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Total: 6532
Small molecule
Approved
Unknown
Unknown
Unknown
Bile acids sequestering agent
Small molecule
Approved
OTHER
INTRAVENOUS; ORAL
Acute Kidney Injury; Alzheimer Disease; Ankle Fractures; Bipolar Disorder; Glycogen Storage Disease Type III; Hypotension, Orthostatic; Malaria; Muscular Dystrophy, Duchenne; Osteoarthritis, Knee; Premature Birth; Rhinitis, Allergic, Seasonal; Uveal Melanoma; Brachial Plexus Neuritis; Bronchopulmonary Dysplasia; Cognitive Dysfunction; Depressive Disorder, Major; Diabetes Mellitus, Type 1; Emphysema; Enuresis; Epilepsies, Partial; Epilepsy; Glioma; Granulomatous Disease, Chronic; Hemorrhage; Hypertension; Kidney Neoplasms; Muscular Diseases; Pancreatitis; Periodontitis; Pre-Eclampsia; Retinopathy of Prematurity; Sinusitis; Spondylarthropathies; Spondylosis; Stomatitis, Aphthous; Sunburn; Temporomandibular Joint Disorders; Tension-Type Headache; Tooth Diseases; Tuberculosis; Wounds and Injuries; Altitude Sickness; Breast Neoplasms; Burns; Causalgia; Cerebral Palsy; Chronic Pain; Fractures, Bone; HIV Infections; Hypospadias; Infections; Low Back Pain; Mucopolysaccharidosis I; Multiple Sclerosis; Neck Pain; Peptic Ulcer; Pulpitis; Respiratory Distress Syndrome; Shock, Septic; Sleep Apnea, Obstructive; Sprains and Strains; Tibial Fractures; Vasculitis; Acute Pain; Arthralgia; Arthritis; Arthritis, Juvenile; Arthritis, Rheumatoid; Back Pain; Cardiovascular Diseases; Common Cold; Ductus Arteriosus, Patent; Dysmenorrhea; Fever; Headache; Influenza, Human; Migraine Disorders; Muscle Cramp; Myalgia; Osteoarthritis; Pain; Pharyngitis; Rheumatic Diseases; Toothache; Vaginitis
Cyclooxygenase inhibitor
Small molecule
Approved
OTHER
INJECTION; ORAL
Bacterial Infections
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
OPHTHALMIC
Myopia; Urinary Incontinence; Dry Eye Syndromes; Presbyopia; Glaucoma; Glaucoma, Angle-Closure; Glaucoma, Open-Angle; Miosis; Ocular Hypertension; Sjogren's Syndrome; Xerostomia
Muscarinic acetylcholine receptor M1 agonist
Small molecule
Approved
OTHER
ORAL
Unknown
Dihydropteroate synthetase inhibitor
Small molecule
Approved
Unknown
Unknown
Cocaine-Related Disorders; Attention Deficit Disorder with Hyperactivity
Unknown
Small molecule
Approved
OTHER; UROLOGY AND KIDNEY
TRANSDERMAL
Paget Disease, Extramammary; Rhinitis, Allergic, Seasonal; Sialorrhea; Sleep Apnea, Obstructive; Sleep Apnea Syndromes; Breast Neoplasms; Enuresis; Hyperhidrosis; Polyneuropathies; Urinary Bladder, Neurogenic; Polyuria; Urinary Bladder, Overactive; Urinary Incontinence; Urinary Incontinence, Urge
Muscarinic acetylcholine receptor M2 antagonist
Small molecule
Approved
OTHER
ORAL
Amyotrophic Lateral Sclerosis; Angelman Syndrome; Asthma; Diabetic Retinopathy; Hypertension; Hypotension, Orthostatic; Tobacco Use Disorder; Albinism; Albinism, Oculocutaneous; Aphasia; Attention Deficit Disorder with Hyperactivity; Back Pain; Chronic Pain; Cocaine-Related Disorders; Fibromyalgia; Macular Degeneration; Multiple Sclerosis; Pain; Retinitis Pigmentosa; Schizophrenia; Spinal Cord Injuries; Amblyopia; Dysautonomia, Familial; Stroke; Parkinson Disease; Parkinson Disease, Postencephalitic; Parkinson Disease, Secondary; Wounds and Injuries
DOPA decarboxylase inhibitor
Small molecule
Approved
OTHER
INJECTION; ORAL
Angioedemas, Hereditary; Cytomegalovirus Infections; Depressive Disorder; Depressive Disorder, Major; Diabetes Mellitus; Diabetes Mellitus, Type 2; Epilepsy; Essential Hypertension; Head and Neck Neoplasms; Hepatitis B, Chronic; Hepatitis C; HIV Infections; Infections; Inflammation; Influenza, Human; Leukemia, Myeloid, Acute; Melanoma; Myelodysplastic Syndromes; Nausea; Neoplasms; Obesity; Pain; Pulmonary Disease, Chronic Obstructive; Substance-Related Disorders; von Hippel-Lindau Disease; Arthritis, Rheumatoid; Breast Neoplasms; Carcinoma, Non-Small-Cell Lung; Keratosis, Actinic; Non-alcoholic Fatty Liver Disease; Pancreatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Sarcoma, Kaposi; Arrhythmias, Cardiac; Tachycardia, Supraventricular; Atrial Fibrillation; Cardiovascular Diseases; Heart Failure
Sodium/potassium-transporting ATPase inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Dopamine transporter releasing agent
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER
INJECTION; INTRAMUSCULAR; SUBCUTANEOUS
Pregnancy; Premature Birth
Progesterone receptor agonist
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; MUSCULOSKELETAL; OTHER; PREGNANCY AND GYNECOLOGY; RHEUMATOLOGY
ORAL; TOPICAL; TRANSDERMAL; VAGINAL
Blood Coagulation Disorders; Cerebral Arterial Diseases; Diabetes Mellitus; Diabetes Mellitus, Type 1; Diabetes Mellitus, Type 2; Polycystic Ovary Syndrome; Aging; Alzheimer Disease; Atherosclerosis; Bulimia Nervosa; Carcinoid Tumor; Depression, Postpartum; Depressive Disorder; Dry Eye Syndromes; Hereditary Breast and Ovarian Cancer Syndrome; HIV Infections; Migraine Disorders; Prostatic Neoplasms; Psychotic Disorders; Schizophrenia; Severe Acute Respiratory Syndrome; Triple Negative Breast Neoplasms; Urinary Tract Infections; Amenorrhea; Anorexia Nervosa; Bone Diseases, Metabolic; Coronary Disease; Dysmenorrhea; Endometriosis; Heart Diseases; Hot Flashes; Infertility; Multiple Sclerosis; Myocardial Ischemia; Non-alcoholic Fatty Liver Disease; Obesity; Pain; Prostatic Neoplasms, Castration-Resistant; Sexual Dysfunction, Physiological; Stress Disorders, Post-Traumatic; Turner Syndrome; Atrophic Vaginitis; Atrophy; Breast Neoplasms; Dyspareunia; Hypogonadism; Menopause; Osteoporosis; Osteoporosis, Postmenopausal; Primary Ovarian Insufficiency
Estrogen receptor alpha agonist
Small molecule
Approved
OTHER
TOPICAL
Dermatitis, Atopic; Oral Submucous Fibrosis; Lichen Planus, Oral; Sinusitis; Gout; Periarthritis; Infections; Psoriasis; Skin Diseases
Glucocorticoid receptor agonist
Small molecule
Approved
OTHER
INJECTION
Breast Neoplasms; Colonic Neoplasms; Lung Neoplasms; Thyroid Neoplasms; Neuroendocrine Tumors; Leiomyosarcoma; Lymphoma; Lymphoma, T-Cell, Peripheral; Neuroblastoma; Sarcoma; Sarcoma, Alveolar Soft Part; Sarcoma, Synovial; Skin Neoplasms; Uveal Melanoma; Hodgkin Disease; Melanoma; Neoplasms
DNA inhibitor
Small molecule
Approved
OTHER
ORAL; TOPICAL; VAGINAL
Anemia, Sickle Cell; Kidney Diseases; Folliculitis; Candidiasis, Oral; Candidiasis, Vulvovaginal; HIV Infections; Otomycosis; Vaginal Discharge; Vaginitis; Vaginosis, Bacterial; Candidiasis; Infections; Mycoses; Pruritus; Skin Diseases, Infectious; Tinea; Tinea Cruris; Tinea Pedis
Cytochrome P450 51 inhibitor
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
ORAL
Burning Mouth Syndrome; Neuralgia; Marijuana Abuse; REM Sleep Behavior Disorder; Anxiety; Dementia; Depressive Disorder; Epilepsia Partialis Continua; Epilepsy, Tonic-Clonic; Pain; Schizophrenia; Status Epilepticus; Epilepsy; Panic Disorder; Seizures
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
Unknown
Unknown
Unknown
Dopamine transporter releasing agent
Small molecule
Approved
OTHER; RESPIRATORY
INHALATION; OPHTHALMIC
Bronchopulmonary Dysplasia; Diabetic Foot; Dry Eye Syndromes; Osteomyelitis; Renal Insufficiency, Chronic; Sinusitis; Bronchiectasis; Pneumonia, Bacterial; Blepharitis; Cataract; Conjunctivitis, Bacterial; Fractures, Bone; Pneumonia; Pseudomonas Infections; Bacterial Infections; Conjunctivitis, Allergic; Cystic Fibrosis; Eye Infections; Infections; Inflammation; Respiratory Tract Infections
70S ribosome inhibitor
Small molecule
Approved
Unknown
Unknown
Asthma; Pulmonary Disease, Chronic Obstructive; Tobacco Use Disorder; Migraine Disorders; Neuralgia; Anxiety; Delirium; Bipolar Disorder; Mental Disorders; Psychomotor Agitation; Psychotic Disorders; Schizophrenia
D2-like dopamine receptor antagonist
Small molecule
Approved
OTHER
ORAL
Unknown
GABA-A receptor; anion channel positive modulator
Small molecule
Approved
Unknown
Unknown
Arthralgia; Myalgia; Rheumatic Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Periodontal Pocket; Acanthamoeba Keratitis; Carcinoma, Non-Small-Cell Lung; Diabetic Foot; Neonatal Sepsis; Peri-Implantitis; Periodontal Diseases; Pneumonia, Ventilator-Associated; Pulmonary Disease, Chronic Obstructive; Severe Acute Respiratory Syndrome; Stomatitis; Bacteremia; Bacterial Infections; Communicable Diseases; Dental Caries; Gingivitis; Neutropenia; Periodontitis; Pharyngitis; Pneumonia; Staphylococcal Infections; Eye Infections; Infections
Unknown
Small molecule
Approved
OTHER
ORAL
Bone Neoplasms; Breast Neoplasms; Glioma; Kidney Neoplasms; Lung Neoplasms; Lymphoma; Lymphoma, AIDS-Related; Lymphoma, Non-Hodgkin; Melanoma; Neoplasm Metastasis; Pancreatic Neoplasms; Sarcoma; Spinal Cord Neoplasms; Uveal Melanoma; Astrocytoma; Central Nervous System Neoplasms; Glioblastoma; Gliosarcoma; Leukemia, Myeloid, Acute; Medulloblastoma; Multiple Myeloma; Neoplasms, Plasma Cell; Paraganglioma; Brain Neoplasms; Hodgkin Disease; Neoplasms
DNA inhibitor
Small molecule
Approved
OTHER
ORAL
Anemia, Aplastic; Dyskeratosis Congenita; Fanconi Anemia; Endometrial Neoplasms; Mastodynia; Myelodysplastic Syndromes; Purpura, Thrombocytopenic, Idiopathic; Purpura, Thrombotic Thrombocytopenic; Infertility; Endometriosis; Fibrocystic Breast Disease
Androgen Receptor agonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Intestinal Obstruction; Pain; Breast Neoplasms; Clostridium Infections; Eczema; Neoplasms; Paget Disease, Extramammary; Carcinoma, Non-Small-Cell Lung; Diarrhea; Fecal Incontinence
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Sepsis; Infections; Bacterial Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
INJECTION; OPHTHALMIC
Herpes Simplex; Eye Infections; Virus Diseases
Human herpesvirus 1 DNA polymerase inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Astringent
Small molecule
Approved
Unknown
Unknown
Breast Neoplasms; Neoplasms; Brain Neoplasms; Hyperemia
Unknown
Small molecule
Approved
Unknown
Unknown
Hemorrhoids; Pruritus
Unknown
Small molecule
Approved
OTHER
TOPICAL
Unknown
DNA inhibitor