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Central Nervous System Neoplasms; Endometrial Neoplasms; Fallopian Tube Neoplasms; Ganglioneuroblastoma; Glioblastoma; Gliosarcoma; Hodgkin Disease; Insulinoma; Ischemia; Kidney Neoplasms; Leukemia; Leukemia, Myeloid, Acute; Liver Neoplasms; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Non-Hodgkin; Melanoma; Multiple Myeloma; Multiple Sclerosis, Relapsing-Remitting; Myelodysplastic Syndromes; Neuroblastoma; Osteosarcoma; Ovarian Neoplasms; Peripheral Arterial Disease; Prostatic Neoplasms, Castration-Resistant; Retroviridae Infections; Sarcoma; Small Cell Lung Carcinoma; Somatostatinoma; Thyroid Neoplasms; Urinary Bladder Neoplasms; Breast Neoplasms; Hepatoblastoma; Lymphoma; Lymphoma, Mantle-Cell; Neoplasm Metastasis; Rhabdomyosarcoma, Alveolar; Rhabdomyosarcoma, Embryonal; Carcinoma, Renal Cell; Neoplasms

FK506-binding protein 1A inhibitor


Small molecule Approved Unknown Unknown Unknown Unknown


Small molecule Approved OTHER INTRAVENOUS Astrocytoma; Gliosarcoma; Head and Neck Neoplasms; Breast Neoplasms, Male; Burkitt Lymphoma; Carcinoma, Non-Small-Cell Lung; Carcinoma, Renal Cell; Carcinoma, Verrucous; Colorectal Neoplasms; Fallopian Tube Neoplasms; Hypopharyngeal Neoplasms; Leukemia; Lung Neoplasms; Lymphoma; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Large-Cell, Anaplastic; Lymphoma, Mantle-Cell; Melanoma; Oropharyngeal Neoplasms; Ovarian Neoplasms; Pancreatic Neoplasms; Peritoneal Neoplasms; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Retroviridae Infections; Sarcoma; Squamous Cell Carcinoma of Head and Neck; Stomach Neoplasms; Tongue Neoplasms; Urethral Neoplasms; Urinary Bladder Neoplasms; Endometrial Neoplasms; Breast Neoplasms; Neoplasms Tubulin inhibitor

Small molecule

Approved

OTHER

INTRAVENOUS

Astrocytoma; Gliosarcoma; Head and Neck Neoplasms; Breast Neoplasms, Male; Burkitt Lymphoma; Carcinoma, Non-Small-Cell Lung; Carcinoma, Renal Cell; Carcinoma, Verrucous; Colorectal Neoplasms; Fallopian Tube Neoplasms; Hypopharyngeal Neoplasms; Leukemia; Lung Neoplasms; Lymphoma; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Large-Cell, Anaplastic; Lymphoma, Mantle-Cell; Melanoma; Oropharyngeal Neoplasms; Ovarian Neoplasms; Pancreatic Neoplasms; Peritoneal Neoplasms; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Retroviridae Infections; Sarcoma; Squamous Cell Carcinoma of Head and Neck; Stomach Neoplasms; Tongue Neoplasms; Urethral Neoplasms; Urinary Bladder Neoplasms; Endometrial Neoplasms; Breast Neoplasms; Neoplasms

Tubulin inhibitor


Small molecule Approved Unknown Unknown Breast Neoplasms; Parkinson Disease; Scleroderma, Systemic; Leukemia, Myelogenous, Chronic, BCR-ABL Positive Bcr/Abl fusion protein


Small molecule Approved Unknown Unknown Heart Failure; Hypertension; Alzheimer Disease; Autistic Disorder; Hypertension, Portal; Lesch-Nyhan Syndrome; Liver Cirrhosis; Phenylketonurias; Pulmonary Disease, Chronic Obstructive; Renal Insufficiency, Chronic Unknown


Small molecule Approved Unknown Unknown Colorectal Neoplasms; Asthma; Dermatitis; Dermatitis, Atopic; Eczema; Rhinitis; Rhinitis, Allergic, Perennial; Rhinitis, Allergic, Seasonal; Rhinitis, Vasomotor; Urticaria; Hypersensitivity Unknown


Small molecule Approved IMMUNE SYSTEM; OTHER ORAL Hypertriglyceridemia; AIDS Dementia Complex; Arthritis, Rheumatoid; Cognitive Dysfunction; Graft vs Host Disease; Hematologic Neoplasms; Hodgkin Disease; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Myelodysplastic Syndromes; Sarcoma, Kaposi; Severe Acute Respiratory Syndrome; Stroke; Acquired Immunodeficiency Syndrome; Infections; Autoimmune Diseases; HIV Infections; Virus Diseases C-C chemokine receptor type 5 antagonist

Small molecule

Approved

IMMUNE SYSTEM; OTHER

ORAL

Hypertriglyceridemia; AIDS Dementia Complex; Arthritis, Rheumatoid; Cognitive Dysfunction; Graft vs Host Disease; Hematologic Neoplasms; Hodgkin Disease; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Myelodysplastic Syndromes; Sarcoma, Kaposi; Severe Acute Respiratory Syndrome; Stroke; Acquired Immunodeficiency Syndrome; Infections; Autoimmune Diseases; HIV Infections; Virus Diseases

C-C chemokine receptor type 5 antagonist


Small molecule Approved CARDIOVASCULAR; OTHER; RESPIRATORY ORAL Anemia, Sickle Cell; Altitude Sickness; Asthma; Hypoplastic Left Heart Syndrome; Severe Acute Respiratory Syndrome; Idiopathic Pulmonary Fibrosis; Vascular Diseases; Familial Primary Pulmonary Hypertension; Hypertension; Hypertension, Pulmonary; Pulmonary Arterial Hypertension Endothelin receptor, ET-A/ET-B antagonist


Small molecule Unknown Unknown Unknown Staphylococcal Infections; Infections; Impetigo 70S ribosome inhibitor


Small molecule Approved NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER ORAL Carcinoma, Non-Small-Cell Lung; Head and Neck Neoplasms; Esophageal Neoplasms; Glioma; Multiple Sclerosis; Neoplasms; Schizophrenia; Sleep Initiation and Maintenance Disorders; Stroke; Brain Injuries; Depressive Disorder; Disorders of Excessive Somnolence; Fatigue; Obesity; Attention Deficit Disorder with Hyperactivity; Narcolepsy; Sleep Apnea, Obstructive; Sleep Wake Disorders Dopamine transporter inhibitor

Small molecule

Approved

NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER

ORAL

Carcinoma, Non-Small-Cell Lung; Head and Neck Neoplasms; Esophageal Neoplasms; Glioma; Multiple Sclerosis; Neoplasms; Schizophrenia; Sleep Initiation and Maintenance Disorders; Stroke; Brain Injuries; Depressive Disorder; Disorders of Excessive Somnolence; Fatigue; Obesity; Attention Deficit Disorder with Hyperactivity; Narcolepsy; Sleep Apnea, Obstructive; Sleep Wake Disorders

Dopamine transporter inhibitor


Small molecule Approved OTHER ORAL Head and Neck Neoplasms; Paraparesis, Tropical Spastic; Hepatitis C; Leukemia, Biphenotypic, Acute; HTLV-I Infections; Liver Cirrhosis, Biliary; Multiple Sclerosis, Relapsing-Remitting; Acquired Immunodeficiency Syndrome; HIV Infections; Infections; Virus Diseases Unknown


Small molecule Approved Unknown Unknown Amphetamine-Related Disorders; Cocaine-Related Disorders; Multiple Sclerosis; Bipolar Disorder; Depressive Disorder; Feeding and Eating Disorders; Attention Deficit Disorder with Hyperactivity Unknown


Small molecule Approved Unknown Unknown Hypertension; Stroke Renin inhibitor


Small molecule Approved Unknown ORAL Urinary Bladder Neoplasms; Carcinoma, Renal Cell; Endometrial Neoplasms; Prostatic Neoplasms, Castration-Resistant; Renal Insufficiency, Chronic; Thyroid Neoplasms; Adenocarcinoma; Brain Neoplasms; Carcinoma, Ductal; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Colorectal Neoplasms; Esophageal Neoplasms; Glioma; Melanoma; Ovarian Neoplasms; Pancreatic Neoplasms; Peritoneal Neoplasms; Pituitary Neoplasms; Stomach Neoplasms; Uterine Cervical Neoplasms; Brain Diseases; Breast Neoplasms; Head and Neck Neoplasms; Sarcoma; Neoplasms Unknown

Small molecule

Approved

Unknown

ORAL

Urinary Bladder Neoplasms; Carcinoma, Renal Cell; Endometrial Neoplasms; Prostatic Neoplasms, Castration-Resistant; Renal Insufficiency, Chronic; Thyroid Neoplasms; Adenocarcinoma; Brain Neoplasms; Carcinoma, Ductal; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Colorectal Neoplasms; Esophageal Neoplasms; Glioma; Melanoma; Ovarian Neoplasms; Pancreatic Neoplasms; Peritoneal Neoplasms; Pituitary Neoplasms; Stomach Neoplasms; Uterine Cervical Neoplasms; Brain Diseases; Breast Neoplasms; Head and Neck Neoplasms; Sarcoma; Neoplasms

Unknown


Small molecule Approved NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER; PEDIATRICS ORAL Pain; Epilepsy; Lennox Gastaut Syndrome; Seizures Sodium channel alpha subunit blocker


Small molecule Approved HEMATOLOGY; OTHER ORAL Myelodysplastic Syndromes; Anemia, Aplastic; Hepatitis C, Chronic; Purpura, Thrombocytopenic, Idiopathic; Thrombocytopenia Thrombopoietin receptor agonist


Small molecule Approved Unknown Unknown Arthritis; Back Pain; Bursitis; Contusions; Muscle Cramp; Myalgia; Pain; Sprains and Strains; Tendinopathy; Wounds and Injuries Unknown


Small molecule Approved Unknown Unknown Brain Injuries; Multiple Myeloma; Nasopharyngeal Neoplasms; Genital Neoplasms, Female; Nausea; Neoplasms; Postoperative Nausea and Vomiting Unknown


Small molecule Approved MUSCULOSKELETAL; OTHER ORAL Tourette Syndrome; Movement Disorders; Huntington Disease Synaptic vesicular amine transporter inhibitor


Small molecule Approved Unknown IV (INFUSION) Hematologic Neoplasms; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Leukemia, Plasma Cell; Myelodysplastic Syndromes; Amyloidosis, Familial; Breast Neoplasms; Hodgkin Disease; Leukemia; Leukemia, Hairy Cell; Lymphoma, B-Cell, Marginal Zone; Lymphoma, T-Cell, Peripheral; Multiple Myeloma; Ovarian Neoplasms; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Waldenstrom Macroglobulinemia; Immunoblastic Lymphadenopathy; Leukemia, Lymphocytic, Chronic, B-Cell; Lymphoma; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Lymphoma, Non-Hodgkin; Neoplasms Unknown

Small molecule

Approved

Unknown

IV (INFUSION)

Hematologic Neoplasms; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Leukemia, Plasma Cell; Myelodysplastic Syndromes; Amyloidosis, Familial; Breast Neoplasms; Hodgkin Disease; Leukemia; Leukemia, Hairy Cell; Lymphoma, B-Cell, Marginal Zone; Lymphoma, T-Cell, Peripheral; Multiple Myeloma; Ovarian Neoplasms; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Waldenstrom Macroglobulinemia; Immunoblastic Lymphadenopathy; Leukemia, Lymphocytic, Chronic, B-Cell; Lymphoma; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Lymphoma, Non-Hodgkin; Neoplasms

Unknown


Small molecule Approved OTHER ORAL Prostatitis; Kidney Calculi; Prostatic Neoplasms, Castration-Resistant; Prostatic Hyperplasia Alpha-1a adrenergic receptor antagonist


Small molecule Approved Unknown ORAL Back Pain; Chronic Pain; Diabetic Neuropathies; Hallux Valgus; Joint Diseases; Low Back Pain; Neoplasms; Neuralgia; Osteoarthritis; Osteoarthritis, Hip; Osteoarthritis, Knee; Pain Unknown


Small molecule Unknown Unknown Unknown Fallopian Tube Neoplasms; Ileus; Ovarian Neoplasms; Peritoneal Neoplasms; Urinary Bladder Neoplasms; Constipation Mu opioid receptor antagonist


Small molecule Unknown Unknown Unknown Colonic Polyps Unknown


Small molecule Approved Unknown Unknown Unknown Diagnostic agent


Small molecule Approved OTHER ORAL Fibromyalgia; Hepatitis C, Chronic; Depressive Disorder; Depressive Disorder, Major Norepinephrine transporter inhibitor


Small molecule Approved Unknown Unknown Coronary Disease Unknown


Small molecule Approved Unknown Unknown Intestinal Obstruction; Kidney Diseases; Liver Diseases; Opioid-Related Disorders; Gastroparesis; Pancreatitis; Constipation; Ileus Unknown


Small molecule Approved Unknown INTRAVENOUS Colonic Neoplasms; Rectal Neoplasms; Esophageal Neoplasms; Anemia; Colorectal Neoplasms; Osteosarcoma Unknown


Small molecule Approved CARDIOVASCULAR; OTHER INTRAVENOUS Vascular Diseases; Scoliosis; Hypertension; Hypertension, Malignant; Cardiovascular Diseases Voltage-gated L-type calcium channel blocker


Small molecule Approved EYE OPHTHALMIC Dry Eye Syndromes; Cataract; Panuveitis; Uveitis; Inflammation; Uveitis, Anterior Glucocorticoid receptor agonist

Small molecule

Approved

Unknown

Diabetic Neuropathies; Tobacco Use Disorder; Deglutition Disorders; Hypertension; Stomach Neoplasms; Arthralgia; Arthritis; Asthma; Back Pain; Bronchitis; Burns; Bursitis; Common Cold; Contusions; Cough; Eczema; Headache; Hemorrhoids; Herpes Labialis; Insect Bites and Stings; Muscle Cramp; Myalgia; Nasal Obstruction; Oral Ulcer; Osteoarthritis; Pain; Pharyngitis; Pruritus; Sprains and Strains; Sunburn; Tendinopathy; Wounds and Injuries

Transient receptor potential cation channel subfamily A member 1 opener