Display Options:
Total: 6532
Small molecule
Approved
OTHER
BUCCAL; ORAL; SUBLINGUAL
Menopause; Breast Neoplasms; Hypogonadism; Orchitis
Androgen Receptor agonist
Small molecule
Approved
Unknown
Unknown
Hypersensitivity; Pruritus
Unknown
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Tuberculosis, Multidrug-Resistant; Tuberculosis; Bacterial Infections; Eye Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Common Cold; Cough; Headache; Nasal Obstruction
Adrenergic receptor alpha-1 agonist
Small molecule
Approved
OTHER
INJECTION; ORAL
Depressive Disorder; Diabetes Mellitus, Type 2; Obesity; Adenoma, Islet Cell; Hyperinsulinism; Hypertension; Hypoglycemia
Potassium channel, inwardly rectifying, subfamily J, member 11 opener
Small molecule
Approved
Unknown
Unknown
Melanoma; Obesity; Fractures, Bone; Wounds and Injuries; Arrhythmias, Cardiac; Bacteremia; Cellulitis; Clostridium Infections; Gram-Positive Bacterial Infections; Infections; Laryngeal Neoplasms; Osteomyelitis; Prostatic Neoplasms, Castration-Resistant; Skin Diseases; Staphylococcal Infections; Bacterial Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Lung Diseases, Obstructive
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL; VAGINAL
Prostatic Neoplasms, Castration-Resistant; Neoplasms
Estrogen receptor alpha agonist
Small molecule
Approved
Unknown
Unknown
Attention Deficit Disorder with Hyperactivity; Psychotic Disorders
Unknown
Small molecule
Approved
Unknown
Unknown
Diabetes Mellitus, Type 1; Neuralgia; Purpura, Thrombocytopenic, Idiopathic; Asthma; Pulmonary Disease, Chronic Obstructive; Lung Diseases, Obstructive
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Diabetic Cardiomyopathies; Heart Failure; Heart Failure, Diastolic; Cardiomyopathy, Hypertrophic; Cardiovascular Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Breast Carcinoma In Situ; Breast Neoplasms, Male; Carcinoma, Pancreatic Ductal; Castleman Disease; Hematologic Diseases; Immunoglobulin Light-chain Amyloidosis; Lymphoma, B-Cell; Lymphoma, Primary Effusion; Lymphoma, T-Cell, Cutaneous; Melanoma; Thymoma; Urethral Neoplasms; Adrenal Cortex Neoplasms; Astrocytoma; Blast Crisis; Blastic Plasmacytoid Dendritic Cell Neoplasm; Bone Neoplasms; Burkitt Lymphoma; Carcinoma, Adenoid Cystic; Carcinoma, Intraductal, Noninfiltrating; Carcinoma, Non-Small-Cell Lung; Carcinoma, Ovarian Epithelial; Carcinoma, Renal Cell; Carcinosarcoma; Cholangiocarcinoma; Glioblastoma; Glioma; Hemangiosarcoma; Hematologic Neoplasms; Hereditary Breast and Ovarian Cancer Syndrome; Leukemia, Lymphoid; Leukemia, Myeloid, Acute; Leukemia, Plasma Cell; Liposarcoma; Lung Neoplasms; Lymphoma, AIDS-Related; Lymphoma, Large-Cell, Anaplastic; Lymphoma, T-Cell; Mesothelioma; Mouth Neoplasms; Myelodysplastic Syndromes; Nasopharyngeal Neoplasms; Neoplasm Metastasis; Neoplasms, Plasma Cell; Neuroendocrine Tumors; Oligodendroglioma; Optic Nerve Glioma; Pancreatic Neoplasms; Paraganglioma; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Rhabdomyosarcoma; Salivary Gland Neoplasms; Stomach Neoplasms; Thyroid Neoplasms; Uterine Cervical Neoplasms; Wilms Tumor; Brain Neoplasms; Breast Neoplasms; Carcinoma; Carcinoma, Hepatocellular; Choroid Plexus Neoplasms; Desmoid Tumors; Endometrial Neoplasms; Fallopian Tube Neoplasms; Ganglioneuroblastoma; Granuloma, Lethal Midline; Hepatoblastoma; Hodgkin Disease; Immunoblastic Lymphadenopathy; Inflammatory Breast Neoplasms; Kidney Neoplasms; Leiomyosarcoma; Leukemia; Leukemia, Biphenotypic, Acute; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia-Lymphoma, Adult T-Cell; Liver Neoplasms; Lymphohistiocytosis, Hemophagocytic; Lymphoma; Lymphoma, B-Cell, Marginal Zone; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Lymphoma, Non-Hodgkin; Lymphoma, T-Cell, Peripheral; Multiple Myeloma; Neuroblastoma; Neutropenia; Osteosarcoma; Ovarian Neoplasms; Peritoneal Neoplasms; Postoperative Nausea and Vomiting; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Precursor T-Cell Lymphoblastic Leukemia-Lymphoma; Retinoblastoma; Sarcoma; Sarcoma, Ewing; Sarcoma, Kaposi; Small Cell Lung Carcinoma; Triple Negative Breast Neoplasms; Urinary Bladder Neoplasms; Waldenstrom Macroglobulinemia; Neoplasms
Unknown
Small molecule
Approved
IMMUNE SYSTEM; PREGNANCY AND GYNECOLOGY
BUCCAL; INJECTION
Intertrigo; Stomatitis; HIV Infections; Otomycosis; Infections; Mycoses; Pruritus; Tinea; Tinea Pedis
Cytochrome P450 51 inhibitor
Small molecule
Approved
Unknown
Unknown
Multiple Sclerosis; Fever; Tachycardia, Ventricular; Wounds and Injuries
Unknown
Small molecule
Approved
OTHER
INJECTION
Unknown
Unknown
Small molecule
Approved
OTHER
TOPICAL
Skin Diseases
Glucocorticoid receptor agonist
Small molecule
Approved
Unknown
Unknown
Bacterial Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Myopia; Miosis
Unknown
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Gram-Positive Bacterial Infections; Mastitis; Enterobacteriaceae Infections; Staphylococcal Infections; Bacterial Infections
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Bacterial Infections
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
OTHER
ORAL
Neoplasms; Prostatic Neoplasms, Castration-Resistant; Small Cell Lung Carcinoma; Carcinoma, Squamous Cell; Hypertension; Laryngeal Neoplasms; Leukemia, Lymphocytic, Chronic, B-Cell; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Prostatic Neoplasms; Angina, Stable
Osmotic agent
Small molecule
Approved
OTHER
ORAL; TRANSDERMAL
Brain Ischemia; Cocaine-Related Disorders; Dermatitis, Atopic; Hemorrhage; Heroin Dependence; Hypotension, Orthostatic; Orthostatic Intolerance; Anxiety; Back Pain; Brain Injuries; Breast Neoplasms; Child Development Disorders, Pervasive; Diabetic Neuropathies; Low Back Pain; Marijuana Abuse; Musculoskeletal Diseases; Opioid-Related Disorders; Sialorrhea; Stomatitis; Substance-Related Disorders; Attention Deficit Disorder with Hyperactivity; Cardiovascular Diseases; Delirium; Dwarfism, Pituitary; Fecal Incontinence; Genital Neoplasms, Male; Hyperemesis Gravidarum; Neonatal Abstinence Syndrome; Pain; Postoperative Complications; Pregnancy; Scoliosis; Stress Disorders, Post-Traumatic; Glaucoma; Hypertension; Migraine Disorders; Neoplasms; Neuralgia
Adrenergic receptor alpha-2 agonist
Small molecule
Approved
OTHER
TOPICAL
Lice Infestations; Ectoparasitic Infestations
GABA-A receptor negative allosteric modulator
Small molecule
Approved
Unknown
Unknown
Depressive Disorder; Diabetes Mellitus; Cognitive Dysfunction; Heart Failure; Premature Birth; Hernias, Diaphragmatic, Congenital; Parkinson Disease; Shock; Shock, Septic; Cardiovascular Diseases
Unknown
Small molecule
Approved
OTHER
INJECTION
Unknown
Unknown
Small molecule
Approved
IMMUNE SYSTEM; OTHER; PEDIATRICS
ORAL
Astrocytoma; Brain Neoplasms; Central Serous Chorioretinopathy; Cholangitis, Sclerosing; Diarrhea; Glioblastoma; Inflammation; Obesity; Obesity, Morbid; Osteomyelitis; Postoperative Complications; Pregnancy; Prostatic Neoplasms, Castration-Resistant; Tooth Diseases; Asthma; Bacteremia; Buruli Ulcer; Chlamydia Infections; Colitis, Ulcerative; Head and Neck Neoplasms; Lymphoma; Lymphoma, B-Cell, Marginal Zone; Mastitis; Periapical Periodontitis; Periodontal Diseases; Pneumonia, Bacterial; Pseudomyxoma Peritonei; Tuberculosis; Tuberculosis, Pulmonary; Vaginosis, Bacterial; Bronchitis; Bronchitis, Chronic; Cholecystitis; Clostridium Infections; Communicable Diseases; Cystitis, Hemorrhagic; Dyspepsia; Endocarditis; Enterobacteriaceae Infections; Fever; Gastritis; Helicobacter Infections; Hemorrhage; Hepatitis, Alcoholic; Hernia; Hypersensitivity; Influenza, Human; Liver Diseases, Alcoholic; Low Back Pain; Lymphoma, Non-Hodgkin; Malaria, Falciparum; Malnutrition; Neutropenia; Otitis Media, Suppurative; Pain; Periodontitis; Pyelonephritis; Severe Acute Respiratory Syndrome; Stomach Ulcer; Urinary Bladder Neoplasms; Bacterial Infections; Duodenal Ulcer; Gonorrhea; Infections; Otitis Media; Pharyngitis; Pneumonia; Respiratory Tract Infections; Sinusitis; Soft Tissue Infections; Tonsillitis; Urinary Tract Infections
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
Unknown
Unknown
Diabetes Mellitus, Type 2; Diabetes Mellitus
Acyl coenzyme A:cholesterol acyltransferase 1 inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Carnitine O-palmitoyltransferase 1, muscle isoform inhibitor
Small molecule
Approved
Unknown
Unknown
Hypersensitivity
Unknown
Small molecule
Approved
OTHER
ORAL
Glioma; Hookworm Infections; Pruritus; Anemia; Colorectal Neoplasms; Necatoriasis; Helminthiasis
Tubulin inhibitor
Small molecule
Approved
OTHER
INTRAVENOUS; ORAL
Acute Kidney Injury; Alzheimer Disease; Ankle Fractures; Bipolar Disorder; Glycogen Storage Disease Type III; Hypotension, Orthostatic; Malaria; Muscular Dystrophy, Duchenne; Osteoarthritis, Knee; Premature Birth; Rhinitis, Allergic, Seasonal; Uveal Melanoma; Brachial Plexus Neuritis; Bronchopulmonary Dysplasia; Cognitive Dysfunction; Depressive Disorder, Major; Diabetes Mellitus, Type 1; Emphysema; Enuresis; Epilepsies, Partial; Epilepsy; Glioma; Granulomatous Disease, Chronic; Hemorrhage; Hypertension; Kidney Neoplasms; Muscular Diseases; Pancreatitis; Periodontitis; Pre-Eclampsia; Retinopathy of Prematurity; Sinusitis; Spondylarthropathies; Spondylosis; Stomatitis, Aphthous; Sunburn; Temporomandibular Joint Disorders; Tension-Type Headache; Tooth Diseases; Tuberculosis; Wounds and Injuries; Altitude Sickness; Breast Neoplasms; Burns; Causalgia; Cerebral Palsy; Chronic Pain; Fractures, Bone; HIV Infections; Hypospadias; Infections; Low Back Pain; Mucopolysaccharidosis I; Multiple Sclerosis; Neck Pain; Peptic Ulcer; Pulpitis; Respiratory Distress Syndrome; Shock, Septic; Sleep Apnea, Obstructive; Sprains and Strains; Tibial Fractures; Vasculitis; Acute Pain; Arthralgia; Arthritis; Arthritis, Juvenile; Arthritis, Rheumatoid; Back Pain; Cardiovascular Diseases; Common Cold; Ductus Arteriosus, Patent; Dysmenorrhea; Fever; Headache; Influenza, Human; Migraine Disorders; Muscle Cramp; Myalgia; Osteoarthritis; Pain; Pharyngitis; Rheumatic Diseases; Toothache; Vaginitis
Cyclooxygenase inhibitor
Small molecule
Approved
OTHER
INJECTION
Atrophic Vaginitis
Androgen Receptor agonist