Display Options:
Total: 1496
Small molecule
Approved
OTHER
INTRAVITREAL; OTIC; TOPICAL
Glaucoma; Macular Degeneration; Retinal Diseases; Uveitis, Posterior; Otitis Externa; Dermatitis, Atopic; Dermatitis, Seborrheic; Eye Diseases; Hemorrhoids; Infections; Macular Edema; Melanosis; Psoriasis; Skin Diseases; Uveitis
Glucocorticoid receptor agonist
Small molecule
Approved
OTHER
ORAL
Rhinitis, Allergic, Seasonal
Histamine H1 receptor antagonist
Small molecule
Approved
OTHER
INJECTION; ORAL; RECTAL
Landau-Kleffner Syndrome; Low Back Pain; Rotator Cuff Injuries; Wounds and Injuries; Dementia; Depressive Disorder; Epilepsy, Complex Partial; Pain; Schizophrenia; Seizures; Status Epilepticus; Anxiety; Anxiety Disorders; Cerebral Palsy; Epilepsy; Mental Disorders; Psychomotor Agitation; Stiff-Person Syndrome
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
OTHER
OPHTHALMIC
Leukemia; Eye Infections; Virus Diseases
DNA inhibitor
Small molecule
Approved
OTHER
ORAL
Cardiovascular Diseases
Thiazide-sensitive sodium-chloride cotransporter inhibitor
Small molecule
Approved
DERMATOLOGY; IMMUNE SYSTEM; OTHER; PREGNANCY AND GYNECOLOGY
INJECTION; ORAL; TOPICAL; VAGINAL
Osteomyelitis; Vaginitis; Central Serous Chorioretinopathy; Cholangitis, Sclerosing; Periapical Periodontitis; Appendicitis; Brain Diseases; Carcinoma, Non-Small-Cell Lung; Clostridium Infections; Colitis, Ulcerative; Leukemia, Lymphocytic, Chronic, B-Cell; Lichen Planus, Oral; Malnutrition; Pilonidal Sinus; Rectal Neoplasms; Tuberculosis, Multidrug-Resistant; Uterine Cervical Neoplasms; Abscess; Blepharitis; Candidiasis; Colorectal Neoplasms; Crohn Disease; Diarrhea; Enterocolitis, Pseudomembranous; Fecal Incontinence; Gingivitis; Helicobacter Infections; Hemorrhoids; HIV Infections; Kidney Calculi; Lymphoma, Non-Hodgkin; Mycoses; Pelvic Inflammatory Disease; Periodontitis; Skin Diseases; Trichomonas Vaginitis; Vaginal Discharge; Bacterial Infections; Duodenal Ulcer; Infections; Intraabdominal Infections; Pneumonia; Rosacea; Sepsis; Trichomonas Infections; Uterine Cervicitis; Vaginosis, Bacterial
DNA inhibitor
Small molecule
Approved
OTHER
ORAL
Osteomyelitis; Acne Vulgaris; Bacterial Infections; Eye Infections
Bacterial 70S ribosome inhibitor
Small molecule
Approved
OTHER
ORAL
Osteomyelitis; Pulmonary Disease, Chronic Obstructive; Tourette Syndrome; Anxiety; Sleep Apnea Syndromes; Agoraphobia; Alcohol Drinking; Bipolar Disorder; Brain Injuries; Cocaine-Related Disorders; Depressive Disorder, Major; Low Back Pain; Opioid-Related Disorders; Psychotic Disorders; Stroke; Substance-Related Disorders; Tobacco Use Disorder; Asperger Syndrome; Autistic Disorder; Obsessive-Compulsive Disorder; Pain; Panic Disorder; Phobia, Social; Phobic Disorders; Schizophrenia; Smoking Cessation; Stress Disorders, Post-Traumatic; Tuberculosis
Alanine racemase inhibitor
Small molecule
Approved
OTHER
ORAL
Cataract; Diabetes Mellitus
Sulfonylurea receptor 1, Kir6.2 blocker
Small molecule
Approved
OTHER
INJECTION; ORAL
Aortic Diseases; Rosacea; Craniosynostoses; Inflammation; Hemorrhage
Plasminogen inhibitor
Small molecule
Approved
OTHER
ORAL
Neoplasms, Neuroepithelial; Anemia; beta-Thalassemia; Blast Crisis; Central Nervous System Neoplasms; Chordoma; Crohn Disease; Fallopian Tube Neoplasms; Neoplasms, Germ Cell and Embryonal; Oligodendroglioma; Peritoneal Neoplasms; Adenoma, Islet Cell; Anemia, Aplastic; Brain Neoplasms; Breast Neoplasms, Male; Bronchiectasis; Burkitt Lymphoma; Carcinoma, Neuroendocrine; Carcinoma, Renal Cell; Ganglioneuroblastoma; Graft vs Host Disease; Granuloma, Lethal Midline; Hematologic Diseases; Hematologic Neoplasms; Hemoglobinuria, Paroxysmal; Histiocytosis; Histiocytosis, Langerhans-Cell; Hodgkin Disease; Immunoblastic Lymphadenopathy; Inflammatory Breast Neoplasms; Kidney Neoplasms; Leukemia, Erythroblastic, Acute; Leukemia, Hairy Cell; Leukemia, Large Granular Lymphocytic; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia-Lymphoma, Adult T-Cell; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myelomonocytic, Chronic; Leukemia, Myelomonocytic, Juvenile; Leukemia, Plasma Cell; Liver Neoplasms; Lymphoma, Large-Cell, Anaplastic; Lymphoma, Non-Hodgkin; Lymphoma, T-Cell; Lymphoma, T-Cell, Peripheral; Medulloblastoma; Multiple Sclerosis, Relapsing-Remitting; Myasthenia Gravis; Mycosis Fungoides; Myelodysplastic-Myeloproliferative Diseases; Myeloproliferative Disorders; Neuromyelitis Optica; Opsoclonus-Myoclonus Syndrome; Plasmacytoma; Polycythemia Vera; Polyradiculoneuropathy, Chronic Inflammatory Demyelinating; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Primary Myelofibrosis; Prostatic Neoplasms, Castration-Resistant; Severe Combined Immunodeficiency; Sezary Syndrome; Shwachman-Diamond Syndrome; Stiff-Person Syndrome; Testicular Neoplasms; Thalassemia; Waldenstrom Macroglobulinemia; Wiskott-Aldrich Syndrome; Amyloidosis; Amyloidosis, Familial; Anemia, Sickle Cell; Breast Neoplasms; Colorectal Neoplasms; Leukemia; Leukemia, Myeloid, Acute; Lymphoma; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Melanoma; Myelodysplastic Syndromes; Neuroblastoma; Ovarian Neoplasms; Retinoblastoma; Sarcoma; Sarcoma, Ewing; Smoldering Multiple Myeloma; Carcinoma; Multiple Myeloma; Neoplasms
DNA inhibitor
Small molecule
Approved
OTHER
FOR RX COMPOUNDING; OPHTHALMIC; ORAL; TOPICAL
Osteomyelitis; Erectile Dysfunction; Hepatitis C; Leukemia, Lymphocytic, Chronic, B-Cell; Renal Insufficiency; Bulimia Nervosa; Colorectal Neoplasms; Gastroparesis; Pulmonary Disease, Chronic Obstructive; Stomach Neoplasms; Carcinoma, Non-Small-Cell Lung; Chlamydia Infections; Epidermolysis Bullosa; Gastrointestinal Hemorrhage; Hematemesis; HIV Infections; Pneumonia; Acne Vulgaris; Bacterial Infections; Eye Infections
Bacterial 70S ribosome inhibitor
Small molecule
Approved
OTHER
ORAL
Psoriasis
DNA inhibitor
Small molecule
Approved
OTHER
ORAL
Unknown
Androgen Receptor agonist
Small molecule
Approved
OTHER
ORAL
Osteomyelitis; Bacterial Infections
Bacterial DNA gyrase inhibitor
Protein
Approved
OTHER
INJECTION
Central Nervous System Neoplasms; Melanoma; Brain Neoplasms; Choriocarcinoma; Choroid Plexus Neoplasms; Gestational Trophoblastic Disease; Hydatidiform Mole; Kidney Neoplasms; Leukemia; Lymphoma; Mesenchymoma; Rhabdomyosarcoma; Rhabdomyosarcoma, Alveolar; Rhabdomyosarcoma, Embryonal; Sarcoma; Sarcoma, Ewing; Neoplasms; Wilms Tumor
DNA inhibitor
Small molecule
Approved
OTHER
ORAL
Fanconi Anemia; Malnutrition; Burns; Klinefelter Syndrome; Rotator Cuff Injuries; Neoplasms; Pressure Ulcer; Turner Syndrome
Androgen Receptor agonist
Small molecule
Approved
OTHER
ORAL; TOPICAL; VAGINAL
Dental Caries; Kidney Diseases; Bacteremia; Burns; Graft vs Host Disease; Pneumonia; Stomatitis, Denture; Candidiasis, Oral; HIV Infections; Leukemia; Multiple Myeloma; Myelodysplastic Syndromes; Myeloproliferative Disorders; Stomatitis; Tobacco Use Disorder; Vaginosis, Bacterial; Candidiasis; Infections
Ergosterol sequestering agent
Small molecule
Approved
OTHER
ORAL
Atherosclerosis; Coronary Disease; Death, Sudden, Cardiac; Diabetes Mellitus, Type 2; Hypercholesterolemia; Cardiovascular Diseases; Edema; Heart Failure; Hyperaldosteronism; Hypertension; Liver Cirrhosis; Nephrotic Syndrome; Toxemia
Amiloride-sensitive sodium channel, ENaC blocker
Small molecule
Approved
OTHER
INJECTION; ORAL; TOPICAL
Leishmaniasis, Cutaneous; Aspergillosis, Allergic Bronchopulmonary; Candidiasis, Chronic Mucocutaneous; Candidiasis, Invasive; Fuchs' Endothelial Dystrophy; Intracranial Hypertension; Leukemia, Myeloid, Acute; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Blastomycosis; Candidiasis, Vulvovaginal; Leishmaniasis; Leishmaniasis, Mucocutaneous; Leukemia; Lung Diseases; Multiple Myeloma; Myelodysplastic Syndromes; Myeloproliferative Disorders; Neoplasms; Vaginosis, Bacterial; Aspergillosis; Candidiasis; Cryptococcosis; Histoplasmosis; Infections; Leishmaniasis, Visceral; Meningitis, Cryptococcal; Mucormycosis; Mycoses; Sporotrichosis; Zygomycosis
Ergosterol sequestering agent
Small molecule
Approved
OTHER
ORAL
Unknown
Unknown
Small molecule
Approved
OTHER
INHALATION; INJECTION; INTRAMUSCULAR; INTRAOCULAR; INTRAVENOUS; SUBCUTANEOUS
Depressive Disorder; Diabetes Mellitus; Parathyroid Neoplasms; Skin Neoplasms; Infections; Acute Lung Injury; Appendicitis; Breast Neoplasms; Cognitive Dysfunction; Death, Sudden, Cardiac; Hemoptysis; Hypospadias; Osteoarthritis, Knee; Rotator Cuff Injuries; Shock; Tachycardia, Ventricular; Ventricular Fibrillation; Wounds and Injuries; Bronchiolitis; Carcinoma, Non-Small-Cell Lung; Gastrointestinal Hemorrhage; Heart Failure; Myoma; Neoplasms; Pain; Pulpitis; Rhinitis, Allergic, Perennial; Stomach Neoplasms; Angioedema; Asthma; Bronchial Spasm; Cardiovascular Diseases; Glaucoma; Heart Arrest; Hemorrhage; Hypersensitivity; Lung Diseases, Obstructive; Muscle Cramp; Mydriasis; Nasal Obstruction; Rhinitis, Allergic, Seasonal; Serum Sickness; Shock, Septic; Sinusitis; Urticaria
Adrenergic receptor agonist
Small molecule
Approved
OTHER
ORAL
Osteomyelitis; Tuberculosis, Multidrug-Resistant; Tuberculosis
Enoyl-[acyl-carrier-protein] reductase inhibitor
Small molecule
Approved
OTHER
INJECTION
Cystic Fibrosis; Neoplasms; Pain; Cataract; Malaria; Urinary Tract Infections; Acidosis
Unknown
Small molecule
Approved
OTHER
TOPICAL
Renal Insufficiency, Chronic; Skin Diseases
Glucocorticoid receptor agonist
Small molecule
Approved
OTHER
ORAL
HIV Infections; Tobacco Use Disorder; Dementia; Depressive Disorder; Schizophrenia; Anxiety; Anxiety Disorders; Mental Disorders
GABA-A receptor; anion channel positive allosteric modulator
Protein
Approved
OTHER
INJECTION
Unknown
Insulin receptor agonist
Small molecule
Approved
OTHER
ORAL
Polycythemia Vera; Neoplasms
DNA inhibitor
Small molecule
Approved
OTHER
ORAL
Bacterial Infections
Bacterial dihydropteroate synthase inhibitor
Small molecule
Approved
OTHER
ORAL
Lymphoma, Non-Hodgkin; Glioblastoma; Histiocytosis, Langerhans-Cell; Hodgkin Disease; Leukemia, Lymphoid; Anemia, Refractory; Anemia, Refractory, with Excess of Blasts; Brain Neoplasms; Leukemia; Leukemia, Basophilic, Acute; Leukemia, Biphenotypic, Acute; Leukemia, Erythroblastic, Acute; Leukemia, Megakaryoblastic, Acute; Leukemia, Monocytic, Acute; Leukemia, Myeloid, Acute; Leukemia, Myelomonocytic, Acute; Leukemia, Myelomonocytic, Chronic; Lymphoma; Myelodysplastic Syndromes; Myeloproliferative Disorders; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Precursor T-Cell Lymphoblastic Leukemia-Lymphoma; Neoplasms
DNA inhibitor
Protein
Approved
OTHER
INJECTION
Unknown
Insulin receptor agonist
Small molecule
Approved
OTHER
INJECTION; ORAL
Premature Birth; Diabetes Mellitus; Dyspnea; Edema; Leukemia; Leukemia, Myeloid, Acute; Schizophrenia; Acute Kidney Injury; Acute Lung Injury; Bronchopulmonary Dysplasia; Hypertension, Pregnancy-Induced; Keratosis, Actinic; Nasal Polyps; Neoplasms; Renal Insufficiency, Chronic; Atherosclerosis; Bronchiolitis; Coronary Disease; Diabetes Mellitus, Type 2; Essential Hypertension; Hypercholesterolemia; Kidney Diseases; Lung Diseases; Myocardial Infarction; Pre-Eclampsia; Pulmonary Embolism; Renal Insufficiency; Tachypnea; Warts; Cardiovascular Diseases; Fibrosis; Heart Failure; Hypertension; Liver Cirrhosis; Nephrotic Syndrome; Pulmonary Edema; Syndrome
Sodium-(potassium)-chloride cotransporter 2 inhibitor
Small molecule
Approved
OTHER
ORAL
Inflammatory Bowel Diseases; Leukemia, Biphenotypic, Acute; Osteoarthritis; Tuberculosis; Angina, Stable; Diabetes Mellitus; Essential Hypertension; Fallopian Tube Neoplasms; Hand-Foot Syndrome; Heart Failure; Kidney Calculi; Leishmaniasis; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Myeloid, Acute; Metabolic Syndrome; Multiple Myeloma; Myelodysplastic Syndromes; Myeloproliferative Disorders; Ovarian Neoplasms; Peritoneal Neoplasms; Renal Insufficiency, Chronic; Bipolar Disorder; Cardiovascular Diseases; Colitis, Ulcerative; Diabetes Mellitus, Type 2; Heart Diseases; Hernias, Diaphragmatic, Congenital; Hypertension; Hyperuricemia; Lymphoma, Non-Hodgkin; Obesity; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Sprains and Strains; Tumor Lysis Syndrome; Gout; Leukemia; Lymphoma; Neoplasms; Response Evaluation Criteria in Solid Tumors
Xanthine dehydrogenase inhibitor
Small molecule
Approved
OTHER
ORAL
Diabetes Mellitus; Diabetes Mellitus, Type 2
Sulfonylurea receptor 1, Kir6.2 blocker
Small molecule
Approved
OTHER
INJECTION; ORAL
Anxiety; Dementia; Depressive Disorder; Schizophrenia; Psychotic Disorders
Dopamine D2 receptor antagonist