Display Options:
Total: 6532
Small molecule
Approved
Unknown
Unknown
Acquired Immunodeficiency Syndrome; HIV Infections
Human immunodeficiency virus type 1 integrase inhibitor
Small molecule
Unknown
Unknown
Unknown
Unknown
Progesterone receptor agonist
Small molecule
Approved
Unknown
ORAL
Kidney Diseases; HIV Infections; Virus Diseases
Reverse transcriptase negative allosteric modulator
Small molecule
Approved
Unknown
INHALATION
Kidney Diseases; Liver Diseases; Lung Diseases, Obstructive; Pulmonary Disease, Chronic Obstructive
Muscarinic acetylcholine receptor M3 antagonist
Small molecule
Approved
Unknown
Unknown
Cocaine-Related Disorders; Heroin Dependence; Liver Failure; Marijuana Abuse; Opioid-Related Disorders; Substance-Related Disorders
Unknown
Small molecule
Approved
Unknown
Unknown
Carcinoma, Non-Small-Cell Lung; Kidney Diseases; Liver Diseases; Blast Crisis; Myelodysplastic Syndromes; Leukemia, Myeloid, Acute; Neoplasms
Tyrosine-protein kinase receptor FLT3 inhibitor
Small molecule
Unknown
Unknown
Unknown
Smallpox; Virus Diseases
Envelope phospholipase F13 (p37) inhibitor
Small molecule
Approved
Unknown
ORAL
Dermatitis, Allergic Contact; Graft vs Host Disease; Sjogren's Syndrome; Diabetes Mellitus, Type 1; Diabetic Nephropathies; Giant Cell Arteritis; Liver Cirrhosis, Biliary; Myositis; Pneumonia; Psoriasis; Vitiligo; Alopecia Areata; Arthritis, Juvenile; Dermatitis, Atopic; Dermatomyositis; Lupus Erythematosus, Systemic; Severe Acute Respiratory Syndrome; Uveitis; Arthritis, Rheumatoid; Immune System Diseases
Tyrosine-protein kinase JAK1 inhibitor
Small molecule
Approved
Unknown
ORAL
Purpura, Thrombocytopenic, Idiopathic; Hemorrhage; Thrombocytopenia
Thrombopoietin receptor agonist
Small molecule
Approved
Unknown
ORAL
Kidney Diseases; Neuroblastoma; Lymphoma, Large-Cell, Anaplastic; Carcinoma, Non-Small-Cell Lung; Lymphoma; Neoplasms
ALK tyrosine kinase receptor inhibitor
Small molecule
Approved
Unknown
ORAL
Influenza, Human; Virus Diseases
Polymerase acidic protein inhibitor
Small molecule
Approved
Unknown
Unknown
Nausea; Vomiting
Neurokinin 1 receptor antagonist
Small molecule
Approved
Unknown
ORAL
Leukemia, Myeloid, Acute
Smoothened homolog antagonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
ORAL
Brain Neoplasms; Carcinoma; Colonic Neoplasms; Gastrointestinal Stromal Tumors; Leukemia; Liver Diseases; Lung Neoplasms; Rectal Neoplasms; Arthritis, Rheumatoid; Breast Neoplasms; Carcinoma, Non-Small-Cell Lung; Cardiomegaly; Colorectal Neoplasms; Leukemia, Hairy Cell; Multiple Myeloma; Pancreatic Neoplasms; Thyroid Neoplasms; Fallopian Tube Neoplasms; Ovarian Neoplasms; Peritoneal Neoplasms; Melanoma; Neoplasms
Dual specificity mitogen-activated protein kinase kinase 1 inhibitor
Small molecule
Approved
Unknown
ORAL
Infections; Elephantiasis, Filarial; Strongyloidiasis; Helminthiasis; Onchocerciasis
Unknown
Small molecule
Approved
Unknown
Unknown
Hematologic Neoplasms; Lymphoma; Ovarian Neoplasms; Pneumonia; Anemia, Hemolytic, Autoimmune; Glomerulonephritis, IGA; Lymphoma, Large B-Cell, Diffuse; Primary Myelofibrosis; Severe Acute Respiratory Syndrome; Arthritis, Rheumatoid; Purpura, Thrombocytopenic, Idiopathic; Hemorrhage
Tyrosine-protein kinase SYK inhibitor
Small molecule
Approved
Unknown
ORAL
Lymphoma, Large B-Cell, Diffuse; Carcinoma, Squamous Cell; Liver Diseases; Melanoma; Mycosis Fungoides; Sezary Syndrome; Arthritis, Rheumatoid; Asthma; Hematologic Neoplasms; Leukemia; Lymphoma, Non-Hodgkin; Lymphoma, T-Cell, Peripheral; Severe Acute Respiratory Syndrome; Leukemia, Lymphocytic, Chronic, B-Cell; Lymphoma; Lymphoma, Follicular; Neoplasms
PI3-kinase p110-delta subunit inhibitor
Small molecule
Approved
Unknown
ORAL
Botulism; Multiple Sclerosis; Lambert-Eaton Myasthenic Syndrome
Voltage-gated potassium channel blocker
Small molecule
Approved
Unknown
Unknown
Renal Insufficiency; Renal Insufficiency, Chronic; Pyelonephritis; Bacterial Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Acne Vulgaris; Bacterial Infections
Unknown
Small molecule
Approved
Unknown
ORAL
Liver Diseases; Myelodysplastic Syndromes; Chondrosarcoma; Glioma; Cholangiocarcinoma; Leukemia, Myeloid, Acute; Neoplasms
Isocitrate dehydrogenase [NADP] cytoplasmic inhibitor
Small molecule
Approved
Unknown
ORAL
Hyperoxaluria, Primary; Epilepsies, Myoclonic; Epilepsy; Seizures
Unknown
Small molecule
Approved
Unknown
ORAL
Carcinoma, Non-Small-Cell Lung; Colorectal Neoplasms; Leukemia, Hairy Cell; Multiple Myeloma; Pancreatic Neoplasms; Thyroid Neoplasms; Melanoma; Neoplasms
Serine/threonine-protein kinase B-raf inhibitor
Small molecule
Approved
Unknown
Unknown
Anemia, Aplastic; Blood Platelet Disorders; Liver Diseases; Purpura, Thrombocytopenic, Idiopathic; Thrombocytopenia; Hemorrhage
Thrombopoietin receptor agonist
Small molecule
Approved
Unknown
Unknown
Polycystic Ovary Syndrome; Endometriosis; Leiomyoma
Gonadotropin-releasing hormone receptor antagonist
Small molecule
Approved
Unknown
Unknown
Glioma; Neoplasms
Neurotrophic tyrosine kinase receptor inhibitor
Small molecule
Approved
Unknown
Unknown
Acute Pain; Substance-Related Disorders
Opioid receptors; mu/kappa/delta agonist
Small molecule
Approved
Unknown
ORAL
Disorders of Excessive Somnolence; Narcolepsy; Sleep Apnea, Obstructive; Attention Deficit Disorder with Hyperactivity
Unknown
Small molecule
Approved
Unknown
Unknown
Pneumonia; Bacterial Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Disorders of Excessive Somnolence; Narcolepsy; Sleep Apnea, Obstructive; Sleep Apnea Syndromes
Unknown
Small molecule
Approved
Unknown
ORAL
Liver Diseases; Substance-Related Disorders; Parkinson Disease
Adenosine A2a receptor antagonist
Small molecule
Approved
Unknown
INTRAVENOUS
Severe Acute Respiratory Syndrome
Supplement
Small molecule
Approved
Unknown
Unknown
Schizophrenia
Unknown
Small molecule
Approved
Unknown
Unknown
Migraine Disorders
Calcitonin gene-related peptide type 1 receptor antagonist