Display Options:
Total: 6532
Small molecule
Approved
Unknown
Unknown
Burns; Acute Lung Injury; Brain Injuries; Shock; Shock, Septic; Heart Failure; Cardiovascular Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL; TOPICAL
Attention Deficit Disorder with Hyperactivity; Carcinoma, Non-Small-Cell Lung; Central Nervous System Neoplasms; Crohn Disease; Familial Hypophosphatemic Rickets; Melanoma; Mouth Neoplasms; Neoplasms; Opioid-Related Disorders; Osteoporosis, Postmenopausal; Prediabetic State; Rickets, Hypophosphatemic; Acute Kidney Injury; Breast Neoplasms; Carcinoma, Basal Cell; Cholangiocarcinoma; Chronic Kidney Disease-Mineral and Bone Disorder; Diabetes Mellitus, Type 1; Hyperparathyroidism, Secondary; Hypertension; Klinefelter Syndrome; Lupus Erythematosus, Systemic; Myelodysplastic Syndromes; Pancreatic Neoplasms; Prostatic Neoplasms; Sepsis; Severe Acute Respiratory Syndrome; Adenomatous Polyposis Coli; Diabetic Nephropathies; Fibroma; Osteopetrosis; Osteoporosis; Prostatic Neoplasms, Castration-Resistant; Hypocalcemia; Hypoparathyroidism; Kidney Failure, Chronic; Psoriasis
Vitamin D receptor agonist
Small molecule
Approved
OTHER
INJECTION
Osteomyelitis
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Cyclooxygenase inhibitor
Small molecule
Approved
OTHER
OPHTHALMIC; ORAL
Optic Neuropathy, Ischemic; Low Tension Glaucoma; Corneal Edema; Hemangioma; Hypertension, Portal; Glaucoma; Glaucoma, Open-Angle; Ocular Hypertension
Beta-1 adrenergic receptor antagonist
Small molecule
Approved
OTHER
ORAL
Substance-Related Disorders; Anxiety; Dementia; Depressive Disorder; Schizophrenia; Sleep Initiation and Maintenance Disorders
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
OTHER
INJECTION
Unknown
Diagnostic agent
Small molecule
Approved
Unknown
Unknown
Dermatitis, Atopic; HIV Infections; Neoplasms; Psoriasis; Takotsubo Cardiomyopathy; Arrhythmias, Cardiac; beta-Thalassemia; Death, Sudden, Cardiac; Heart Arrest; Heart Diseases; Obesity; Orthostatic Intolerance; Prader-Willi Syndrome; Premature Birth; Tachycardia, Ventricular; Vascular Diseases; Ventricular Fibrillation; Atherosclerosis; Atrial Fibrillation; Breast Neoplasms; Coronary Disease; Diabetes Mellitus, Type 2; Heart Failure; Hypercholesterolemia; Hypertension; Myocardial Infarction; Non-ST Elevated Myocardial Infarction; Respiratory Distress Syndrome; ST Elevation Myocardial Infarction; Cardiovascular Diseases
Unknown
Small molecule
Approved
OTHER
INJECTION
Sexual Dysfunction, Physiological; Diabetic Neuropathies; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Hypogonadism; Neoplasms; Orchitis
Androgen Receptor agonist
Small molecule
Approved
OTHER
INJECTION
Carcinoma, Basal Cell; Carcinoma, Endometrioid; Cystadenoma, Serous; Digestive System Neoplasms; Genital Neoplasms, Female; Kidney Diseases; Klatskin Tumor; Liver Diseases; Neoplasms, Cystic, Mucinous, and Serous; Neuroendocrine Tumors; Primary Myelofibrosis; Rhabdomyosarcoma; Xerostomia; Bile Duct Neoplasms; Carcinoid Tumor; Carcinoma, Islet Cell; Carcinoma, Large Cell; Carcinoma, Merkel Cell; Carcinoma, Neuroendocrine; Carcinoma, Pancreatic Ductal; Carcinoma, Renal Cell; Carcinoma, Verrucous; Digestive System Diseases; Esthesioneuroblastoma, Olfactory; Gastrointestinal Stromal Tumors; Glioblastoma; Glioma; Granuloma, Lethal Midline; Immunoblastic Lymphadenopathy; Kidney Neoplasms; Leukemia; Leukemia-Lymphoma, Adult T-Cell; Lymphoma, AIDS-Related; Lymphoma, Large-Cell, Anaplastic; Mesothelioma, Malignant; Myelodysplastic Syndromes; Nausea; Neoplasm Metastasis; Paraganglioma; Penile Neoplasms; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Salivary Gland Neoplasms; Thymoma; Thyroid Neoplasms; Tongue Neoplasms; Uveal Melanoma; Adenocarcinoma; Adenocarcinoma of Lung; Adrenal Cortex Neoplasms; Anemia; Anus Neoplasms; Biliary Tract Neoplasms; Brain Neoplasms; Breast Neoplasms; Carcinoma; Carcinoma, Embryonal; Carcinoma, Hepatocellular; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Central Nervous System Neoplasms; Cholangiocarcinoma; Choriocarcinoma; Choroid Plexus Neoplasms; Colorectal Neoplasms; Endodermal Sinus Tumor; Endometrial Neoplasms; Ependymoma; Esophageal Neoplasms; Fallopian Tube Neoplasms; Gallbladder Neoplasms; Ganglioneuroblastoma; Gestational Trophoblastic Disease; Head and Neck Neoplasms; Hepatoblastoma; Hodgkin Disease; Hypopharyngeal Neoplasms; Inflammatory Breast Neoplasms; Laryngeal Neoplasms; Liver Neoplasms; Lung Neoplasms; Lymphoma; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Lymphoma, Non-Hodgkin; Lymphoma, T-Cell, Peripheral; Malaria; Mediastinal Neoplasms; Medulloblastoma; Melanoma; Mesothelioma; Mouth Neoplasms; Mucositis; Multiple Myeloma; Nasopharyngeal Carcinoma; Nasopharyngeal Neoplasms; Neoplasms, Germ Cell and Embryonal; Neuroblastoma; Neuroectodermal Tumors, Primitive; Oropharyngeal Neoplasms; Osteosarcoma; Ovarian Neoplasms; Pancreatic Neoplasms; Paranasal Sinus Neoplasms; Peritoneal Neoplasms; Pharyngeal Neoplasms; Pleural Effusion; Postoperative Nausea and Vomiting; Retinoblastoma; Sarcoma; Seminoma; Sex Cord-Gonadal Stromal Tumors; Skin Neoplasms; Small Cell Lung Carcinoma; Squamous Cell Carcinoma of Head and Neck; Stomach Neoplasms; Stomatitis; Teratoma; Testicular Neoplasms; Thymus Neoplasms; Triple Negative Breast Neoplasms; Urethral Neoplasms; Urinary Bladder Neoplasms; Urogenital Neoplasms; Uterine Cervical Neoplasms; Uterine Neoplasms; Vulvar Neoplasms; Neoplasms
DNA inhibitor
Small molecule
Approved
Unknown
Unknown
Tuberculosis, Pulmonary; Bacterial Infections; Infections; Pharyngitis
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Mu opioid receptor agonist
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Lung Diseases; Bacterial Infections
Unknown
Small molecule
Approved
OTHER
ORAL
Breast Neoplasms; Carcinoma, Squamous Cell; Desmoid Tumors; Fragile X Syndrome; Leukemia, Myeloid, Acute; Melanoma; Adenomatous Polyposis Coli; Colorectal Neoplasms; Precancerous Conditions; Arthritis, Rheumatoid; Osteoarthritis; Rheumatic Diseases; Spondylitis
Cyclooxygenase inhibitor
Small molecule
Approved
OTHER
OPHTHALMIC
Sturge-Weber Syndrome; Hemangioma; Macular Degeneration; Migraine Disorders; Telangiectasia, Hereditary Hemorrhagic; Varicose Ulcer; Wet Macular Degeneration; Wounds and Injuries; Exfoliation Syndrome; Melanoma; Paronychia; Cardiovascular Diseases; Glaucoma; Glaucoma, Open-Angle; Ocular Hypertension
Beta-1 adrenergic receptor antagonist
Small molecule
Approved
OTHER
OPHTHALMIC
Mycoses; Acanthamoeba Keratitis; Eye Infections; Infections
Ergosterol sequestering agent
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
ORAL
Astrocytoma; Brain Injuries; Burkitt Lymphoma; Carcinoma, Non-Small-Cell Lung; Central Nervous System Neoplasms; Colorectal Neoplasms; Epilepsies, Partial; Lung Neoplasms; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Medulloblastoma; Melanoma; Nasopharyngeal Carcinoma; Neoplasms; Ovarian Neoplasms; Paraganglioma; Sarcoma; Shock; Urinary Bladder Neoplasms; Wounds and Injuries; Alopecia; Brain Neoplasms; Breast Neoplasms; Carcinoma, Squamous Cell; Ependymoma; Glioblastoma; Glioma; Head and Neck Neoplasms; HIV Infections; Leukemia; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Lymphoma; Myelodysplastic Syndromes; Neuralgia; Pancreatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Retinitis Pigmentosa; Small Cell Lung Carcinoma; Supranuclear Palsy, Progressive; Thyroid Neoplasms; Uveal Melanoma; Alcoholism; Alzheimer Disease; Anxiety; Autistic Disorder; Dementia; Depressive Disorder; Migraine Disorders; Muscular Atrophy, Spinal; Paraparesis, Tropical Spastic; Psychomotor Agitation; Schizophrenia; Status Epilepticus; Bipolar Disorder; Epilepsy; Epilepsy, Absence; Epilepsy, Complex Partial; Mitochondrial Diseases; Seizures
Succinate semialdehyde dehydrogenase inhibitor
Small molecule
Approved
Unknown
Unknown
Adenomyosis; Alzheimer Disease; Anorexia Nervosa; Diabetes Mellitus, Type 1; Intellectual Disability; Obesity; Ovarian Hyperstimulation Syndrome; Peripartum Cardiomyopathy; Parkinson Disease
Unknown
Small molecule
Approved
OTHER
INTRAVESICAL
HIV Infections; Melanoma; Neoplasms; Osteoarthritis; Contracture; Cystitis, Interstitial; Reflex, Abnormal; Urinary Bladder, Overactive; Urinary Incontinence; Urinary Incontinence, Urge; Arthralgia; Cystitis; Infections; Myalgia
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Anxiety; Pain
Unknown
Small molecule
Approved
OTHER
INHALATION
Heart Diseases; Opioid-Related Disorders; Respiratory Distress Syndrome; Subarachnoid Hemorrhage; Substance-Related Disorders; Hernia, Inguinal; Respiratory Insufficiency; Severe Acute Respiratory Syndrome
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
Unknown
Unknown
Dry Eye Syndromes; Eye Manifestations; Nasal Obstruction
Unknown
Small molecule
Approved
Unknown
Unknown
Hematologic Neoplasms; Leukemia, Biphenotypic, Acute; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Polycythemia Vera; Primary Myelofibrosis; Thrombocythemia, Essential; Anemia, Refractory; Leukemia, Lymphoid; Myelodysplastic Syndromes; Hepatitis B, Chronic; Leukemia; Leukemia, Myeloid; Lymphoma, Non-Hodgkin; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Precursor T-Cell Lymphoblastic Leukemia-Lymphoma; Sarcoma, Kaposi; Leukemia, Myeloid, Acute; Neoplasms
DNA inhibitor
Small molecule
Approved
Unknown
Unknown
Alzheimer Disease; Dementia; Phobia, Social; Renal Colic; Amyotrophic Lateral Sclerosis; Bipolar Disorder; Depressive Disorder; Depressive Disorder, Major; Pain; Motion Sickness; Nausea; Postoperative Nausea and Vomiting
Muscarinic acetylcholine receptor M1 antagonist
Small molecule
Approved
Unknown
Unknown
Anemia, Refractory; Anemia, Refractory, with Excess of Blasts; Leukemia; Leukemia, Basophilic, Acute; Leukemia, Biphenotypic, Acute; Leukemia, Erythroblastic, Acute; Leukemia, Megakaryoblastic, Acute; Leukemia, Monocytic, Acute; Leukemia, Myeloid, Acute; Leukemia, Myelomonocytic, Acute; Leukemia, Myelomonocytic, Chronic; Leukemia, Promyelocytic, Acute; Lymphoma; Myelodysplastic Syndromes; Myeloproliferative Disorders; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Precursor T-Cell Lymphoblastic Leukemia-Lymphoma; Sarcoma; Sarcoma, Myeloid; Leukemia, Lymphoid
DNA inhibitor
Small molecule
Approved
Unknown
Unknown
Lung Diseases, Obstructive
Unknown
Small molecule
Approved
OTHER
ORAL; TOPICAL
Carcinoma, Non-Small-Cell Lung; Lung Diseases; Pemphigoid, Benign Mucous Membrane; Pemphigus; Pulmonary Fibrosis; Rosacea; Sarcoidosis; Stroke; Fever; HIV Infections; Malaria; Malaria, Falciparum; Malaria, Vivax; Pneumonia, Pneumocystis; Severe Acute Respiratory Syndrome; Acne Vulgaris; Dermatitis Herpetiformis; Leprosy
Dihydropteroate synthase 1 inhibitor
Small molecule
Approved
Unknown
Unknown
Rheumatic Diseases
Cyclooxygenase inhibitor
Small molecule
Approved
Unknown
Unknown
Hypotension, Orthostatic; Orthostatic Intolerance; Prostatic Neoplasms, Castration-Resistant; Hyperemesis Gravidarum; Hypoglycemia; Intestinal Obstruction; Myelodysplastic Syndromes; Pain; Wounds and Injuries; Gastroenteritis; Gastrointestinal Hemorrhage; Gastroparesis; Gastroschisis; Headache; HIV Infections; Migraine Disorders; Nausea; Neoplasms; Postoperative Nausea and Vomiting; Sepsis; Vomiting; Digestive System Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Hemorrhage; Postpartum Hemorrhage
Prostanoid FP receptor agonist
Small molecule
Approved
Unknown
Unknown
Anxiety; Dementia; Schizophrenia; Depressive Disorder
Unknown
Small molecule
Approved
OTHER
TOPICAL
Unknown
Glucocorticoid receptor agonist