Display Options:
Total: 6532
Small molecule
Approved
Unknown
Unknown
Hepatitis; Hepatitis B, Chronic; Hepatitis C, Chronic; Hepatitis D; Liver Cirrhosis, Biliary; HIV Infections; Severe Acute Respiratory Syndrome; Virus Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Endometritis; Appendicitis; Pyelonephritis; Renal Insufficiency, Chronic; Tuberculosis; Tuberculosis, Pulmonary; Diabetic Foot; Gonorrhea; Infections; Osteomyelitis; Pneumonia; Urinary Tract Infections; Bacterial Infections
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
DERMATOLOGY
TOPICAL
Netherton Syndrome; Dermatitis, Seborrheic; Dry Eye Syndromes; Lichen Planus, Oral; Lichen Sclerosus et Atrophicus; Vitiligo; Dermatitis; Dermatitis, Perioral; Lichen Planus; Dermatitis, Atopic; Eczema
FK506-binding protein 1A inhibitor
Small molecule
Approved
EYE; OTHER
OPHTHALMIC
Exfoliation Syndrome; Glaucoma; Glaucoma, Open-Angle; Ocular Hypertension
Prostanoid FP receptor agonist
Small molecule
Approved
Unknown
Unknown
Pain; Migraine Disorders
Unknown
Small molecule
Approved
IMMUNE SYSTEM; OTHER
ORAL
Hepatitis C; Hepatitis, Chronic; Insulin Resistance; Lymphoma; Parkinson Disease; Tuberculosis; Communicable Diseases; Hepatitis D; Lipodystrophy; Liver Cirrhosis, Biliary; Multiple Sclerosis; Acquired Immunodeficiency Syndrome; Severe Acute Respiratory Syndrome; Hepatitis B, Chronic; HIV Infections; Infections; Liver Diseases
Human immunodeficiency virus type 1 reverse transcriptase inhibitor
Small molecule
Approved
OTHER; RESPIRATORY
INHALATION
Lung Neoplasms; Tobacco Use Disorder; Asthma; Bronchial Spasm; Bronchitis, Chronic; Emphysema; Pulmonary Disease, Chronic Obstructive
Beta-2 adrenergic receptor agonist
Small molecule
Approved
Unknown
ORAL
Obesity; Bulimia; Bulimia Nervosa; Depressive Disorder; Hidradenitis Suppurativa; Premenstrual Syndrome; Dysmenorrhea; Polycystic Ovary Syndrome; Acne Vulgaris
Mineralocorticoid receptor antagonist
Small molecule
Approved
OTHER; PREGNANCY AND GYNECOLOGY
ORAL
Osteoarthritis, Knee; Pancreatitis; Pain; Pharyngitis; Arthritis, Rheumatoid; Dysmenorrhea; Osteoarthritis; Rheumatic Diseases
Cyclooxygenase-2 inhibitor
Small molecule
Approved
Unknown
Unknown
Hypotension, Orthostatic; Lecithin Cholesterol Acyltransferase Deficiency; Memory; Obesity; Subarachnoid Hemorrhage; Cocaine-Related Disorders; HIV Infections; Psychotic Disorders; Tobacco Use Disorder; Alzheimer Disease; Anxiety; Autistic Disorder; Dementia, Vascular; Depressive Disorder; Lewy Body Disease; Schizophrenia; Dementia
Unknown
Small molecule
Approved
CANCER; DIABETES DRUGS & ENDOCRINOLOGY; MUSCULOSKELETAL; OTHER
INJECTION; INTRAVENOUS; IV (INFUSION)
Adenocarcinoma; Anemia, Sickle Cell; Chondrosarcoma; Menopause; Neuroblastoma; beta-Thalassemia; Bone Resorption; Carcinoma, Intraductal, Noninfiltrating; Complex Regional Pain Syndromes; Kidney Neoplasms; Leiomyosarcoma; Low Back Pain; Macular Degeneration; Mesothelioma; Nasopharyngeal Neoplasms; Osteosarcoma; Pancreatic Neoplasms; Primary Myelofibrosis; Progeria; Urogenital Neoplasms; Uterine Cervical Neoplasms; Arthritis, Rheumatoid; Bone Diseases, Metabolic; Bone Neoplasms; Breast Neoplasms; Carcinoma, Hepatocellular; Carcinoma, Non-Small-Cell Lung; Giant Cell Tumors; Lung Neoplasms; Lymphoma; Lymphoma, Non-Hodgkin; Neoplasms, Plasma Cell; Osteoarthritis, Hip; Osteogenesis Imperfecta; Osteonecrosis; Pain; Plasmacytoma; Sarcoma; Sarcoma, Ewing; Spinal Cord Injuries; Bone Diseases; Fractures, Bone; Hypercalcemia; Multiple Myeloma; Neoplasm Metastasis; Osteitis Deformans; Osteoporosis; Osteoporosis, Postmenopausal; Prostatic Neoplasms
Farnesyl diphosphate synthase inhibitor
Small molecule
Approved
IMMUNE SYSTEM; OTHER
ORAL
Urinary Tract Infections; Bronchitis, Chronic; Infections; Pharyngitis; Tonsillitis
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
Unknown
Unknown
Attention Deficit Disorder with Hyperactivity
Unknown
Small molecule
Approved
IMMUNE SYSTEM; OTHER; RESPIRATORY
ORAL
Lecithin Cholesterol Acyltransferase Deficiency; Carcinoma, Non-Small-Cell Lung; Common Cold; Conjunctivitis, Allergic; Dermatitis; Eczema; Multiple Sclerosis; Multiple Sclerosis, Chronic Progressive; Pruritus; Hypersensitivity; Rhinitis, Allergic, Perennial; Rhinitis, Allergic, Seasonal; Urticaria
Histamine H1 receptor antagonist
Small molecule
Approved
Unknown
Unknown
Cardiovascular Diseases; Opioid-Related Disorders; Substance-Related Disorders; Autistic Disorder; Borderline Personality Disorder; Depressive Disorder, Major; Mood Disorders; Phobia, Social; Anxiety; Bipolar Disorder; Dementia; Depressive Disorder; Schizophrenia; Psychotic Disorders
Unknown
Small molecule
Approved
Unknown
Unknown
Alzheimer Disease; Bronchiolitis Obliterans; Hypersensitivity; Respiratory Distress Syndrome; Severe Acute Respiratory Syndrome; Asthma; Bronchiectasis; Bronchitis; Emphysema; Pulmonary Disease, Chronic Obstructive; Lung Diseases, Obstructive
Unknown
Small molecule
Approved
Unknown
Unknown
Acute Lung Injury; Carcinoma, Renal Cell; Carcinoma, Squamous Cell; Colorectal Neoplasms; Desmoplastic Small Round Cell Tumor; Fibrosarcoma; Head and Neck Neoplasms; Hematologic Neoplasms; Liver Cirrhosis; Lymphoma, Large-Cell, Anaplastic; Lymphoma, Non-Hodgkin; Pancreatic Neoplasms; Rhinitis, Allergic, Seasonal; Thymoma; Arthritis, Rheumatoid; Breast Neoplasms; Chordoma; Colonic Neoplasms; Desmoid Tumors; Fibroma; Glioblastoma; Hypereosinophilic Syndrome; Leukemia, Lymphoid; Leukemia, Myeloid, Acute; Lung Neoplasms; Malaria, Falciparum; Melanoma; Scleroderma, Systemic; Spinal Cord Injuries; Stomach Neoplasms; Thyroid Neoplasms; Tuberculosis; Gastrointestinal Stromal Tumors; Graft vs Host Disease; Hypertension, Pulmonary; Influenza, Human; Leukemia; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid; Neoplasms; Pneumonia; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Sarcoma; Severe Acute Respiratory Syndrome; Stroke
Unknown
Small molecule
Approved
OTHER; UROLOGY AND KIDNEY
ORAL
Aging; Amyotrophic Lateral Sclerosis; Bulbo-Spinal Atrophy, X-Linked; Prostatitis; Severe Acute Respiratory Syndrome; Alopecia; Hypogonadism; Prostatic Neoplasms, Castration-Resistant; Prostatic Hyperplasia; Prostatic Neoplasms
Steroid 5-alpha-reductase inhibitor
Small molecule
Approved
OTHER
ORAL
Cystic Fibrosis; Diabetes Mellitus, Type 2; Hepatitis B, Chronic; Hepatitis C; Hepatitis C, Chronic; HIV Infections; Infertility, Female; Leukemia, Lymphocytic, Chronic, B-Cell; Non-alcoholic Fatty Liver Disease; Obesity; Bulimia; Bulimia Nervosa; Depressive Disorder; Endometrial Neoplasms; Hidradenitis Suppurativa; Hyperandrogenism; Metrorrhagia; Osteoporosis; Premenstrual Syndrome; Amenorrhea; Anorexia Nervosa; Bone Diseases, Metabolic; Breast Neoplasms; Dysmenorrhea; Endometriosis; Migraine Disorders; Neural Tube Defects; Polycystic Ovary Syndrome; Pregnancy; Turner Syndrome; Acne Vulgaris; Neoplasms
Estrogen receptor alpha agonist
Small molecule
Approved
Unknown
Unknown
Arthritis, Juvenile; Breast Neoplasms; Fatty Liver; Hepatitis B, Chronic; Hypertension, Pulmonary; Lymphoma; Neoplasms; Non-alcoholic Fatty Liver Disease; Asthma; Autistic Disorder; Child Development Disorders, Pervasive; Cystic Fibrosis; Dyspepsia; Eosinophilic Esophagitis; Neuralgia; Digestive System Diseases; Duodenal Ulcer; Esophageal Neoplasms; Esophagitis, Peptic; Gastritis; Gastroesophageal Reflux; Gastrointestinal Hemorrhage; Helicobacter Infections; Hemorrhage; Nausea; Osteoarthritis; Peptic Ulcer; Pre-Eclampsia; Stomach Ulcer; Ulcer
Unknown
Small molecule
Approved
Unknown
Unknown
HIV Infections; Metrorrhagia; Pregnancy
Progesterone receptor agonist
Small molecule
Approved
Unknown
Unknown
Migraine Disorders
Unknown
Small molecule
Approved
IMMUNE SYSTEM; OTHER; PEDIATRICS
ORAL
HIV Infections; Irritable Bowel Syndrome; Kidney Diseases; Liver Diseases; Bronchiolitis; Crohn Disease; Diabetes Mellitus, Type 2; Gastroenteritis; Hepatitis B, Chronic; Hepatitis C; Hepatitis C, Chronic; Malnutrition; Periodontitis; Sexually Transmitted Diseases; Tuberculosis; Arthritis, Rheumatoid; Brain Diseases; Clostridium Infections; Cryptosporidiosis; Dyspepsia; Enterocolitis, Pseudomembranous; Helicobacter Infections; Influenza, Human; Peritonitis; Respiratory Tract Diseases; Severe Acute Respiratory Syndrome; Amebiasis; Diarrhea
Pyruvate:ferredoxin oxidoreductase inhibitor
Small molecule
Approved
IMMUNE SYSTEM; OTHER
ORAL
Hepatitis, Chronic; Cytomegalovirus Infections; HIV Infections; Hepatitis B, Chronic; Virus Diseases
DNA polymerase/reverse transcriptase inhibitor
Small molecule
Approved
Unknown
Unknown
Amphetamine-Related Disorders; Cocaine-Related Disorders; Diabetes Mellitus, Type 1; Orthostatic Intolerance; Parkinson Disease; Tobacco Use Disorder; Alcoholism; Cognitive Dysfunction; Hypotension, Orthostatic; Marijuana Abuse; Opioid-Related Disorders; Phobia, Social; Sleep Apnea, Obstructive; Sleep Apnea Syndromes; Substance-Related Disorders; Syncope, Vasovagal; Tourette Syndrome; Autistic Disorder; Neoplasms; Schizophrenia; Attention Deficit Disorder with Hyperactivity
Unknown
Small molecule
Approved
CANCER
INTRAMUSCULAR
Carcinoma, Ductal; Carcinoma, Squamous Cell; Colorectal Neoplasms; Hereditary Breast and Ovarian Cancer Syndrome; Lymphoma; Lymphoma, Non-Hodgkin; Mesothelioma; Pancreatic Neoplasms; Small Cell Lung Carcinoma; Urinary Bladder Neoplasms; Carcinoma; Carcinoma, Intraductal, Noninfiltrating; Carcinoma, Non-Small-Cell Lung; Endometrial Neoplasms; Fibrous Dysplasia, Polyostotic; Genital Neoplasms, Female; Hypertension, Pulmonary; Lung Neoplasms; Lupus Erythematosus, Systemic; Ovarian Neoplasms; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Puberty, Precocious; Sarcoma, Endometrial Stromal; Carcinoma, Lobular; Neoplasm Metastasis; Breast Neoplasms; Neoplasms
Estrogen receptor alpha antagonist
Small molecule
Approved
OTHER
ORAL
HIV Infections; Prostatic Neoplasms, Castration-Resistant; Hepatitis C, Chronic; Hepatitis D; Non-alcoholic Fatty Liver Disease; Aortic Valve Stenosis; Atherosclerosis; Coronary Disease; Diabetes Mellitus; Diabetes Mellitus, Type 2; Hypertension; Hypertriglyceridemia; Lipid Metabolism Disorders; Metabolic Syndrome; Metabolism, Inborn Errors; Myocardial Infarction; Cardiovascular Diseases; Hypercholesterolemia; Hyperlipidemias; Hyperlipoproteinemia Type II
Niemann-Pick C1-like protein 1 inhibitor
Small molecule
Approved
Unknown
Unknown
Alzheimer Disease; Hepatitis C; Premature Ejaculation; Aphasia; Borderline Personality Disorder; Cocaine-Related Disorders; Digestive System Diseases; Fibromyalgia; Panic Disorder; Phobia, Social; Phobic Disorders; Renal Insufficiency, Chronic; Stress Disorders, Post-Traumatic; Stroke; Substance-Related Disorders; Anxiety; Anxiety Disorders; Arthritis, Rheumatoid; Bipolar Disorder; Burning Mouth Syndrome; Carcinoma; Dementia; Hypertension, Pulmonary; Neoplasms; Obsessive-Compulsive Disorder; Schizophrenia; Depressive Disorder; Depressive Disorder, Major
Unknown
Small molecule
Approved
OTHER
INTRAMUSCULAR; ORAL; ORALLY DISINTEGRATING
Amphetamine-Related Disorders; Asperger Syndrome; Attention Deficit Disorder with Hyperactivity; Cocaine-Related Disorders; Fragile X Syndrome; Obsessive-Compulsive Disorder; Trichotillomania; Alcoholism; Alzheimer Disease; Anorexia Nervosa; Anxiety; Child Development Disorders, Pervasive; Dementia; Depression, Postpartum; Mental Disorders; Stress Disorders, Post-Traumatic; Tic Disorders; Aggression; Autistic Disorder; Bipolar Disorder; Depressive Disorder; Depressive Disorder, Major; Psychomotor Agitation; Psychotic Disorders; Schizophrenia; Tourette Syndrome
Dopamine D2 receptor partial agonist
Small molecule
Approved
CANCER; OTHER
INJECTION; INTRAVENOUS
Digestive System Diseases; Gastrointestinal Stromal Tumors; Glioblastoma; Gliosarcoma; Hematologic Neoplasms; Leukemia; Leukemia, Myeloid, Acute; Liver Diseases; Lymphoma, T-Cell, Cutaneous; Melanoma; Myelodysplastic Syndromes; Neuroblastoma; Triple Negative Breast Neoplasms; Anus Neoplasms; Bile Duct Neoplasms; Breast Neoplasms; Carcinoid Tumor; Carcinoma, Islet Cell; Carcinoma, Neuroendocrine; Carcinoma, Ovarian Epithelial; Carcinoma, Renal Cell; Carcinoma, Transitional Cell; Central Nervous System Neoplasms; Digestive System Neoplasms; Endometrial Neoplasms; Fallopian Tube Neoplasms; Head and Neck Neoplasms; Hodgkin Disease; Klatskin Tumor; Leukemia-Lymphoma, Adult T-Cell; Lung Neoplasms; Lymphoma, Follicular; Lymphoma, T-Cell, Peripheral; Mesothelioma; Nasopharyngeal Carcinoma; Nasopharyngeal Neoplasms; Neoplasms, Germ Cell and Embryonal; Neuroendocrine Tumors; Ovarian Neoplasms; Peripheral Nervous System Diseases; Peritoneal Neoplasms; Prostatic Neoplasms, Castration-Resistant; Small Cell Lung Carcinoma; Urinary Bladder Neoplasms; Uterine Cervical Neoplasms; Uterine Neoplasms; Adenocarcinoma; Biliary Tract Neoplasms; Carcinoma; Carcinoma, Hepatocellular; Carcinoma, Non-Small-Cell Lung; Carcinoma, Pancreatic Ductal; Carcinoma, Squamous Cell; Cholangiocarcinoma; Colonic Neoplasms; Colorectal Neoplasms; Colorectal Neoplasms, Hereditary Nonpolyposis; Esophageal Neoplasms; Gallbladder Neoplasms; Granuloma, Lethal Midline; Hepatoblastoma; Liver Neoplasms; Lymphoma; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Non-Hodgkin; Neoplasm Metastasis; Pancreatic Neoplasms; Pulmonary Disease, Chronic Obstructive; Rectal Neoplasms; Stomach Neoplasms; Teratoma; Testicular Neoplasms; Neoplasms
DNA inhibitor
Small molecule
Approved
CARDIOVASCULAR; OTHER
ORAL
Diabetes Mellitus, Type 2; Atrial Fibrillation; Breast Neoplasms; Central Serous Chorioretinopathy; Diabetic Nephropathies; Hyperparathyroidism, Primary; Cardiomyopathies; Essential Hypertension; Muscular Dystrophy, Duchenne; Renal Insufficiency, Chronic; Cardiovascular Diseases; Heart Failure; Hypertension; Myocardial Infarction; Stroke
Mineralocorticoid receptor antagonist
Small molecule
Approved
Unknown
Unknown
Migraine with Aura; Migraine without Aura; Migraine Disorders
Unknown
Small molecule
Approved
Unknown
Unknown
Glomerulonephritis; Atherosclerosis; Diabetic Nephropathies; Essential Hypertension; Kidney Diseases; Proteinuria; Cardiovascular Diseases; Diabetes Mellitus; Heart Failure; Hypertension; Myocardial Infarction; Stroke
Type-1 angiotensin II receptor antagonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Dyspepsia; Gastroesophageal Reflux; Constipation
Unknown