Display Options:
Total: 6532
Small molecule
Approved
Unknown
Unknown
Hepatitis B, Chronic; Infections; Renal Insufficiency, Chronic; Hepatitis C; Hepatitis C, Chronic; Severe Acute Respiratory Syndrome; Virus Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Hyperkalemia
Potassium chelating agent
Small molecule
Approved
Unknown
INTRAVENOUS
Acute Coronary Syndrome; Coronary Disease; ST Elevation Myocardial Infarction; Ischemia; Myocardial Infarction; Percutaneous Coronary Intervention; Thrombosis
Purinergic receptor P2Y12 inhibitor
Small molecule
Approved
Unknown
Unknown
Lung Neoplasms; Carcinoma, Non-Small-Cell Lung
Epidermal growth factor receptor erbB1 inhibitor
Small molecule
Approved
Unknown
Unknown
Brain Neoplasms; Adenocarcinoma; Adenocarcinoma of Lung; Carcinoma; Carcinoma, Squamous Cell; Colorectal Neoplasms; Glioblastoma; Carcinoma, Non-Small-Cell Lung; Lung Neoplasms; Neoplasms
Epidermal growth factor receptor erbB1 inhibitor
Small molecule
Approved
Unknown
ORAL
Familial Primary Pulmonary Hypertension; Hypertension, Pulmonary; Pulmonary Arterial Hypertension; Thrombosis
Prostanoid IP receptor agonist
Small molecule
Approved
Unknown
SUBCUTANEOUS
Neurofibroma; Neurofibromatosis 1; Obesity; Lipoma; Pain
Cell membrane disrupting agent
Small molecule
Approved
Unknown
Unknown
Severe Acute Respiratory Syndrome; Aortic Valve Insufficiency; Cardiomyopathy, Hypertrophic; Essential Hypertension; Peripheral Arterial Disease; Chagas Cardiomyopathy; Hypertension; Hypertension, Pulmonary; Myocardial Infarction; ST Elevation Myocardial Infarction; Heart Failure
Neprilysin inhibitor
Small molecule
Approved
Unknown
INHALATION
Anxiety; Autistic Disorder; Bell Palsy; Brain Diseases; Carcinoma, Non-Small-Cell Lung; Central Nervous System Neoplasms; Diabetes Mellitus, Type 2; Erectile Dysfunction; Hypoplastic Left Heart Syndrome; Hypovolemia; Hypoxia; Ileus; Inflammatory Bowel Diseases; Ischemia; Lung Diseases; Lung Neoplasms; Neuralgia; Osteonecrosis; Reperfusion Injury; Respiratory Insufficiency; Retinitis Pigmentosa; Spinal Cord Injuries; Aging; Angina, Stable; Brain Concussion; Brain Injuries; Brain Neoplasms; Breast Neoplasms; Carcinoma, Squamous Cell; Child Development Disorders, Pervasive; Colitis, Ulcerative; Cystitis, Hemorrhagic; Death, Sudden, Cardiac; Endocarditis; Gliosarcoma; Hypoadrenocorticism, Familial; Idiopathic Pulmonary Fibrosis; Laryngeal Neoplasms; Lymphedema; Migraine Disorders; Multiple Myeloma; Myocardial Infarction; Myocardial Ischemia; Neoplasms; Opioid-Related Disorders; Osteoradionecrosis; Pulmonary Fibrosis; Severe Acute Respiratory Syndrome; Sleep Apnea, Obstructive; Status Asthmaticus; Stress Disorders, Post-Traumatic; Stroke; Tinea Pedis; Tonsillitis; Wounds and Injuries; Xerostomia; Acute Kidney Injury; Anemia, Sickle Cell; Bronchiolitis; Burns; Carbon Monoxide Poisoning; Complex Regional Pain Syndromes; Coronary Disease; Diabetes Mellitus; Fractures, Bone; Heart Failure; Hypertension, Pulmonary; Infections; Ischemic Stroke; Optic Neuropathy, Ischemic; Pain; Pneumonia; Post-Acute COVID-19 Syndrome; Postoperative Nausea and Vomiting; Pregnancy; Premature Birth; Pulmonary Disease, Chronic Obstructive; Pulmonary Embolism; Pyoderma; Respiratory Distress Syndrome; Retinopathy of Prematurity; Schizophrenia; Sepsis; Shock; Ulcer; Vascular Diseases
Essential for cellular homeostasis
Small molecule
Approved
Unknown
Unknown
Neoplasms; Pulmonary Disease, Chronic Obstructive; Carcinoma, Squamous Cell; Colonic Neoplasms; Nasopharyngeal Neoplasms; Pancreatic Neoplasms; Rectal Neoplasms; Small Cell Lung Carcinoma; Stomach Neoplasms; Colorectal Neoplasms
Thymidine phosphorylase inhibitor
Small molecule
Approved
Unknown
ORAL
Acquired Immunodeficiency Syndrome; Hepatitis B; Hepatitis B, Chronic; HIV Infections
Human immunodeficiency virus type 1 reverse transcriptase inhibitor
Small molecule
Approved
Unknown
Unknown
Hepatitis C, Chronic
Nonstructural protein 5A inhibitor
Small molecule
Approved
Unknown
Unknown
Carcinoma, Hepatocellular; Glioblastoma; Glioma; Liver Diseases; Brain Neoplasms; Bronchial Neoplasms; Cholangiocarcinoma; Colorectal Neoplasms; Digestive System Neoplasms; Head and Neck Neoplasms; Hematologic Neoplasms; Intestinal Neoplasms; Lung Neoplasms; Lymphoma, Large-Cell, Anaplastic; Melanoma; Neuroendocrine Tumors; Ovarian Neoplasms; Pancreatic Neoplasms; Respiratory Tract Diseases; Respiratory Tract Neoplasms; Salivary Gland Neoplasms; Sarcoma; Thyroid Neoplasms; Carcinoma, Non-Small-Cell Lung; Neoplasms
Unknown
Small molecule
Approved
Unknown
INTRAMUSCULAR
Psychotic Disorders; Schizophrenia
Dopamine D2 receptor partial agonist
Small molecule
Approved
Unknown
INHALATION
Status Asthmaticus; Pulmonary Disease, Chronic Obstructive
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
INTRAVENOUS
Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Lymphoid; Sarcoma, Ewing; Breast Neoplasms; Carcinoma, Ovarian Epithelial; Chondrosarcoma, Mesenchymal; Endocrine Gland Neoplasms; Fallopian Tube Neoplasms; Hereditary Breast and Ovarian Cancer Syndrome; Liposarcoma, Myxoid; Meningioma; Mesothelioma; Paget Disease, Extramammary; Pancreatic Neoplasms; Peritoneal Neoplasms; Prostatic Neoplasms, Castration-Resistant; Soft Tissue Neoplasms; Leiomyosarcoma; Liposarcoma; Neoplasms; Ovarian Neoplasms; Sarcoma
DNA inhibitor
Small molecule
Approved
Unknown
Unknown
Carcinoma, Non-Small-Cell Lung; Neoplasms; Breast Neoplasms; Cholangiocarcinoma; Colonic Neoplasms; Pancreatic Neoplasms; Rectal Neoplasms; Stomach Neoplasms; Urinary Bladder Neoplasms; Colorectal Neoplasms
Unknown
Small molecule
Approved
Unknown
Unknown
Adenocarcinoma; Carcinoma, Pancreatic Ductal; Esophageal Neoplasms; Leukemia, Myeloid, Acute; Multiple Myeloma; Ovarian Neoplasms; Pancreatic Neoplasms; Sarcoma; Skin Neoplasms; Stomach Neoplasms; Breast Neoplasms; Carcinoma, Non-Small-Cell Lung; Craniopharyngioma; Gallbladder Neoplasms; Hematologic Neoplasms; Intracranial Arteriovenous Malformations; Leukemia, Myelomonocytic, Chronic; Thyroid Neoplasms; Colorectal Neoplasms; Melanoma; Neoplasms
Dual specificity mitogen-activated protein kinase kinase 1 inhibitor
Small molecule
Approved
Unknown
ORAL
Diarrhea; Irritable Bowel Syndrome
Mu opioid receptor agonist
Small molecule
Approved
Unknown
Unknown
Blood Coagulation Disorders; Coronary Disease; Hemorrhage; Ischemic Stroke; Liver Cirrhosis; Myocardial Infarction; Peripheral Arterial Disease; Aortic Valve Stenosis; Atrial Fibrillation; Heart Diseases; Severe Acute Respiratory Syndrome; Stroke; Venous Thromboembolism; Thrombosis
Unknown
Small molecule
Approved
Unknown
ORAL
Gout; Hyperuricemia
Solute carrier family 22 member 12 inhibitor
Small molecule
Approved
Unknown
Unknown
Postoperative Nausea and Vomiting; Nausea
Unknown
Small molecule
Approved
Unknown
Unknown
Anemia, Sickle Cell; Carcinoma, Hepatocellular; Carcinoma, Non-Small-Cell Lung; Colonic Neoplasms; HIV Infections; Leukemia, Myelomonocytic, Chronic; Liver Neoplasms; Lung Neoplasms; Lymphoma, Mantle-Cell; Melanoma; Nasopharyngeal Neoplasms; Neoplasms, Plasma Cell; Paraganglioma; Polycythemia Vera; Primary Myelofibrosis; Prostatic Neoplasms; Rectal Neoplasms; Skin Neoplasms; Breast Neoplasms; Bronchiolitis Obliterans Syndrome; Carcinoma, Renal Cell; Colorectal Neoplasms; Diffuse Intrinsic Pontine Glioma; Glioblastoma; Glioma; Graft vs Host Disease; Hematologic Neoplasms; Leukemia; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Leukemia, Plasma Cell; Lymphoma; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Non-Hodgkin; Lymphoma, T-Cell, Cutaneous; Myelodysplastic Syndromes; Neuroendocrine Tumors; Pancreatic Neoplasms; Plasmacytoma; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Prostatic Neoplasms, Castration-Resistant; Stomach Neoplasms; Thyroid Neoplasms; Waldenstrom Macroglobulinemia; Hodgkin Disease; Multiple Myeloma; Neoplasms
Unknown
Small molecule
Approved
Unknown
ORAL
Prostatic Neoplasms; Sexual Dysfunctions, Psychological
Unknown
Small molecule
Approved
Unknown
Unknown
Renal Insufficiency; Systemic Inflammatory Response Syndrome; Gram-Negative Bacterial Infections; Urinary Tract Infections; Bacterial Infections; Infections; Pneumonia; Pyelonephritis
Unknown
Small molecule
Approved
Unknown
Unknown
Carcinoma, Hepatocellular; Esophageal Neoplasms; Graft vs Host Disease; Liver Diseases; Ovarian Neoplasms; Pancreatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Breast Neoplasms; Carcinoma, Basal Cell; Leukemia; Medulloblastoma; Multiple Myeloma; Neoplasms
Unknown
Small molecule
Approved
Unknown
ORAL
Smith-Lemli-Opitz Syndrome; Fatty Liver; Digestive System Diseases; Liver Diseases; Metabolism, Inborn Errors; Peroxisomal Disorders
Unknown
Small molecule
Approved
Unknown
ORAL
Heart Failure, Diastolic; Heart Failure, Systolic; Hypotension; Hypotension, Orthostatic; Lymphoma; Multiple Organ Failure; Non-ST Elevated Myocardial Infarction; Post-Acute COVID-19 Syndrome; Aging; Angina, Stable; Atrial Fibrillation; Coronary Disease; Diabetic Nephropathies; Mitral Valve Stenosis; Neoplasms; Orthostatic Intolerance; Shock, Septic; Tachycardia; Cardiovascular Diseases; Heart Failure
Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 4 blocker
Small molecule
Approved
Unknown
INHALATION
Bipolar Disorder; Cystic Fibrosis; Depressive Disorder, Major; Severe Acute Respiratory Syndrome; Death, Sudden, Cardiac; Heart Failure; Obsessive-Compulsive Disorder; Pulmonary Disease, Chronic Obstructive; Reperfusion Injury; Stress Disorders, Post-Traumatic; Tinea Pedis; Burns; Colorectal Neoplasms; Keratosis, Actinic; Respiratory Insufficiency
Unknown
Small molecule
Approved
Unknown
ORAL
Alcoholism; Borderline Personality Disorder; Alzheimer Disease; Bipolar Disorder; Depressive Disorder; Mental Disorders; Psychomotor Agitation; Sleep Wake Disorders; Stress Disorders, Post-Traumatic; Depressive Disorder, Major; Psychotic Disorders; Schizophrenia
Dopamine D2 receptor partial agonist
Small molecule
Approved
Unknown
Unknown
Anxiety Disorders; Bipolar Disorder; Child Development Disorders, Pervasive; Depressive Disorder; Depressive Disorder, Major; Schizophrenia; Psychotic Disorders
Unknown
Small molecule
Approved
Unknown
ORAL
Melanoma
Dual specificity mitogen-activated protein kinase kinase 1 inhibitor
Small molecule
Approved
Unknown
Unknown
Carcinoma, Pancreatic Ductal; Central Nervous System Neoplasms; Glioblastoma; Kidney Diseases; Liver Diseases; Lymphoma; Rectal Neoplasms; Adenocarcinoma; Adenocarcinoma, Follicular; Adenocarcinoma of Lung; Adrenal Cortex Neoplasms; Biliary Tract Neoplasms; Breast Neoplasms; Carcinoma, Adenoid Cystic; Carcinoma, Merkel Cell; Carcinoma, Neuroendocrine; Kidney Neoplasms; Liver Neoplasms; Meningeal Carcinomatosis; Mesothelioma; Neuroendocrine Tumors; Osteosarcoma; Ovarian Neoplasms; Paraganglioma; Retroviridae Infections; Sarcoma; Sarcoma, Kaposi; Small Cell Lung Carcinoma; Stomach Neoplasms; Thymoma; Uterine Cervical Neoplasms; Vulvar Neoplasms; Carcinoma, Hepatocellular; Carcinoma, Non-Small-Cell Lung; Carcinoma, Renal Cell; Carcinoma, Squamous Cell; Cholangiocarcinoma; Colorectal Neoplasms; Endometrial Neoplasms; Esophageal Neoplasms; Melanoma; Thyroid Neoplasms; Urinary Bladder Neoplasms; Neoplasms
Unknown
Small molecule
Approved
Unknown
Unknown
Amyotrophic Lateral Sclerosis; Insulin Resistance; Hepatitis D; Leukemia, Lymphocytic, Chronic, B-Cell; Weight Gain; Acquired Immunodeficiency Syndrome; Hepatitis B, Chronic; HIV Infections; Severe Acute Respiratory Syndrome; Virus Diseases
Human immunodeficiency virus type 1 reverse transcriptase inhibitor