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Total: 6532
Small molecule
Approved
Unknown
Unknown
Endocarditis; Infections; Intraabdominal Infections; Pneumonia; Sepsis; Urinary Tract Infections
Renal dipeptidase inhibitor
Small molecule
Approved
Unknown
Unknown
Irritable Bowel Syndrome; Blepharospasm; Charcot-Marie-Tooth Disease; Chronic Pain; Dystonic Disorders; Death, Sudden, Cardiac; Myocardial Infarction; Myotonic Dystrophy; Ventricular Fibrillation; Arrhythmias, Cardiac
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Azoospermia; Endocardial Cushion Defects; Heart Septal Defects, Ventricular; Infertility; Acquired Immunodeficiency Syndrome; beta-Thalassemia; Carbon Monoxide Poisoning; Diabetes Mellitus, Type 2; Heart Failure; Muscle Cramp; Neoplasms; Non-alcoholic Fatty Liver Disease; Poisoning; Polycystic Ovary Syndrome; Renal Insufficiency, Chronic; Shock, Septic; Spinal Cord Injuries; Acute Kidney Injury; Arthritis, Rheumatoid; Asthma; Atrial Fibrillation; Cytomegalovirus Infections; Gastrointestinal Stromal Tumors; HIV Infections; Hyperthyroidism; Hypotension; Lipid Metabolism Disorders; Multiple Sclerosis; Muscular Atrophy, Spinal; Pancreatic Neoplasms; Postpoliomyelitis Syndrome; Pyelonephritis; Brain Diseases; Kidney Failure, Chronic; Muscle Weakness
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Radiographic contrast agent
Small molecule
Approved
OTHER
ORAL
Obsessive-Compulsive Disorder; Fibromyalgia; Marijuana Abuse; Muscle Spasticity; Neuralgia; Obesity; Suicidal Ideation; Diabetic Neuropathies; Parkinson Disease; Nausea; Neoplasms; Postoperative Nausea and Vomiting
Cannabinoid CB1 receptor agonist
Small molecule
Approved
Unknown
Unknown
Multiple Sclerosis; Acidosis, Lactic; Heart Arrest; Huntington Disease; Respiratory Insufficiency; Heart Failure; Hyperemesis Gravidarum; Sepsis; Shock, Septic; Anemia; Brain Diseases; Kidney Failure, Chronic; Thiamine Deficiency
Unknown
Small molecule
Approved
OTHER
ORAL
Adenocarcinoma of Lung; Amebiasis; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Glioblastoma; HIV Infections; Small Cell Lung Carcinoma; Leukemia; Leukemia, Lymphocytic, Chronic, B-Cell; Ovarian Neoplasms; Pain; Tuberculosis; Arthritis, Rheumatoid; Rheumatic Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Barrett Esophagus; Erectile Dysfunction; Ischemia; Renal Insufficiency, Chronic; Cerebral Hemorrhage; Diabetes Mellitus, Type 1; Essential Hypertension; Glomerulonephritis, IGA; Heart Diseases; Melanoma; Pseudohypoaldosteronism; Stroke; Vascular Diseases; Cardiomyopathies; Cardiotoxicity; Chagas Cardiomyopathy; Coronary Disease; Heart Failure; Hematologic Neoplasms; Hypertension; Influenza, Human; Leukemia, Lymphoid; Leukemia, Myeloid, Acute; Lymphoma; Multiple Myeloma; Myocardial Ischemia; Neoplasms; Pneumonia; Severe Acute Respiratory Syndrome; ST Elevation Myocardial Infarction; Cardiovascular Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Glaucoma
Unknown
Small molecule
Approved
GASTROINTESTINAL; IMMUNE SYSTEM; OTHER
INHALATION; ORAL
Breast Neoplasms; Neoplasms; Diabetes Mellitus, Type 1; Encephalitis, Japanese; Hemorrhagic Fever with Renal Syndrome; Hepatitis D; Influenza, Human; Lassa Fever; Leukemia, Myeloid, Acute; Thrombocytopenia; Depressive Disorder; Hepatitis; Hepatitis B, Chronic; Hepatitis C; HIV Infections; Infections; Respiratory Syncytial Virus Infections; Severe Acute Respiratory Syndrome; Fibrosis; Hepatitis C, Chronic; Liver Cirrhosis; Virus Diseases
Inosine-5'-monophosphate dehydrogenase 1 inhibitor
Small molecule
Approved
Unknown
Unknown
Coronary Disease; Amyloidosis, Familial; Hemorrhagic Fever, Ebola; Severe Acute Respiratory Syndrome; Tachycardia, Supraventricular; Atrial Fibrillation; Atrial Flutter; Cardiomyopathies; Death, Sudden, Cardiac; Heart Arrest; Heart Diseases; Heart Failure; Myocardial Infarction; Tachycardia, Ventricular; Ventricular Fibrillation; Arrhythmias, Cardiac
Unknown
Small molecule
Approved
OTHER
TOPICAL
Unknown
Unknown
Small molecule
Approved
OTHER
OPHTHALMIC
Rheumatic Diseases
Cyclooxygenase inhibitor
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Hematologic Neoplasms; Lung Diseases; Bacterial Infections; Enterobacteriaceae Infections; Pneumonia, Bacterial; Pneumonia, Ventilator-Associated; Pyelonephritis; Endocarditis; Infections; Intraabdominal Infections; Pneumonia; Sepsis; Urinary Tract Infections
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Sepsis; Hematologic Neoplasms; Infections; Bacterial Infections; Pneumonia, Bacterial; Pneumonia, Ventilator-Associated; Pyelonephritis; Urinary Tract Infections
Renal dipeptidase inhibitor
Small molecule
Approved
OTHER
INJECTION; ORAL; RECTAL; URETHRAL
Breast Neoplasms; Fabry Disease; HIV Infections; Neoplasms; Renal Insufficiency; Acute Kidney Injury; Kidney Diseases; Myocardial Ischemia
Diagnostic agent
Small molecule
Approved
Unknown
Unknown
Anemia; Arthritis, Rheumatoid; Asthma; Infertility; Ovarian Neoplasms; Pancreatic Neoplasms; Penile Induration; Acute Kidney Injury; Adrenoleukodystrophy; Asthenozoospermia; Atherosclerosis; Brain Diseases; Burns; Cardiovascular Diseases; Carotid Artery Diseases; Diabetes Mellitus, Type 2; Endometriosis; Fibrosis; Friedreich Ataxia; Heart Diseases; Heart Failure; Heavy Metal Poisoning; Infertility, Male; Intracranial Arteriosclerosis; Lung Neoplasms; Mastodynia; Neoplasms; Neuromuscular Diseases; Peripheral Nervous System Diseases; Polycystic Ovary Syndrome; Renal Insufficiency, Chronic; Reperfusion Injury; Stomatitis; Tobacco Use Disorder; Wounds and Injuries; Alzheimer Disease; Amyotrophic Lateral Sclerosis; Breast Neoplasms; Cataract; Cerebrovascular Disorders; Colorectal Neoplasms; Coronary Disease; Delirium; Depressive Disorder; Fatty Liver; Gaucher Disease; Glaucoma; Head and Neck Neoplasms; Hypobetalipoproteinemias; Infections; Kidney Diseases; Liver Cirrhosis; Liver Diseases; Macular Degeneration; Menopause; Migraine Disorders; Myocardial Infarction; Myocardial Ischemia; Non-alcoholic Fatty Liver Disease; Osteonecrosis; Pain; Parkinson Disease; Prostatic Neoplasms, Castration-Resistant; Psoriasis; Pulmonary Disease, Chronic Obstructive; Rectal Neoplasms; Retinitis Pigmentosa; Schizophrenia; Urinary Bladder Neoplasms; Vascular Diseases
Unknown
Small molecule
Approved
OTHER
VAGINAL
Bacterial Infections
Bacterial dihydropteroate synthase inhibitor
Small molecule
Approved
OTHER
ORAL
Hepatolenticular Degeneration; Alcoholism; Feeding and Eating Disorders; Obesity; Bipolar Disorder; Lung Neoplasms; Neoplasms; Smoking; Smoking Cessation; Tobacco Use Disorder; Depressive Disorder; Depressive Disorder, Major; Mood Disorders; Seasonal Affective Disorder
Dopamine transporter inhibitor
Small molecule
Approved
OTHER
ORAL
Sleep Initiation and Maintenance Disorders
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
Unknown
NASAL
Alzheimer Disease; Amnesia; Amyotrophic Lateral Sclerosis; Anemia; Anemia, Sickle Cell; Anti-Neutrophil Cytoplasmic Antibody-Associated Vasculitis; Arthritis, Rheumatoid; Aspergillosis; Atherosclerosis; Burns; Carcinoma, Non-Small-Cell Lung; Cardiovascular Diseases; Chronic Pain; Cocaine-Related Disorders; Colitis, Ulcerative; Communicable Diseases; Cough; Crohn Disease; Cystic Fibrosis; Dermatitis, Atopic; Diabetes Mellitus, Type 2; Endometriosis; Gastrointestinal Stromal Tumors; Heart Failure; Hepatitis B, Chronic; Hepatitis C; Hepatitis C, Chronic; Hernia, Inguinal; HIV Infections; Infections; Influenza, Human; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Myeloid, Acute; Low Back Pain; Lung Neoplasms; Lymphoma, Non-Hodgkin; Malaria; Melanoma; Mesothelioma; Mitochondrial Diseases; Multiple Myeloma; Muscular Atrophy, Spinal; Myositis Ossificans; Nausea; Neck Pain; Neoplasm Metastasis; Neoplasms; Neuralgia; Non-alcoholic Fatty Liver Disease; Obesity; Osteoporosis, Postmenopausal; Parkinson Disease; Polycystic Kidney, Autosomal Dominant; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Pruritus; Psoriasis; Psychotic Disorders; Pulmonary Disease, Chronic Obstructive; Renal Insufficiency; Respiratory Syncytial Virus Infections; Sepsis; Severe Acute Respiratory Syndrome; Skin Diseases; Substance-Related Disorders; Suicidal Ideation; Tobacco Use Disorder; Trypanosomiasis; Tuberculosis; Urinary Tract Infections; Aggression; Bipolar Disorder; Borderline Personality Disorder; Breast Neoplasms; Cataract; Complex Regional Pain Syndromes; Depressive Disorder, Major; Depressive Disorder, Treatment-Resistant; Fractures, Multiple; Hypotension; Ischemic Stroke; Obsessive-Compulsive Disorder; Seizures; Stress Disorders, Post-Traumatic; Subarachnoid Hemorrhage; Tonsillitis; Tuberculosis, Pulmonary; Anxiety; Brain Injuries; Breech Presentation; Delirium; Dementia; Dental Anxiety; Depressive Disorder; Fluoride Poisoning; Fractures, Bone; Hemorrhage; Hypertension; Infertility; Liver Cirrhosis; Lung Diseases; Multiple Sclerosis, Relapsing-Remitting; Pain; Postoperative Nausea and Vomiting; Respiratory Insufficiency; Schizophrenia; Shock, Septic; Wounds and Injuries; Epilepsy; Status Epilepticus
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
Unknown
Unknown
Anemia, Sickle Cell; Amyotrophic Lateral Sclerosis; Anemia, Neonatal; Heart Failure; Huntington Disease; Asthma; Multiple Sclerosis; Anemia; Anemia, Iron-Deficiency; Diabetes Mellitus, Type 2; Kidney Failure, Chronic
Unknown
Small molecule
Approved
OTHER
ORAL
Alcoholism; Bipolar Disorder; Cognitive Dysfunction; Diabetes Mellitus, Type 2; Essential Tremor; Joint Diseases; Mental Disorders; Schizophrenia; Substance-Related Disorders; Alcohol Drinking; Amyotrophic Lateral Sclerosis; Anemia, Sickle Cell; Arthritis, Psoriatic; Arthritis, Rheumatoid; Child Development Disorders, Pervasive; Chronic Pain; Dementia; HIV Infections; Irritable Bowel Syndrome; Marijuana Abuse; Migraine with Aura; Migraine without Aura; Multiple Sclerosis; Neuralgia; Opioid-Related Disorders; Pain; Sleep Apnea, Obstructive; Stress Disorders, Post-Traumatic; Torticollis; Tourette Syndrome; Trichotillomania; Anorexia Nervosa; Osteoarthritis, Knee; Anorexia; Nausea; Neoplasms; Vomiting
Cannabinoid CB1 receptor agonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Alzheimer Disease; Anemia, Sickle Cell; Bipolar Disorder; Carcinoma, Non-Small-Cell Lung; Diabetes Mellitus, Type 2; Head and Neck Neoplasms; Leukemia, Lymphocytic, Chronic, B-Cell; Melanoma; Mitochondrial Diseases; Neoplasms; Prostatic Neoplasms, Castration-Resistant; Sexual Dysfunction, Physiological; Alcoholism; Amphetamine-Related Disorders; Cocaine-Related Disorders; Crohn Disease; Huntington Disease; Marijuana Abuse; Restless Legs Syndrome; Substance-Related Disorders; Anxiety; Attention Deficit Disorder with Hyperactivity; Dementia; Depressive Disorder, Treatment-Resistant; Obesity; Schizophrenia; Smoking Cessation; Tobacco Use Disorder; Depressive Disorder; Depressive Disorder, Major
Unknown
Small molecule
Approved
OTHER
ORAL
Bacterial Infections; Cryptosporidiosis; Lung Diseases; Tuberculosis, Multidrug-Resistant; Crohn Disease; Mycobacterium avium-intracellulare Infection; Tuberculosis; Tuberculosis, Pulmonary; Leprosy
DNA inhibitor
Small molecule
Approved
MUSCULOSKELETAL; OTHER; RHEUMATOLOGY
ORAL
Kidney Calculi; Renal Colic; Multiple Sclerosis; Paget Disease, Extramammary; Periodontitis; Bursitis; Inflammation; Low Back Pain; Migraine Disorders; Osteoarthritis, Knee; Postoperative Nausea and Vomiting; Sprains and Strains; Tendinopathy; Wounds and Injuries; Acute Pain; Arthralgia; Arthritis, Rheumatoid; Dysmenorrhea; Myalgia; Osteoarthritis; Rheumatic Diseases
Cyclooxygenase inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Asthma
Unknown
Small molecule
Approved
OTHER
OPHTHALMIC; ORAL
Osteomyelitis; Hermanski-Pudlak Syndrome; Cystitis, Hemorrhagic; Esophageal and Gastric Varices; Liver Cirrhosis; Peritonitis; Bacterial Infections; Eye Infections
Bacterial DNA gyrase inhibitor
Small molecule
Approved
Unknown
Unknown
Carcinoma, Non-Small-Cell Lung; Colorectal Neoplasms; Fibrosis; Glycogen Storage Disease Type III; HIV Infections; Leukemia, Hairy Cell; Lupus Erythematosus, Systemic; Melanoma; Mesothelioma; Neoplasms; Psoriasis; Thyroid Neoplasms; Anemia, Sickle Cell; Breast Carcinoma In Situ; Breast Neoplasms; Eosinophilic Esophagitis; Immunoglobulin G4-Related Disease; Movement Disorders; Schizophrenia; Stomach Neoplasms; Gastrointestinal Hemorrhage; Severe Acute Respiratory Syndrome; Arthritis, Rheumatoid; Chest Pain; Duodenal Ulcer; Esophagitis; Gastroesophageal Reflux; Heartburn; Osteoarthritis; Peptic Ulcer; Stomach Ulcer; Ulcer
Histamine H2 receptor antagonist
Small molecule
Approved
Unknown
Unknown
Lung Diseases, Obstructive
Unknown
Small molecule
Approved
Unknown
Unknown
Common Cold; Fecal Incontinence; Hypotension, Orthostatic; Presbyopia; Rhinitis, Allergic, Seasonal; Erythema; Rosacea; Eye Manifestations; Nasal Obstruction
Unknown