Display Options:
Total: 6532
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Pain
Mu opioid receptor agonist
Small molecule
Approved
GASTROINTESTINAL
ORAL
Carcinoma, Medullary; Esophagitis, Peptic; Hypotension, Orthostatic; Immune System Diseases; Neoplasms; Breast Carcinoma In Situ; Breast Neoplasms; Carcinoma, Renal Cell; Helicobacter Infections; Job Syndrome; Leukemia, T-Cell; Postpartum Hemorrhage; Precursor T-Cell Lymphoblastic Leukemia-Lymphoma; Barrett Esophagus; Cough; Multiple Sclerosis; Stomach Ulcer; Gastroesophageal Reflux; Peptic Ulcer
Histamine H2 receptor antagonist
Small molecule
Approved
Unknown
Unknown
Unknown
Neutralises acid
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Bacterial Infections; Eye Infections
Unknown
Small molecule
Approved
OTHER
ORAL
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Bacterial Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Cardiovascular Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Constipation; Urinary Tract Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
TOPICAL; VAGINAL
Unknown
Cytochrome P450 51 inhibitor
Small molecule
Approved
OTHER
INJECTION; ORAL
Fallopian Tube Neoplasms; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Plasma Cell; Lymphoma, Primary Effusion; Myelodysplastic-Myeloproliferative Diseases; Neoplasms, Neuroepithelial; Neuroendocrine Tumors; Peritoneal Neoplasms; Sarcoma, Kaposi; Acquired Immunodeficiency Syndrome; Astrocytoma; Carcinoid Tumor; Carcinoma, Hepatocellular; Carcinoma, Islet Cell; Carcinoma, Large Cell; Carcinoma, Merkel Cell; Carcinoma, Neuroendocrine; Castleman Disease; Esthesioneuroblastoma, Olfactory; Glioblastoma; Glioma; Gliosarcoma; Graft vs Host Disease; Hematologic Diseases; Hematologic Neoplasms; Leukemia, Lymphocytic, Chronic, B-Cell; Lymphoma, AIDS-Related; Lymphoma, B-Cell, Marginal Zone; Lymphoma, Large-Cell, Anaplastic; Lymphoma, T-Cell; Multiple Sclerosis, Relapsing-Remitting; Myasthenia Gravis; Neoplasms, Plasma Cell; Neuromyelitis Optica; Neutropenia; Oligodendroglioma; Opsoclonus-Myoclonus Syndrome; Optic Nerve Glioma; Oropharyngeal Neoplasms; Pancreatic Neoplasms; Paraganglioma; Polyradiculoneuropathy, Chronic Inflammatory Demyelinating; Prostatic Neoplasms; Rhabdomyosarcoma, Alveolar; Rhabdomyosarcoma, Embryonal; Severe Acute Respiratory Syndrome; Stiff-Person Syndrome; Thymoma; Waldenstrom Macroglobulinemia; Adenocarcinoma of Lung; Adrenal Cortex Neoplasms; Anemia, Refractory; Anemia, Refractory, with Excess of Blasts; Brain Neoplasms; Breast Neoplasms; Burkitt Lymphoma; Carcinoma; Carcinoma, Embryonal; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Central Nervous System Neoplasms; Choriocarcinoma; Choroid Plexus Neoplasms; Colorectal Neoplasms; Endodermal Sinus Tumor; Ependymoma; Ganglioneuroblastoma; Gestational Trophoblastic Disease; Granuloma, Lethal Midline; Hepatoblastoma; HIV Infections; Hodgkin Disease; Kidney Neoplasms; Leukemia; Leukemia, Basophilic, Acute; Leukemia, Biphenotypic, Acute; Leukemia, Erythroblastic, Acute; Leukemia, Lymphoid; Leukemia-Lymphoma, Adult T-Cell; Leukemia, Megakaryoblastic, Acute; Leukemia, Monocytic, Acute; Leukemia, Myeloid, Acute; Leukemia, Myelomonocytic, Acute; Leukemia, Myelomonocytic, Chronic; Lymphohistiocytosis, Hemophagocytic; Lymphoma; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Lymphoma, Non-Hodgkin; Lymphoma, T-Cell, Peripheral; Mediastinal Neoplasms; Medulloblastoma; Multiple Myeloma; Myelodysplastic Syndromes; Myeloproliferative Disorders; Neoplasms, Germ Cell and Embryonal; Neuroblastoma; Neuroectodermal Tumors, Primitive; Osteosarcoma; Ovarian Neoplasms; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Precursor T-Cell Lymphoblastic Leukemia-Lymphoma; Prostatic Neoplasms, Castration-Resistant; Retinoblastoma; Rhabdomyosarcoma; Sarcoma; Sarcoma, Ewing; Sarcoma, Myeloid; Seminoma; Sex Cord-Gonadal Stromal Tumors; Stomach Neoplasms; Teratoma; Testicular Neoplasms; Thymus Neoplasms; Wilms Tumor; Carcinoma, Small Cell; Lung Neoplasms; Neoplasms; Small Cell Lung Carcinoma
DNA topoisomerase II inhibitor
Small molecule
Approved
Unknown
Unknown
Pain
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Pancreatic Neoplasms; Atherosclerosis; Renal Insufficiency, Chronic; Diabetes Mellitus; Diabetes Mellitus, Type 2
Sulfonylurea receptor 1, Kir6.2 blocker
Small molecule
Approved
Unknown
Unknown
Arthralgia; Eye Diseases; Myalgia
Xanthine dehydrogenase inhibitor
Small molecule
Approved
OTHER
ORAL
Amyotrophic Lateral Sclerosis; Anxiety; Dementia; Depressive Disorder; Schizophrenia; Psychotic Disorders; Tics; Tourette Syndrome
Dopamine receptor antagonist
Small molecule
Approved
Unknown
Unknown
Carcinoma, Hepatocellular; Hodgkin Disease; Kidney Diseases; Pancreatic Neoplasms; Colorectal Neoplasms; Diabetes Mellitus, Type 1; Leishmaniasis; Lymphoma, AIDS-Related; Melanoma; Trypanosomiasis; Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Alpha-1a adrenergic receptor agonist
Small molecule
Approved
OTHER
INJECTION
Unknown
Phosphodiesterase 3A inhibitor
Small molecule
Approved
Unknown
Unknown
Astrocytoma; Bacterial Infections; Brain Neoplasms; Diarrhea; Glioblastoma; Obesity; Osteomyelitis; Respiratory Tract Infections; Sepsis; Asthma; Buruli Ulcer; Cocaine-Related Disorders; Depressive Disorder, Major; Erectile Dysfunction; Head and Neck Neoplasms; Mastitis; Periapical Periodontitis; Pneumonia, Bacterial; Tobacco Use Disorder; Tuberculosis; Tuberculosis, Pulmonary; Bronchitis; Bronchitis, Chronic; Cholecystitis; Clostridium Infections; Cystitis, Hemorrhagic; Enterobacteriaceae Infections; Helicobacter Infections; Hernia; Infections; Influenza, Human; Otitis Media; Otitis Media, Suppurative; Pneumonia; Severe Acute Respiratory Syndrome; Sinusitis; Urinary Bladder Neoplasms; Urinary Tract Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Depressive Disorder; Smoking; Tobacco Use Disorder
Neuronal acetylcholine receptor; alpha4/beta2 agonist
Small molecule
Approved
Unknown
Unknown
Delirium; Chronic Pain; Pulpitis; Back Pain; Pain; Pregnancy; Wounds and Injuries
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
INHALATION
Unknown
Beta-2 adrenergic receptor agonist
Small molecule
Approved
Unknown
Unknown
Unknown
Monoamine transporter inhibitor
Small molecule
Approved
Unknown
Unknown
Depressive Disorder
Unknown
Small molecule
Approved
Unknown
Unknown
Sepsis; Mastitis; Periapical Periodontitis; Tuberculosis; Enterobacteriaceae Infections; Pyelonephritis; Infections; Otitis Media; Pneumonia; Respiratory Tract Infections; Sinusitis; Soft Tissue Infections; Urinary Tract Infections
Bacterial beta-lactamase TEM inhibitor
Small molecule
Approved
Unknown
Unknown
Constipation; Kidney Neoplasms; Opioid-Related Disorders; Wounds and Injuries; Anemia, Sickle Cell; Cancer Pain; Chronic Pain; Heroin Dependence; Ileus; Low Back Pain; Mucositis; Osteoarthritis, Hip; Osteoarthritis, Knee; Pain
Unknown
Small molecule
Approved
Unknown
Unknown
Arrhythmias, Cardiac
Unknown
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; HEMATOLOGY; OTHER
ORAL
Angina, Stable; Ischemic Stroke; Spinal Cord Injuries; Brain Injuries; Diabetes Mellitus, Type 1; Stroke; Diabetes, Gestational; Diabetes Mellitus; Diabetes Mellitus, Type 2
Sulfonylurea receptor 1, Kir6.2 blocker
Small molecule
Approved
Unknown
Unknown
Constipation; Fractures, Bone; Heart Arrest; Heroin Dependence; Restless Legs Syndrome; Rheumatic Diseases; Blood Coagulation Disorders; Fractures, Multiple; Hemorrhage; Mucositis; Neuralgia; Postoperative Complications; Premature Birth; Respiratory Insufficiency; Rotator Cuff Injuries; Stomatitis; Tonsillitis; Anemia, Sickle Cell; Back Pain; Cancer Pain; Chronic Pain; Dyspnea; Kidney Calculi; Leukemia; Leukemia, Myeloid, Acute; Myocardial Infarction; Neonatal Abstinence Syndrome; Neoplasms; Obesity; Opioid-Related Disorders; Pregnancy; Prostatic Neoplasms, Castration-Resistant; Pruritus; Pulmonary Disease, Chronic Obstructive; Renal Colic; Rib Fractures; Scoliosis; Sleep Apnea, Obstructive; Wounds and Injuries; Pain
Unknown
Small molecule
Approved
Unknown
Unknown
Lung Diseases, Obstructive
Unknown
Small molecule
Approved
OTHER
ORAL
Peripheral Nerve Injuries; Clostridium Infections; Crohn Disease; Colonic Neoplasms; Colorectal Neoplasms; Diabetes Mellitus; Hepatitis C; Hepatitis C, Chronic; Constipation
Osmotic laxative
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Bacterial Infections
Unknown