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Total: 1496
Small molecule
Approved
EYE; OTHER
OPHTHALMIC
Carcinoma, Non-Small-Cell Lung; Stomach Neoplasms; Breast Neoplasms; Cholangiocarcinoma; Colonic Neoplasms; Rectal Neoplasms; Esophageal Neoplasms; Colorectal Neoplasms; Eye Infections; Herpes Simplex; Keratoconjunctivitis; Neoplasms
DNA inhibitor
Protein
Approved
OTHER
INJECTION
Diabetes Mellitus
Insulin receptor agonist
Small molecule
Approved
OTHER
ORAL
Osteomyelitis; Bacterial Infections
Bacterial DNA gyrase inhibitor
Small molecule
Approved
OTHER
ORAL
Acute Kidney Injury; Severe Acute Respiratory Syndrome; Sleep Apnea, Obstructive; Vitamin D Deficiency; Myocardial Infarction; Hyperparathyroidism, Secondary; Parathyroid Diseases; Renal Insufficiency, Chronic
Vitamin D receptor agonist
Protein
Approved
OTHER
INJECTION
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Alzheimer Disease; Anemia; Diabetes Mellitus, Type 2; HIV Infections; Hypertriglyceridemia; Multiple Sclerosis; Neoplasms; Alcoholism; Myocardial Ischemia; Parkinson Disease; Smoking Cessation; Tobacco Use Disorder; Abdominal Pain; Cardiovascular Diseases; Coronary Disease
Peroxisome proliferator-activated receptor alpha agonist
Small molecule
Approved
OTHER
INHALATION; NASAL
Rhinitis, Allergic, Perennial; Asthma; Lung Diseases, Obstructive; Nasal Obstruction; Rhinitis
Glucocorticoid receptor agonist
Small molecule
Approved
OTHER
INJECTION
Breast Neoplasms
Unknown
Small molecule
Approved
OTHER; RESPIRATORY
INHALATION
Ciliary Motility Disorders; Depressive Disorder, Major; Diabetes Mellitus; Glycogen Storage Disease Type II; Idiopathic Pulmonary Fibrosis; Lymphangioleiomyomatosis; Myasthenic Syndromes, Congenital; Tachypnea; Bronchiolitis; Cough; Familial Primary Pulmonary Hypertension; Hypersensitivity; Memory Disorders; Pulmonary Edema; Respiratory Insufficiency; Spinal Cord Injuries; Status Asthmaticus; Abdominal Pain; Dysautonomia, Familial; Heart Failure; Hypertension, Pulmonary; Lung Diseases; Organophosphate Poisoning; Rhinitis, Allergic, Seasonal; Asthma, Exercise-Induced; Bronchial Spasm; Lung Diseases, Obstructive; Pulmonary Disease, Chronic Obstructive
Beta-2 adrenergic receptor agonist
Small molecule
Approved
CARDIOVASCULAR; GASTROINTESTINAL; OTHER
INJECTION; INTRA-ANAL; SUBLINGUAL; TRANSDERMAL
Colorectal Neoplasms; Hypertension, Pulmonary; Hypotension; Infections; Inflammation; Peripheral Arterial Disease; Phlebitis; Rectal Neoplasms; Carcinoma, Non-Small-Cell Lung; Diabetic Neuropathies; Erectile Dysfunction; Hot Flashes; Lung Neoplasms; Pulmonary Edema; Shock; Tendinopathy; Anus Diseases; Arthritis, Rheumatoid; Bone Diseases, Metabolic; Heart Diseases; Muscle Cramp; Myocardial Ischemia; Osteoporosis; Raynaud Disease; Reperfusion Injury; Scleroderma, Localized; Stroke; Wounds and Injuries; Angina Pectoris; Cardiovascular Diseases; Coronary Artery Disease; Heart Failure; Hemorrhoids; Hypertension; Myocardial Infarction; Pain
Soluble guanylate cyclase activator
Small molecule
Approved
OTHER
ORAL
Lung Diseases, Obstructive
Adenosine receptor antagonist
Small molecule
Approved
OTHER
INJECTION; TOPICAL
Kidney Failure, Chronic; Leukemia; Myopia; Neoplasm Metastasis; Appendiceal Neoplasms; Biliary Tract Neoplasms; Carcinoma, Squamous Cell; Cholangiocarcinoma; Cholangitis, Sclerosing; Corneal Opacity; Esophageal Stenosis; Glaucoma, Neovascular; Glaucoma, Open-Angle; Keratoconus; Liver Neoplasms; Pterygium; Sarcoma; Urethral Stricture; Anus Neoplasms; Breast Neoplasms; Carcinoma; Carcinoma, Hepatocellular; Carcinoma in Situ; Carcinoma, Non-Small-Cell Lung; Carcinoma, Transitional Cell; Colorectal Neoplasms; Head and Neck Neoplasms; Lung Neoplasms; Mesothelioma; Nasopharyngeal Carcinoma; Pancreatic Neoplasms; Stomach Neoplasms; Urinary Bladder Neoplasms; Uterine Cervical Neoplasms; Adenocarcinoma; Glaucoma; Neoplasms
DNA inhibitor
Small molecule
Approved
OTHER
INJECTION; ORAL
Orthostatic Intolerance; Osteoporosis; Stress Disorders, Post-Traumatic; Atrial Fibrillation; Cerebrovascular Disorders; Essential Hypertension; Heart Diseases; Heart Failure; Hemangioma; Hypertrophy, Left Ventricular; Marfan Syndrome; Mitral Valve Stenosis; Myocardial Ischemia; Vascular Diseases; Angina Pectoris; Cardiovascular Diseases; Coronary Artery Disease; Diabetes Mellitus; Hypertension; Myocardial Infarction; Stroke
Beta-1 adrenergic receptor antagonist
Small molecule
Approved
OTHER
ORAL
Hypersensitivity; Multiple Sclerosis; Sunburn; Angioedema; Conjunctivitis, Allergic; Rhinitis, Allergic, Perennial; Rhinitis, Allergic, Seasonal; Rhinitis, Vasomotor; Urticaria
Histamine H1 receptor antagonist
Small molecule
Approved
CARDIOVASCULAR; DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Diabetes Mellitus, Type 2; Glioblastoma; Hypertension, Pulmonary; Neoplasms; Primary Myelofibrosis; Heart Diseases; Pneumonia; Diabetes Mellitus, Type 1; Essential Hypertension; Severe Acute Respiratory Syndrome; Cardiovascular Diseases; Collagen Diseases; Diabetic Nephropathies; Diabetic Retinopathy; Heart Failure; Hypertension; Myocardial Infarction; Renal Insufficiency; Ventricular Dysfunction, Left
Angiotensin-converting enzyme inhibitor
Small molecule
Approved
OTHER
ORAL
Anxiety
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
OTHER
ORAL
Anxiety; Dementia; Depressive Disorder; Pulmonary Disease, Chronic Obstructive; Schizophrenia; Sleep Initiation and Maintenance Disorders
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
IMMUNE SYSTEM; OTHER
ORAL; TOPICAL
Alzheimer Disease; Asthma; Diabetes Mellitus, Type 2; Erectile Dysfunction; Essential Hypertension; Gastroparesis; Glioblastoma; Hematologic Neoplasms; Hepatitis C; Immune System Diseases; Insulin Resistance; Leukemia, Lymphocytic, Chronic, B-Cell; Lymphoma; Lymphoma, Non-Hodgkin; Melanoma; Multiple Sclerosis; Nausea; Neuroblastoma; Onychomycosis; Osteoporosis; Premature Birth; Pulmonary Disease, Chronic Obstructive; Tinea Versicolor; Breast Neoplasms; Burns; Hypogonadism; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Neoplasms; Prostatic Neoplasms; Psoriasis; Acne Vulgaris; Candidiasis, Vulvovaginal; Dermatitis; Prostatic Neoplasms, Castration-Resistant; Respiratory Distress Syndrome; Vaginosis, Bacterial; Adrenal Gland Diseases; Blastomycosis; Cushing Syndrome; Dermatitis, Seborrheic; Tinea; Tinea Pedis
Cytochrome P450 51 inhibitor
Small molecule
Approved
CARDIOVASCULAR; OTHER; UROLOGY AND KIDNEY
INJECTION; URETHRAL
Acute Kidney Injury; Arteriosclerosis Obliterans; Optic Neuropathy, Ischemic; Peripheral Arterial Disease; Peripheral Vascular Diseases; Respiratory Distress Syndrome; Severe Acute Respiratory Syndrome; Sexual Dysfunction, Physiological; Heart Failure; Macular Degeneration; Prostatic Neoplasms, Castration-Resistant; Cardiovascular Diseases; Ductus Arteriosus, Patent; Erectile Dysfunction
Prostanoid EP1 receptor agonist
Small molecule
Approved
OTHER
ORAL
Adrenal Hyperplasia, Congenital; Substance-Related Disorders; Anus Diseases; Epilepsies, Partial; Epilepsy; Fissure in Ano; Proteinuria; Renal Insufficiency, Chronic; Diabetic Nephropathies; Hypertension, Pulmonary; Kidney Calculi; Myocardial Ischemia; Placenta Previa; Pre-Eclampsia; Premature Birth; Raynaud Disease; Cardiovascular Diseases; Coronary Vasospasm; Hypertension
Voltage-gated L-type calcium channel blocker
Small molecule
Approved
OTHER
ORAL
Asthma; Diabetes Mellitus, Type 1; Migraine Disorders; Phobia, Social; Substance-Related Disorders; Dental Anxiety; Epilepsy; Stress Disorders, Post-Traumatic; Dementia; Depressive Disorder; Schizophrenia; Seizures; Anxiety; Anxiety Disorders; Panic Disorder
GABA-A receptor; anion channel positive allosteric modulator
Unknown
Approved
OTHER
ORAL
Eosinophilic Esophagitis; Hemorrhage; Esophagitis; Duodenal Ulcer; Gastroesophageal Reflux; Peptic Ulcer
Glycoproteins cross-linking agent
Small molecule
Approved
OTHER
TOPICAL
Unknown
Cell membrane inhibitor
Small molecule
Approved
OTHER
ORAL
Arthritis, Rheumatoid; Colonic Neoplasms; Leukemia, Myeloid, Acute; Prostatic Neoplasms, Castration-Resistant; Adenomatous Polyposis Coli; Colorectal Neoplasms; Prostatic Neoplasms; Diabetic Nephropathies; Severe Acute Respiratory Syndrome; Helminthiasis
DNA inhibitor
Small molecule
Approved
OTHER
ORAL
Osteomyelitis
Bacterial 70S ribosome inhibitor
Small molecule
Approved
OTHER
ORAL
Unknown
Glucocorticoid receptor agonist
Small molecule
Approved
OTHER
TOPICAL
Stomatitis
Bacterial 70S ribosome inhibitor
Small molecule
Approved
OTHER
ORAL
Epilepsy
Voltage-gated T-type calcium channel blocker
Small molecule
Approved
OTHER
TOPICAL
Unknown
Glucocorticoid receptor agonist
Protein
Approved
OTHER
INJECTION
Atherosclerosis; Coronary Disease; Diabetes Mellitus; Diabetes Mellitus, Type 1; Diabetes Mellitus, Type 2; Hypercholesterolemia; Hyperglycemia; Hypertension
Insulin receptor agonist
Small molecule
Approved
OTHER
ORAL
Bacterial Infections
Penicillin-binding protein inhibitor
Small molecule
Approved
OTHER
INJECTION
Anxiety; Dementia; Depressive Disorder; Schizophrenia; Psychotic Disorders
D2-like dopamine receptor antagonist
Small molecule
Approved
OTHER
ORAL
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Anxiety
GABA-A receptor; anion channel positive allosteric modulator
Protein
Approved
OTHER
INJECTION
Unknown
Unknown