Display Options:
Total: 6532
Small molecule
Approved
Unknown
Unknown
Intestinal Obstruction; Kidney Diseases; Liver Diseases; Opioid-Related Disorders; Gastroparesis; Pancreatitis; Constipation; Enteral Nutrition; Ileus
Unknown
Small molecule
Approved
EYE
OPHTHALMIC
Dry Eye Syndromes; Cataract; Keratitis; Panuveitis; Uveitis; Eye Diseases; Inflammation; Uveitis, Anterior
Glucocorticoid receptor agonist
Small molecule
Approved
Unknown
Unknown
Diabetic Neuropathies; Tobacco Use Disorder; Deglutition Disorders; Hypertension; Stomach Neoplasms; Arthralgia; Arthritis; Asthma; Back Pain; Bronchitis; Burns; Bursitis; Common Cold; Contusions; Cough; Eczema; Headache; Hemorrhoids; Herpes Labialis; Insect Bites and Stings; Muscle Cramp; Myalgia; Nasal Obstruction; Oral Ulcer; Osteoarthritis; Pain; Pharyngitis; Pruritus; Sprains and Strains; Sunburn; Tendinopathy; Wounds and Injuries
Transient receptor potential cation channel subfamily A member 1 opener
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER; PEDIATRICS
ORAL
Pain; Epilepsy; Lennox Gastaut Syndrome; Seizures
Sodium channel alpha subunit blocker
Small molecule
Approved
IMMUNE SYSTEM; OTHER
ORAL
Infections; Acquired Immunodeficiency Syndrome; Friedreich Ataxia; HIV; HIV Infections; Virus Diseases
Human immunodeficiency virus type 1 reverse transcriptase inhibitor
Small molecule
Approved
CANCER
SUBCUTANEOUS
beta-Thalassemia; Blood Platelet Disorders; Diabetes Mellitus, Type 1; Diabetic Foot; End Stage Liver Disease; Glioblastoma; Graft vs Host Disease; Kidney Diseases; Leukemia; Leukemia, Biphenotypic, Acute; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Myeloid, Acute; Lymphoma, Follicular; Lymphoma, Mantle-Cell; Myelodysplastic Syndromes; Neutropenia; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Sarcoma; Syndrome; Thalassemia; Anemia, Sickle Cell; Fanconi Anemia; Gliosarcoma; Granulomatous Disease, Chronic; Head and Neck Neoplasms; Hematologic Neoplasms; Hodgkin Disease; Lymphoma, Large B-Cell, Diffuse; Lymphoma, T-Cell; Lymphopenia; Pancreatic Neoplasms; Scleroderma, Systemic; Hematopoietic Stem Cell Transplantation; Lymphoma; Lymphoma, Non-Hodgkin; Multiple Myeloma; Neoplasms
C-X-C chemokine receptor type 4 partial agonist
Small molecule
Approved
Unknown
ORAL
Anemia; Liver Cirrhosis; Multiple Myeloma; Osteosarcoma; Blood Platelet Disorders; Fanconi Anemia; Graft vs Host Disease; Leukemia; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Myeloid, Acute; Liver Diseases; Lymphoma; Myelodysplastic Syndromes; Wiskott-Aldrich Syndrome; Anemia, Aplastic; Hemorrhage; Hepatitis C; Hepatitis C, Chronic; Neoplasms; Purpura, Thrombocytopenic, Idiopathic; Thrombocytopenia
Unknown
Small molecule
Approved
OTHER
ORAL
Premature Ejaculation; Prostatitis; Kidney Calculi; Prostatic Neoplasms, Castration-Resistant; Urolithiasis; Prostatic Hyperplasia
Alpha-1a adrenergic receptor antagonist
Small molecule
Approved
Unknown
Unknown
Angina, Stable; Hypertension; Kidney Calculi; Kidney Diseases; Non-alcoholic Fatty Liver Disease; Cardiovascular Diseases; Tumor Lysis Syndrome; Arthritis, Gouty; Gout; Hyperuricemia
Xanthine dehydrogenase inhibitor
Small molecule
Approved
Unknown
Unknown
Influenza, Human; Metabolic Syndrome; Renal Insufficiency; Breast Neoplasms; Coronary Disease; Diabetes Mellitus, Type 1; Diabetes Mellitus, Type 2; Hypercholesterolemia; Hyperlipidemias; Lipid Metabolism Disorders; Cardiovascular Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Rhinitis, Allergic, Perennial; Conjunctivitis, Allergic; Pruritus
Histamine H1 receptor antagonist
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM
TOPICAL
Amyotrophic Lateral Sclerosis; Brain Injuries; Cough; Migraine Disorders; Pruritus; Stroke; Cardiovascular Diseases; Facial Pain; HIV Infections; Hypertension, Pulmonary; Morton Neuroma; Myofascial Pain Syndromes; Nausea; Neuralgia, Postherpetic; Neuroma; Tennis Elbow; Vomiting; Angina, Stable; Breast Neoplasms; Common Cold; Diabetic Neuropathies; Head and Neck Neoplasms; Herpes Zoster; Osteoarthritis, Knee; Peripheral Nervous System Diseases; Arthralgia; Arthritis; Back Pain; Bursitis; Contusions; Muscle Cramp; Myalgia; Neuralgia; Osteoarthritis; Pain; Sprains and Strains; Tendinopathy
Vanilloid receptor opener
Small molecule
Approved
OTHER
SUBLINGUAL
Psychotic Disorders; Stuttering; Bipolar Disorder; Schizophrenia
Dopamine D2 receptor antagonist
Small molecule
Approved
OTHER
ORAL
Liver Diseases; Stress Disorders, Post-Traumatic; Bipolar Disorder; Psychotic Disorders; Schizophrenia
Dopamine D2 receptor antagonist
Small molecule
Approved
Unknown
Unknown
HIV Infections; Schistosomiasis haematobia; Fever; Malaria, Falciparum; Malaria, Vivax; Malaria
Ferriprotoporphyrin IX inhibitor
Small molecule
Approved
Unknown
ORAL
Arrhythmias, Cardiac; Atrial Fibrillation; Atrial Flutter; Heart Failure
Unknown
Small molecule
Approved
Unknown
ORAL
Motor Activity; Diabetes Mellitus, Type 1; Glucose Intolerance; Diabetes Mellitus; Diabetes Mellitus, Type 2; Myocardial Infarction; Polycystic Ovary Syndrome
Unknown
Small molecule
Approved
OTHER; PEDIATRICS
ORAL
Tourette Syndrome; Alcoholism; Amphetamine-Related Disorders; Cocaine-Related Disorders; Obesity; Tuberous Sclerosis; Epilepsies, Partial; Epilepsy; Epilepsy, Complex Partial; Spasms, Infantile
Gamma-amino-N-butyrate transaminase inhibitor
Small molecule
Approved
Unknown
Unknown
Irritable Bowel Syndrome; Low Back Pain; Neuralgia; Fibromyalgia; Peripheral Nervous System Diseases; Depressive Disorder
Unknown
Small molecule
Approved
Unknown
SUBLINGUAL; TRANSDERMAL
Bipolar Disorder; Psychotic Disorders; Schizophrenia
Unknown
Small molecule
Approved
CANCER; OTHER
INJECTION; INTRAVENOUS
Fallopian Tube Neoplasms; Lymphoma, Large-Cell, Anaplastic; Lymphoma, T-Cell, Cutaneous; Multiple Myeloma; Mycosis Fungoides; Ovarian Neoplasms; Peritoneal Neoplasms; Sezary Syndrome; Breast Neoplasms; Carcinoma, Non-Small-Cell Lung; Head and Neck Neoplasms; Leukemia-Lymphoma, Adult T-Cell; Lung Neoplasms; Lymphoma; Lymphoma, T-Cell; Lymphoma, T-Cell, Peripheral; Neoplasms
Dihydrofolate reductase inhibitor
Small molecule
Approved
CANCER; IMMUNE SYSTEM; OTHER; UROLOGY AND KIDNEY
ORAL
Acute Coronary Syndrome; Adenocarcinoma; Aging; Breast Neoplasms, Male; Carcinoma, Ovarian Epithelial; Central Nervous System Neoplasms; Esophageal Neoplasms; Fallopian Tube Neoplasms; Gastrointestinal Stromal Tumors; Hamartoma Syndrome, Multiple; Hematologic Diseases; Leukemia; Leukemia, Lymphoid; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Lymphoma, Non-Hodgkin; Nasopharyngeal Neoplasms; Neoplasm Metastasis; Neoplasms, Plasma Cell; Peritoneal Neoplasms; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Progeria; Sarcoma, Synovial; Uterine Cervical Neoplasms; Adenoma, Islet Cell; Bile Duct Neoplasms; Brain Neoplasms; Carcinoma, Adenoid Cystic; Carcinoma, Hepatocellular; Carcinoma, Medullary; Carcinoma, Neuroendocrine; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Carcinoma, Transitional Cell; Cholangiocarcinoma; Chondrosarcoma; Colonic Neoplasms; Colorectal Neoplasms; Diffuse Intrinsic Pontine Glioma; Endometrial Neoplasms; Ependymoma; Epilepsy; Gallbladder Neoplasms; Glioblastoma; Glioma; Head and Neck Neoplasms; Hepatitis C; Hodgkin Disease; Hyperaldosteronism; Kidney Diseases; Leukemia, Myeloid, Acute; Liver Neoplasms; Lung Neoplasms; Lymphangioleiomyomatosis; Lymphoma; Lymphoma, B-Cell, Marginal Zone; Lymphoma, Mantle-Cell; Lymphoma, T-Cell, Cutaneous; Macular Degeneration; Mastocytosis, Systemic; Melanoma; Meningioma; Mesothelioma; Multiple Myeloma; Myelodysplastic Syndromes; Neoplasms, Germ Cell and Embryonal; Neurilemmoma; Neurofibromatosis 1; Neurofibromatosis 2; Oligodendroglioma; Osteosarcoma; Ovarian Neoplasms; Paraganglioma; Peutz-Jeghers Syndrome; Polycystic Kidney Diseases; Sarcoma; Sarcoma, Kaposi; Small Cell Lung Carcinoma; Sturge-Weber Syndrome; Thymus Neoplasms; Thyroid Neoplasms; Triple Negative Breast Neoplasms; Tuberculosis; Urinary Bladder Neoplasms; Uterine Neoplasms; Uveal Melanoma; Uveitis; Waldenstrom Macroglobulinemia; Carcinoid Tumor; Carcinoma; Coronary Disease; Coronary Restenosis; Cytomegalovirus Infections; Endocardial Cushion Defects; Graft vs Host Disease; Infections; Kidney Failure, Chronic; Kidney Neoplasms; Lymphoma, Large B-Cell, Diffuse; Malignant Carcinoid Syndrome; Polycystic Kidney, Autosomal Dominant; Prostatic Neoplasms, Castration-Resistant; Renal Insufficiency; Renal Insufficiency, Chronic; Skin Neoplasms; Stomach Neoplasms; Angiomyolipoma; Astrocytoma; Breast Neoplasms; Carcinoma, Renal Cell; Neoplasms; Neuroendocrine Tumors; Pancreatic Neoplasms; Tuberous Sclerosis
FK506-binding protein 1A inhibitor
Small molecule
Approved
Unknown
Unknown
Breast Neoplasms; Carcinoma, Intraductal, Noninfiltrating; Osteoporosis, Postmenopausal; Menopause; Osteoporosis
Unknown
Small molecule
Approved
OTHER
ORAL
Barrett Esophagus; Esophagitis, Peptic; Esophagitis; Gastroesophageal Reflux; Heartburn; Peptic Ulcer
Potassium-transporting ATPase inhibitor
Small molecule
Approved
Unknown
Unknown
HIV Infections; Neoplasms; Schistosomiasis haematobia; Fever; Malaria, Falciparum; Malaria, Vivax; Malaria
Ferriprotoporphyrin IX inhibitor
Small molecule
Approved
Unknown
Unknown
Cataract; Conjunctivitis, Bacterial; Eye Infections
Unknown
Small molecule
Approved
OTHER
TOPICAL
Ectoparasitic Infestations; Lice Infestations; Otitis Externa
Unknown
Small molecule
Approved
Unknown
Unknown
Rhinitis, Allergic, Seasonal; Conjunctivitis, Allergic; Dermatitis; Rhinitis, Allergic, Perennial
Unknown
Small molecule
Approved
HEMATOLOGY; OTHER
ORAL
Carcinoma; Kidney Diseases; Kidney Failure, Chronic; Dyspnea; Edema, Cardiac; Liver Cirrhosis; Cardiovascular Diseases; Heart Failure; Hyponatremia; Inappropriate ADH Syndrome; Polycystic Kidney, Autosomal Dominant; Polycystic Kidney Diseases
Vasopressin V2 receptor antagonist
Small molecule
Approved
Unknown
Unknown
Carcinoma, Hepatocellular; Colorectal Neoplasms; Corneal Neovascularization; Glioblastoma; Lymphoma; Psoriasis; Breast Neoplasms; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Central Nervous System Neoplasms; Chondrosarcoma; Dermatofibrosarcoma; Fallopian Tube Neoplasms; Gastrointestinal Stromal Tumors; Gliosarcoma; Hemangiosarcoma; Kidney Neoplasms; Leiomyosarcoma; Leukemia, Myeloid, Acute; Liposarcoma; Lung Neoplasms; Lymphedema; Macular Degeneration; Melanoma; Neoplasms, Germ Cell and Embryonal; Neuroendocrine Tumors; Osteosarcoma; Pancreatic Neoplasms; Paraganglioma; Peritoneal Neoplasms; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Salivary Gland Neoplasms; Sarcoma, Alveolar Soft Part; Small Cell Lung Carcinoma; Solitary Fibrous Tumors; Stomach Neoplasms; Telangiectasia, Hereditary Hemorrhagic; Thyroid Neoplasms; Urinary Bladder Neoplasms; Uterine Cervical Neoplasms; Carcinoma, Renal Cell; Neoplasms; Ovarian Neoplasms; Sarcoma
Unknown
Small molecule
Approved
Unknown
Unknown
HIV Infections; Asthma; Cardiovascular Diseases; Heart Diseases; Acute Coronary Syndrome; Anemia, Sickle Cell; Atrial Fibrillation; Coronary Disease; Influenza, Human; Kidney Failure, Chronic; Myocardial Infarction; Pneumonia; Severe Acute Respiratory Syndrome; ST Elevation Myocardial Infarction; Thrombosis
Unknown
Small molecule
Approved
IMMUNE SYSTEM; OTHER; RESPIRATORY
INJECTION
Renal Insufficiency, Chronic; Gram-Positive Bacterial Infections; Infections; Bacteremia; Bacterial Infections; Pneumonia, Bacterial; Staphylococcal Skin Infections
Unknown