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Total: 6532
Small molecule
Approved
OTHER; RESPIRATORY
INHALATION
Ciliary Motility Disorders; Depressive Disorder, Major; Diabetes Mellitus; Glycogen Storage Disease Type II; Idiopathic Pulmonary Fibrosis; Lymphangioleiomyomatosis; Myasthenic Syndromes, Congenital; Tachypnea; Bronchiolitis; Cough; Familial Primary Pulmonary Hypertension; Hypersensitivity; Memory Disorders; Pulmonary Edema; Respiratory Insufficiency; Spinal Cord Injuries; Status Asthmaticus; Abdominal Pain; Dysautonomia, Familial; Heart Failure; Hypertension, Pulmonary; Lung Diseases; Organophosphate Poisoning; Rhinitis, Allergic, Seasonal; Asthma, Exercise-Induced; Bronchial Spasm; Lung Diseases, Obstructive; Pulmonary Disease, Chronic Obstructive
Beta-2 adrenergic receptor agonist
Small molecule
Approved
CARDIOVASCULAR; OTHER; UROLOGY AND KIDNEY
INJECTION; URETHRAL
Acute Kidney Injury; Arteriosclerosis Obliterans; Optic Neuropathy, Ischemic; Peripheral Arterial Disease; Peripheral Vascular Diseases; Respiratory Distress Syndrome; Severe Acute Respiratory Syndrome; Sexual Dysfunction, Physiological; Heart Failure; Macular Degeneration; Prostatic Neoplasms, Castration-Resistant; Cardiovascular Diseases; Ductus Arteriosus, Patent; Erectile Dysfunction
Prostanoid EP1 receptor agonist
Small molecule
Approved
OTHER
ORAL
Hypersensitivity; Multiple Sclerosis; Sunburn; Angioedema; Conjunctivitis, Allergic; Rhinitis, Allergic, Perennial; Rhinitis, Allergic, Seasonal; Rhinitis, Vasomotor; Urticaria
Histamine H1 receptor antagonist
Small molecule
Approved
OTHER
ORAL
Anxiety; Dementia; Depressive Disorder; Pulmonary Disease, Chronic Obstructive; Schizophrenia; Sleep Initiation and Maintenance Disorders
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
OTHER
ORAL
Asthma; Diabetes Mellitus, Type 1; Migraine Disorders; Phobia, Social; Substance-Related Disorders; Dental Anxiety; Epilepsy; Stress Disorders, Post-Traumatic; Dementia; Depressive Disorder; Schizophrenia; Seizures; Anxiety; Anxiety Disorders; Panic Disorder
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Otitis Media; Appendicitis; Communicable Diseases; Graft vs Host Disease; Abscess; Cholecystitis, Acute; Diabetic Foot; Enterobacteriaceae Infections; Hematologic Neoplasms; Infections; Influenza, Human; Pneumonia; Pneumonia, Bacterial; Pneumonia, Ventilator-Associated; Pseudomonas Infections; Sepsis; Severe Acute Respiratory Syndrome; Shock, Septic; Urinary Tract Infections; Bacterial Infections
Unknown
Small molecule
Approved
OTHER
ORAL
Alzheimer Disease; Anemia; Diabetes Mellitus, Type 2; HIV Infections; Hypertriglyceridemia; Multiple Sclerosis; Neoplasms; Alcoholism; Myocardial Ischemia; Parkinson Disease; Smoking Cessation; Tobacco Use Disorder; Abdominal Pain; Cardiovascular Diseases; Coronary Disease
Peroxisome proliferator-activated receptor alpha agonist
Small molecule
Approved
Unknown
Unknown
Hypotension, Orthostatic; Orthostatic Intolerance; Depressive Disorder; Hypotension; Myocardial Infarction; Hypertension
Unknown
Small molecule
Approved
Unknown
Unknown
Anemia; HIV Infections; Malaria; Malaria, Falciparum; Malaria, Vivax; Pneumonia, Pneumocystis; Pregnancy; Premature Birth
Dihydropteroate synthetase inhibitor
Small molecule
Approved
IMMUNE SYSTEM; OTHER
ORAL; TOPICAL
Alzheimer Disease; Asthma; Diabetes Mellitus, Type 2; Erectile Dysfunction; Essential Hypertension; Gastroparesis; Glioblastoma; Hematologic Neoplasms; Hepatitis C; Immune System Diseases; Insulin Resistance; Leukemia, Lymphocytic, Chronic, B-Cell; Lymphoma; Lymphoma, Non-Hodgkin; Melanoma; Multiple Sclerosis; Nausea; Neuroblastoma; Onychomycosis; Osteoporosis; Premature Birth; Pulmonary Disease, Chronic Obstructive; Tinea Versicolor; Breast Neoplasms; Burns; Hypogonadism; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Neoplasms; Prostatic Neoplasms; Psoriasis; Acne Vulgaris; Candidiasis, Vulvovaginal; Dermatitis; Prostatic Neoplasms, Castration-Resistant; Respiratory Distress Syndrome; Vaginosis, Bacterial; Adrenal Gland Diseases; Blastomycosis; Cushing Syndrome; Dermatitis, Seborrheic; Tinea; Tinea Pedis
Cytochrome P450 51 inhibitor
Small molecule
Approved
OTHER
ORAL
Lung Diseases, Obstructive
Adenosine receptor antagonist
Small molecule
Approved
CARDIOVASCULAR; GASTROINTESTINAL; OTHER
INJECTION; INTRA-ANAL; SUBLINGUAL; TRANSDERMAL
Colorectal Neoplasms; Hypertension, Pulmonary; Hypotension; Infections; Inflammation; Peripheral Arterial Disease; Phlebitis; Rectal Neoplasms; Carcinoma, Non-Small-Cell Lung; Diabetic Neuropathies; Erectile Dysfunction; Hot Flashes; Lung Neoplasms; Pulmonary Edema; Shock; Tendinopathy; Anus Diseases; Arthritis, Rheumatoid; Bone Diseases, Metabolic; Heart Diseases; Muscle Cramp; Myocardial Ischemia; Osteoporosis; Raynaud Disease; Reperfusion Injury; Scleroderma, Localized; Stroke; Wounds and Injuries; Angina Pectoris; Cardiovascular Diseases; Coronary Artery Disease; Heart Failure; Hemorrhoids; Hypertension; Myocardial Infarction; Pain
Soluble guanylate cyclase activator
Small molecule
Approved
OTHER
INJECTION; TOPICAL
Kidney Failure, Chronic; Leukemia; Myopia; Neoplasm Metastasis; Appendiceal Neoplasms; Biliary Tract Neoplasms; Carcinoma, Squamous Cell; Cholangiocarcinoma; Cholangitis, Sclerosing; Corneal Opacity; Esophageal Stenosis; Glaucoma, Neovascular; Glaucoma, Open-Angle; Keratoconus; Liver Neoplasms; Pterygium; Sarcoma; Urethral Stricture; Anus Neoplasms; Breast Neoplasms; Carcinoma; Carcinoma, Hepatocellular; Carcinoma in Situ; Carcinoma, Non-Small-Cell Lung; Carcinoma, Transitional Cell; Colorectal Neoplasms; Head and Neck Neoplasms; Lung Neoplasms; Mesothelioma; Nasopharyngeal Carcinoma; Pancreatic Neoplasms; Stomach Neoplasms; Urinary Bladder Neoplasms; Uterine Cervical Neoplasms; Adenocarcinoma; Glaucoma; Neoplasms
DNA inhibitor
Small molecule
Approved
CARDIOVASCULAR; DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Diabetes Mellitus, Type 2; Glioblastoma; Hypertension, Pulmonary; Neoplasms; Primary Myelofibrosis; Heart Diseases; Pneumonia; Diabetes Mellitus, Type 1; Essential Hypertension; Severe Acute Respiratory Syndrome; Cardiovascular Diseases; Collagen Diseases; Diabetic Nephropathies; Diabetic Retinopathy; Heart Failure; Hypertension; Myocardial Infarction; Renal Insufficiency; Ventricular Dysfunction, Left
Angiotensin-converting enzyme inhibitor
Small molecule
Approved
Unknown
Unknown
Osteomyelitis
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
OTHER
INHALATION; NASAL
Rhinitis, Allergic, Perennial; Asthma; Lung Diseases, Obstructive; Nasal Obstruction; Rhinitis
Glucocorticoid receptor agonist
Small molecule
Approved
Unknown
Unknown
Hepatitis C; Amphetamine-Related Disorders; Anemia, Sickle Cell; Carcinoma, Squamous Cell; Rotator Cuff Injuries; Schizophrenia; Stress Disorders, Post-Traumatic; Toothache; Back Pain; Cocaine-Related Disorders; Depressive Disorder; Depressive Disorder, Major; Heroin Dependence; HIV Infections; Intervertebral Disc Degeneration; Low Back Pain; Morphine Dependence; Neonatal Abstinence Syndrome; Neuralgia; Osteoarthritis; Substance Withdrawal Syndrome; Acute Pain; Chronic Pain; Drug Overdose; Opioid-Related Disorders; Pain; Substance-Related Disorders
Kappa opioid receptor agonist
Small molecule
Approved
OTHER
INJECTION; ORAL
Orthostatic Intolerance; Osteoporosis; Stress Disorders, Post-Traumatic; Atrial Fibrillation; Cerebrovascular Disorders; Essential Hypertension; Heart Diseases; Heart Failure; Hemangioma; Hypertrophy, Left Ventricular; Marfan Syndrome; Mitral Valve Stenosis; Myocardial Ischemia; Vascular Diseases; Angina Pectoris; Cardiovascular Diseases; Coronary Artery Disease; Diabetes Mellitus; Hypertension; Myocardial Infarction; Stroke
Beta-1 adrenergic receptor antagonist
Small molecule
Approved
Unknown
Unknown
Crohn Disease; Diabetes Mellitus, Type 2; Hemorrhage; Hodgkin Disease; Ischemic Stroke; Osteoarthritis, Knee; Respiratory Syncytial Virus Infections; Substance-Related Disorders; Pain; Severe Acute Respiratory Syndrome; Arrhythmias, Cardiac; Atrial Fibrillation; Bipolar Disorder; Diabetes Mellitus, Type 1; Heart Failure; Cardiovascular Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Attention Deficit Disorder with Hyperactivity; Cystic Fibrosis; Coronary Disease; Demyelinating Diseases; Hyperparathyroidism, Primary; Migraine with Aura; Multiple Sclerosis, Chronic Progressive; Optic Neuritis; Hypertension; Cardiovascular Diseases
Unknown
Small molecule
Approved
OTHER
ORAL
Adrenal Hyperplasia, Congenital; Substance-Related Disorders; Anus Diseases; Epilepsies, Partial; Epilepsy; Fissure in Ano; Proteinuria; Renal Insufficiency, Chronic; Diabetic Nephropathies; Hypertension, Pulmonary; Kidney Calculi; Myocardial Ischemia; Placenta Previa; Pre-Eclampsia; Premature Birth; Raynaud Disease; Cardiovascular Diseases; Coronary Vasospasm; Hypertension
Voltage-gated L-type calcium channel blocker
Small molecule
Approved
OTHER
ORAL
Anxiety
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
CARDIOVASCULAR; DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Depressive Disorder; Depressive Disorder, Major; Cardiovascular Diseases
Beta-1 adrenergic receptor partial agonist
Small molecule
Approved
OTHER
ORAL
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Bacterial Infections
Unknown
Small molecule
Approved
OTHER
TOPICAL
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
INJECTION
Unknown
Prostanoid FP receptor agonist
Small molecule
Approved
Unknown
Unknown
Schistosomiasis mansoni; Cysticercosis; Schistosomiasis haematobia; Helminthiasis; Infections; Opisthorchiasis; Schistosomiasis
Voltage-activated calcium channel beta 1 subunit blocker
Small molecule
Approved
OTHER
VAGINAL
Hidradenitis Suppurativa; Candidiasis, Oral; HIV Infections
DNA inhibitor
Small molecule
Approved
Unknown
Unknown
Fecal Incontinence; Urinary Incontinence; Cardiovascular Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown