Display Options:
Total: 6532
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Sodium channel alpha subunit blocker
Small molecule
Approved
OTHER
INJECTION
Arrhythmias, Cardiac; Ventricular Fibrillation
Norepinephrine transporter substrate
Small molecule
Approved
Unknown
Unknown
Asthma
Unknown
Small molecule
Approved
OTHER
OPHTHALMIC; ORAL
Osteomyelitis; Hermanski-Pudlak Syndrome; Cystitis, Hemorrhagic; Esophageal and Gastric Varices; Liver Cirrhosis; Peritonitis; Bacterial Infections; Eye Infections
Bacterial DNA gyrase inhibitor
Small molecule
Approved
Unknown
Unknown
Cognitive Dysfunction; Ovarian Cysts; Shock, Septic; Diabetic Foot; Hypertension
Beta-1 adrenergic receptor antagonist
Small molecule
Approved
Unknown
Unknown
Lung Diseases, Obstructive
Unknown
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Chorioamnionitis; Cleft Palate; Infections; Urinary Tract Infections; Bacterial Infections
Unknown
Small molecule
Approved
OTHER; PREGNANCY AND GYNECOLOGY
INJECTION; INTRAVENOUS; ORAL
Back Pain; Hypotension; Liver Cirrhosis; Skin Neoplasms; Spinal Cord Neoplasms; Cerebral Hemorrhage; Epistaxis; Intervertebral Disc Degeneration; Osteoarthritis, Knee; Shock, Septic; Subarachnoid Hemorrhage; Urinary Bladder Neoplasms; Anemia; Angioedemas, Hereditary; Aortic Aneurysm, Abdominal; Astrocytoma; Blood Coagulation Disorders; Bone Neoplasms; Brain Injuries; Brain Neoplasms; Burns; Coronary Disease; Femoral Neck Fractures; Fractures, Bone; Gastrointestinal Hemorrhage; Genital Neoplasms, Female; Head and Neck Neoplasms; Hematologic Neoplasms; Hematoma; Hematoma, Subdural, Intracranial; Hemoptysis; Hip Fractures; Ileus; Inflammation; Joint Diseases; Leiomyoma; Melanoma; Melanosis; Meningioma; Nasal Polyps; Neoplasms; Osteoarthritis; Pain; Paraganglioma; Pelvic Organ Prolapse; Placenta Accreta; Placenta Previa; Postpartum Hemorrhage; Prostatic Neoplasms, Castration-Resistant; Scoliosis; Sepsis; Severe Acute Respiratory Syndrome; Shock; Shoulder Impingement Syndrome; Telangiectasia, Hereditary Hemorrhagic; Thrombocytopenia; von Willebrand Diseases; Wounds and Injuries; Hemophilia A; Hemorrhage; Menorrhagia
Plasminogen inhibitor
Small molecule
Approved
OTHER
ORAL
Anemia; Anemia, Sickle Cell; Arthritis, Rheumatoid; Diabetes Mellitus, Type 2; Fractures, Bone; HIV Infections; Mitochondrial Diseases; Low Back Pain; Periodontitis; Pain; Pharyngitis; Arthralgia; Eye Diseases; Miosis; Myalgia; Rheumatic Diseases
Cyclooxygenase inhibitor
Small molecule
Approved
Unknown
Unknown
Common Cold; Fecal Incontinence; Hypotension, Orthostatic; Presbyopia; Rhinitis, Allergic, Seasonal; Erythema; Rosacea; Eye Manifestations; Nasal Obstruction
Unknown
Small molecule
Approved
Unknown
Unknown
Carcinoma, Non-Small-Cell Lung; Colorectal Neoplasms; Fibrosis; Glycogen Storage Disease Type III; HIV Infections; Leukemia, Hairy Cell; Lupus Erythematosus, Systemic; Melanoma; Mesothelioma; Neoplasms; Psoriasis; Thyroid Neoplasms; Anemia, Sickle Cell; Breast Carcinoma In Situ; Breast Neoplasms; Eosinophilic Esophagitis; Immunoglobulin G4-Related Disease; Movement Disorders; Schizophrenia; Stomach Neoplasms; Gastrointestinal Hemorrhage; Severe Acute Respiratory Syndrome; Arthritis, Rheumatoid; Chest Pain; Duodenal Ulcer; Esophagitis; Gastroesophageal Reflux; Heartburn; Osteoarthritis; Peptic Ulcer; Stomach Ulcer; Ulcer
Histamine H2 receptor antagonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
INJECTION
Delirium; Schizophrenia
D2-like dopamine receptor inverse agonist
Small molecule
Approved
Unknown
Unknown
Dyspepsia; Scleroderma, Systemic; Attention Deficit Disorder with Hyperactivity; Autistic Disorder; Child Development Disorders, Pervasive; Cocaine-Related Disorders; Depressive Disorder, Major; Gastroparesis; Marijuana Abuse; Sexual Dysfunction, Physiological; Spinal Cord Injuries; Anxiety Disorders; Apnea; Dementia; Depressive Disorder; Ischemic Stroke; Parkinson Disease; Schizophrenia; Anxiety
Unknown
Small molecule
Approved
Unknown
Unknown
Arrhythmias, Cardiac
Unknown
Small molecule
Approved
Unknown
Unknown
Status Asthmaticus; Pulmonary Disease, Chronic Obstructive
Unknown
Small molecule
Approved
OTHER
ORAL
Psoriasis
Retinoid receptor agonist
Small molecule
Approved
Unknown
Unknown
Polyuria; Urinary Incontinence
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER; RESPIRATORY
INHALATION; INJECTION
Carcinoma, Non-Small-Cell Lung; Osteomyelitis; Renal Insufficiency; Gonorrhea; Gram-Negative Bacterial Infections; Enterobacteriaceae Infections; Skin Diseases; Bacterial Infections; Cystic Fibrosis; Infections; Intraabdominal Infections; Pneumonia; Pyelonephritis; Sepsis; Urinary Tract Infections
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Muscarinic acetylcholine receptor antagonist
Small molecule
Approved
Unknown
Unknown
Rectal Neoplasms; Cystitis; Infections; Otitis Externa; Pyelonephritis; Urinary Tract Infections
Bacterial DNA gyrase inhibitor
Small molecule
Approved
GASTROINTESTINAL; OTHER; RESPIRATORY
INJECTION; ORAL; OTIC
Arthritis, Rheumatoid; Carcinoma, Pancreatic Ductal; Diabetic Foot; Dysentery, Bacillary; Erectile Dysfunction; Gastroenteritis; Hearing Loss; Hepatitis, Alcoholic; Hepatitis C; Leukemia, Myeloid, Acute; Liver Cirrhosis, Alcoholic; Lung Diseases; Lymphoma; Neoplasms; Osteomyelitis; Periapical Periodontitis; Pseudomonas Infections; Purpura, Thrombocytopenic, Idiopathic; Rhinoscleroma; Amyotrophic Lateral Sclerosis; Anthrax; Cataract; Corneal Ulcer; Crohn Disease; Cystic Fibrosis; Endophthalmitis; Leukemia, Lymphocytic, Chronic, B-Cell; Pancreatic Neoplasms; Breast Neoplasms; Bronchiectasis; Communicable Diseases; Diarrhea; Digestive System Diseases; Fever; Hypertriglyceridemia; Kidney Calculi; Lipid Metabolism Disorders; Liver Abscess; Neutropenia; Otitis Media; Peritonitis; Plague; Pneumonia; Prostatic Neoplasms, Castration-Resistant; Pulmonary Disease, Chronic Obstructive; Sepsis; Urinary Bladder Neoplasms; Urolithiasis; Bacterial Infections; Bronchitis, Chronic; Cystitis; Eye Infections; Gonorrhea; Infections; Intraabdominal Infections; Otitis Externa; Prostatitis; Pyelonephritis; Sinusitis; Typhoid Fever; Urinary Tract Infections
Bacterial DNA gyrase inhibitor
Small molecule
Approved
OTHER
IMPLANTATION; INHALATION; NASAL; TOPICAL
Alopecia Areata; Hypersensitivity; Otitis Media with Effusion; Spinal Cord Injuries; Anemia, Sickle Cell; Dermatitis, Atopic; Eosinophilic Esophagitis; Pemphigoid, Bullous; Psoriasis; Radiodermatitis; Breast Neoplasms; Hypertrophy; Pulmonary Disease, Chronic Obstructive; Rhinitis, Allergic, Perennial; Severe Acute Respiratory Syndrome; Sinusitis; Sleep Apnea, Obstructive; Asthma; Lung Diseases, Obstructive; Nasal Obstruction; Nasal Polyps; Rhinitis, Allergic; Rhinitis, Allergic, Seasonal; Skin Diseases
Glucocorticoid receptor agonist
Small molecule
Approved
Unknown
Unknown
Cardiovascular Diseases
Unknown
Small molecule
Approved
OTHER
VAGINAL
Vaginitis; Candidiasis, Vulvovaginal
Cytochrome P450 51 inhibitor
Small molecule
Approved
DERMATOLOGY; OTHER
TOPICAL
Bacterial Infections; Osteomyelitis; Sinusitis; Cystic Fibrosis; Hemangioma; Radiodermatitis; Epistaxis; Infections; Staphylococcal Infections; Telangiectasia, Hereditary Hemorrhagic; Impetigo; Nasal Obstruction
Isoleucyl-tRNA synthetase inhibitor
Small molecule
Approved
OTHER
ORAL
Unknown
Cyclooxygenase-2 inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER; RESPIRATORY
ORAL
Osteomyelitis; Bronchitis, Chronic; Infections; Maxillary Sinusitis; Otitis Media; Pharyngitis; Sinusitis; Tonsillitis; Urinary Tract Infections
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown