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Therapeutic Area
CANCER (51)
CARDIOVASCULAR (45)
DENTISTRY (2)
DERMATOLOGY (31)
DIABETES DRUGS & ENDOCRINOLOGY (61)
EMERGENCY MEDICINE (3)
ENT (5)
EYE (23)
GASTROINTESTINAL (29)
HEMATOLOGY (23)
MUSCULOSKELETAL (28)
NEUROLOGY DRUGS & NERVOUS SYSTEM (50)
PEDIATRICS (27)
PHARMACOLOGY (8)
PREGNANCY AND GYNECOLOGY (30)
RESPIRATORY (42)
RHEUMATOLOGY (19)
OTHER (1482)
Therapeutic Indication
Adverse Reaction (System Organ Classification)
Mechanism of Action
Primary Target
Target Level
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Level 5
Level 6
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Display Options:
Drug type
Therapeutic Area
Route of administration
Mechanism of Action
Indication
Status
Total:
10647
ARQ-736
1
Small molecule
Investigational
Unknown
Unknown
Neoplasms
Serine/threonine-protein kinase B-raf inhibitor
ARQ-736
×
Maximum Phase:
1
First Approval:
None
UNII:
Y2H4S74Y8U
Molecule Type:
Small molecule
Molecular Formula:
Molecular Weight:
AlogP:
PSA:
HBD:
HBA:
#RotB:
Source:
LS 11
1
Unknown
Investigational
Unknown
Unknown
Unknown
Unknown
LS 11
×
Maximum Phase:
1
First Approval:
None
UNII:
Molecule Type:
Unknown
Molecular Formula:
Molecular Weight:
AlogP:
PSA:
HBD:
HBA:
#RotB:
Source:
BUTANE
1
Small molecule
Investigational
Unknown
Unknown
Essential Hypertension
Unknown
BUTANE
×
Maximum Phase:
1
First Approval:
None
UNII:
6LV4FOR43R
Molecule Type:
Small molecule
Molecular Formula:
C4H10
Molecular Weight:
58.12
AlogP:
1.81
PSA:
0.0
HBD:
0.0
HBA:
#RotB:
1.0
Source:
ATU027
1
Unknown
Investigational
Unknown
Unknown
Unknown
Unknown
ATU027
×
Maximum Phase:
1
First Approval:
None
UNII:
Molecule Type:
Unknown
Molecular Formula:
Molecular Weight:
AlogP:
PSA:
HBD:
HBA:
#RotB:
Source:
BENZOYLPHENYLUREA
1
Small molecule
Investigational
Unknown
Unknown
Neoplasms
Unknown
BENZOYLPHENYLUREA
×
Maximum Phase:
1
First Approval:
None
UNII:
None
Molecule Type:
Small molecule
Molecular Formula:
C14H12N2O2
Molecular Weight:
240.26
AlogP:
2.41
PSA:
63.4
HBD:
1.0
HBA:
#RotB:
2.0
Source:
IMD-2560
1
Small molecule
Investigational
Unknown
Unknown
Unknown
Inhibitor of nuclear factor kappa B kinase beta subunit inhibitor
IMD-2560
×
Maximum Phase:
1
First Approval:
None
UNII:
None
Molecule Type:
Small molecule
Molecular Formula:
Molecular Weight:
AlogP:
PSA:
HBD:
HBA:
#RotB:
Source:
GS-441524
1
Small molecule
Investigational
Unknown
Unknown
Severe Acute Respiratory Syndrome
Unknown
GS-441524
×
Maximum Phase:
1
First Approval:
None
UNII:
1BQK176DT6
Molecule Type:
Small molecule
Molecular Formula:
C12H13N5O4
Molecular Weight:
291.27
AlogP:
-1.86
PSA:
149.92
HBD:
4.0
HBA:
#RotB:
2.0
Source:
ANX-042
1
Protein
Investigational
Unknown
Unknown
Unknown
Unknown
ANX-042
×
Maximum Phase:
1
First Approval:
None
UNII:
ZV0MCR055T
Molecule Type:
Protein
Molecular Formula:
C189H312N58O53S4
Molecular Weight:
4373.2
AlogP:
None
PSA:
None
HBD:
None
HBA:
#RotB:
None
Source:
MINT-1526A
1
Unknown
Investigational
Unknown
Unknown
Neoplasms
Unknown
MINT-1526A
×
Maximum Phase:
1
First Approval:
None
UNII:
H6BAM62K4Q
Molecule Type:
Unknown
Molecular Formula:
Molecular Weight:
AlogP:
PSA:
HBD:
HBA:
#RotB:
Source:
PALOMID-529
1
Small molecule
Investigational
Unknown
Unknown
Macular Degeneration
Serine/threonine-protein kinase mTOR inhibitor
PALOMID-529
×
Maximum Phase:
1
First Approval:
None
UNII:
XV9409EWG4
Molecule Type:
Small molecule
Molecular Formula:
C24H22O6
Molecular Weight:
406.43
AlogP:
4.6
PSA:
78.13
HBD:
1.0
HBA:
#RotB:
6.0
Source:
PF-03814735
1
Small molecule
Investigational
Unknown
Unknown
Neoplasms
Serine/threonine-protein kinase Aurora-A inhibitor
PF-03814735
×
Maximum Phase:
1
First Approval:
None
UNII:
6V5T4O5758
Molecule Type:
Small molecule
Molecular Formula:
Molecular Weight:
AlogP:
PSA:
HBD:
HBA:
#RotB:
Source:
LU AF-82422
1
Unknown
Investigational
Unknown
Unknown
Parkinson Disease
Unknown
LU AF-82422
×
Maximum Phase:
1
First Approval:
None
UNII:
52V6AS6U0A
Molecule Type:
Unknown
Molecular Formula:
Molecular Weight:
AlogP:
PSA:
HBD:
HBA:
#RotB:
Source:
HUA33
1
Antibody
Investigational
Unknown
Unknown
Colorectal Neoplasms
Cell surface A33 antigen binding agent
HUA33
×
Maximum Phase:
1
First Approval:
None
UNII:
None
Molecule Type:
Antibody
Molecular Formula:
Molecular Weight:
AlogP:
PSA:
HBD:
HBA:
#RotB:
Source:
INULINE
1
Small molecule
Investigational
Unknown
Unknown
Unknown
Unknown
INULINE
×
Maximum Phase:
1
First Approval:
None
UNII:
None
Molecule Type:
Small molecule
Molecular Formula:
C32H46N2O8
Molecular Weight:
586.73
AlogP:
1.72
PSA:
132.94
HBD:
3.0
HBA:
#RotB:
8.0
Source:
LY-2780301
1
Small molecule
Investigational
Unknown
Unknown
Lymphoma; Neoplasm Metastasis
Ribosomal protein S6 kinase (P70S6K) inhibitor
LY-2780301
×
Maximum Phase:
1
First Approval:
None
UNII:
None
Molecule Type:
Small molecule
Molecular Formula:
Molecular Weight:
AlogP:
PSA:
HBD:
HBA:
#RotB:
Source:
CHF4227
1
Small molecule
Investigational
Unknown
Unknown
Unknown
Estrogen receptor modulator
CHF4227
×
Maximum Phase:
1
First Approval:
None
UNII:
1O98089Q9M
Molecule Type:
Small molecule
Molecular Formula:
C30H33NO4
Molecular Weight:
471.6
AlogP:
5.81
PSA:
51.16
HBD:
1.0
HBA:
#RotB:
8.0
Source:
AZD-9977
1
Small molecule
Investigational
Unknown
Unknown
Cardiovascular Diseases; Heart Failure; Kidney Diseases
Mineralocorticoid receptor modulator
AZD-9977
×
Maximum Phase:
1
First Approval:
None
UNII:
6C9UKZ0CYE
Molecule Type:
Small molecule
Molecular Formula:
C20H18FN3O5
Molecular Weight:
399.38
AlogP:
1.7
PSA:
96.97
HBD:
2.0
HBA:
#RotB:
3.0
Source:
IPI-493
1
Unknown
Investigational
Unknown
Unknown
Unknown
Unknown
IPI-493
×
Maximum Phase:
1
First Approval:
None
UNII:
Molecule Type:
Unknown
Molecular Formula:
Molecular Weight:
AlogP:
PSA:
HBD:
HBA:
#RotB:
Source:
MBX-400
1
Small molecule
Investigational
Unknown
Unknown
Unknown
Unknown
MBX-400
×
Maximum Phase:
1
First Approval:
None
UNII:
Molecule Type:
Small molecule
Molecular Formula:
Molecular Weight:
AlogP:
PSA:
HBD:
HBA:
#RotB:
Source:
MBC-11
1
Small molecule
Investigational
Unknown
Unknown
Neoplasm Metastasis
Unknown
MBC-11
×
Maximum Phase:
1
First Approval:
None
UNII:
None
Molecule Type:
Small molecule
Molecular Formula:
C11H20N3O14P3
Molecular Weight:
511.21
AlogP:
-2.39
PSA:
281.42
HBD:
8.0
HBA:
#RotB:
8.0
Source:
PF-03732010
1
Antibody
Investigational
Unknown
Unknown
Neoplasms
Cadherin-3 inhibitor
PF-03732010
×
Maximum Phase:
1
First Approval:
None
UNII:
LPW79O1J5Z
Molecule Type:
Antibody
Molecular Formula:
Molecular Weight:
AlogP:
PSA:
HBD:
HBA:
#RotB:
Source:
MSC2499550A
1
Small molecule
Investigational
Unknown
Unknown
Unknown
Unknown
MSC2499550A
×
Maximum Phase:
1
First Approval:
None
UNII:
Molecule Type:
Small molecule
Molecular Formula:
Molecular Weight:
AlogP:
PSA:
HBD:
HBA:
#RotB:
Source:
AV-380
1
Unknown
Investigational
Unknown
Unknown
Cachexia
Unknown
AV-380
×
Maximum Phase:
1
First Approval:
None
UNII:
None
Molecule Type:
Unknown
Molecular Formula:
Molecular Weight:
AlogP:
PSA:
HBD:
HBA:
#RotB:
Source:
PF-00562271
1
Small molecule
Investigational
Unknown
Unknown
Unknown
Focal adhesion kinase 1 inhibitor
PF-00562271
×
Maximum Phase:
1
First Approval:
None
UNII:
K5BX8ZA7UF
Molecule Type:
Small molecule
Molecular Formula:
C21H20F3N7O3S
Molecular Weight:
507.5
AlogP:
3.14
PSA:
129.21
HBD:
3.0
HBA:
#RotB:
7.0
Source:
PHI-101
1
Small molecule
Investigational
Unknown
Unknown
Leukemia, Myeloid, Acute
Unknown
PHI-101
×
Maximum Phase:
1
First Approval:
None
UNII:
None
Molecule Type:
Small molecule
Molecular Formula:
C19H19FN4O2S
Molecular Weight:
386.45
AlogP:
2.26
PSA:
96.25
HBD:
4.0
HBA:
#RotB:
3.0
Source:
ETHASELEN
1
Small molecule
Investigational
Unknown
Unknown
Carcinoma, Non-Small-Cell Lung
Unknown
ETHASELEN
×
Maximum Phase:
1
First Approval:
None
UNII:
4Q2EZS1IWG
Molecule Type:
Small molecule
Molecular Formula:
C16H12N2O2Se2
Molecular Weight:
422.2
AlogP:
None
PSA:
None
HBD:
None
HBA:
#RotB:
None
Source:
ERAGIDOMIDE
1
Unknown
Investigational
Unknown
Unknown
Leukemia, Myeloid, Acute
Unknown
ERAGIDOMIDE
×
Maximum Phase:
1
First Approval:
None
UNII:
None
Molecule Type:
Unknown
Molecular Formula:
Molecular Weight:
AlogP:
PSA:
HBD:
HBA:
#RotB:
Source:
LEXANERSEN
1
Oligonucleotide
Investigational
Unknown
Unknown
Huntington Disease
Unknown
LEXANERSEN
×
Maximum Phase:
1
First Approval:
None
UNII:
None
Molecule Type:
Oligonucleotide
Molecular Formula:
Molecular Weight:
AlogP:
PSA:
HBD:
HBA:
#RotB:
Source:
DAROVASERTIB
1
Small molecule
Investigational
Unknown
Unknown
Unknown
Unknown
DAROVASERTIB
×
Maximum Phase:
1
First Approval:
None
UNII:
E0YF0M8O09
Molecule Type:
Small molecule
Molecular Formula:
C22H23F3N8O
Molecular Weight:
472.48
AlogP:
3.1
PSA:
135.94
HBD:
3.0
HBA:
#RotB:
4.0
Source:
HUPAM4
1
Antibody
Investigational
Unknown
Unknown
Unknown
Mucin-1 binding agent
HUPAM4
×
Maximum Phase:
1
First Approval:
None
UNII:
None
Molecule Type:
Antibody
Molecular Formula:
Molecular Weight:
AlogP:
PSA:
HBD:
HBA:
#RotB:
Source:
SGN-CD33A
1
Antibody
Investigational
Unknown
Unknown
Unknown
Unknown
SGN-CD33A
×
Maximum Phase:
1
First Approval:
None
UNII:
Molecule Type:
Antibody
Molecular Formula:
Molecular Weight:
AlogP:
PSA:
HBD:
HBA:
#RotB:
Source:
ASTX-660
1
Small molecule
Investigational
Unknown
Unknown
Leukemia, Myeloid, Acute; Lymphoma
Unknown
ASTX-660
×
Maximum Phase:
1
First Approval:
None
UNII:
2LHZ9ZC3YO
Molecule Type:
Small molecule
Molecular Formula:
C30H42FN5O3
Molecular Weight:
539.7
AlogP:
2.31
PSA:
81.17
HBD:
2.0
HBA:
#RotB:
7.0
Source:
MONEPANTEL
1
Small molecule
Investigational
Unknown
Unknown
Motor Neuron Disease
Unknown
MONEPANTEL
×
Maximum Phase:
1
First Approval:
None
UNII:
82MA79VJ33
Molecule Type:
Small molecule
Molecular Formula:
C20H13F6N3O2S
Molecular Weight:
473.4
AlogP:
5.28
PSA:
85.91
HBD:
1.0
HBA:
#RotB:
6.0
Source:
DI-LEU16-IL2
1
Unknown
Investigational
Unknown
Unknown
Lymphoma, Follicular
Unknown
DI-LEU16-IL2
×
Maximum Phase:
1
First Approval:
None
UNII:
None
Molecule Type:
Unknown
Molecular Formula:
Molecular Weight:
AlogP:
PSA:
HBD:
HBA:
#RotB:
Source:
AG-24322
1
Small molecule
Investigational
Unknown
Unknown
Lymphoma, Non-Hodgkin
Cyclin-dependent kinase 1 inhibitor
AG-24322
×
Maximum Phase:
1
First Approval:
None
UNII:
926F8X7TNO
Molecule Type:
Small molecule
Molecular Formula:
C23H20F2N6
Molecular Weight:
418.45
AlogP:
2.95
PSA:
73.7
HBD:
3.0
HBA:
#RotB:
4.0
Source:
1
2
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Compound Properties
Molecular Formula
Molecular Weight
ALogP
PSA