Display Options:
Total: 6532
Small molecule
Approved
OTHER
INJECTION
Astrocytoma; Glioblastoma; Glioma; Multiple Sclerosis, Chronic Progressive; Paraganglioma; Central Nervous System Diseases
Diagnostic agent
Small molecule
Approved
Unknown
Unknown
Cardiovascular Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Asthma; Eye Manifestations; Lung Diseases, Obstructive; Nasal Obstruction
Unknown
Small molecule
Approved
IMMUNE SYSTEM; OTHER
TOPICAL
Hepatitis B, Chronic; Mycoses; Colitis, Ulcerative; Crohn Disease; Tinea Pedis; Onychomycosis; Tinea
Squalene monooxygenase inhibitor
Small molecule
Approved
Unknown
Unknown
Bacterial Infections
Unknown
Small molecule
Approved
OTHER
ORAL
Osteomyelitis; Otitis Media
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
CANCER; OTHER; RESPIRATORY
INJECTION; IV (INFUSION)
Anus Neoplasms; Brain Neoplasms; Carcinoid Tumor; Carcinoma, Intraductal, Noninfiltrating; Carcinoma, Renal Cell; Carcinoma, Small Cell; Carcinoma, Verrucous; Coronary Restenosis; Glioblastoma; Gliosarcoma; Hodgkin Disease; Leukemia, Lymphocytic, Chronic, B-Cell; Liver Neoplasms; Mesothelioma; Neoplasms, Cystic, Mucinous, and Serous; Rectal Neoplasms; Thyroid Carcinoma, Anaplastic; Vaginal Neoplasms; Adenocarcinoma, Bronchiolo-Alveolar; Adrenal Cortex Neoplasms; Arthritis, Rheumatoid; Bone Neoplasms; Breast Carcinoma In Situ; Carcinoma, Ductal; Carcinoma, Endometrioid; Carcinoma, Hepatocellular; Carcinoma, Merkel Cell; Carcinoma, Neuroendocrine; Carcinoma, Ovarian Epithelial; Central Nervous System Neoplasms; Cholangiocarcinoma; Colorectal Neoplasms; Constriction, Pathologic; Cystadenoma, Serous; Digestive System Diseases; Gallbladder Neoplasms; Gastrointestinal Stromal Tumors; Glioma; Hemangiosarcoma; Hereditary Breast and Ovarian Cancer Syndrome; Hypopharyngeal Neoplasms; Keratosis, Actinic; Kidney Neoplasms; Leukemia; Lymphoma; Mouth Neoplasms; Multiple Myeloma; Neoplasms, Complex and Mixed; Neoplasms, Germ Cell and Embryonal; Oropharyngeal Neoplasms; Penile Neoplasms; Peripheral Vascular Diseases; Prostatic Hyperplasia; Prostatic Neoplasms; Psoriasis; Salivary Gland Neoplasms; Small Cell Lung Carcinoma; Thymoma; Uterine Cervical Dysplasia; Uveal Melanoma; Vulvar Neoplasms; Adenocarcinoma; Adenocarcinoma of Lung; Anemia; Biliary Tract Neoplasms; Breast Neoplasms, Male; Carcinoma, Large Cell; Carcinoma, Pancreatic Ductal; Carcinoma, Squamous Cell; Endometrial Neoplasms; Esophageal Neoplasms; Fallopian Tube Neoplasms; Genital Neoplasms, Female; Gestational Trophoblastic Disease; Head and Neck Neoplasms; HIV Infections; Hypersensitivity; Inflammatory Breast Neoplasms; Ischemia; Lung Neoplasms; Lymphoma, Non-Hodgkin; Melanoma; Nasopharyngeal Carcinoma; Nasopharyngeal Neoplasms; Neoplasm Metastasis; Pain; Paraganglioma; Peripheral Arterial Disease; Peripheral Nervous System Diseases; Peritoneal Neoplasms; Prostatic Neoplasms, Castration-Resistant; Retroviridae Infections; Sarcoma; Sex Cord-Gonadal Stromal Tumors; Squamous Cell Carcinoma of Head and Neck; Stomach Neoplasms; Teratoma; Testicular Neoplasms; Thyroid Neoplasms; Triple Negative Breast Neoplasms; Urethral Neoplasms; Urinary Bladder Neoplasms; Urogenital Neoplasms; Uterine Cervical Neoplasms; Uterine Neoplasms; Breast Neoplasms; Carcinoma; Carcinoma, Non-Small-Cell Lung; Neoplasms; Ovarian Neoplasms; Pancreatic Neoplasms; Sarcoma, Kaposi
Tubulin inhibitor
Small molecule
Approved
OTHER
ORAL
HIV Infections; Virus Diseases
Human immunodeficiency virus type 1 reverse transcriptase inhibitor
Small molecule
Approved
Unknown
Unknown
Melanosis; Skin Neoplasms; Sunburn
Unknown
Small molecule
Approved
Unknown
Unknown
Lecithin Cholesterol Acyltransferase Deficiency; Essential Hypertension; Proteinuria; Angina Pectoris; Angina Pectoris, Variant; Angina, Stable; Coronary Artery Disease; Diabetes Mellitus; Heart Failure; Hypercholesterolemia; Hyperlipidemias; Hyperlipoproteinemia Type II; Hypertension; Myocardial Infarction; Osteoarthritis; Stroke
Voltage-gated L-type calcium channel blocker
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Dystonic Disorders; Low Back Pain; Marijuana Abuse; Obesity; Prostatic Neoplasms; Autistic Disorder; Parkinson Disease; Substance-Related Disorders; Anxiety; Attention Deficit Disorder with Hyperactivity; Dementia; Depressive Disorder; Schizophrenia; Sleep Initiation and Maintenance Disorders; Sleep Wake Disorders
Unknown
Small molecule
Approved
Unknown
Unknown
Breast Neoplasms; Erectile Dysfunction; HIV Infections; Hyperlipidemias; Kidney Diseases; Neoplasms; Pancreatitis; Aortic Aneurysm, Abdominal; Aortic Valve Insufficiency; beta-Thalassemia; Cardiomyopathy, Hypertrophic; Dystonic Disorders; Heart Diseases; Hyperaldosteronism; Liver Diseases; Raynaud Disease; Thalassemia; Vascular Diseases; Atherosclerosis; Coronary Disease; Depressive Disorder; Diabetes Mellitus; Diabetes Mellitus, Type 2; Essential Hypertension; Heart Failure; Hypercholesterolemia; Hypertension; Myocardial Infarction; Myocardial Ischemia; Cardiovascular Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Melanosis; Skin Neoplasms; Sunburn
Unknown
Small molecule
Approved
OTHER
ORAL
Carcinoma, Non-Small-Cell Lung; Gastroesophageal Reflux; Leukemia, Myeloid, Acute; Infections; Severe Acute Respiratory Syndrome; Toxoplasmosis, Cerebral; Malaria, Falciparum; Amebiasis; Malaria; Pneumocystis Infections; Pneumonia, Pneumocystis
Cytochrome b inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Lecithin Cholesterol Acyltransferase Deficiency; Acute Coronary Syndrome; Muscular Dystrophy, Duchenne; Hypertension
Beta-1 adrenergic receptor antagonist
Small molecule
Approved
DERMATOLOGY; DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Hyperplasia; Hypogonadism; Acne Vulgaris; Carcinoma, Non-Small-Cell Lung; Prostatic Neoplasms, Castration-Resistant; Retinal Diseases; Alopecia; Prostatic Hyperplasia; Prostatic Neoplasms
Steroid 5-alpha-reductase 2 inhibitor
Small molecule
Approved
OTHER
OPHTHALMIC
Unknown
Unknown
Small molecule
Approved
CARDIOVASCULAR
ORAL
Bronchopulmonary Dysplasia
Unknown
Small molecule
Approved
OTHER
INTRAMUSCULAR; ORAL; SUBCUTANEOUS
Dyskinesia, Drug-Induced; Huntington Disease; Lecithin Cholesterol Acyltransferase Deficiency; Opioid-Related Disorders; Schizotypal Personality Disorder; Amphetamine-Related Disorders; Child Development Disorders, Pervasive; Cocaine-Related Disorders; Obsessive-Compulsive Disorder; Stress Disorders, Post-Traumatic; Substance-Related Disorders; Tourette Syndrome; Alzheimer Disease; Anxiety; Asperger Syndrome; Attention Deficit and Disruptive Behavior Disorders; Conduct Disorder; Dementia; Dementia, Vascular; Depressive Disorder; Depressive Disorder, Major; Developmental Disabilities; Intellectual Disability; Mental Disorders; Neurodevelopmental Disorders; Rett Syndrome; Aggression; Autistic Disorder; Bipolar Disorder; Psychotic Disorders; Schizophrenia
Dopamine D2 receptor antagonist
Small molecule
Approved
Unknown
Unknown
Digestive System Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Corneal Ulcer; Hyperopia; Multiple Sclerosis; Muscular Diseases; Uterine Cervical Neoplasms; Acidosis, Lactic; Brain Concussion; Chronic Pain; Heart Failure; Myocardial Infarction; Myopia; Psoriasis; Refractive Errors; Diabetic Neuropathies; Hematologic Diseases; Keratoconus; Stroke; Anemia; Anemia, Iron-Deficiency; Eye Diseases; Folic Acid Deficiency; Kidney Failure, Chronic
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Central Nervous System Neoplasms; Graft vs Host Disease; Multiple Myeloma; Myeloproliferative Disorders; Neoplasms, Plasma Cell; Cholangitis, Sclerosing; Histiocytosis; Histiocytosis, Langerhans-Cell; Leukemia, Biphenotypic, Acute; Leukemia, Myeloid; Lymphoma, B-Cell, Marginal Zone; Lymphoma, Mantle-Cell; Mastocytosis, Systemic; Multiple Sclerosis, Chronic Progressive; Myelodysplastic Syndromes; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Leukemia; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Myeloid, Acute; Lymphoma; Lymphoma, T-Cell, Peripheral; Multiple Sclerosis, Relapsing-Remitting; Anemia; Immune System Diseases; Leukemia, Hairy Cell; Multiple Sclerosis; Neoplasms
DNA inhibitor
Small molecule
Approved
Unknown
Unknown
Amebiasis
Unknown
Small molecule
Approved
OTHER
INJECTION
Colorectal Neoplasms; Pancreatic Neoplasms; Sarcoma; Pneumonia, Pneumocystis
Dihydrofolate reductase inhibitor
Small molecule
Approved
Unknown
Unknown
Amphetamine-Related Disorders; Stress Disorders, Post-Traumatic; Substance-Related Disorders; Alzheimer Disease; Aortic Aneurysm, Abdominal; Breast Neoplasms; Neoplasms; Cardiomyopathy, Dilated; Diabetes Mellitus, Type 2; Hypertension; Marfan Syndrome; Cardiovascular Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Arthritis, Rheumatoid; Dermatitis, Atopic; Lymphoma; Multiple Myeloma; Multiple Sclerosis; Back Pain; Breast Neoplasms; Eosinophilic Esophagitis; Lymphangioleiomyomatosis; Severe Acute Respiratory Syndrome; Asthma; Hypersensitivity; Pruritus; Rhinitis, Allergic, Perennial; Rhinitis, Allergic, Seasonal; Urticaria
Histamine H1 receptor antagonist
Small molecule
Approved
Unknown
Unknown
Depressive Disorder
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Diabetes Mellitus, Type 2; Pre-Eclampsia; Cardiovascular Diseases; Heart Failure; Hypertension; Myocardial Infarction; Stroke
Sodium-(potassium)-chloride cotransporter 2 inhibitor
Small molecule
Approved
Unknown
Unknown
Kidney Diseases; Osteomyelitis; Otitis Media; Appendicitis; Communicable Diseases; Graft vs Host Disease; Abscess; Cholecystitis, Acute; Diabetic Foot; Enterobacteriaceae Infections; Hematologic Neoplasms; Infections; Influenza, Human; Lung Diseases; Pneumonia; Pneumonia, Bacterial; Pneumonia, Ventilator-Associated; Pseudomonas Infections; Pyelonephritis; Sepsis; Severe Acute Respiratory Syndrome; Shock, Septic; Urinary Tract Infections; Bacterial Infections
Unknown
Small molecule
Approved
OTHER
ORAL
Bipolar Disorder; Anemia; Epilepsy; Seizures
Glutamate [NMDA] receptor antagonist
Small molecule
Approved
Unknown
Unknown
Dysmenorrhea; Pulpitis; Stomach Ulcer; Toothache; Acute Pain; Arthritis, Rheumatoid; Migraine Disorders; Osteoarthritis; Pain
Cyclooxygenase inhibitor
Small molecule
Approved
OTHER
INJECTION
Unknown
Diagnostic agent