Display Options:
Total: 6532
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Psychotic Disorders; Schizophrenia; Appendicitis; Bipolar Disorder; Borrelia Infections; Cholangitis; Colitis, Ulcerative; Dysentery, Bacillary; Endocarditis; Endometritis; Malnutrition; Parkinson Disease; Pelvic Inflammatory Disease; Amyotrophic Lateral Sclerosis; Gonorrhea; Infections; Influenza, Human; Lyme Disease; Peritonitis; Pneumonia; Pneumonia, Bacterial; Sepsis; Severe Acute Respiratory Syndrome; Urinary Tract Infections; Bacterial Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Bacterial Infections
Unknown
Small molecule
Approved
OTHER
INJECTION
Bacterial Infections
Bacterial penicillin-binding protein 2 inhibitor
Small molecule
Approved
Unknown
Unknown
Sepsis; Mastitis; Periapical Periodontitis; Tuberculosis; Enterobacteriaceae Infections; Pyelonephritis; Infections; Otitis Media; Pneumonia; Respiratory Tract Infections; Sinusitis; Soft Tissue Infections; Urinary Tract Infections
Bacterial beta-lactamase TEM inhibitor
Small molecule
Approved
OTHER
INHALATION
Unknown
Beta-2 adrenergic receptor agonist
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM
INTRAMUSCULAR
Anorexia Nervosa; Bulimia; Bulimia Nervosa; Child Development Disorders, Pervasive; Dermatitis, Atopic; Melanoma; Mental Disorders; Psoriasis; Schizophrenia; Smoking Cessation; Alcohol Drinking; Alcohol-Related Disorders; Back Pain; Breast Neoplasms; Colitis, Ulcerative; Coronavirus Infections; Crohn Disease; Cystitis, Interstitial; Depressive Disorder, Major; Diabetic Neuropathies; Dry Eye Syndromes; Fatigue; Fibromyalgia; Low Back Pain; Marijuana Abuse; Migraine Disorders; Obsessive-Compulsive Disorder; Post-Acute COVID-19 Syndrome; Respiratory Distress Syndrome; Severe Acute Respiratory Syndrome; Trichotillomania; Amphetamine-Related Disorders; Borderline Personality Disorder; Chronic Pain; Cocaine-Related Disorders; Depressive Disorder; Endometriosis; Gambling; Heroin Dependence; HIV Infections; Multiple Sclerosis; Obesity; Opioid-Related Disorders; Pain; Stress Disorders, Post-Traumatic; Substance-Related Disorders; Tobacco Use Disorder; Alcoholism
Opioid receptors; mu/kappa/delta antagonist
Small molecule
Approved
OTHER
INJECTION
Unknown
Phosphodiesterase 3A inhibitor
Small molecule
Approved
OTHER
INJECTION
Bacterial Infections
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Arthralgia; Eye Diseases; Myalgia
Xanthine dehydrogenase inhibitor
Small molecule
Approved
OTHER
NASAL; ORAL; TRANSDERMAL
Aging; Attention Deficit Disorder with Hyperactivity; Cocaine-Related Disorders; Memory Disorders; Sarcoidosis; Sarcoidosis, Pulmonary; Schizophrenia; Substance-Related Disorders; Alcohol Drinking; Carcinoma; Cognitive Dysfunction; Depressive Disorder; Parkinson Disease; Postoperative Nausea and Vomiting; Sarcoma; Wounds and Injuries; Heart Failure; Lung Neoplasms; Marijuana Abuse; Pulmonary Disease, Chronic Obstructive; Severe Acute Respiratory Syndrome; Smoking; Smoking Cessation; Uterine Cervical Neoplasms; Tobacco Use Disorder
Neuronal acetylcholine receptor; alpha4/beta2 agonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Constipation; Fractures, Bone; Heart Arrest; Heroin Dependence; Restless Legs Syndrome; Rheumatic Diseases; Blood Coagulation Disorders; Fractures, Multiple; Hemorrhage; Mucositis; Neuralgia; Postoperative Complications; Premature Birth; Respiratory Insufficiency; Rotator Cuff Injuries; Stomatitis; Tonsillitis; Anemia, Sickle Cell; Back Pain; Cancer Pain; Chronic Pain; Dyspnea; Kidney Calculi; Leukemia; Leukemia, Myeloid, Acute; Myocardial Infarction; Neonatal Abstinence Syndrome; Neoplasms; Obesity; Opioid-Related Disorders; Pregnancy; Prostatic Neoplasms, Castration-Resistant; Pruritus; Pulmonary Disease, Chronic Obstructive; Renal Colic; Rib Fractures; Scoliosis; Sleep Apnea, Obstructive; Wounds and Injuries; Pain
Unknown
Small molecule
Approved
Unknown
Unknown
Endocarditis; Infections; Intraabdominal Infections; Pneumonia; Sepsis; Urinary Tract Infections
Renal dipeptidase inhibitor
Small molecule
Approved
Unknown
Unknown
Barrett Esophagus; Erectile Dysfunction; Ischemia; Renal Insufficiency, Chronic; Cerebral Hemorrhage; Diabetes Mellitus, Type 1; Essential Hypertension; Glomerulonephritis, IGA; Heart Diseases; Melanoma; Pseudohypoaldosteronism; Stroke; Vascular Diseases; Cardiomyopathies; Cardiotoxicity; Chagas Cardiomyopathy; Coronary Disease; Heart Failure; Hematologic Neoplasms; Hypertension; Influenza, Human; Leukemia, Lymphoid; Leukemia, Myeloid, Acute; Lymphoma; Multiple Myeloma; Myocardial Ischemia; Neoplasms; Pneumonia; Severe Acute Respiratory Syndrome; ST Elevation Myocardial Infarction; Cardiovascular Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Opioid receptors; mu/kappa/delta agonist
Small molecule
Approved
Unknown
Unknown
Amyloidosis, Familial; Atrial Fibrillation; Chagas Cardiomyopathy; Heart Failure; Arrhythmias, Cardiac; Tachycardia, Ventricular; Ventricular Fibrillation
HERG blocker
Small molecule
Approved
Unknown
Unknown
Unknown
Diagnostic
Small molecule
Approved
OTHER
INJECTION; ORAL
Azoospermia; Endocardial Cushion Defects; Heart Septal Defects, Ventricular; Infertility; Acquired Immunodeficiency Syndrome; beta-Thalassemia; Carbon Monoxide Poisoning; Diabetes Mellitus, Type 2; Heart Failure; Muscle Cramp; Neoplasms; Non-alcoholic Fatty Liver Disease; Poisoning; Polycystic Ovary Syndrome; Renal Insufficiency, Chronic; Shock, Septic; Spinal Cord Injuries; Acute Kidney Injury; Arthritis, Rheumatoid; Asthma; Atrial Fibrillation; Cytomegalovirus Infections; Gastrointestinal Stromal Tumors; HIV Infections; Hyperthyroidism; Hypotension; Lipid Metabolism Disorders; Multiple Sclerosis; Muscular Atrophy, Spinal; Pancreatic Neoplasms; Postpoliomyelitis Syndrome; Pyelonephritis; Brain Diseases; Kidney Failure, Chronic; Muscle Weakness
Unknown
Small molecule
Approved
OTHER
INJECTION
Cystic Fibrosis; Osteomyelitis; Esophageal Achalasia; Meningitis, Bacterial; Enterobacteriaceae Infections; Skin Diseases; Staphylococcal Skin Infections; Bacterial Infections; Infections; Intraabdominal Infections; Parametritis; Peritonitis; Pneumonia; Pyelonephritis; Urinary Tract Infections
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
OTHER
ORAL
Adenocarcinoma of Lung; Amebiasis; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Glioblastoma; HIV Infections; Small Cell Lung Carcinoma; Leukemia; Leukemia, Lymphocytic, Chronic, B-Cell; Ovarian Neoplasms; Pain; Tuberculosis; Arthritis, Rheumatoid; Rheumatic Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Irritable Bowel Syndrome; Blepharospasm; Charcot-Marie-Tooth Disease; Chronic Pain; Dystonic Disorders; Death, Sudden, Cardiac; Myocardial Infarction; Myotonic Dystrophy; Ventricular Fibrillation; Arrhythmias, Cardiac
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Cheilitis; Erythema; Stomatitis; Skin Diseases; Eye Diseases; Skin Ulcer
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Diagnostic agent
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Sepsis; Hematologic Neoplasms; Infections; Bacterial Infections; Pneumonia, Bacterial; Pneumonia, Ventilator-Associated; Pyelonephritis; Urinary Tract Infections
Renal dipeptidase inhibitor
Small molecule
Approved
Unknown
Unknown
Anemia, Sickle Cell; Amyotrophic Lateral Sclerosis; Anemia, Neonatal; Heart Failure; Huntington Disease; Asthma; Multiple Sclerosis; Anemia; Anemia, Iron-Deficiency; Diabetes Mellitus, Type 2; Kidney Failure, Chronic
Unknown
Small molecule
Approved
OTHER
TOPICAL
Tinea Pedis
Cytochrome P450 51 inhibitor
Small molecule
Approved
Unknown
Unknown
Nausea; Neoplasms; Pulmonary Alveolar Proteinosis; Atherosclerosis; Attention Deficit Disorder with Hyperactivity; Colorectal Neoplasms; Epilepsy; Fatty Liver, Alcoholic; Heart Diseases; Heart Failure; Hepatitis, Alcoholic; HIV Infections; Lymphoma; Multiple Myeloma; Myocardial Infarction; Myocardial Ischemia; Psychotic Disorders; Tuberculosis, Pulmonary; Vomiting; Alzheimer Disease; Hand-Foot Syndrome; Movement Disorders; Non-alcoholic Fatty Liver Disease; Spasms, Infantile; Tuberculosis; Anemia; Diabetes Mellitus, Type 2; Kidney Failure, Chronic; Osteoporosis; Postoperative Nausea and Vomiting
Unknown
Small molecule
Approved
OTHER
ORAL
Obsessive-Compulsive Disorder; Fibromyalgia; Marijuana Abuse; Muscle Spasticity; Neuralgia; Obesity; Suicidal Ideation; Diabetic Neuropathies; Parkinson Disease; Nausea; Neoplasms; Postoperative Nausea and Vomiting
Cannabinoid CB1 receptor agonist
Small molecule
Approved
Unknown
Unknown
Multiple Sclerosis; Acidosis, Lactic; Heart Arrest; Huntington Disease; Respiratory Insufficiency; Heart Failure; Hyperemesis Gravidarum; Sepsis; Shock, Septic; Anemia; Brain Diseases; Kidney Failure, Chronic; Thiamine Deficiency
Unknown
Small molecule
Approved
Unknown
Unknown
Anemia; Arthritis, Rheumatoid; Asthma; Infertility; Ovarian Neoplasms; Pancreatic Neoplasms; Penile Induration; Acute Kidney Injury; Adrenoleukodystrophy; Asthenozoospermia; Atherosclerosis; Brain Diseases; Burns; Cardiovascular Diseases; Carotid Artery Diseases; Diabetes Mellitus, Type 2; Endometriosis; Fibrosis; Friedreich Ataxia; Heart Diseases; Heart Failure; Heavy Metal Poisoning; Infertility, Male; Intracranial Arteriosclerosis; Lung Neoplasms; Mastodynia; Neoplasms; Neuromuscular Diseases; Peripheral Nervous System Diseases; Polycystic Ovary Syndrome; Renal Insufficiency, Chronic; Reperfusion Injury; Stomatitis; Tobacco Use Disorder; Wounds and Injuries; Alzheimer Disease; Amyotrophic Lateral Sclerosis; Breast Neoplasms; Cataract; Cerebrovascular Disorders; Colorectal Neoplasms; Coronary Disease; Delirium; Depressive Disorder; Fatty Liver; Gaucher Disease; Glaucoma; Head and Neck Neoplasms; Hypobetalipoproteinemias; Infections; Kidney Diseases; Liver Cirrhosis; Liver Diseases; Macular Degeneration; Menopause; Migraine Disorders; Myocardial Infarction; Myocardial Ischemia; Non-alcoholic Fatty Liver Disease; Osteonecrosis; Pain; Parkinson Disease; Prostatic Neoplasms, Castration-Resistant; Psoriasis; Pulmonary Disease, Chronic Obstructive; Rectal Neoplasms; Retinitis Pigmentosa; Schizophrenia; Urinary Bladder Neoplasms; Vascular Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
GASTROINTESTINAL; IMMUNE SYSTEM; OTHER
INHALATION; ORAL
Breast Neoplasms; Neoplasms; Diabetes Mellitus, Type 1; Encephalitis, Japanese; Hemorrhagic Fever with Renal Syndrome; Hepatitis D; Influenza, Human; Lassa Fever; Leukemia, Myeloid, Acute; Thrombocytopenia; Depressive Disorder; Hepatitis; Hepatitis B, Chronic; Hepatitis C; HIV Infections; Infections; Respiratory Syncytial Virus Infections; Severe Acute Respiratory Syndrome; Fibrosis; Hepatitis C, Chronic; Liver Cirrhosis; Virus Diseases
Inosine-5'-monophosphate dehydrogenase 1 inhibitor