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Total: 6532
Small molecule
Approved
OTHER
ORAL
Unknown
Unknown
Small molecule
Approved
EMERGENCY MEDICINE; GASTROINTESTINAL; OTHER
INJECTION; ORAL
Brain Diseases; Brain Injuries; Dyspnea; Lecithin Cholesterol Acyltransferase Deficiency; Neuralgia; Opioid-Related Disorders; Pruritus; Small Cell Lung Carcinoma; Amphetamine-Related Disorders; Breast Neoplasms; Cholecystitis; Cocaine-Related Disorders; Dementia; Gastroparesis; Glioma; Hallucinations; Lymphoma, Follicular; Lymphoma, Non-Hodgkin; Obsessive-Compulsive Disorder; Pancreatic Neoplasms; Sarcoma; Tobacco Use Disorder; Tonsillitis; Alcoholism; Gastroenteritis; Genital Neoplasms, Female; HIV Infections; Hypotension; Irritable Bowel Syndrome; Pain; Schizophrenia; Syncope; Uterine Cervical Neoplasms; Vomiting; Nausea; Neoplasms; Postoperative Nausea and Vomiting
Serotonin 3a (5-HT3a) receptor antagonist
Small molecule
Approved
OTHER
ORAL
Amyotrophic Lateral Sclerosis; Osteomyelitis; Bacterial Infections
DNA gyrase inhibitor
Small molecule
Approved
IMMUNE SYSTEM; OTHER; RESPIRATORY
ORAL
Anovulation; Depressive Disorder, Major; HIV Infections; Neoplasm Metastasis; Neoplasms; Osteomyelitis; Parkinson Disease; Prostatic Neoplasms, Castration-Resistant; Venous Thromboembolism; Buruli Ulcer; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Cystic Fibrosis; Disorders of Excessive Somnolence; Idiopathic Hypersomnia; Leukemia, Lymphocytic, Chronic, B-Cell; Lung Diseases; Lymphoma; Lymphoma, B-Cell, Marginal Zone; Narcolepsy; Periodontitis; Pseudomyxoma Peritonei; Toxoplasmosis, Cerebral; Asthma; Bronchiolitis Obliterans; Bronchopulmonary Dysplasia; Crohn Disease; Gastritis; Heart Diseases; Helicobacter Infections; Hemorrhage; Lymphoma, Non-Hodgkin; Multiple Myeloma; Mycobacterium avium-intracellulare Infection; Pneumonia, Bacterial; Sepsis; Shock, Septic; Stomach Neoplasms; Stomach Ulcer; Tuberculosis; Bacterial Infections; Bronchitis, Chronic; Duodenal Ulcer; Infections; Maxillary Sinusitis; Otitis Media; Pharyngitis; Pneumonia; Sinusitis; Tonsillitis
Bacterial 70S ribosome inhibitor
Small molecule
Approved
OTHER
INJECTION
Anxiety; Dental Anxiety; Disorders of Excessive Somnolence; Fragile X Syndrome; Idiopathic Hypersomnia; Narcolepsy; Parkinson Disease; Sleep Initiation and Maintenance Disorders; Alcoholism; Obsessive-Compulsive Disorder; Substance-Related Disorders
GABA-A receptor; anion channel allosteric antagonist
Small molecule
Approved
Unknown
Unknown
IgA Vasculitis; Lecithin Cholesterol Acyltransferase Deficiency; Nephritis, Hereditary; Kidney Diseases; Diabetes Mellitus; Hypertension; Renal Insufficiency; Stroke
Angiotensin-converting enzyme inhibitor
Small molecule
Approved
EYE; IMMUNE SYSTEM; OTHER
INJECTION; OPHTHALMIC; ORAL
Anemia, Sickle Cell; Graves Ophthalmopathy; Hemorrhagic Fever, Ebola; Immune System Diseases; Obesity; Osteomyelitis; Respiratory Distress Syndrome; Sepsis; Toxoplasmosis, Cerebral; Communicable Diseases; Crohn Disease; Dysentery, Bacillary; Eye Diseases; Gastrointestinal Hemorrhage; Gastroparesis; Multiple Sclerosis; Neoplasms; Obsessive-Compulsive Disorder; Onchocerciasis; Periodontitis; Respiratory Syncytial Virus Infections; Sarcoidosis; Tuberculosis; Virus Diseases; Whooping Cough; Abdominal Pain; Acne Vulgaris; Arthritis, Reactive; Asthma; Blepharitis; Bronchial Diseases; Bronchiectasis; Bronchiolitis Obliterans; Bronchitis; Bronchopulmonary Dysplasia; Cardiovascular Diseases; Chlamydia Infections; Chronic Periodontitis; Conjunctivitis, Inclusion; Coronary Disease; Coronavirus Infections; Cough; Diarrhea; Digestive System Diseases; Fever; Gonorrhea; Heart Diseases; Inflammation; Lung Diseases; Malaria; Malaria, Falciparum; Malnutrition; Maxillary Sinusitis; Mycobacterium avium-intracellulare Infection; Mycobacterium Infections; Mycoses; Myocardial Infarction; Neonatal Sepsis; Otitis Media, Suppurative; Pneumonia, Viral; Pregnancy; Premature Birth; Respiratory Insufficiency; Severe Acute Respiratory Syndrome; Spotted Fever Group Rickettsiosis; Syphilis; Vomiting; Yaws; Bacterial Infections; Bronchitis, Chronic; Conjunctivitis, Bacterial; Cystic Fibrosis; Eye Infections; HIV Infections; Infections; Otitis Media; Pelvic Inflammatory Disease; Pharyngitis; Pneumonia; Pulmonary Disease, Chronic Obstructive; Sinusitis; Tonsillitis; Urethritis; Uterine Cervicitis
Bacterial 70S ribosome inhibitor
Small molecule
Approved
OTHER
TOPICAL
Psoriasis; Candidiasis; Eczema; Tinea Pedis; Skin Diseases
Glucocorticoid receptor agonist
Small molecule
Approved
OTHER
INJECTION
Anemia, Aplastic; Anemia, Sickle Cell; Kidney Neoplasms; Lymphoma, B-Cell; Bronchiolitis Obliterans Syndrome; Leukemia; Lymphoma; Graft vs Host Disease; Leukemia, Lymphocytic, Chronic, B-Cell; Anemia; Leukemia, Hairy Cell; Neoplasms
Adenosine deaminase inhibitor
Small molecule
Approved
Unknown
Unknown
Low Back Pain; Osteoporosis; Breast Neoplasms; Multiple Myeloma; Bone Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Pain
Unknown
Small molecule
Approved
Unknown
Unknown
Lupus Erythematosus, Systemic; Nephritis, Hereditary; Atherosclerosis; Coronary Disease; Diabetes Mellitus; Diabetes Mellitus, Type 2; Hypercholesterolemia; Hypertension; Cardiovascular Diseases
Unknown
Small molecule
Approved
OTHER
ORAL
Hepatolenticular Degeneration; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Myelodysplastic Syndromes; Asperger Syndrome; Autistic Disorder
Lead chelating agent
Small molecule
Approved
Unknown
Unknown
Metabolic Syndrome; Arthritis, Rheumatoid; Kidney Diseases; Lupus Erythematosus, Systemic; Severe Acute Respiratory Syndrome; Albuminuria; Atherosclerosis; Atrial Fibrillation; Atrial Flutter; Diabetes Mellitus, Type 1; Diabetes Mellitus, Type 2; Diabetic Nephropathies; Glomerulonephritis; Glucose Intolerance; Heart Diseases; Hypercholesterolemia; Metabolic Diseases; Myocardial Ischemia; Renal Insufficiency, Chronic; Stuttering; Cardiovascular Diseases; Coronary Artery Disease; Diabetes Mellitus; Heart Failure; Hypertension; Myocardial Infarction; Stroke
Angiotensin-converting enzyme inhibitor
Small molecule
Approved
CARDIOVASCULAR; OTHER
ORAL
Alopecia Areata; Arthritis, Rheumatoid; Choroideremia; Chronic Pain; Cystic Fibrosis; Dental Caries; Dental Pulp Exposure; Endotoxemia; Epilepsy; Heart Failure; Hemangioma; Hemangioma, Cavernous, Central Nervous System; Hepatitis B, Chronic; HIV Infections; Leukemia, Lymphocytic, Chronic, B-Cell; Lupus Erythematosus, Systemic; Lymphoma; Neoplasms; Obesity; Ovarian Neoplasms; Pancreatitis, Chronic; Sleep Wake Disorders; Vascular Diseases; Anemia, Sickle Cell; Atrial Fibrillation; Bipolar Disorder; Breast Neoplasms; Carcinoma, Hepatocellular; Carcinoma, Non-Small-Cell Lung; Cardiomyopathy, Dilated; Carotid Artery Diseases; Cerebral Hemorrhage; Diabetes Mellitus, Type 1; Hypertension, Pulmonary; Intermittent Claudication; Leiomyoma; Lung Neoplasms; Migraine Disorders; Mucositis; Multiple Myeloma; Pancreatic Neoplasms; Pancreatitis; Parkinson Disease; Periodontitis; Peripheral Arterial Disease; Prediabetic State; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Rectal Neoplasms; Sepsis; Shock, Septic; Sinusitis; Small Cell Lung Carcinoma; Smith-Lemli-Opitz Syndrome; Smoking Cessation; Urinary Bladder Neoplasms; Uveitis; Vitiligo; Waldenstrom Macroglobulinemia; Acute Coronary Syndrome; Alzheimer Disease; Aortic Valve Stenosis; Asthma; Atherosclerosis; Cholangitis, Sclerosing; Colorectal Neoplasms; Depressive Disorder, Treatment-Resistant; Diabetes Mellitus; Diabetes Mellitus, Type 2; Diabetic Nephropathies; Diabetic Retinopathy; Essential Hypertension; Graves Ophthalmopathy; Hyperlipidemia, Familial Combined; Hypertension; Hypertension, Portal; Hypertriglyceridemia; Inflammation; Influenza, Human; Intestinal Neoplasms; Ischemic Stroke; Lipid Metabolism Disorders; Liver Cirrhosis; Multiple Sclerosis; Multiple Sclerosis, Chronic Progressive; Multiple Sclerosis, Relapsing-Remitting; Myocardial Ischemia; Noonan Syndrome; Optic Neuritis; Pneumonia; Polycystic Ovary Syndrome; Pulmonary Disease, Chronic Obstructive; Renal Insufficiency, Chronic; Severe Acute Respiratory Syndrome; Stomach Neoplasms; Subarachnoid Hemorrhage; Cardiovascular Diseases; Coronary Artery Disease; Coronary Disease; Dyslipidemias; Hypercholesterolemia; Hyperlipidemias; Hyperlipoproteinemia Type II; Myocardial Infarction; Stroke
HMG-CoA reductase inhibitor
Small molecule
Approved
OTHER
ORAL
Osteomyelitis; Bacterial Infections
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
Unknown
Unknown
Acute Kidney Injury; Arthritis, Rheumatoid; HIV Infections; Leukemia; Pneumonia; Breast Neoplasms; Carcinoma; Cardiomyopathies; Fibrosis; Lupus Erythematosus, Systemic; Mucocutaneous Lymph Node Syndrome; Progeria; Tuberculosis; Tuberculosis, Pulmonary; Carcinoma, Hepatocellular; Diabetes Mellitus; Heart Failure; Hypercholesterolemia; Hyperlipidemia, Familial Combined; Hyperlipidemias; Hyperlipoproteinemia Type III; Hypertension; Ischemic Stroke; Lipid Metabolism Disorders; Multiple Sclerosis, Relapsing-Remitting; Myocardial Infarction; Myocardial Ischemia; Polycystic Kidney, Autosomal Dominant; Pre-Eclampsia; Renal Insufficiency, Chronic; Cardiovascular Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Acute Coronary Syndrome; Oligodendroglioma; Renal Insufficiency, Chronic; Rhabdomyosarcoma; Calcinosis; Dermatomyositis; Glioma; Head and Neck Neoplasms; Hearing Loss; Mesothelioma; Myositis; Severe Acute Respiratory Syndrome; Hepatoblastoma; Medulloblastoma; Ototoxicity
Unknown
Small molecule
Approved
Unknown
Unknown
Coronary Disease; Familial Primary Pulmonary Hypertension; Hemorrhage; Lecithin Cholesterol Acyltransferase Deficiency; Breast Neoplasms; Atrial Fibrillation; Hypertension; Cardiovascular Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
INJECTION
Astrocytoma; Glioblastoma; Glioma; Multiple Sclerosis, Chronic Progressive; Paraganglioma; Central Nervous System Diseases
Diagnostic agent
Small molecule
Approved
Unknown
Unknown
Anovulation; Fibromyalgia; Idiopathic Pulmonary Fibrosis; Myocardial Infarction; Tinnitus; Agoraphobia; Alcoholism; Anxiety; Anxiety Disorders; Arthritis, Rheumatoid; Bipolar Disorder; Dementia; Diabetes Mellitus, Type 2; Hepatitis C, Chronic; Neuralgia; Obsessive-Compulsive Disorder; Panic Disorder; Parkinson Disease; Phobia, Social; Premature Ejaculation; Schizophrenia; Stress Disorders, Post-Traumatic; Depressive Disorder; Depressive Disorder, Major
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Bacterial DNA gyrase inhibitor
Small molecule
Approved
IMMUNE SYSTEM; OTHER
INJECTION; ORAL
Alzheimer Disease; Amyotrophic Lateral Sclerosis; Anti-Neutrophil Cytoplasmic Antibody-Associated Vasculitis; Asthma; Bacterial Infections; Cachexia; Celiac Disease; Cystic Fibrosis; Diabetic Foot; Erectile Dysfunction; Esophageal Neoplasms; Glioblastoma; Heart Failure; Hepatitis B, Chronic; Hepatitis C, Chronic; Infections; Inflammatory Bowel Diseases; Lymphoma; Lymphoma, Non-Hodgkin; Malaria; Melanoma; Multiple Myeloma; Muscular Atrophy, Spinal; Myelodysplastic Syndromes; Neoplasm Metastasis; Neuralgia; Obesity; Pain; Polycystic Ovary Syndrome; Primary Myelofibrosis; Pulmonary Disease, Chronic Obstructive; Renal Insufficiency, Chronic; Respiratory Syncytial Virus Infections; Severe Acute Respiratory Syndrome; Sporotrichosis; Thrombosis; Burns; Carcinoma, Basal Cell; Carcinoma, Non-Small-Cell Lung; Coccidioidomycosis; Crohn Disease; Hematologic Diseases; Leukemia, Myeloid, Acute; Lung Neoplasms; Meningitis, Cryptococcal; Mycetoma; Opioid-Related Disorders; Ovarian Neoplasms; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Sinusitis; Skin Neoplasms; Tinea Pedis; Tinea Versicolor; Aspergillosis, Allergic Bronchopulmonary; Bronchiectasis; Cryptococcosis; Histoplasmosis; Neoplasms; Aspergillosis; Blastomycosis; Candidiasis; Lung Diseases; Mycoses; Onychomycosis
Cytochrome P450 51 inhibitor
Small molecule
Approved
OTHER
ORAL
Osteomyelitis; Lung Diseases; Tuberculosis, Pulmonary; Crohn Disease; Infections; Mycobacterium Infections; Mycoses; HIV Infections; Mycobacterium avium-intracellulare Infection; Tuberculosis
Bacterial DNA-directed RNA polymerase inhibitor
Small molecule
Approved
Unknown
Unknown
Arrhythmias, Cardiac; Atrial Fibrillation; Death, Sudden, Cardiac; Heart Diseases; Heart Failure; Myocardial Infarction; Tachycardia, Ventricular; Ventricular Fibrillation; Cardiovascular Diseases
Unknown
Small molecule
Approved
OTHER
TOPICAL
Prostatic Neoplasms, Castration-Resistant; Neoplasms
Insulin-like growth factor I receptor inhibitor
Small molecule
Approved
Unknown
Unknown
Melanosis
Sunscreen
Small molecule
Approved
Unknown
Unknown
Sleep Apnea, Central; Amenorrhea; Hemorrhage; Infertility; Polycystic Ovary Syndrome
Progesterone receptor agonist
Small molecule
Approved
Unknown
Unknown
Asthma; Eye Manifestations; Lung Diseases, Obstructive; Nasal Obstruction
Unknown
Small molecule
Approved
Unknown
Unknown
Obesity; Pain; Migraine with Aura; Migraine without Aura; Migraine Disorders
Serotonin 1b (5-HT1b) receptor agonist
Small molecule
Approved
Unknown
Unknown
Cardiovascular Diseases
Unknown
Small molecule
Approved
IMMUNE SYSTEM; OTHER
TOPICAL
Hepatitis B, Chronic; Mycoses; Colitis, Ulcerative; Crohn Disease; Tinea Pedis; Onychomycosis; Tinea
Squalene monooxygenase inhibitor
Small molecule
Approved
Unknown
Unknown
Melanosis; Skin Neoplasms; Sunburn
Unknown
Small molecule
Approved
Unknown
Unknown
Lecithin Cholesterol Acyltransferase Deficiency; Essential Hypertension; Proteinuria; Angina Pectoris; Angina Pectoris, Variant; Angina, Stable; Coronary Artery Disease; Diabetes Mellitus; Heart Failure; Hypercholesterolemia; Hyperlipidemias; Hyperlipoproteinemia Type II; Hypertension; Myocardial Infarction; Osteoarthritis; Stroke
Voltage-gated L-type calcium channel blocker