Display Options:
Total: 6532
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Bacterial Infections
Bacterial DNA gyrase inhibitor
Small molecule
Approved
Unknown
Unknown
Desmoid Tumors; Ovarian Neoplasms; Prostatic Neoplasms, Castration-Resistant; Severe Acute Respiratory Syndrome; Breast Neoplasms; Fractures, Bone; Mastodynia; Neoplasms; Prostatic Intraepithelial Neoplasia
Unknown
Small molecule
Approved
OTHER
ORAL
Lecithin Cholesterol Acyltransferase Deficiency; Multiple Sclerosis; Alcoholism; Anxiety; Anxiety Disorders; Borderline Personality Disorder; Brain Concussion; Dementia; Depressive Disorder; Neurotic Disorders; Obsessive-Compulsive Disorder; Phobia, Social; Psychomotor Agitation; Psychotic Disorders; Stress Disorders, Post-Traumatic; Bipolar Disorder; Depressive Disorder, Major; Schizophrenia
Dopamine D2 receptor antagonist
Small molecule
Approved
OTHER; RESPIRATORY
INTRAPLEURAL
Carcinoma, Non-Small-Cell Lung; Osteoarthritis, Hip; Osteoarthritis, Knee; Radius Fractures; Pleural Effusion
Unknown
Small molecule
Approved
Unknown
Unknown
Carcinoma, Renal Cell; Colorectal Neoplasms; Glioblastoma; Lung Neoplasms; Lymphoma; Neoplasms; Pancreatic Neoplasms; Paraganglioma; Sepsis; Uterine Cervical Neoplasms; Vulvar Neoplasms; Carcinoma, Non-Small-Cell Lung; Lupus Erythematosus, Systemic; Multiple Myeloma; Uterine Cervical Dysplasia; Acquired Immunodeficiency Syndrome; Carcinoma; Diarrhea; HIV Infections; Virus Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Hyperprolactinemia; Cocaine-Related Disorders; Fibromyalgia; Stroke; Unverricht-Lundborg Syndrome; Restless Legs Syndrome; Parkinson Disease
Unknown
Small molecule
Approved
Unknown
Unknown
Amyotrophic Lateral Sclerosis; Chronic Pain; Cocaine-Related Disorders; Renal Colic; Substance-Related Disorders; Alzheimer Disease; Bipolar Disorder; Depressive Disorder, Major; Fibromyalgia; Obsessive-Compulsive Disorder; Depressive Disorder; Essential Tremor; Feeding and Eating Disorders; Psychotic Disorders; Restless Legs Syndrome; Schizophrenia; Tourette Syndrome; Parkinson Disease
Unknown
Small molecule
Approved
Unknown
Unknown
Kidney Diseases; Essential Hypertension; Severe Acute Respiratory Syndrome; Cardiovascular Diseases
Unknown
Small molecule
Approved
OTHER
ORAL
Unknown
Unknown
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Anemia, Sickle Cell; Arthritis, Rheumatoid; Gastrointestinal Stromal Tumors; Malaria; Mitochondrial Diseases; Neoplasms; Parkinson Disease; Prostatic Neoplasms, Castration-Resistant; Atherosclerosis; Coronary Disease; Cystic Fibrosis; Hypercholesterolemia; Hypertension; Diabetes Mellitus; Diabetes Mellitus, Type 2
Sulfonylurea receptor 1, Kir6.2 blocker
Small molecule
Approved
OTHER
TOPICAL
Skin Diseases
Glucocorticoid receptor agonist
Small molecule
Approved
Unknown
Unknown
HIV Infections; Virus Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Otosclerosis; Bone Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Voltage-gated T-type calcium channel blocker
Small molecule
Approved
ENT; OTHER; PHARMACOLOGY; RESPIRATORY
ORAL
Appendicitis; Osteomyelitis; Mastitis; Bacterial Infections; Bronchitis, Chronic; Infections; Otitis Media; Pharyngitis; Pneumonia; Tonsillitis
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
Unknown
Unknown
HIV Infections
Human immunodeficiency virus type 1 reverse transcriptase inhibitor
Small molecule
Approved
DERMATOLOGY; IMMUNE SYSTEM; OTHER
TOPICAL
Astrocytoma; Brain Neoplasms; Carcinoma, Squamous Cell; Cheilitis; Colorectal Neoplasms; Diffuse Intrinsic Pontine Glioma; Ependymoma; Glioblastoma; Glioma; Influenza in Birds; Lymphoma, T-Cell, Cutaneous; Malaria, Falciparum; Medulloblastoma; Mouth Neoplasms; Mycosis Fungoides; Neoplasms; Osteosarcoma; Paraganglioma; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Sarcoma; Bowen's Disease; Breast Neoplasms; Carcinoma in Situ; Carcinoma, Non-Small-Cell Lung; Hemangioma; Hepatitis B, Chronic; Keloid; Leukemia; Leukemia, Lymphocytic, Chronic, B-Cell; Liver Cirrhosis; Melanoma; Port-Wine Stain; Renal Insufficiency; Uterine Cervical Neoplasms; Influenza, Human; Leishmaniasis, Cutaneous; Paget Disease, Extramammary; Papillomavirus Infections; Scleroderma, Localized; Squamous Intraepithelial Lesions; Uterine Cervical Dysplasia; Vulvar Neoplasms; Carcinoma, Basal Cell; Condylomata Acuminata; Keratosis; Keratosis, Actinic; Virus Diseases
Toll-like receptor 7 agonist
Small molecule
Approved
Unknown
Unknown
Infections
Diagnostic agent
Small molecule
Approved
Unknown
Unknown
Presbyopia; Macular Degeneration; Cataract; Conjunctivitis, Allergic; Dry Eye Syndromes; Inflammation; Macular Edema; Eye Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Epilepsy; Colonic Neoplasms; Myocardial Infarction; Neoplasms
Diagnostic
Small molecule
Approved
Unknown
Unknown
Acute Kidney Injury; Hypertension
Dopamine D1 receptor agonist
Small molecule
Approved
Unknown
Unknown
Central Nervous System Neoplasms; Glioblastoma; Cardiovascular Diseases
Unknown
Small molecule
Approved
IMMUNE SYSTEM; OTHER; PHARMACOLOGY
ORAL
Unknown
Bacterial DNA gyrase inhibitor
Small molecule
Approved
Unknown
Unknown
Myeloproliferative Disorders; Polycythemia Vera; Thrombocythemia, Essential; Neoplasms
Unknown
Small molecule
Approved
Unknown
Unknown
Erectile Dysfunction; Hyperplasia; Kidney Calculi; Postoperative Complications; Premature Ejaculation; Prostatic Neoplasms, Castration-Resistant; Ureterolithiasis; Urinary Retention; Urinary Tract Infections; Urolithiasis; Prostatic Hyperplasia
Unknown
Small molecule
Approved
Unknown
Unknown
Prostatic Neoplasms; Alzheimer Disease; Endometrial Neoplasms; Menopause; Severe Acute Respiratory Syndrome; Bone Diseases, Metabolic; Breast Neoplasms; Cognitive Dysfunction; Osteoporosis; Osteoporosis, Postmenopausal; Polycystic Ovary Syndrome; Psychotic Disorders; Schizophrenia
Estrogen receptor modulator
Small molecule
Approved
Unknown
Unknown
Depressive Disorder, Major; Diabetes Mellitus, Type 2; Head and Neck Neoplasms; Lupus Erythematosus, Systemic; Asthma; Cardiovascular Diseases; Heart Diseases; HIV Infections; Hypertension, Pulmonary; Intermittent Claudication; Peripheral Vascular Diseases; Pneumonia, Viral; Polycythemia Vera; Pregnancy; Respiratory Insufficiency; Scleroderma, Systemic; Venous Thromboembolism; Acute Coronary Syndrome; Angina, Stable; Aortic Valve Stenosis; Arteriosclerosis; Atherosclerosis; Atrial Fibrillation; Brain Infarction; Carotid Stenosis; Coronary Disease; Gastrointestinal Hemorrhage; Heart Defects, Congenital; Heart Failure; Hemorrhage; Influenza, Human; Intracranial Aneurysm; Intracranial Arteriosclerosis; Ischemia; Ischemic Attack, Transient; Ischemic Stroke; Kidney Failure, Chronic; Macular Degeneration; Myocardial Infarction; Myocardial Ischemia; Pancreatic Neoplasms; Peripheral Arterial Disease; Pneumonia; Pulmonary Disease, Chronic Obstructive; Renal Insufficiency, Chronic; Severe Acute Respiratory Syndrome; ST Elevation Myocardial Infarction; Stroke; Thrombophilia; Vascular Diseases; Thrombosis
Unknown
Small molecule
Approved
Unknown
Unknown
Cardiovascular Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Bacterial Infections
Unknown
Small molecule
Approved
OTHER; PHARMACOLOGY
INJECTION
Macular Degeneration
Alcohol dehydrogenase class I inhibitor
Small molecule
Approved
Unknown
Unknown
Gingivitis; Hypersensitivity; Mucositis; Periodontal Diseases; Periodontitis
Bacterial enoyl-[acyl-carrier-protein] reductase inhibitor
Small molecule
Approved
OTHER
ORAL
Sarcoma; Diabetes Mellitus
Peroxisome proliferator-activated receptor gamma agonist
Small molecule
Approved
Unknown
Unknown
Eye Manifestations
Unknown
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
NASAL; ORAL
Migraine Disorders
Serotonin 1b (5-HT1b) receptor agonist
Small molecule
Approved
Unknown
Unknown
Fibromyalgia; Nausea
Unknown