Display Options:
Total: 6532
Small molecule
Approved
Unknown
Unknown
Hypotension, Orthostatic; Orthostatic Intolerance; Prostatic Neoplasms, Castration-Resistant; Hyperemesis Gravidarum; Hypoglycemia; Intestinal Obstruction; Myelodysplastic Syndromes; Pain; Wounds and Injuries; Gastroenteritis; Gastrointestinal Hemorrhage; Gastroparesis; Gastroschisis; Headache; HIV Infections; Migraine Disorders; Nausea; Neoplasms; Postoperative Nausea and Vomiting; Sepsis; Vomiting; Digestive System Diseases
Unknown
Small molecule
Approved
OTHER
INJECTION
Obesity; Premenstrual Syndrome
Estrogen receptor alpha agonist
Small molecule
Approved
OTHER
ORAL
Psychotic Disorders; Hypertension; Pheochromocytoma
Tyrosine 3-hydroxylase inhibitor
Small molecule
Approved
Unknown
Unknown
Rheumatic Diseases
Cyclooxygenase inhibitor
Small molecule
Approved
OTHER
TOPICAL
Unknown
Glucocorticoid receptor agonist
Small molecule
Approved
OTHER
ORAL; TOPICAL
Carcinoma, Non-Small-Cell Lung; Lung Diseases; Pemphigoid, Benign Mucous Membrane; Pemphigus; Pulmonary Fibrosis; Rosacea; Sarcoidosis; Stroke; Fever; HIV Infections; Malaria; Malaria, Falciparum; Malaria, Vivax; Pneumonia, Pneumocystis; Severe Acute Respiratory Syndrome; Acne Vulgaris; Dermatitis Herpetiformis; Leprosy
Dihydropteroate synthase 1 inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Anxiety; Dementia; Schizophrenia; Depressive Disorder
Unknown
Small molecule
Approved
Unknown
Unknown
Hemorrhage; Postpartum Hemorrhage
Prostanoid FP receptor agonist
Small molecule
Approved
Unknown
Unknown
Cardiovascular Diseases
Unknown
Small molecule
Approved
OTHER
ORAL
Asthma; Smoking Cessation; Hemangioma; Angina Pectoris; Cardiovascular Diseases; Hypertension; Myocardial Infarction; Stroke
Beta-1 adrenergic receptor antagonist
Small molecule
Approved
DERMATOLOGY; OTHER
ORAL; TOPICAL
Acne Vulgaris; Ovarian Neoplasms; Alopecia; Hypertension
Sulfonylurea receptor 2, Kir6.2 opener
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Arthralgia; Myalgia; Rheumatic Diseases
Cyclooxygenase inhibitor
Small molecule
Approved
EYE; OTHER
OPHTHALMIC
Carcinoma, Non-Small-Cell Lung; Stomach Neoplasms; Breast Neoplasms; Cholangiocarcinoma; Colonic Neoplasms; Rectal Neoplasms; Esophageal Neoplasms; Colorectal Neoplasms; Eye Infections; Herpes Simplex; Keratoconjunctivitis; Neoplasms
DNA inhibitor
Small molecule
Approved
Unknown
Unknown
Glaucoma
Unknown
Small molecule
Approved
Unknown
Unknown
Arthralgia; Myalgia; Rheumatic Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Brain Neoplasms; Glioblastoma; Anxiety; Dementia; Schizophrenia; Depressive Disorder
Unknown
Small molecule
Approved
OTHER
ORAL
Helminthiasis
DNA inhibitor
Small molecule
Approved
OTHER
ORAL
Prostatic Neoplasms, Castration-Resistant; Breast Neoplasms; Neoplasms
Cytochrome P450 11A1 inhibitor
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Bacterial Infections
Unknown
Small molecule
Approved
OTHER
ORAL
Acute Kidney Injury; Severe Acute Respiratory Syndrome; Sleep Apnea, Obstructive; Vitamin D Deficiency; Myocardial Infarction; Hyperparathyroidism, Secondary; Parathyroid Diseases; Renal Insufficiency, Chronic
Vitamin D receptor agonist
Small molecule
Approved
Unknown
Unknown
Ischemic Stroke; Cardiovascular Diseases
Unknown
Small molecule
Approved
OTHER
ORAL
Osteomyelitis; Bacterial Infections
Bacterial DNA gyrase inhibitor
Small molecule
Approved
OTHER
ORAL
Depressive Disorder
Dopamine receptor antagonist
Small molecule
Approved
Unknown
Unknown
Rheumatic Diseases
Unknown
Small molecule
Approved
OTHER
INJECTION; TOPICAL
Kidney Failure, Chronic; Leukemia; Myopia; Neoplasm Metastasis; Appendiceal Neoplasms; Biliary Tract Neoplasms; Carcinoma, Squamous Cell; Cholangiocarcinoma; Cholangitis, Sclerosing; Corneal Opacity; Esophageal Stenosis; Glaucoma, Neovascular; Glaucoma, Open-Angle; Keratoconus; Liver Neoplasms; Pterygium; Sarcoma; Urethral Stricture; Anus Neoplasms; Breast Neoplasms; Carcinoma; Carcinoma, Hepatocellular; Carcinoma in Situ; Carcinoma, Non-Small-Cell Lung; Carcinoma, Transitional Cell; Colorectal Neoplasms; Head and Neck Neoplasms; Lung Neoplasms; Mesothelioma; Nasopharyngeal Carcinoma; Pancreatic Neoplasms; Stomach Neoplasms; Urinary Bladder Neoplasms; Uterine Cervical Neoplasms; Adenocarcinoma; Glaucoma; Neoplasms
DNA inhibitor
Small molecule
Approved
Unknown
Unknown
Attention Deficit Disorder with Hyperactivity; Cystic Fibrosis; Coronary Disease; Demyelinating Diseases; Hyperparathyroidism, Primary; Migraine with Aura; Multiple Sclerosis, Chronic Progressive; Optic Neuritis; Hypertension; Cardiovascular Diseases
Unknown
Small molecule
Approved
CARDIOVASCULAR; OTHER; UROLOGY AND KIDNEY
INJECTION; URETHRAL
Acute Kidney Injury; Arteriosclerosis Obliterans; Optic Neuropathy, Ischemic; Peripheral Arterial Disease; Peripheral Vascular Diseases; Respiratory Distress Syndrome; Severe Acute Respiratory Syndrome; Sexual Dysfunction, Physiological; Heart Failure; Macular Degeneration; Prostatic Neoplasms, Castration-Resistant; Cardiovascular Diseases; Ductus Arteriosus, Patent; Erectile Dysfunction
Prostanoid EP1 receptor agonist
Small molecule
Approved
OTHER
INJECTION
Breast Neoplasms
Unknown
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Bacterial Infections
Unknown
Small molecule
Approved
OTHER; RESPIRATORY
INHALATION
Ciliary Motility Disorders; Depressive Disorder, Major; Diabetes Mellitus; Glycogen Storage Disease Type II; Idiopathic Pulmonary Fibrosis; Lymphangioleiomyomatosis; Myasthenic Syndromes, Congenital; Tachypnea; Bronchiolitis; Cough; Familial Primary Pulmonary Hypertension; Hypersensitivity; Memory Disorders; Pulmonary Edema; Respiratory Insufficiency; Spinal Cord Injuries; Status Asthmaticus; Abdominal Pain; Dysautonomia, Familial; Heart Failure; Hypertension, Pulmonary; Lung Diseases; Organophosphate Poisoning; Rhinitis, Allergic, Seasonal; Asthma, Exercise-Induced; Bronchial Spasm; Lung Diseases, Obstructive; Pulmonary Disease, Chronic Obstructive
Beta-2 adrenergic receptor agonist
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Pulmonary Disease, Chronic Obstructive; Urinary Tract Infections; Lung Diseases; Pneumonia; Tuberculosis; Cystic Fibrosis; Mycobacterium Infections; Pneumonia, Bacterial; Pneumonia, Ventilator-Associated; Bacterial Infections; Eye Infections
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Orthostatic Intolerance; Osteoporosis; Stress Disorders, Post-Traumatic; Atrial Fibrillation; Cerebrovascular Disorders; Essential Hypertension; Heart Diseases; Heart Failure; Hemangioma; Hypertrophy, Left Ventricular; Marfan Syndrome; Mitral Valve Stenosis; Myocardial Ischemia; Vascular Diseases; Angina Pectoris; Cardiovascular Diseases; Coronary Artery Disease; Diabetes Mellitus; Hypertension; Myocardial Infarction; Stroke
Beta-1 adrenergic receptor antagonist
Small molecule
Approved
OTHER
ORAL
Lung Diseases, Obstructive
Adenosine receptor antagonist