Display Options:
Total: 6532
Small molecule
Approved
Unknown
Unknown
Infections; Bacteremia; Gram-Positive Bacterial Infections; Osteomyelitis; Bacterial Infections
Unknown
Small molecule
Approved
OTHER
ORAL
Pain
Mu opioid receptor agonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Astrocytoma; Brain Neoplasms; Carcinoma, Hepatocellular; Colorectal Neoplasms; Digestive System Neoplasms; Glioblastoma; Gliosarcoma; Neoplasms; Oligodendroglioma; Intracranial Hypertension; Meningitis, Cryptococcal; Candidiasis; Infections; Meningitis
Thymidylate synthase inhibitor
Small molecule
Approved
OTHER
OPHTHALMIC; TOPICAL
Corneal Opacity; Dry Eye Syndromes; Acne Vulgaris; Eye Diseases; Hemorrhoids; Inflammation
Glucocorticoid receptor agonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
CARDIOVASCULAR; DIABETES DRUGS & ENDOCRINOLOGY; OTHER
BUCCAL; IMPLANTATION; INJECTION; NASAL; TRANSDERMAL
Aging; Cerebral Arterial Diseases; Dyspareunia; Insulin Resistance; Kallmann Syndrome; Pain; Penile Induration; Polycystic Ovary Syndrome; Acquired Immunodeficiency Syndrome; Anorexia Nervosa; Carcinoma, Intraductal, Noninfiltrating; Dwarfism; Heart Failure; Hereditary Breast and Ovarian Cancer Syndrome; Multiple Sclerosis; Muscle Weakness; Obesity; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Sarcopenia; Spinal Cord Injuries; Testicular Neoplasms; Coronary Disease; Disorders of Sex Development; Erectile Dysfunction; Hip Fractures; Infertility; Kidney Failure, Chronic; Menopause; Metabolic Syndrome; Hypogonadism; Klinefelter Syndrome; Neoplasms; Orchitis; Sexual Dysfunctions, Psychological
Androgen Receptor agonist
Small molecule
Approved
EMERGENCY MEDICINE; NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
INJECTION
Aortic Coarctation; Brain Neoplasms; Hernia, Ventral; HIV Infections; Lung Diseases; Neuralgia; Obesity, Morbid; Prostatic Neoplasms, Castration-Resistant; Sarcoma; Sinusitis; Stress Disorders, Post-Traumatic; Subarachnoid Hemorrhage; Vasospasm, Intracranial; Abdominal Pain; Appendicitis; Atrial Fibrillation; Blepharoptosis; Blood Coagulation Disorders; Cleft Palate; Complex Regional Pain Syndromes; Dupuytren Contracture; Fasciitis, Plantar; Femoral Neck Fractures; Headache; Hemorrhage; Hernia, Umbilical; Hip Fractures; Hypospadias; Hypotension; Lacrimal Apparatus Diseases; Low Back Pain; Mucositis; Musculoskeletal Diseases; Osteoarthritis, Hip; Pregnancy; Pulpitis; Rib Fractures; Shoulder Pain; Spinal Stenosis; Analgesia; Ankle Fractures; Breast Neoplasms; Breech Presentation; Carcinoma, Non-Small-Cell Lung; Chronic Pain; Cough; Fractures, Bone; Genital Neoplasms, Female; Hallux Valgus; Hemorrhoids; Hernia, Inguinal; Ileus; Liver Diseases; Lung Neoplasms; Migraine Disorders; Neoplasms; Osteoarthritis; Osteoarthritis, Knee; Pancreatic Neoplasms; Pancreatitis, Chronic; Peritoneal Neoplasms; Postoperative Nausea and Vomiting; Radiculopathy; Radius Fractures; Rotator Cuff Injuries; Toothache; Urethral Stricture; Wounds and Injuries; Acute Pain; Hernia; Pain
Sodium channel protein type IV alpha subunit blocker
Small molecule
Approved
OTHER
INJECTION
Psoriasis
Dopamine D2 receptor antagonist
Small molecule
Approved
Unknown
Unknown
Aortic Valve Stenosis; Neoplasms; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant
Unknown
Small molecule
Approved
OTHER
ORAL
Anxiety; Anxiety Disorders; Seizures
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
OTHER
INHALATION
Unknown
GABA-A receptor; anion channel positive modulator
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Bacterial Infections
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Postoperative Nausea and Vomiting; Vertigo; Hypersensitivity
Histamine H1 receptor antagonist
Small molecule
Approved
OTHER
ORAL
Unknown
Androgen Receptor agonist
Small molecule
Approved
DERMATOLOGY; OTHER
TOPICAL
Dermatitis, Atopic; Eye Diseases; Skin Diseases
Glucocorticoid receptor agonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
INTRAOCULAR
Presbyopia; Cataract; Glaucoma; Miosis
Muscarinic acetylcholine receptor M3 agonist
Small molecule
Approved
OTHER
INJECTION
Unknown
Muscle-type nicotinic acetylcholine receptor antagonist
Small molecule
Approved
OTHER
ORAL
Anemia; Astrocytoma; Brain Neoplasms; Glioblastoma; Granulomatosis with Polyangiitis; Kidney Diseases; Leukemia; Leukemia, Biphenotypic, Acute; Macular Degeneration; Neoplasms; Osteomyelitis; Pulmonary Disease, Chronic Obstructive; Cystic Fibrosis; Dermatitis; Diabetes Mellitus, Type 1; Eczema; Epidermolysis Bullosa; Lymphoma, AIDS-Related; Skin Diseases; Abscess; HIV Infections; Idiopathic Pulmonary Fibrosis; Malaria; Measles; Pneumonia; Pyelonephritis; Sepsis; Staphylococcal Infections; Toxoplasmosis, Ocular; Tuberculosis; Bacterial Infections; Infections; Otitis Media; Pneumonia, Pneumocystis; Urinary Tract Infections
Bacterial dihydrofolate reductase inhibitor
Small molecule
Approved
OTHER
ORAL
Heart Diseases; Substance-Related Disorders; Brain Injuries; Status Epilepticus; Sleep Initiation and Maintenance Disorders
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Renal Insufficiency, Chronic; Cardiovascular Diseases; Heart Failure; Hypertension; Toxemia
Thiazide-sensitive sodium-chloride cotransporter inhibitor
Small molecule
Approved
Unknown
Unknown
Infections; Osteomyelitis; Burns
Bacterial dihydropteroate synthase inhibitor
Small molecule
Approved
OTHER
INJECTION; ORAL; VAGINAL
Prostatic Neoplasms, Castration-Resistant; Neoplasms
Estrogen receptor alpha agonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Hypersensitivity; Pruritus
Unknown
Small molecule
Approved
Unknown
Unknown
Keratitis, Herpetic
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Substance-Related Disorders; Asthma
Beta-2 adrenergic receptor agonist
Small molecule
Approved
OTHER
ORAL
Attention Deficit Disorder with Hyperactivity; Cocaine-Related Disorders; Narcolepsy; Obesity
Monoamine transporter inhibitor
Small molecule
Approved
OTHER
ORAL
Astrocytoma; Brain Neoplasms; Glioblastoma; Granulomatosis with Polyangiitis; Kidney Diseases; Leukemia; Leukemia, Biphenotypic, Acute; Macular Degeneration; Neoplasms; Osteomyelitis; Pulmonary Disease, Chronic Obstructive; Cystic Fibrosis; Dermatitis; Diabetes Mellitus, Type 1; Eczema; Lymphoma, AIDS-Related; Skin Diseases; Abscess; HIV Infections; Idiopathic Pulmonary Fibrosis; Malaria; Measles; Pneumonia; Pyelonephritis; Sepsis; Staphylococcal Infections; Toxoplasmosis, Ocular; Tuberculosis; Bacterial Infections; Infections; Pneumonia, Pneumocystis; Urinary Tract Infections
Bacterial dihydropteroate synthase inhibitor
Small molecule
Approved
Unknown
Unknown
Adenoma; Carcinoma, Renal Cell; Colorectal Neoplasms; Hashimoto Disease; Lung Neoplasms; Lymphoma, Follicular; Prostatic Neoplasms, Castration-Resistant
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Depressive Disorder; Diabetes Mellitus, Type 2; Obesity; Adenoma, Islet Cell; Hyperinsulinism; Hypertension; Hypoglycemia
Potassium channel, inwardly rectifying, subfamily J, member 11 opener