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Total: 6532
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Adenocarcinoma; Carcinoma; Central Nervous System Neoplasms; Diffuse Intrinsic Pontine Glioma; Esophageal Neoplasms; Glioma; Neuroblastoma; Paraganglioma; Pheochromocytoma; Rectal Neoplasms; Adenocarcinoma, Follicular; Astrocytoma; Breast Neoplasms; Carcinoma, Hepatocellular; Carcinoma, Renal Cell; Carcinoma, Squamous Cell; Colorectal Neoplasms; Fallopian Tube Neoplasms; Gastrointestinal Stromal Tumors; Glioblastoma; Gliosarcoma; Head and Neck Neoplasms; Kidney Neoplasms; Leukemia, Myeloid, Acute; Mesothelioma; Multiple Myeloma; Neoplasm Metastasis; Oligodendroglioma; Ovarian Neoplasms; Pancreatic Neoplasms; Peritoneal Neoplasms; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Small Cell Lung Carcinoma; Stomach Neoplasms; Ureteral Neoplasms; Urethral Neoplasms; Urinary Bladder Neoplasms; Carcinoma, Non-Small-Cell Lung; Lung Neoplasms; Carcinoma, Medullary; Neoplasms; Thyroid Neoplasms
Ephrin receptor inhibitor
Small molecule
Approved
Unknown
Unknown
Marijuana Abuse; Memory Disorders; Anxiety Disorders; Depressive Disorder
Unknown
Small molecule
Approved
OTHER
INTRAVENOUS
Arthritis, Rheumatoid; Cystitis, Interstitial; Genital Neoplasms, Female; Heart Failure; Urinary Bladder Neoplasms; Uterine Cervical Neoplasms; Neoplasms; Central Nervous System Diseases
Diagnostic agent
Small molecule
Approved
Unknown
Unknown
Alcohol Drinking; Anxiety; Arthritis, Rheumatoid; Celiac Disease; Gingivitis; Otitis Media with Effusion; Acne Vulgaris; Amyotrophic Lateral Sclerosis; Burns; Chemical and Drug Induced Liver Injury; Hidradenitis Suppurativa; Ileus; Intervertebral Disc Degeneration; Melanoma; Severe Acute Respiratory Syndrome; Tinea Pedis; Cardiovascular Diseases; Dental Caries; Hemorrhoids; Infections; Pain; Periodontitis; Tension-Type Headache; Tooth Diseases
Unknown
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY
ORAL
Adenocarcinoma; Carcinoma, Non-Small-Cell Lung; Esophageal Neoplasms; Hypertension; Renal Insufficiency; Schizophrenia; Stomach Neoplasms; Respiratory Tract Diseases; Severe Acute Respiratory Syndrome; Diabetes Mellitus; Diabetes Mellitus, Type 2
Dipeptidyl peptidase IV inhibitor
Small molecule
Approved
Unknown
Unknown
Brain Diseases; Depressive Disorder, Major; Lymphoma; Neoplasms; Nervous System Diseases; Obesity; Peripheral Nervous System Diseases; Schizophrenia; Cognitive Dysfunction; Dementia; Dermatitis; Dermatitis, Seborrheic; Diabetes Mellitus, Type 2; Fragile X Syndrome; Non-alcoholic Fatty Liver Disease; Respiratory Distress Syndrome; Rosacea; Asthma; Bronchiectasis; Dermatitis, Atopic; Diabetic Nephropathies; Bronchitis, Chronic; Lung Diseases, Obstructive; Psoriasis; Pulmonary Disease, Chronic Obstructive
Phosphodiesterase 4 inhibitor
Small molecule
Approved
Unknown
Unknown
Heart Arrest
Unknown
Small molecule
Approved
Unknown
Unknown
Cardiovascular Diseases; Essential Hypertension; Hypertension
Unknown
Small molecule
Approved
Unknown
Unknown
Alzheimer Disease; Dementia; Lewy Body Disease; Movement Disorders; Multiple System Atrophy; Parkinson Disease; Parkinsonian Disorders; Radionuclide Imaging; Tomography, Emission-Computed, Single-Photon
Diagnostic agent
Small molecule
Approved
OTHER
INHALATION
Asthma; Lung Diseases; Bronchitis, Chronic; Emphysema; Pulmonary Disease, Chronic Obstructive
Beta-2 adrenergic receptor agonist
Small molecule
Approved
Unknown
Unknown
Osteoarthritis, Knee
Unknown
Small molecule
Approved
OTHER
TOPICAL
Lice Infestations
Nicotinic acetylcholine receptor agonist
Small molecule
Approved
CARDIOVASCULAR; OTHER
ORAL
Hypertension; Stroke
Type-1 angiotensin II receptor antagonist
Small molecule
Approved
Unknown
Unknown
Lung Diseases; Asthma; Heart Failure; Pulmonary Disease, Chronic Obstructive; Lung Diseases, Obstructive
Unknown
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER; PEDIATRICS
ORAL
Alcoholism; Bipolar Disorder; Depressive Disorder, Major; Torticollis; Amyotrophic Lateral Sclerosis; Diabetic Neuropathies; Essential Tremor; Migraine Disorders; Neuralgia; Small Fiber Neuropathy; Epilepsy, Tonic-Clonic; Lennox Gastaut Syndrome; Parkinson Disease; Epilepsies, Partial; Epilepsy; Seizures
Glutamate receptor ionotropic AMPA antagonist
Small molecule
Approved
RESPIRATORY
ORAL
Liver Diseases; Sinusitis; Bronchitis, Chronic; Ciliary Motility Disorders; Pulmonary Disease, Chronic Obstructive; Cystic Fibrosis; Respiratory Tract Diseases
Cystic fibrosis transmembrane conductance regulator positive modulator
Small molecule
Approved
GASTROINTESTINAL
ORAL
Breast Neoplasms; Irritable Bowel Syndrome; Diarrhea
Anoctamin-1 blocker
Small molecule
Approved
OTHER; UROLOGY AND KIDNEY
ORAL
Esophageal Achalasia; Kidney Diseases; Liver Diseases; Polycystic Ovary Syndrome; Cerebral Hemorrhage; Heart Failure; Hypertrophy, Left Ventricular; Pain; Prediabetic State; Urinary Bladder, Neurogenic; Cystitis, Interstitial; Kidney Calculi; Polyuria; Urinary Bladder, Overactive; Urinary Incontinence; Urinary Incontinence, Urge
Beta-3 adrenergic receptor agonist
Small molecule
Approved
Unknown
ORAL
Dermatomyositis; Granuloma Annulare; Granulomatous Disease, Chronic; Kidney Diseases; Lupus Erythematosus, Cutaneous; Lupus Erythematosus, Systemic; Myasthenia Gravis; Renal Insufficiency, Chronic; Sarcoidosis; Stevens-Johnson Syndrome; Alopecia Areata; Colitis; Crohn Disease; Down Syndrome; Dry Eye Syndromes; Granuloma, Lethal Midline; Leishmaniasis, Cutaneous; Myocarditis; Myositis; Pneumonia; Pouchitis; Scleroderma, Systemic; Sjogren's Syndrome; Wounds and Injuries; Arthritis, Juvenile; Arthritis, Psoriatic; Arthritis, Rheumatoid; Colitis, Ulcerative; Glioblastoma; Polymyalgia Rheumatica; Psoriasis; Severe Acute Respiratory Syndrome; Spondylitis, Ankylosing; Takayasu Arteritis
Unknown
Small molecule
Approved
CARDIOVASCULAR
ORAL
Breast Neoplasms; Lipid Metabolism Disorders; Adenoma; Alzheimer Disease; Colonic Neoplasms; Non-alcoholic Fatty Liver Disease; Cardiovascular Diseases; Severe Acute Respiratory Syndrome; Dyslipidemias; Hypertriglyceridemia; Pancreatitis
Unknown
Small molecule
Approved
MUSCULOSKELETAL; OTHER
ORAL
Celiac Disease; Kidney Diseases; Paraparesis, Tropical Spastic; Purpura, Thrombocytopenic, Idiopathic; Multiple Sclerosis, Chronic Progressive; Multiple Sclerosis; Multiple Sclerosis, Relapsing-Remitting
Dihydroorotate dehydrogenase inhibitor
Small molecule
Approved
CANCER
ORAL
Primary Myelofibrosis; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Skin Neoplasms; Triple Negative Breast Neoplasms; Basal Cell Nevus Syndrome; Breast Neoplasms; Bronchiolitis Obliterans Syndrome; Carcinoma, Pancreatic Ductal; Chondrosarcoma, Clear Cell; Chondrosarcoma, Mesenchymal; Glioblastoma; Gliosarcoma; Idiopathic Pulmonary Fibrosis; Leukemia, Myeloid, Acute; Medulloblastoma; Meningioma; Multiple Myeloma; Ovarian Neoplasms; Pancreatic Neoplasms; Paraganglioma; Small Cell Lung Carcinoma; Stomach Neoplasms; Carcinoma, Basal Cell; Neoplasms
Smoothened homolog inhibitor
Small molecule
Approved
Unknown
Unknown
Liver Diseases; Lung Diseases; Mycobacterium avium-intracellulare Infection; Leprosy; Tuberculosis, Multidrug-Resistant; Tuberculosis, Pulmonary; Tuberculosis
Unknown
Small molecule
Approved
OTHER
INTRAVENOUS
Prostatic Neoplasms
Diagnostic agent
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
CANCER; OTHER; UROLOGY AND KIDNEY
ORAL
Blast Crisis; Breast Neoplasms; Carcinoma; Endometriosis; Gliosarcoma; Mesothelioma; Neoplasm Metastasis; Stomach Neoplasms; Adrenal Cortex Neoplasms; Biliary Tract Neoplasms; Carcinoid Tumor; Carcinoma, Adenoid Cystic; Carcinoma, Hepatocellular; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Colorectal Neoplasms; Endometrial Neoplasms; Gastrointestinal Stromal Tumors; Glioblastoma; Leukemia, Myeloid, Acute; Liver Neoplasms; Lung Neoplasms; Melanoma; Myelodysplastic Syndromes; Nasopharyngeal Neoplasms; Pancreatic Neoplasms; Paraganglioma; Pheochromocytoma; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Salivary Gland Neoplasms; Sarcoma; Sarcoma, Alveolar Soft Part; Skin Neoplasms; Solitary Fibrous Tumors; Thyroid Neoplasms; Carcinoma, Pancreatic Ductal; Kidney Neoplasms; Carcinoma, Renal Cell; Neoplasms
Vascular endothelial growth factor receptor inhibitor
Small molecule
Approved
Unknown
Unknown
Cardiovascular Diseases; Hyperlipoproteinemia Type II
Unknown
Small molecule
Approved
OTHER
ORAL
Insulin Resistance; Acquired Immunodeficiency Syndrome; HIV Infections; Virus Diseases
Human immunodeficiency virus type 1 integrase inhibitor
Small molecule
Approved
Unknown
Unknown
Cardiovascular Diseases; Kidney Diseases; Liver Diseases; Marijuana Abuse; Substance-Related Disorders; Cocaine-Related Disorders; Opioid-Related Disorders; Peripheral Nervous System Diseases; Tobacco Use Disorder; Obesity
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Myelodysplastic Syndromes; Adenocarcinoma of Lung; Blast Crisis; Carcinoma, Medullary; Carcinoma, Non-Small-Cell Lung; Gastrointestinal Stromal Tumors; Glioblastoma; Leukemia; Leukemia, Myeloid, Acute; Small Cell Lung Carcinoma; Thyroid Neoplasms; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Neoplasms; Precursor Cell Lymphoblastic Leukemia-Lymphoma
Unknown
Small molecule
Approved
OTHER
ORAL
Carcinoma, Non-Small-Cell Lung; Carcinoma, Pancreatic Ductal; Insulin Resistance; Leukemia, Biphenotypic, Acute; Malaria; Pancreatic Neoplasms; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Leukemia, Myeloid, Acute; Neoplasms; Acquired Immunodeficiency Syndrome; Pneumonia, Pneumocystis; Severe Acute Respiratory Syndrome; HIV Infections; Infections
Cytochrome P450 3A inhibitor
Small molecule
Approved
GASTROINTESTINAL; OTHER; UROLOGY AND KIDNEY
ORAL
Bone Neoplasms; Leukemia, Myeloid, Acute; Myelodysplastic Syndromes; Rhabdomyosarcoma; Small Cell Lung Carcinoma; Bile Duct Neoplasms; Biliary Tract Neoplasms; Carcinoma, Adenoid Cystic; Carcinoma, Renal Cell; Cholangiocarcinoma; Digestive System Neoplasms; Fallopian Tube Neoplasms; Glioblastoma; Hemangiosarcoma; Liposarcoma; Macular Degeneration; Melanoma; Meningioma; Osteosarcoma; Ovarian Neoplasms; Pancreatic Neoplasms; Pulmonary Disease, Chronic Obstructive; Rectal Neoplasms; Sarcoma; Stomach Neoplasms; Thyroid Neoplasms; Carcinoma, Hepatocellular; Colonic Neoplasms; Esophageal Neoplasms; Gastrointestinal Stromal Tumors; Colorectal Neoplasms; Neoplasms
Discoidin domain-containing receptor 2 inhibitor
Small molecule
Approved
Unknown
Unknown
Pulmonary Disease, Chronic Obstructive
Unknown