DrugMapper


Display Options: Drug type Therapeutic Area Route of administration Mechanism of Action Indication Status		Total: 6532


Small molecule Approved CARDIOVASCULAR; OTHER INTRAVENOUS Vascular Diseases; Scoliosis; Hypertension; Hypertension, Malignant; Cardiovascular Diseases Voltage-gated L-type calcium channel blocker


Small molecule Approved EYE OPHTHALMIC Dry Eye Syndromes; Cataract; Panuveitis; Uveitis; Inflammation; Uveitis, Anterior Glucocorticoid receptor agonist


Small molecule Approved Unknown INTRAVENOUS Colonic Neoplasms; Rectal Neoplasms; Esophageal Neoplasms; Anemia; Colorectal Neoplasms; Osteosarcoma Unknown


Small molecule Approved Unknown Unknown Diabetic Neuropathies; Tobacco Use Disorder; Deglutition Disorders; Hypertension; Stomach Neoplasms; Arthralgia; Arthritis; Asthma; Back Pain; Bronchitis; Burns; Bursitis; Common Cold; Contusions; Cough; Eczema; Headache; Hemorrhoids; Herpes Labialis; Insect Bites and Stings; Muscle Cramp; Myalgia; Nasal Obstruction; Oral Ulcer; Osteoarthritis; Pain; Pharyngitis; Pruritus; Sprains and Strains; Sunburn; Tendinopathy; Wounds and Injuries Transient receptor potential cation channel subfamily A member 1 opener

Small molecule

Approved

Unknown

Diabetic Neuropathies; Tobacco Use Disorder; Deglutition Disorders; Hypertension; Stomach Neoplasms; Arthralgia; Arthritis; Asthma; Back Pain; Bronchitis; Burns; Bursitis; Common Cold; Contusions; Cough; Eczema; Headache; Hemorrhoids; Herpes Labialis; Insect Bites and Stings; Muscle Cramp; Myalgia; Nasal Obstruction; Oral Ulcer; Osteoarthritis; Pain; Pharyngitis; Pruritus; Sprains and Strains; Sunburn; Tendinopathy; Wounds and Injuries

Transient receptor potential cation channel subfamily A member 1 opener


Small molecule Approved Unknown Unknown Unknown Unknown


Small molecule Approved OTHER; UROLOGY AND KIDNEY ORAL Urinary Incontinence; Urinary Bladder, Overactive; Urinary Incontinence, Urge Muscarinic acetylcholine receptor M2 antagonist


Small molecule Approved OTHER INTRAVENOUS Anemia, Sickle Cell; Retinal Artery Occlusion; Coronary Disease; Cardiovascular Diseases Adenosine A2a receptor agonist


Small molecule Approved CANCER SUBCUTANEOUS Diabetes Mellitus, Type 1; Diabetic Foot; End Stage Liver Disease; Graft vs Host Disease; Kidney Diseases; Leukemia; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Myeloid, Acute; Lymphoma, Follicular; Lymphoma, Mantle-Cell; Myelodysplastic Syndromes; Neutropenia; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Sarcoma; Thalassemia; Anemia, Sickle Cell; Fanconi Anemia; Gliosarcoma; Granulomatous Disease, Chronic; Head and Neck Neoplasms; Hematologic Neoplasms; Hodgkin Disease; Lymphoma; Lymphoma, Large B-Cell, Diffuse; Lymphoma, T-Cell; Lymphopenia; Neoplasms; Pancreatic Neoplasms; Scleroderma, Systemic; Lymphoma, Non-Hodgkin; Multiple Myeloma C-X-C chemokine receptor type 4 partial agonist

Small molecule

Approved

CANCER

SUBCUTANEOUS

Diabetes Mellitus, Type 1; Diabetic Foot; End Stage Liver Disease; Graft vs Host Disease; Kidney Diseases; Leukemia; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Myeloid, Acute; Lymphoma, Follicular; Lymphoma, Mantle-Cell; Myelodysplastic Syndromes; Neutropenia; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Sarcoma; Thalassemia; Anemia, Sickle Cell; Fanconi Anemia; Gliosarcoma; Granulomatous Disease, Chronic; Head and Neck Neoplasms; Hematologic Neoplasms; Hodgkin Disease; Lymphoma; Lymphoma, Large B-Cell, Diffuse; Lymphoma, T-Cell; Lymphopenia; Neoplasms; Pancreatic Neoplasms; Scleroderma, Systemic; Lymphoma, Non-Hodgkin; Multiple Myeloma

C-X-C chemokine receptor type 4 partial agonist


Small molecule Approved Unknown ORAL Multiple Myeloma; Anemia; Liver Cirrhosis; Osteosarcoma; Blood Platelet Disorders; Fanconi Anemia; Graft vs Host Disease; Leukemia; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Myeloid, Acute; Liver Diseases; Myelodysplastic Syndromes; Wiskott-Aldrich Syndrome; Anemia, Aplastic; Hepatitis C; Hepatitis C, Chronic; Neoplasms; Purpura, Thrombocytopenic, Idiopathic; Thrombocytopenia; Hemorrhage Unknown

Small molecule

Approved

Unknown

ORAL

Multiple Myeloma; Anemia; Liver Cirrhosis; Osteosarcoma; Blood Platelet Disorders; Fanconi Anemia; Graft vs Host Disease; Leukemia; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Myeloid, Acute; Liver Diseases; Myelodysplastic Syndromes; Wiskott-Aldrich Syndrome; Anemia, Aplastic; Hepatitis C; Hepatitis C, Chronic; Neoplasms; Purpura, Thrombocytopenic, Idiopathic; Thrombocytopenia; Hemorrhage

Unknown


Small molecule Approved MUSCULOSKELETAL; OTHER ORAL Tourette Syndrome; Movement Disorders; Huntington Disease Synaptic vesicular amine transporter inhibitor


Small molecule Approved Unknown Unknown Breast Neoplasms; Leukemia; Myelodysplastic Syndromes; Ovarian Neoplasms; Carcinoma, Non-Small-Cell Lung Glutathione reductase


Small molecule Approved Unknown Unknown Carcinoma, Hepatocellular; Colorectal Neoplasms; Corneal Neovascularization; Glioblastoma; Lymphoma; Psoriasis; Breast Neoplasms; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Chondrosarcoma; Dermatofibrosarcoma; Fallopian Tube Neoplasms; Gastrointestinal Stromal Tumors; Glioma; Gliosarcoma; Hemangiosarcoma; Kidney Neoplasms; Leiomyosarcoma; Leukemia, Myeloid, Acute; Liposarcoma; Lung Neoplasms; Lymphedema; Macular Degeneration; Melanoma; Neoplasms, Germ Cell and Embryonal; Neuroendocrine Tumors; Osteosarcoma; Pancreatic Neoplasms; Peritoneal Neoplasms; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Salivary Gland Neoplasms; Sarcoma, Alveolar Soft Part; Small Cell Lung Carcinoma; Solitary Fibrous Tumors; Stomach Neoplasms; Telangiectasia, Hereditary Hemorrhagic; Thyroid Neoplasms; Urinary Bladder Neoplasms; Uterine Cervical Neoplasms; Carcinoma, Renal Cell; Ovarian Neoplasms; Sarcoma; Neoplasms Unknown

Small molecule

Approved

Unknown

Carcinoma, Hepatocellular; Colorectal Neoplasms; Corneal Neovascularization; Glioblastoma; Lymphoma; Psoriasis; Breast Neoplasms; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Chondrosarcoma; Dermatofibrosarcoma; Fallopian Tube Neoplasms; Gastrointestinal Stromal Tumors; Glioma; Gliosarcoma; Hemangiosarcoma; Kidney Neoplasms; Leiomyosarcoma; Leukemia, Myeloid, Acute; Liposarcoma; Lung Neoplasms; Lymphedema; Macular Degeneration; Melanoma; Neoplasms, Germ Cell and Embryonal; Neuroendocrine Tumors; Osteosarcoma; Pancreatic Neoplasms; Peritoneal Neoplasms; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Salivary Gland Neoplasms; Sarcoma, Alveolar Soft Part; Small Cell Lung Carcinoma; Solitary Fibrous Tumors; Stomach Neoplasms; Telangiectasia, Hereditary Hemorrhagic; Thyroid Neoplasms; Urinary Bladder Neoplasms; Uterine Cervical Neoplasms; Carcinoma, Renal Cell; Ovarian Neoplasms; Sarcoma; Neoplasms

Unknown


Small molecule Approved CANCER; IMMUNE SYSTEM; OTHER; UROLOGY AND KIDNEY ORAL Acute Coronary Syndrome; Adenocarcinoma; Breast Neoplasms, Male; Central Nervous System Neoplasms; Colonic Neoplasms; Esophageal Neoplasms; Fallopian Tube Neoplasms; Gallbladder Neoplasms; Gastrointestinal Stromal Tumors; Hamartoma Syndrome, Multiple; Hematologic Diseases; Leukemia; Leukemia, Lymphoid; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Lymphoma, Non-Hodgkin; Nasopharyngeal Neoplasms; Neoplasm Metastasis; Ovarian Neoplasms; Peritoneal Neoplasms; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Progeria; Sarcoma, Synovial; Triple Negative Breast Neoplasms; Uterine Cervical Neoplasms; Adenoma, Islet Cell; Brain Neoplasms; Carcinoma, Adenoid Cystic; Carcinoma, Hepatocellular; Carcinoma, Medullary; Carcinoma, Neuroendocrine; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Carcinoma, Transitional Cell; Cholangiocarcinoma; Chondrosarcoma; Colorectal Neoplasms; Diffuse Intrinsic Pontine Glioma; Endometrial Hyperplasia; Endometrial Neoplasms; Ependymoma; Epilepsy; Glioblastoma; Glioma; Head and Neck Neoplasms; Hepatitis C; Hodgkin Disease; Hyperaldosteronism; Kidney Diseases; Leukemia, Myeloid, Acute; Liver Neoplasms; Lung Neoplasms; Lymphangioleiomyomatosis; Lymphoma; Lymphoma, B-Cell, Marginal Zone; Lymphoma, Mantle-Cell; Lymphoma, T-Cell, Cutaneous; Macular Degeneration; Mastocytosis, Systemic; Melanoma; Meningioma; Mesothelioma; Multiple Myeloma; Myelodysplastic Syndromes; Neoplasms, Germ Cell and Embryonal; Neurilemmoma; Neurofibromatosis 1; Neurofibromatosis 2; Oligodendroglioma; Osteosarcoma; Pancreatic Neoplasms; Peutz-Jeghers Syndrome; Polycystic Kidney Diseases; Sarcoma; Sarcoma, Kaposi; Small Cell Lung Carcinoma; Thymus Neoplasms; Thyroid Neoplasms; Tuberculosis; Urinary Bladder Neoplasms; Uterine Neoplasms; Uveitis; Waldenstrom Macroglobulinemia; Carcinoid Tumor; Carcinoma; Coronary Restenosis; Cytomegalovirus Infections; Endocardial Cushion Defects; Graft vs Host Disease; Infections; Kidney Neoplasms; Lymphoma, Large B-Cell, Diffuse; Malignant Carcinoid Syndrome; Polycystic Kidney, Autosomal Dominant; Prostatic Neoplasms, Castration-Resistant; Renal Insufficiency; Renal Insufficiency, Chronic; Skin Neoplasms; Stomach Neoplasms; Angiomyolipoma; Astrocytoma; Breast Neoplasms; Carcinoma, Renal Cell; Immune System Diseases; Neoplasms; Neuroendocrine Tumors; Tuberous Sclerosis FK506-binding protein 1A inhibitor

Small molecule

Approved

CANCER; IMMUNE SYSTEM; OTHER; UROLOGY AND KIDNEY

ORAL

Acute Coronary Syndrome; Adenocarcinoma; Breast Neoplasms, Male; Central Nervous System Neoplasms; Colonic Neoplasms; Esophageal Neoplasms; Fallopian Tube Neoplasms; Gallbladder Neoplasms; Gastrointestinal Stromal Tumors; Hamartoma Syndrome, Multiple; Hematologic Diseases; Leukemia; Leukemia, Lymphoid; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Lymphoma, Non-Hodgkin; Nasopharyngeal Neoplasms; Neoplasm Metastasis; Ovarian Neoplasms; Peritoneal Neoplasms; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Progeria; Sarcoma, Synovial; Triple Negative Breast Neoplasms; Uterine Cervical Neoplasms; Adenoma, Islet Cell; Brain Neoplasms; Carcinoma, Adenoid Cystic; Carcinoma, Hepatocellular; Carcinoma, Medullary; Carcinoma, Neuroendocrine; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Carcinoma, Transitional Cell; Cholangiocarcinoma; Chondrosarcoma; Colorectal Neoplasms; Diffuse Intrinsic Pontine Glioma; Endometrial Hyperplasia; Endometrial Neoplasms; Ependymoma; Epilepsy; Glioblastoma; Glioma; Head and Neck Neoplasms; Hepatitis C; Hodgkin Disease; Hyperaldosteronism; Kidney Diseases; Leukemia, Myeloid, Acute; Liver Neoplasms; Lung Neoplasms; Lymphangioleiomyomatosis; Lymphoma; Lymphoma, B-Cell, Marginal Zone; Lymphoma, Mantle-Cell; Lymphoma, T-Cell, Cutaneous; Macular Degeneration; Mastocytosis, Systemic; Melanoma; Meningioma; Mesothelioma; Multiple Myeloma; Myelodysplastic Syndromes; Neoplasms, Germ Cell and Embryonal; Neurilemmoma; Neurofibromatosis 1; Neurofibromatosis 2; Oligodendroglioma; Osteosarcoma; Pancreatic Neoplasms; Peutz-Jeghers Syndrome; Polycystic Kidney Diseases; Sarcoma; Sarcoma, Kaposi; Small Cell Lung Carcinoma; Thymus Neoplasms; Thyroid Neoplasms; Tuberculosis; Urinary Bladder Neoplasms; Uterine Neoplasms; Uveitis; Waldenstrom Macroglobulinemia; Carcinoid Tumor; Carcinoma; Coronary Restenosis; Cytomegalovirus Infections; Endocardial Cushion Defects; Graft vs Host Disease; Infections; Kidney Neoplasms; Lymphoma, Large B-Cell, Diffuse; Malignant Carcinoid Syndrome; Polycystic Kidney, Autosomal Dominant; Prostatic Neoplasms, Castration-Resistant; Renal Insufficiency; Renal Insufficiency, Chronic; Skin Neoplasms; Stomach Neoplasms; Angiomyolipoma; Astrocytoma; Breast Neoplasms; Carcinoma, Renal Cell; Immune System Diseases; Neoplasms; Neuroendocrine Tumors; Tuberous Sclerosis

FK506-binding protein 1A inhibitor


Small molecule Approved Unknown Unknown Rhinitis, Allergic, Seasonal; Conjunctivitis, Allergic; Dermatitis; Rhinitis, Allergic, Perennial Unknown


Small molecule Unknown Unknown Unknown Angina, Stable; Hypertension; Kidney Calculi; Kidney Diseases; Non-alcoholic Fatty Liver Disease; Cardiovascular Diseases; Tumor Lysis Syndrome; Gout; Hyperuricemia Xanthine dehydrogenase inhibitor


Small molecule Approved IMMUNE SYSTEM; OTHER; RESPIRATORY INJECTION Renal Insufficiency, Chronic; Gram-Positive Bacterial Infections; Infections; Bacteremia; Pneumonia, Bacterial; Staphylococcal Skin Infections; Bacterial Infections Unknown


Small molecule Approved OTHER TOPICAL Ectoparasitic Infestations; Lice Infestations; Otitis Externa; Pruritus Unknown


Small molecule Approved Unknown Unknown HIV Infections; Asthma; Heart Diseases; Acute Coronary Syndrome; Anemia, Sickle Cell; Atrial Fibrillation; Coronary Disease; Myocardial Infarction; Renal Insufficiency, Chronic; ST Elevation Myocardial Infarction; Thrombosis Unknown


Small molecule Approved OTHER SUBLINGUAL Psychotic Disorders; Bipolar Disorder; Schizophrenia Dopamine D2 receptor antagonist


Small molecule Approved Unknown SUBLINGUAL; TRANSDERMAL Bipolar Disorder; Psychotic Disorders; Schizophrenia Unknown


Small molecule Approved Unknown Unknown Rhinitis, Allergic, Perennial; Conjunctivitis, Allergic; Pruritus Histamine H1 receptor antagonist


Small molecule Approved Unknown Unknown Breast Neoplasms; Carcinoma, Intraductal, Noninfiltrating; Osteoporosis, Postmenopausal; Endometrial Hyperplasia; Menopause; Osteoporosis Unknown


Small molecule Approved NEUROLOGY DRUGS & NERVOUS SYSTEM TOPICAL Amyotrophic Lateral Sclerosis; Brain Injuries; Cough; Migraine Disorders; Pruritus; Stroke; Facial Pain; HIV Infections; Hypertension, Pulmonary; Myofascial Pain Syndromes; Nausea; Neuralgia, Postherpetic; Neuroma; Tennis Elbow; Vomiting; Angina, Stable; Breast Neoplasms; Diabetic Neuropathies; Head and Neck Neoplasms; Herpes Zoster; Osteoarthritis, Knee; Peripheral Nervous System Diseases; Arthralgia; Arthritis; Back Pain; Bursitis; Contusions; Muscle Cramp; Myalgia; Neuralgia; Osteoarthritis; Pain; Sprains and Strains; Tendinopathy Vanilloid receptor opener

Small molecule

Approved

NEUROLOGY DRUGS & NERVOUS SYSTEM

TOPICAL

Amyotrophic Lateral Sclerosis; Brain Injuries; Cough; Migraine Disorders; Pruritus; Stroke; Facial Pain; HIV Infections; Hypertension, Pulmonary; Myofascial Pain Syndromes; Nausea; Neuralgia, Postherpetic; Neuroma; Tennis Elbow; Vomiting; Angina, Stable; Breast Neoplasms; Diabetic Neuropathies; Head and Neck Neoplasms; Herpes Zoster; Osteoarthritis, Knee; Peripheral Nervous System Diseases; Arthralgia; Arthritis; Back Pain; Bursitis; Contusions; Muscle Cramp; Myalgia; Neuralgia; Osteoarthritis; Pain; Sprains and Strains; Tendinopathy

Vanilloid receptor opener


Small molecule Approved Unknown ORAL Atrial Fibrillation; Atrial Flutter; Heart Failure; Arrhythmias, Cardiac Unknown


Small molecule Approved OTHER ORAL Liver Diseases; Stress Disorders, Post-Traumatic; Bipolar Disorder; Psychotic Disorders; Schizophrenia Dopamine D2 receptor antagonist


Small molecule Approved OTHER ORAL Barrett Esophagus; Esophagitis, Peptic; Duodenal Ulcer; Esophagitis; Gastroesophageal Reflux; Heartburn; Peptic Ulcer; Stomach Ulcer Potassium-transporting ATPase inhibitor


Small molecule Approved Unknown Unknown Irritable Bowel Syndrome; Low Back Pain; Neuralgia; Fibromyalgia; Peripheral Nervous System Diseases; Depressive Disorder Unknown

Small molecule

Approved

CANCER; OTHER

INJECTION; INTRAVENOUS

Fallopian Tube Neoplasms; Lymphoma, Large-Cell, Anaplastic; Lymphoma, T-Cell, Cutaneous; Multiple Myeloma; Mycosis Fungoides; Ovarian Neoplasms; Peritoneal Neoplasms; Sezary Syndrome; Breast Neoplasms; Carcinoma, Non-Small-Cell Lung; Head and Neck Neoplasms; Leukemia-Lymphoma, Adult T-Cell; Lung Neoplasms; Lymphoma; Lymphoma, T-Cell; Lymphoma, T-Cell, Peripheral; Neoplasms

Dihydrofolate reductase inhibitor


Small molecule Approved Unknown Unknown HIV Infections; Schistosomiasis haematobia; Fever; Malaria, Falciparum; Malaria, Vivax; Malaria Ferriprotoporphyrin IX inhibitor


Small molecule Approved OTHER; PEDIATRICS ORAL Tourette Syndrome; Alcoholism; Amphetamine-Related Disorders; Cocaine-Related Disorders; Obesity; Tuberous Sclerosis; Epilepsy; Epilepsy, Complex Partial; Spasms, Infantile Gamma-amino-N-butyrate transaminase inhibitor


Small molecule Approved HEMATOLOGY; OTHER ORAL Kidney Calculi; Carcinoma; Kidney Diseases; Renal Insufficiency, Chronic; Dyspnea; Edema, Cardiac; Inappropriate ADH Syndrome; Liver Cirrhosis; Polycystic Kidney, Autosomal Dominant; Cardiovascular Diseases; Heart Failure; Hyponatremia; Polycystic Kidney Diseases Vasopressin V2 receptor antagonist


Small molecule Approved Unknown Unknown Cataract; Conjunctivitis, Bacterial; Eye Infections Unknown


Small molecule Approved Unknown ORAL Diabetes Mellitus, Type 1; Glucose Intolerance; Diabetes Mellitus, Type 2; Myocardial Infarction; Polycystic Ovary Syndrome; Diabetes Mellitus Unknown


Small molecule Approved Unknown Unknown Influenza, Human; Metabolic Syndrome; Renal Insufficiency; Breast Neoplasms; Coronary Disease; Diabetes Mellitus, Type 1; Diabetes Mellitus, Type 2; Hypercholesterolemia; Hyperlipidemias; Ischemic Stroke; Lipid Metabolism Disorders; Cardiovascular Diseases Unknown


Small molecule Approved Unknown Unknown HIV Infections; Neoplasms; Schistosomiasis haematobia; Fever; Malaria, Falciparum; Malaria, Vivax; Malaria Ferriprotoporphyrin IX inhibitor