Display Options:
Total: 6532
Small molecule
Approved
Unknown
Unknown
Lymphoma, Follicular; Sarcoma
Histone-lysine N-methyltransferase EZH2 inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
GABA-B receptor agonist
Small molecule
Approved
Unknown
Unknown
Neoplasms; Leukemia, Myeloid, Acute; Myelodysplastic Syndromes
Cytidine deaminase inhibitor
Small molecule
Approved
Unknown
Unknown
Dwarfism, Pituitary
Growth hormone receptor agonist
Small molecule
Approved
Unknown
Unknown
Alzheimer Disease; Chronic Traumatic Encephalopathy; Cognitive Dysfunction
Diagnostic agent
Small molecule
Approved
Unknown
Unknown
Lice Infestations
Copper sequestering agent
Small molecule
Approved
Unknown
Unknown
Carcinoma, Non-Small-Cell Lung
Hepatocyte growth factor receptor inhibitor
Small molecule
Approved
Unknown
Unknown
Liver Diseases; Severe Acute Respiratory Syndrome; Colitis, Ulcerative; Crohn Disease; Multiple Sclerosis; Immune System Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
HIV Infections; Virus Diseases
Envelope polyprotein GP160 inhibitor
Small molecule
Approved
Unknown
Unknown
Anorexia Nervosa; Depressive Disorder, Major; Obsessive-Compulsive Disorder; Renal Insufficiency, Chronic; Bipolar Disorder; Nausea; Anxiety; Dementia; Depressive Disorder; Schizophrenia; Postoperative Nausea and Vomiting; Psychotic Disorders
Dopamine receptors; D2 & D3 antagonist
Small molecule
Approved
Unknown
Unknown
Alopecia; Acne Vulgaris
Androgen Receptor antagonist
Small molecule
Approved
Unknown
Unknown
Parkinson Disease
Catechol O-methyltransferase inhibitor
Small molecule
Approved
Unknown
Unknown
Liver Diseases; Epilepsies, Partial; Epilepsy; Seizures
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
Unknown
Unknown
Astrocytoma; Central Nervous System Neoplasms; Colorectal Neoplasms; Gliosarcoma; Head and Neck Neoplasms; Lymphoma; Breast Neoplasms; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Liver Neoplasms; Ovarian Neoplasms; Urethral Neoplasms; Urinary Bladder Neoplasms; Carcinoma, Non-Small-Cell Lung; Hepatitis D; Leukemia, Myelomonocytic, Chronic; Myelodysplastic Syndromes; Neoplasm Metastasis; Progeria
Protein farnesyltransferase inhibitor
Small molecule
Approved
Unknown
Unknown
Constipation
Osmotic agent
Small molecule
Approved
Unknown
Unknown
Kidney Diseases; Liver Diseases; Cushing Syndrome; Essential Hypertension; Hyperaldosteronism; Hypertension; Pituitary ACTH Hypersecretion; Adrenal Gland Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Hypertension; Irritable Bowel Syndrome; Urinary Bladder, Overactive; Urinary Incontinence; Urinary Incontinence, Urge
Beta-3 adrenergic receptor agonist
Small molecule
Approved
Unknown
Unknown
Migraine Disorders
Calcitonin gene-related peptide type 1 receptor antagonist
Small molecule
Approved
Unknown
Unknown
Glycogen Storage Disease Type I; Migraine Disorders; Amyotrophic Lateral Sclerosis; Ataxia Telangiectasia; Glycogen Storage Disease; Glycogen Storage Disease Type VII; Hemiplegia; Huntington Disease; Rett Syndrome
Supplement
Small molecule
Approved
Unknown
Unknown
Kidney Diseases; Liver Diseases; Sleep Apnea, Obstructive; Sleep Disorders, Circadian Rhythm; Sleep Initiation and Maintenance Disorders
Orexin receptor 1 antagonist
Small molecule
Approved
Unknown
Unknown
Astrocytoma; Biliary Tract Neoplasms; Cholangiocarcinoma; Colonic Neoplasms; Kidney Neoplasms; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Optic Nerve Glioma; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Rectal Neoplasms; Sarcoma, Kaposi; Triple Negative Breast Neoplasms; Urinary Bladder Neoplasms; Adenocarcinoma; Adenocarcinoma, Follicular; Breast Neoplasms; Carcinoma, Hepatocellular; Carcinoma, Squamous Cell; Colorectal Neoplasms; Gallbladder Neoplasms; Liver Neoplasms; Lung Neoplasms; Lymphoma, Large B-Cell, Diffuse; Melanoma; Multiple Myeloma; Neurofibroma, Plexiform; Neurofibromatosis 1; Pancreatic Neoplasms; Sarcoma; Stomach Neoplasms; Carcinoma, Non-Small-Cell Lung; Thyroid Neoplasms; Neoplasms
Dual specificity mitogen-activated protein kinase kinase 1 inhibitor
Small molecule
Unknown
Unknown
Unknown
Carcinoma, Non-Small-Cell Lung
Unknown
Small molecule
Unknown
Unknown
Unknown
Cholangiocarcinoma
Fibroblast growth factor receptor inhibitor
Small molecule
Approved
Unknown
Unknown
Breast Neoplasms; Carcinoma, Non-Small-Cell Lung; Cholangiocarcinoma; Carcinoma, Hepatocellular; Colorectal Neoplasms; Fallopian Tube Neoplasms; Glioblastoma; Ovarian Neoplasms; Prostatic Neoplasms, Castration-Resistant; Sarcoma; Carcinoma, Renal Cell; Neoplasms
Vascular endothelial growth factor receptor inhibitor
Small molecule
Approved
Unknown
Unknown
Diabetic Nephropathies; Heart Failure; Renal Insufficiency, Chronic
Mineralocorticoid receptor antagonist
Small molecule
Unknown
Unknown
Unknown
Bipolar Disorder; Schizophrenia
Delta opioid receptor partial agonist
Small molecule
Approved
Unknown
Unknown
Alagille Syndrome; Biliary Atresia; Liver Diseases
Ileal bile acid transporter inhibitor
Small molecule
Unknown
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Cholestasis; Liver Cirrhosis, Biliary; Non-alcoholic Fatty Liver Disease; Alagille Syndrome; Biliary Atresia; Cholestasis, Intrahepatic; Pruritus
Ileal bile acid transporter inhibitor
Small molecule
Unknown
Unknown
Unknown
Liver Diseases; Graft vs Host Disease; Idiopathic Pulmonary Fibrosis; Psoriasis; Scleroderma, Diffuse
Rho-associated protein kinase 2 inhibitor
Small molecule
Unknown
Unknown
Unknown
Attention Deficit Disorder with Hyperactivity
Dopamine transporter inhibitor
Small molecule
Approved
Unknown
Unknown
Breast Neoplasms; Gastrointestinal Stromal Tumors; Uterine Cervical Neoplasms; Achondroplasia; Glioblastoma; Melanoma; Neoplasms; Osteomalacia; Papillomavirus Infections; Squamous Cell Carcinoma of Head and Neck; Cholangiocarcinoma; Urinary Bladder Neoplasms
Fibroblast growth factor receptor inhibitor
Small molecule
Approved
Unknown
Unknown
Hodgkin Disease; Leukemia, Lymphocytic, Chronic, B-Cell; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Waldenstrom Macroglobulinemia
Unknown
Small molecule
Unknown
Unknown
Unknown
Candidiasis, Vulvovaginal
1,3-beta-glucan synthase inhibitor
Small molecule
Unknown
Unknown
Unknown
Small Cell Lung Carcinoma
Cyclin-dependent kinase 4 inhibitor