Display Options:
Total: 6532
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Pain
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Neoplasms, Neuroepithelial; Fallopian Tube Neoplasms; Graft vs Host Disease; Hematologic Neoplasms; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Plasma Cell; Lymphoma, B-Cell; Myelodysplastic-Myeloproliferative Diseases; Peritoneal Neoplasms; Sarcoma, Kaposi; Acquired Immunodeficiency Syndrome; Astrocytoma; Carcinoid Tumor; Carcinoma, Hepatocellular; Carcinoma, Islet Cell; Carcinoma, Merkel Cell; Carcinoma, Neuroendocrine; Castleman Disease; Glioblastoma; Glioma; Gliosarcoma; Hematologic Diseases; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Lymphoid; Lymphoma, AIDS-Related; Lymphoma, Large-Cell, Anaplastic; Lymphoma, T-Cell; Multiple Sclerosis, Relapsing-Remitting; Myasthenia Gravis; Neuromyelitis Optica; Neutropenia; Oligodendroglioma; Opsoclonus-Myoclonus Syndrome; Optic Nerve Glioma; Oropharyngeal Neoplasms; Pancreatic Neoplasms; Polyradiculoneuropathy, Chronic Inflammatory Demyelinating; Precursor T-Cell Lymphoblastic Leukemia-Lymphoma; Rhabdomyosarcoma, Alveolar; Rhabdomyosarcoma, Embryonal; Severe Acute Respiratory Syndrome; Stiff-Person Syndrome; Thymoma; Waldenstrom Macroglobulinemia; Adenocarcinoma of Lung; Adrenal Cortex Neoplasms; Anemia, Refractory; Anemia, Refractory, with Excess of Blasts; Brain Neoplasms; Breast Neoplasms; Burkitt Lymphoma; Carcinoma; Carcinoma, Embryonal; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Central Nervous System Neoplasms; Choriocarcinoma; Choroid Plexus Neoplasms; Colorectal Neoplasms; Endodermal Sinus Tumor; Ependymoma; Ganglioneuroblastoma; Gestational Trophoblastic Disease; Granuloma, Lethal Midline; Hepatoblastoma; HIV Infections; Hodgkin Disease; Kidney Neoplasms; Leukemia; Leukemia, Basophilic, Acute; Leukemia, Biphenotypic, Acute; Leukemia, Erythroblastic, Acute; Leukemia-Lymphoma, Adult T-Cell; Leukemia, Megakaryoblastic, Acute; Leukemia, Monocytic, Acute; Leukemia, Myeloid, Acute; Leukemia, Myelomonocytic, Acute; Leukemia, Myelomonocytic, Chronic; Lung Neoplasms; Lymphohistiocytosis, Hemophagocytic; Lymphoma; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Lymphoma, Non-Hodgkin; Lymphoma, T-Cell, Peripheral; Mediastinal Neoplasms; Medulloblastoma; Multiple Myeloma; Myelodysplastic Syndromes; Myeloproliferative Disorders; Neoplasms, Germ Cell and Embryonal; Neuroblastoma; Neuroectodermal Tumors, Primitive; Osteosarcoma; Ovarian Neoplasms; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Prostatic Neoplasms, Castration-Resistant; Retinoblastoma; Rhabdomyosarcoma; Sarcoma; Sarcoma, Ewing; Sarcoma, Myeloid; Seminoma; Sex Cord-Gonadal Stromal Tumors; Small Cell Lung Carcinoma; Stomach Neoplasms; Teratoma; Testicular Neoplasms; Thymus Neoplasms; Wilms Tumor; Neoplasms
DNA topoisomerase II inhibitor
Small molecule
Approved
OTHER
TOPICAL; VAGINAL
Unknown
Cytochrome P450 51 inhibitor
Small molecule
Approved
Unknown
Unknown
Migraine Disorders
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
OTHER
INJECTION
HIV Wasting Syndrome; Hip Fractures; Malnutrition; Eye Diseases
Androgen Receptor agonist
Small molecule
Approved
OTHER
ORAL
Irritable Bowel Syndrome; Paraplegia; Xanthomatosis, Cerebrotendinous
Bile acid receptor FXR agonist
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Bacterial Infections; Eye Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Kidney Calculi; Diabetes Mellitus, Type 2; Cardiovascular Diseases; Heart Failure; Hypertension; Toxemia
Thiazide-sensitive sodium-chloride cotransporter inhibitor
Small molecule
Approved
Unknown
Unknown
Constipation; Urinary Tract Infections
Unknown
Small molecule
Approved
GASTROINTESTINAL
ORAL
Carcinoma, Medullary; Esophagitis, Peptic; Hypotension, Orthostatic; Immune System Diseases; Neoplasms; Breast Carcinoma In Situ; Breast Neoplasms; Carcinoma, Renal Cell; Helicobacter Infections; Job Syndrome; Leukemia, T-Cell; Postpartum Hemorrhage; Precursor T-Cell Lymphoblastic Leukemia-Lymphoma; Barrett Esophagus; Cough; Multiple Myeloma; Multiple Sclerosis; Stomach Ulcer; Gastroesophageal Reflux; Peptic Ulcer
Histamine H2 receptor antagonist
Small molecule
Approved
Unknown
Unknown
Dengue; HIV Infections; Infections; Influenza, Human; Leishmaniasis, Cutaneous; Malaria; Malaria, Falciparum; Plague; Respiratory Syncytial Virus Infections; Schistosomiasis; Severe Acute Respiratory Syndrome; Shock; Staphylococcal Infections; Anthrax; Diabetes Mellitus, Type 1; Hookworm Infections; Influenza in Birds; Pneumonia, Pneumococcal; Stomatitis; Tobacco Use Disorder; Heartburn
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
INHALATION
Unknown
Beta-2 adrenergic receptor agonist
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Psychotic Disorders; Schizophrenia; Bipolar Disorder; Cholangitis; Colitis, Ulcerative; Endometritis; Malnutrition; Parkinson Disease; Pelvic Inflammatory Disease; Amyotrophic Lateral Sclerosis; Gonorrhea; Infections; Lyme Disease; Peritonitis; Pneumonia; Pneumonia, Bacterial; Pyelonephritis; Sepsis; Urinary Tract Infections; Bacterial Infections
Unknown
Small molecule
Approved
OTHER
INJECTION
Bacterial Infections
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
OTHER
INJECTION
Bacterial Infections
Bacterial penicillin-binding protein 2 inhibitor
Small molecule
Approved
Unknown
Unknown
Diarrhea; Osteomyelitis; Astrocytoma; Brain Neoplasms; Cocaine-Related Disorders; Glioblastoma; Obesity; Respiratory Tract Infections; Sepsis; Asthma; Depressive Disorder, Major; Erectile Dysfunction; Head and Neck Neoplasms; Mastitis; Periapical Periodontitis; Pneumonia, Bacterial; Tobacco Use Disorder; Tuberculosis; Tuberculosis, Pulmonary; Abscess; Bronchitis, Chronic; Cholecystitis; Enterobacteriaceae Infections; Helicobacter Infections; Infections; Otitis Media; Otitis Media, Suppurative; Pneumonia; Severe Acute Respiratory Syndrome; Sinusitis; Urinary Tract Infections
Unknown
Small molecule
Approved
OTHER
NASAL; ORAL; TRANSDERMAL
Aging; Attention Deficit Disorder with Hyperactivity; Cocaine-Related Disorders; Memory Disorders; Sarcoidosis; Schizophrenia; Alcohol Drinking; Carcinoma in Situ; Cognitive Dysfunction; Depressive Disorder; Parkinson Disease; Postoperative Nausea and Vomiting; Sarcoma; Substance-Related Disorders; Wounds and Injuries; Heart Failure; Lung Neoplasms; Marijuana Abuse; Pulmonary Disease, Chronic Obstructive; Severe Acute Respiratory Syndrome; Smoking Cessation; Tuberculosis; Uterine Cervical Neoplasms; Tobacco Use Disorder
Neuronal acetylcholine receptor; alpha4/beta2 agonist
Small molecule
Approved
Unknown
Unknown
Lung Diseases, Obstructive
Unknown
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Atherosclerosis; Renal Insufficiency, Chronic; Diabetes Mellitus; Diabetes Mellitus, Type 2
Sulfonylurea receptor 1, Kir6.2 blocker
Small molecule
Approved
Unknown
Unknown
Unknown
Monoamine transporter inhibitor
Small molecule
Approved
Unknown
Unknown
Depressive Disorder
Unknown
Small molecule
Approved
Unknown
Unknown
Constipation; Heart Arrest; Heroin Dependence; Restless Legs Syndrome; Rheumatic Diseases; Blood Coagulation Disorders; Chronic Pain; Fractures, Multiple; Hemorrhage; Mucositis; Neuralgia; Postoperative Complications; Premature Birth; Respiratory Insufficiency; Rotator Cuff Injuries; Stomatitis; Tonsillitis; Anemia, Sickle Cell; Back Pain; Dyspnea; Fractures, Bone; Kidney Calculi; Leukemia, Myeloid, Acute; Myocardial Infarction; Neonatal Abstinence Syndrome; Neoplasms; Obesity; Opioid-Related Disorders; Pregnancy; Prostatic Neoplasms, Castration-Resistant; Pruritus; Pulmonary Disease, Chronic Obstructive; Renal Colic; Scoliosis; Sleep Apnea, Obstructive; Wounds and Injuries; Pain
Unknown
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM
INTRAMUSCULAR
Bulimia; Alcohol Drinking; Child Development Disorders, Pervasive; Dermatitis, Atopic; Psoriasis; Schizophrenia; Alcohol-Related Disorders; Amphetamine-Related Disorders; Breast Neoplasms; Colitis, Ulcerative; Coronavirus Infections; Crohn Disease; Cystitis, Interstitial; Depressive Disorder, Major; Diabetic Neuropathies; Dry Eye Syndromes; Fibromyalgia; Low Back Pain; Marijuana Abuse; Migraine Disorders; Obsessive-Compulsive Disorder; Respiratory Distress Syndrome; Severe Acute Respiratory Syndrome; Trichotillomania; Borderline Personality Disorder; Chronic Pain; Cocaine-Related Disorders; Depressive Disorder; Endometriosis; Gambling; Heroin Dependence; HIV Infections; Multiple Sclerosis; Obesity; Opioid-Related Disorders; Pain; Stress Disorders, Post-Traumatic; Substance-Related Disorders; Tobacco Use Disorder; Alcoholism
Opioid receptors; mu/kappa/delta antagonist
Small molecule
Approved
Unknown
Unknown
Arrhythmias, Cardiac
Unknown
Small molecule
Approved
OTHER
ORAL
Peripheral Nerve Injuries; Clostridium Infections; Crohn Disease; Colonic Neoplasms; Colorectal Neoplasms; Diabetes Mellitus; Hepatitis C; Hepatitis C, Chronic; Constipation
Osmotic laxative
Small molecule
Unknown
Unknown
Unknown
Depressive Disorder; Tobacco Use Disorder
Neuronal acetylcholine receptor; alpha4/beta2 agonist
Small molecule
Approved
Unknown
Unknown
Delirium; Chronic Pain; Pulpitis; Wounds and Injuries; Back Pain; Pain; Pregnancy
Unknown
Small molecule
Approved
Unknown
Unknown
Sepsis; Mastitis; Periapical Periodontitis; Tuberculosis; Enterobacteriaceae Infections; Pyelonephritis; Infections; Otitis Media; Pneumonia; Respiratory Tract Infections; Sinusitis; Soft Tissue Infections; Urinary Tract Infections
Bacterial beta-lactamase TEM inhibitor
Small molecule
Approved
Unknown
Unknown
Keratosis, Actinic; Infections; Acne Vulgaris
Releases active oxygen
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Bacterial Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Constipation; Opioid-Related Disorders; Wounds and Injuries; Anemia, Sickle Cell; Chronic Pain; Heroin Dependence; Ileus; Low Back Pain; Mucositis; Neoplasms; Osteoarthritis, Hip; Osteoarthritis, Knee; Pain
Unknown