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Total: 6532
Small molecule
Approved
OTHER
ORAL
Aging; Alcoholism; Depressive Disorder; Fractures, Bone; Neoplasms; Pancreatitis; Periodontitis; Bile Duct Diseases; Carcinoma; Carcinoma, Basal Cell; Mastodynia; Pulmonary Embolism; Wounds and Injuries; Infertility; Osteoarthritis, Hip; Osteoarthritis, Knee; Renal Colic; Spondylitis, Ankylosing; Stomach Ulcer; Toothache; Acute Pain; Arthralgia; Arthritis, Rheumatoid; Cataract; Dysmenorrhea; Eye Diseases; Inflammation; Keratosis, Actinic; Migraine Disorders; Myalgia; Osteoarthritis; Rheumatic Diseases; Sprains and Strains
Cyclooxygenase inhibitor
Small molecule
Approved
OTHER
INJECTION
Multiple Myeloma; Myelodysplastic Syndromes; Myeloproliferative Disorders; Neoplasm Metastasis; Neoplasms, Plasma Cell; Breast Neoplasms; Burkitt Lymphoma; Leukemia, Myeloid, Acute; Lymphoma, AIDS-Related; Lymphoma, B-Cell; Lymphoma, Large-Cell, Anaplastic; Lymphoma, Mantle-Cell; Nasopharyngeal Neoplasms; Pancreatic Neoplasms; Penile Neoplasms; Peritoneal Neoplasms; Rhabdomyosarcoma, Alveolar; Rhabdomyosarcoma, Embryonal; Urethral Neoplasms; Urinary Bladder Neoplasms; Uterine Neoplasms; Wilms Tumor; Carcinoma; Carcinoma, Non-Small-Cell Lung; Central Nervous System Neoplasms; Dermatofibrosarcoma; Endometrial Neoplasms; Fallopian Tube Neoplasms; Fibrosarcoma; Hemangiosarcoma; Histiocytoma; Hodgkin Disease; Kidney Neoplasms; Leiomyosarcoma; Leukemia; Leukemia, Biphenotypic, Acute; Liposarcoma; Lung Neoplasms; Lymphoma; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Non-Hodgkin; Lymphoma, T-Cell, Peripheral; Mediastinal Neoplasms; Neoplasms, Germ Cell and Embryonal; Neurilemmoma; Neuroblastoma; Osteosarcoma; Ovarian Neoplasms; Pheochromocytoma; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Precursor T-Cell Lymphoblastic Leukemia-Lymphoma; Retroviridae Infections; Rhabdomyosarcoma; Sarcoma; Sarcoma, Alveolar Soft Part; Sarcoma, Ewing; Sarcoma, Synovial; Small Cell Lung Carcinoma; Teratoma; Uterine Cervical Neoplasms; Neoplasms; Testicular Neoplasms
DNA inhibitor
Small molecule
Approved
Unknown
Unknown
Gastritis; Gastroparesis; Duodenal Ulcer; Esophagitis; Gastroesophageal Reflux; Heartburn; Peptic Ulcer
Histamine H2 receptor antagonist
Small molecule
Approved
Unknown
Unknown
Onychomycosis; Tinea Pedis
Unknown
Small molecule
Approved
Unknown
Unknown
Bacterial Infections
Unknown
Small molecule
Approved
OTHER
ORAL
Unknown
Beta-1 adrenergic receptor antagonist
Small molecule
Approved
Unknown
Unknown
Cystic Fibrosis; Hepatitis C; HIV Infections; Migraine Disorders; Metrorrhagia; Osteoporosis; Neural Tube Defects; Acne Vulgaris
Progesterone receptor agonist
Small molecule
Approved
EYE; OTHER
IMPLANTATION; OPHTHALMIC; ORAL
Central Nervous System Neoplasms; Kidney Diseases; Melanoma; Mesothelioma; Neuroblastoma; Carcinoma, Hepatocellular; Diabetes Mellitus, Type 1; Fallopian Tube Neoplasms; Glioblastoma; Graft vs Host Disease; Lymphoma; Ovarian Neoplasms; Peritoneal Neoplasms; Conjunctivitis; Cytomegalovirus Infections; Infections; Cytomegalovirus Retinitis; Eye Infections; HIV Infections; Virus Diseases
Human herpesvirus 1 DNA polymerase inhibitor
Small molecule
Approved
OTHER
INJECTION; INTRAVENOUS; IV (INFUSION)
Adenocarcinoma, Follicular; Adrenal Cortex Neoplasms; Anus Neoplasms; Appendiceal Neoplasms; Carcinoma, Renal Cell; Carcinoma, Verrucous; HIV Infections; Hypopharyngeal Neoplasms; Insulinoma; Lymphoma, Large-Cell, Anaplastic; Lymphoma, Mantle-Cell; Multiple Myeloma; Neoplasms, Cystic, Mucinous, and Serous; Neoplasms, Plasma Cell; Neuroendocrine Tumors; Parathyroid Neoplasms; Pericardial Effusion; Pleural Effusion; Skin Diseases; Somatostatinoma; Vaginal Neoplasms; Adenocarcinoma; Adenocarcinoma, Bronchiolo-Alveolar; Bile Duct Neoplasms; Bone Neoplasms; Brain Stem Neoplasms; Breast Neoplasms, Male; Burkitt Lymphoma; Carcinoid Tumor; Carcinoma, Endometrioid; Carcinoma, Intraductal, Noninfiltrating; Carcinoma, Islet Cell; Carcinoma, Merkel Cell; Carcinoma, Neuroendocrine; Carcinosarcoma; Cystadenoma, Serous; Gallbladder Neoplasms; Gastrointestinal Stromal Tumors; Gliosarcoma; Hereditary Breast and Ovarian Cancer Syndrome; Leiomyosarcoma; Leukemia; Leukemia, Myeloid, Acute; Lymphoma, B-Cell; Mesothelioma, Malignant; Myelodysplastic Syndromes; Myeloproliferative Disorders; Nasopharyngeal Neoplasms; Neoplasm Metastasis; Neoplasms, Complex and Mixed; Oligodendroglioma; Osteosarcoma; Pancreatic Neoplasms; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Prostatic Neoplasms; Retinal Neoplasms; Salivary Gland Neoplasms; Stomach Neoplasms; Thrombosis; Thymoma; Ureteral Neoplasms; Uveal Melanoma; Vulvar Neoplasms; Wilms Tumor; Adenocarcinoma of Lung; Anemia; Astrocytoma; Biliary Tract Neoplasms; Brain Neoplasms; Breast Neoplasms; Carcinoma; Carcinoma, Hepatocellular; Carcinoma, Large Cell; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Central Nervous System Neoplasms; Cholangiocarcinoma; Choroid Plexus Neoplasms; Colorectal Neoplasms; Endometrial Neoplasms; Ependymoma; Esophageal Neoplasms; Fallopian Tube Neoplasms; Ganglioneuroblastoma; Genital Neoplasms, Female; Gestational Trophoblastic Disease; Glioblastoma; Glioma; Head and Neck Neoplasms; Hepatoblastoma; Hodgkin Disease; Inflammatory Breast Neoplasms; Kidney Neoplasms; Laryngeal Neoplasms; Leukemia-Lymphoma, Adult T-Cell; Liver Neoplasms; Lung Neoplasms; Lymphoma; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Non-Hodgkin; Medulloblastoma; Melanoma; Mesothelioma; Mouth Neoplasms; Nasopharyngeal Carcinoma; Neoplasms, Germ Cell and Embryonal; Neuroblastoma; Neuroectodermal Tumors, Primitive; Oropharyngeal Neoplasms; Pain; Paraganglioma; Peripheral Nervous System Diseases; Peritoneal Neoplasms; Prostatic Neoplasms, Castration-Resistant; Retinoblastoma; Retroviridae Infections; Sarcoma; Seminoma; Sex Cord-Gonadal Stromal Tumors; Skin Neoplasms; Small Cell Lung Carcinoma; Squamous Cell Carcinoma of Head and Neck; Testicular Neoplasms; Thyroid Neoplasms; Triple Negative Breast Neoplasms; Urethral Neoplasms; Urinary Bladder Neoplasms; Urogenital Neoplasms; Uterine Cervical Neoplasms; Uterine Neoplasms; Carcinoma, Ovarian Epithelial; Neoplasms; Ovarian Neoplasms
DNA inhibitor
Small molecule
Approved
OTHER
ORAL
Anxiety; Bipolar Disorder; Dementia; Depressive Disorder; Developmental Disabilities; Intellectual Disability; Psychotic Disorders; Schizophrenia
Dopamine D2 receptor antagonist
Small molecule
Approved
OTHER; UROLOGY AND KIDNEY
ORAL
Ovarian Neoplasms; Polycystic Ovary Syndrome; Prostatic Neoplasms, Castration-Resistant; Carcinoma; Neoplasms; Prostatic Neoplasms
Androgen Receptor antagonist
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Colorectal Neoplasms; Bacterial Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Atrial Fibrillation; Death, Sudden, Cardiac; Heart Failure; Myocardial Infarction; Ventricular Fibrillation; Arrhythmias, Cardiac
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
INJECTION
Amnesia; Colorectal Neoplasms; Depressive Disorder; Depressive Disorder, Major; Inflammation; Neural Tube Defects; Osteonecrosis; Premature Birth; Psychomotor Agitation; Renal Insufficiency; Renal Insufficiency, Chronic; Scoliosis; Sepsis; Shock; Sleep Initiation and Maintenance Disorders; Spinal Stenosis; Coronary Disease; Depressive Disorder, Treatment-Resistant; Hypotension; Intestinal Polyps; Leukemia; Lung Neoplasms; Migraine Disorders; Obesity, Morbid; Postoperative Nausea and Vomiting; Pulmonary Disease, Chronic Obstructive; Sleep Apnea, Obstructive; Strabismus; Tonsillitis; Wounds and Injuries; Adenomatous Polyposis Coli; Atrial Fibrillation; Back Pain; Brain Injuries; Breast Neoplasms; Cerebral Arterial Diseases; Delirium; Esophageal Neoplasms; Genital Neoplasms, Male; Heart Diseases; Hypertension; Intracranial Aneurysm; Liver Cirrhosis; Neoplasms; Obesity; Pain; Pancreatic Neoplasms; Pruritus; Reperfusion Injury; Respiratory Distress Syndrome; Respiratory Distress Syndrome, Newborn; Respiratory Insufficiency; Severe Acute Respiratory Syndrome; Shock, Septic; Status Epilepticus; Stroke; Subarachnoid Hemorrhage
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
Unknown
Unknown
Chronic Pain; Diabetic Retinopathy; Fallopian Tube Neoplasms; Hypoxia; Ovarian Neoplasms; Peritoneal Neoplasms; Renal Colic; Conjunctivitis, Viral; Heart Diseases; Kidney Neoplasms; Miosis; Musculoskeletal Diseases; Osteoarthritis, Knee; Pancreatitis; Periodontitis; Pre-Eclampsia; Retinopathy of Prematurity; Rotator Cuff Injuries; Scoliosis; Tonsillitis; Abdominal Pain; Back Pain; Breast Neoplasms; Cataract; Deglutition Disorders; Headache; Inflammation; Kidney Calculi; Migraine Disorders; Osteoarthritis; Pain; Wounds and Injuries; Eye Diseases; Rheumatic Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Glaucoma
Unknown
Small molecule
Approved
Unknown
Unknown
Anxiety; Dementia; Obsessive-Compulsive Disorder; Premature Ejaculation; Schizophrenia; Depressive Disorder
Unknown
Small molecule
Approved
Unknown
Unknown
Pain
Kappa opioid receptor antagonist
Small molecule
Approved
OTHER
INJECTION; INTRAVENOUS
Inflammation; Ischemia; Leukemia; Leukemia, Lymphocytic, Chronic, B-Cell; Cardiomyopathies; Coronary Disease; Pain; Respiratory Distress Syndrome; ST Elevation Myocardial Infarction; Takotsubo Cardiomyopathy; Angina, Stable; Atrial Fibrillation; Coronary Stenosis; Myocardial Infarction; Myocardial Ischemia; Neoplasms; Tachycardia, Ventricular; Cardiovascular Diseases; Tachycardia, Paroxysmal; Wolff-Parkinson-White Syndrome
Adenosine receptor agonist
Small molecule
Approved
OTHER
ORAL
Neoplasms; Osteomyelitis; HIV Infections; Liver Abscess; Syphilis; Bacterial Infections; Bronchitis; Bronchitis, Chronic; Gonorrhea; Infections; Otitis Media; Pharyngitis; Tonsillitis; Urinary Tract Infections
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
GASTROINTESTINAL; OTHER
ORAL
Alzheimer Disease; Anemia; Anemia, Sickle Cell; Arthritis, Rheumatoid; Carcinoma, Medullary; Central Serous Chorioretinopathy; Child Development Disorders, Pervasive; Chronic Pain; Clostridium Infections; Colitis, Ulcerative; Communicable Diseases; Crohn Disease; Dermatitis, Atopic; Diabetes Mellitus; Diabetes Mellitus, Type 2; Erectile Dysfunction; Glaucoma; Hepatitis B, Chronic; Hepatitis C; Hepatitis C, Chronic; HIV Infections; Laryngomalacia; Melanoma; Mitochondrial Diseases; Muscular Atrophy, Spinal; Neoplasms; Pancreatic Neoplasms; Prostatic Neoplasms; Psoriasis; Pulmonary Disease, Chronic Obstructive; Breast Neoplasms; Carcinoma, Squamous Cell; Colorectal Neoplasms; Gastrinoma; Gastritis; Granuloma; Head and Neck Neoplasms; Idiopathic Pulmonary Fibrosis; Lymphoma; Lymphoma, B-Cell, Marginal Zone; Prostatic Neoplasms, Castration-Resistant; Squamous Cell Carcinoma of Head and Neck; Squamous Intraepithelial Lesions; Ulcer; Zollinger-Ellison Syndrome; Barrett Esophagus; Cough; Cysticercosis; Diabetes Mellitus, Type 1; Dyspepsia; Esophagitis, Peptic; Exocrine Pancreatic Insufficiency; Gastrointestinal Hemorrhage; Helicobacter Infections; Hemorrhage; Multiple Sclerosis, Relapsing-Remitting; Osteoarthritis; Pain; Peripheral Nervous System Diseases; Spondylitis, Ankylosing; Stomach Neoplasms; Wounds and Injuries; Duodenal Ulcer; Esophagitis; Gastroesophageal Reflux; Heartburn; Infections; Peptic Ulcer; Stomach Ulcer
Potassium-transporting ATPase inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
TRANSDERMAL
Amphetamine-Related Disorders; Schizophrenia; Prostatic Neoplasms; Tobacco Use Disorder; Borderline Personality Disorder; Cocaine-Related Disorders; Depressive Disorder; Depressive Disorder, Major; Parkinson Disease
Monoamine oxidase B inhibitor
Small molecule
Approved
Unknown
Unknown
Glioblastoma; Gliosarcoma; Leukoencephalopathy, Progressive Multifocal; Pneumonia, Viral; Respiratory Insufficiency; Severe Acute Respiratory Syndrome; Malaria, Falciparum; Schistosomiasis haematobia; Malaria
Unknown
Small molecule
Approved
OTHER
ORAL
Hypertension
Sulfonylurea receptor 2, Kir6.2 opener
Small molecule
Approved
Unknown
Unknown
Coronary Artery Disease
Unknown
Small molecule
Approved
Unknown
Unknown
Bacterial Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Erectile Dysfunction; Substance-Related Disorders; Alcoholism; Cardiovascular Diseases; Cocaine-Related Disorders; Heart Diseases; Stress Disorders, Post-Traumatic; Tobacco Use Disorder; Vascular Diseases; Diabetes Mellitus; Heart Failure; Hypercholesterolemia; Kidney Calculi; Myocardial Infarction; Myocardial Ischemia; Paraganglioma; Pheochromocytoma; Prostatic Hyperplasia; Hypertension
Unknown
Small molecule
Approved
Unknown
Unknown
Respiratory Distress Syndrome, Newborn; Respiratory Tract Diseases
Lung surfactant
Small molecule
Approved
Unknown
Unknown
Unknown
Adrenergic receptor beta antagonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Alzheimer Disease; Graft vs Host Disease; Leukemia, Myeloid, Acute; Lymphoma; Non-alcoholic Fatty Liver Disease; Pulmonary Disease, Chronic Obstructive; Respiratory Syncytial Virus Infections; Tinea Versicolor; Urinary Bladder, Overactive; Blastomycosis; Histoplasmosis; Intracranial Hypertension; Premature Birth; Sporotrichosis; Vulvovaginitis; Aspergillosis; Bacterial Infections; Candidemia; Candidiasis, Invasive; Candidiasis, Oral; Coccidioidomycosis; Crohn Disease; HIV Infections; Infections; Inflammatory Bowel Diseases; Leishmaniasis, Cutaneous; Leukopenia; Mycoses; Neoplasms; Tinea Pedis; Vaginal Discharge; Vaginitis; Vaginosis, Bacterial; Candidiasis; Candidiasis, Vulvovaginal; Meningitis, Cryptococcal; Urinary Tract Infections
Cytochrome P450 51 inhibitor
Small molecule
Approved
Unknown
Unknown
Atrial Fibrillation; Arrhythmias, Cardiac
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown