Display Options:
Total: 6532
Small molecule
Approved
Unknown
Unknown
Intestinal Obstruction; Pain; Breast Neoplasms; Clostridium Infections; Eczema; Neoplasms; Paget Disease, Extramammary; Carcinoma, Non-Small-Cell Lung; Diarrhea; Fecal Incontinence
Unknown
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER; PREGNANCY AND GYNECOLOGY
INJECTION; INTRAUTERINE; ORAL; VAGINAL
Amphetamine-Related Disorders; Gliosarcoma; Anorexia Nervosa; Bulimia Nervosa; Cocaine-Related Disorders; Depression, Postpartum; Depressive Disorder; Endometrial Neoplasms; HIV Infections; Marijuana Abuse; Orthostatic Intolerance; Placenta Previa; Polycystic Ovary Syndrome; Pre-Eclampsia; Severe Acute Respiratory Syndrome; Tobacco Use Disorder; Uterine Cervical Dysplasia; Vulvar Lichen Sclerosus; Alzheimer Disease; Angina, Unstable; Bone Diseases; Bone Diseases, Metabolic; Brain Injuries; Breast Neoplasms; Cardiovascular Diseases; Coronary Disease; Diabetes Mellitus; Epilepsy; Hypercholesterolemia; Hypertension; Infertility; Infertility, Female; Leiomyoma; Memory Disorders; Menopause; Myocardial Ischemia; Osteoporosis; Ovarian Hyperstimulation Syndrome; Ovarian Neoplasms; Pregnancy; Premature Birth; Thrombosis; Amenorrhea; Endometrial Hyperplasia; Uterine Hemorrhage
Progesterone receptor agonist
Small molecule
Approved
OTHER
INJECTION; OPHTHALMIC
Herpes Simplex; Eye Infections; Virus Diseases
Human herpesvirus 1 DNA polymerase inhibitor
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Sepsis; Infections; Bacterial Infections
Unknown
Small molecule
Approved
OTHER
ORAL
Bone Neoplasms; Breast Neoplasms; Glioma; Kidney Neoplasms; Lung Neoplasms; Lymphoma; Lymphoma, AIDS-Related; Lymphoma, Non-Hodgkin; Melanoma; Neoplasm Metastasis; Pancreatic Neoplasms; Sarcoma; Spinal Cord Neoplasms; Uveal Melanoma; Astrocytoma; Central Nervous System Neoplasms; Glioblastoma; Gliosarcoma; Leukemia, Myeloid, Acute; Medulloblastoma; Multiple Myeloma; Neoplasms, Plasma Cell; Paraganglioma; Brain Neoplasms; Hodgkin Disease; Neoplasms
DNA inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Endocarditis
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Breast Neoplasms; Neoplasms; Brain Neoplasms; Hyperemia
Unknown
Small molecule
Approved
Unknown
Unknown
Brain Neoplasms
Unknown
Small molecule
Approved
Unknown
Unknown
Arthralgia; Myalgia; Rheumatic Diseases
Unknown
Small molecule
Approved
OTHER
ORAL
Arthritis, Rheumatoid; Osteoarthritis
Cyclooxygenase inhibitor
Small molecule
Approved
OTHER
ORAL; VAGINAL
Atrophy; Hypogonadism; Menopause; Osteoporosis; Primary Ovarian Insufficiency
Estrogen receptor alpha agonist
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; MUSCULOSKELETAL; OTHER
ORAL
Atrophy; Breast Neoplasms; Hypogonadism; Menopause; Primary Ovarian Insufficiency
Estrogen receptor agonist
Small molecule
Approved
OTHER
TOPICAL
Unknown
Glucocorticoid receptor agonist
Small molecule
Approved
OTHER
ORAL
Diabetic Nephropathies; Peripheral Arterial Disease; Hyperlipidemias; Cardiovascular Diseases
ATP-binding cassette sub-family A member 1 inhibitor
Small molecule
Approved
Unknown
Unknown
Brain Neoplasms; Hepatitis C, Chronic; Neoplasms, Cystic, Mucinous, and Serous; Osteosarcoma; Adenoma; Amyotrophic Lateral Sclerosis; Bipolar Disorder; Endometrial Neoplasms; Glioblastoma; Gynecomastia; HIV Infections; Infertility, Male; Lymphoma, Large B-Cell, Diffuse; Neuroendocrine Tumors; Pain; Retroperitoneal Fibrosis; Telangiectasia, Hereditary Hemorrhagic; Urinary Bladder Neoplasms; Uterine Cervical Neoplasms; Breast Neoplasms; Breast Neoplasms, Male; Carcinoma, Intraductal, Noninfiltrating; Cognitive Dysfunction; Coronary Disease; Fallopian Tube Neoplasms; Hot Flashes; Hyperplasia; Hypertension; Infertility; Menopause; Muscular Dystrophy, Duchenne; Myocardial Ischemia; Neoplasm Metastasis; Ovarian Neoplasms; Peritoneal Neoplasms; Prostatic Neoplasms, Castration-Resistant; Neoplasms
Unknown
Small molecule
Approved
Unknown
Unknown
Pseudoxanthoma Elasticum; Bone Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
ENDOCERVICAL; VAGINAL
Abortion, Incomplete; Fetal Growth Retardation; Myoma; Pain; Pregnancy
Prostaglandin E2 receptor agonist
Small molecule
Approved
GASTROINTESTINAL; OTHER
ORAL
Amyotrophic Lateral Sclerosis; Anxiety Disorders; Infections; Pulmonary Disease, Chronic Obstructive; Breast Carcinoma In Situ; Breast Neoplasms; Endometrial Neoplasms; Protoporphyria, Erythropoietic; Dermatitis, Atopic; Gastrointestinal Hemorrhage; Hemorrhage; Ulcer; Duodenal Ulcer; Gastroesophageal Reflux; Heartburn; Peptic Ulcer
Histamine H2 receptor antagonist
Small molecule
Approved
OTHER
INJECTION; ORAL
Alzheimer Disease; Epidermolysis Bullosa; Obsessive-Compulsive Disorder; Substance-Related Disorders; Voice Disorders; Alcoholism; Amphetamine-Related Disorders; Cocaine-Related Disorders; Delirium; Down Syndrome; Epilepsy, Reflex; Pain; Seizures; Substance Withdrawal Syndrome; Dementia; Depressive Disorder; Epilepsia Partialis Continua; Epilepsy; Psychomotor Agitation; Psychotic Disorders; Schizophrenia; Vertigo; Anxiety; Anxiety Disorders; Depression; Status Epilepticus
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
OTHER
ORAL
Unknown
Histamine H1 receptor antagonist
Small molecule
Approved
OTHER
TOPICAL
Psoriasis; Skin Diseases
Glucocorticoid receptor agonist
Small molecule
Approved
Unknown
Unknown
Depressive Disorder; Fibromyalgia; Liver Cirrhosis; Pain; Stress Disorders, Post-Traumatic
Unknown
Small molecule
Approved
Unknown
Unknown
Coronary Artery Disease; Myocardial Infarction
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Atrial Fibrillation; Heart Failure; Arrhythmias, Cardiac
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Multiple Sclerosis; Multiple Sclerosis, Relapsing-Remitting; Optic Neuritis; Schizophrenia; Urticaria; Angioedema; Dermatitis; Williams Syndrome; Hypersensitivity; Pruritus
Unknown
Small molecule
Approved
Unknown
Unknown
Hypersensitivity
Unknown
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER
INJECTION; INTRACRANIAL
Hereditary Breast and Ovarian Cancer Syndrome; Leukemia, Plasma Cell; Lymphoma, T-Cell, Cutaneous; Mycosis Fungoides; Neuroblastoma; Sezary Syndrome; Brain Neoplasms; Colorectal Neoplasms; Gliosarcoma; Graft vs Host Disease; Hematologic Diseases; Leukemia, Lymphocytic, Chronic, B-Cell; Lymphoma, T-Cell, Peripheral; Melanoma; Multiple Sclerosis, Relapsing-Remitting; Myasthenia Gravis; Neoplasms, Plasma Cell; Neuromyelitis Optica; Opsoclonus-Myoclonus Syndrome; Ovarian Neoplasms; Polyradiculoneuropathy, Chronic Inflammatory Demyelinating; Prostatic Neoplasms, Castration-Resistant; Sarcoma; Stiff-Person Syndrome; Breast Neoplasms; Central Nervous System Neoplasms; Leukemia; Lymphoma; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Oligodendroglioma; Paraganglioma; Astrocytoma; Ependymoma; Glioblastoma; Glioma; Hodgkin Disease; Lymphoma, Non-Hodgkin; Medulloblastoma; Multiple Myeloma; Neoplasms
DNA inhibitor
Small molecule
Approved
OTHER; RESPIRATORY
ORAL
Hypersensitivity; Multiple Sclerosis; Multiple Sclerosis, Chronic Progressive; Multiple Sclerosis, Relapsing-Remitting; Common Cold; Rhinitis, Allergic; Rhinitis, Allergic, Seasonal; Urticaria
Histamine H1 receptor antagonist
Small molecule
Approved
OTHER
INTRATHECAL; ORAL
Ataxia Telangiectasia; Autistic Disorder; Liver Cirrhosis, Alcoholic; Obesity; Carcinoma, Hepatocellular; Cocaine-Related Disorders; Fragile X Syndrome; Marijuana Abuse; Paget Disease, Extramammary; Substance-Related Disorders; Tobacco Use Disorder; Alcoholism; Charcot-Marie-Tooth Disease; Gastroesophageal Reflux; Pain; Substance Withdrawal Syndrome; Brain Injuries; Brain Injuries, Traumatic; Cerebral Palsy; Multiple Sclerosis; Muscle Rigidity; Muscle Spasticity; Spinal Cord Diseases; Spinal Cord Injuries
GABA-B receptor agonist