Display Options:
Total: 6532
Small molecule
Investigational
Unknown
Unknown
Arthritis, Rheumatoid; Osteoarthritis
P2X purinoceptor 7 antagonist
Small molecule
Investigational
Unknown
Unknown
Depressive Disorder, Major; Hypercholesterolemia; Obesity; Weight Gain; Vertigo
Histamine H1 receptor agonist
Small molecule
Investigational
Unknown
Unknown
Unknown
Unknown
Small molecule
Investigational
Unknown
Unknown
Unknown
Unknown
Small molecule
Investigational
Unknown
Unknown
Chronic Pain; Neuralgia; Fibromyalgia
Mu opioid receptor agonist
Small molecule
Investigational
Unknown
Unknown
Brain Neoplasms; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Central Nervous System Neoplasms; Colorectal Neoplasms; Head and Neck Neoplasms; Leukemia, Myeloid, Acute; Leukemia, Myelomonocytic, Chronic; Medulloblastoma; Myelodysplastic Syndromes; Neoplasm Metastasis; Neoplasms; Ovarian Neoplasms; Small Cell Lung Carcinoma
Serine/threonine-protein kinase Chk1 inhibitor
Small molecule
Investigational
Unknown
Unknown
Tobacco Use Disorder
Unknown
Small molecule
Investigational
Unknown
Unknown
Adenocarcinoma of Lung; Breast Neoplasms; Carcinoma, Squamous Cell; Colonic Neoplasms; Colorectal Neoplasms; Multiple Myeloma; Neoplasms; Rectal Neoplasms; Carcinoma, Non-Small-Cell Lung; Gastrointestinal Stromal Tumors; Lymphoma; Myeloproliferative Disorders; Stomach Neoplasms
Heat shock protein HSP90 inhibitor
Small molecule
Investigational
Unknown
Unknown
Idiopathic Pulmonary Fibrosis
c-Jun N-terminal kinase 1 inhibitor
Small molecule
Investigational
Unknown
Unknown
Breast Neoplasms; Hemangiosarcoma
Unknown
Small molecule
Investigational
Unknown
Unknown
Unknown
Dopamine D3 receptor agonist
Small molecule
Investigational
Unknown
Unknown
Unknown
Unknown
Small molecule
Investigational
Unknown
Unknown
Hypertension, Pulmonary
Unknown
Small molecule
Investigational
Unknown
Unknown
Unknown
Isocitrate dehydrogenase [NADP] cytoplasmic inhibitor
Small molecule
Investigational
Unknown
Unknown
Aging
Ghrelin receptor agonist
Small molecule
Investigational
Unknown
Unknown
Cardiovascular Diseases; Coronary Disease
Purinergic receptor P2Y12 antagonist
Small molecule
Investigational
Unknown
Unknown
Depressive Disorder; Depressive Disorder, Major; Phobia, Social; Postoperative Nausea and Vomiting; Sleep Initiation and Maintenance Disorders; Sleep Wake Disorders; Tinnitus
Unknown
Small molecule
Investigational
Unknown
Unknown
Atrial Fibrillation; Mucopolysaccharidosis VI
Glycosaminoglycans modulator
Small molecule
Investigational
Unknown
Unknown
Neoplasms; Stomach Neoplasms
Platelet-derived growth factor receptor beta inhibitor
Small molecule
Investigational
Unknown
Unknown
Flushing; Polycystic Ovary Syndrome; Schizophrenia
Neurokinin 3 receptor antagonist
Small molecule
Investigational
Unknown
Unknown
Diabetic Neuropathies; Neuralgia, Postherpetic
Voltage-gated N-type calcium channel alpha-1B subunit blocker
Small molecule
Investigational
Unknown
Unknown
HIV Infections
Unknown
Small molecule
Investigational
Unknown
Unknown
Glioma; Glioblastoma
Unknown
Small molecule
Investigational
Unknown
Unknown
Hepatitis C; Hepatitis C, Chronic
Hepatitis C virus NS5B RNA-dependent RNA polymerase inhibitor
Small molecule
Investigational
Unknown
Unknown
Neoplasms; Breast Neoplasms
Insulin-like growth factor I receptor inhibitor
Small molecule
Investigational
Unknown
Unknown
Heart Failure
Unknown
Small molecule
Investigational
Unknown
Unknown
Myelodysplastic Syndromes; Neoplasms; Small Cell Lung Carcinoma; Glioblastoma; Oligodendroglioma
Serine/threonine protein phosphatase 2A, catalytic subunit, alpha isoform inhibitor
Small molecule
Investigational
Unknown
Unknown
Obesity
Unknown
Small molecule
Investigational
Unknown
Unknown
Psoriasis
Unknown
Small molecule
Investigational
Unknown
Unknown
Hypertension, Pulmonary
Thromboxane A2 receptor antagonist
Small molecule
Investigational
Unknown
Unknown
Constipation
Mu opioid receptor antagonist
Small molecule
Investigational
Unknown
Unknown
Diabetic Neuropathies; Neuralgia, Postherpetic
Angiotensin II type 2 (AT-2) receptor antagonist
Small molecule
Investigational
Unknown
Unknown
Anxiety; Huntington Disease; Mood Disorders; Stress Disorders, Post-Traumatic
Vasopressin V1a receptor antagonist
Small molecule
Investigational
Unknown
Unknown
Unknown
Unknown
Small molecule
Investigational
Unknown
Unknown
Neuralgia
Adenosine A1 receptor agonist