Display Options:
Total: 10647
Small molecule
Approved
OTHER
ORAL
Infections; Rhinitis, Allergic, Seasonal; Postoperative Nausea and Vomiting
Histamine H1 receptor antagonist
Small molecule
Approved
Unknown
Unknown
Alcoholism; Amblyopia; Amyotrophic Lateral Sclerosis; Anemia; Arthritis, Rheumatoid; Chronic Pain; Colitis, Ulcerative; Communicable Diseases; Crohn Disease; Dermatitis, Atopic; Diabetes Mellitus, Type 2; Endotoxemia; Hepatitis C, Chronic; HIV Infections; Hypotension, Orthostatic; Melanoma; Mitochondrial Diseases; Narcolepsy; Neoplasm Metastasis; Neoplasms; Non-alcoholic Fatty Liver Disease; Prostatic Neoplasms, Castration-Resistant; Psoriasis; Severe Acute Respiratory Syndrome; Sexual Dysfunction, Physiological; Spinal Cord Injuries; Substance-Related Disorders; Voice Disorders; Breast Neoplasms; Cocaine-Related Disorders; Dyspnea; Tension-Type Headache; Alzheimer Disease; Atrial Fibrillation; Back Pain; Bronchopulmonary Dysplasia; Common Cold; Coronary Disease; Dysmenorrhea; Headache; Hypoxia; Intermittent Claudication; Low Back Pain; Migraine with Aura; Migraine without Aura; Multiple Sclerosis, Relapsing-Remitting; Neck Pain; Obesity; Parkinson Disease; Toothache; Apnea; Attention Deficit Disorder with Hyperactivity; Migraine Disorders; Pain
Adenosine receptor antagonist
Small molecule
Approved
Unknown
Unknown
Hypersensitivity; Pruritus
Unknown
Small molecule
Approved
OTHER
ORAL
Unknown
Histamine H1 receptor antagonist
Small molecule
Approved
Unknown
Unknown
Hypotension, Orthostatic; Migraine Disorders
Unknown
Small molecule
Approved
DENTISTRY; NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
BUCCAL; ORAL; RECTAL; TOPICAL
Abortion, Spontaneous; Attention Deficit Disorder with Hyperactivity; Brain Neoplasms; Carcinoma, Squamous Cell; Cicatrix; Complex Regional Pain Syndromes; Glioblastoma; Glycogen Storage Disease Type II; Hypertension, Pulmonary; Keratosis, Actinic; Lung Neoplasms; Morton Neuroma; Neoplasms, Cystic, Mucinous, and Serous; Neuroma; Parathyroid Neoplasms; Premature Birth; Radius Fractures; Skin Neoplasms; Spinal Fractures; Thromboembolism; Tinnitus; Anus Diseases; Anxiety; Cancer Pain; Carcinoma; Cocaine-Related Disorders; Cognitive Dysfunction; Cystitis, Interstitial; Diabetic Neuropathies; Dysmenorrhea; Dysphonia; Geographic Atrophy; Heart Diseases; Humeral Fractures; Infertility; Irritable Bowel Syndrome; Leiomyoma; Myofascial Pain Syndromes; Neoplasms; Renal Colic; Rib Fractures; Scleroderma, Localized; Severe Acute Respiratory Syndrome; Shoulder Impingement Syndrome; Shoulder Pain; Skin Diseases; Temporomandibular Joint Disorders; Trigeminal Neuralgia; Urinary Incontinence; Urinary Tract Infections; Analgesia; Breast Neoplasms; Carpal Tunnel Syndrome; Chronic Pain; Colorectal Neoplasms; Common Cold; Cough; Dysuria; Fibromyalgia; Fractures, Bone; Headache; Heart Arrest; Hemorrhage; Ileus; Low Back Pain; Migraine Disorders; Muscular Diseases; Nutrition Disorders; Obesity; Obesity, Morbid; Osteoarthritis, Knee; Osteoporosis, Postmenopausal; Paget Disease, Extramammary; Parathyroid Diseases; Periarthritis; Peripheral Nervous System Diseases; Pharyngitis; Pre-Eclampsia; Pregnancy; Pulpitis; Scoliosis; Shock, Septic; Sinusitis; Stomatitis; Stroke; Tennis Elbow; Urinary Bladder Neoplasms; Urinary Bladder, Overactive; Uterine Cervical Dysplasia; Wounds and Injuries; Arrhythmias, Cardiac; Arthritis; Back Pain; Burns; Bursitis; Hemorrhoids; Inflammation; Insect Bites and Stings; Muscle Cramp; Myalgia; Neuralgia; Neuralgia, Postherpetic; Osteoarthritis; Pain; Premature Ejaculation; Pruritus; Rectal Diseases; Sprains and Strains; Sunburn; Tendinopathy; Urethritis
Sodium channel alpha subunit blocker
Small molecule
Approved
Unknown
Unknown
Diabetes Mellitus, Type 2; Eosinophilic Esophagitis; Pancreatic Neoplasms
Unknown
Small molecule
Approved
Unknown
Unknown
Hypersensitivity
Unknown
Protein
Approved
OTHER
FOR RX COMPOUNDING; INJECTION; OPHTHALMIC; TOPICAL
Osteomyelitis; Paranasal Sinus Diseases; Arrhythmias, Cardiac; Bacterial Infections; Burns; Eye Infections; Infections; Pneumonia
C55-isoprenyl pyrophosphate inhibitor
Small molecule
Approved
Unknown
Unknown
Carcinoma, Intraductal, Noninfiltrating; Gliosarcoma; Neoplasms; Pancreatic Neoplasms; Severe Dengue; Small Cell Lung Carcinoma; Acquired Immunodeficiency Syndrome; Anemia, Sickle Cell; Brain Diseases; Breast Neoplasms; HIV Infections; Influenza, Human; Lupus Erythematosus, Systemic; Multiple Myeloma; Arthritis, Rheumatoid; Glioblastoma; Malaria, Falciparum; Malaria, Vivax; Pregnancy; Severe Acute Respiratory Syndrome; Malaria
Unknown
Small molecule
Approved
OTHER
TOPICAL
Unknown
Bacterial enoyl-[acyl-carrier-protein] reductase inhibitor
Small molecule
Approved
Unknown
Unknown
Bacterial Infections
Bacterial dihydropteroate synthase inhibitor
Small molecule
Approved
OTHER
TOPICAL
Scabies
Unknown
Small molecule
Approved
Unknown
Unknown
Hodgkin Disease; Lichen Planus; Lymphoma, T-Cell, Cutaneous; Lymphoma; Mycosis Fungoides; Neoplasms
DNA inhibitor
Small molecule
Approved
OTHER
ORAL
Epilepsy
Voltage-gated T-type calcium channel blocker
Small molecule
Approved
Unknown
Unknown
Dystonic Disorders; Parkinson Disease
Unknown
Small molecule
Approved
Unknown
Unknown
Infections; Loiasis; Elephantiasis, Filarial; Helminthiasis
Unknown
Small molecule
Approved
OTHER
INJECTION; OPHTHALMIC; ORAL; OTIC; TOPICAL
Osteomyelitis; Acne Vulgaris; Bacterial Infections; Eye Infections
Bacterial 70S ribosome inhibitor
Small molecule
Approved
Unknown
Unknown
Pain
Mu opioid receptor agonist
Small molecule
Approved
Unknown
Unknown
Digestive System Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Depressive Disorder; Hypotension, Orthostatic; Inflammation; Ischemic Stroke; Obesity; Radiodermatitis; Acute Lung Injury; Brain Injuries; Cognitive Dysfunction; Heart Diseases; Hepatorenal Syndrome; Hernias, Diaphragmatic, Congenital; Hypotension; Sepsis; Shock; Shock, Septic; Stroke; Syndrome; Cardiovascular Diseases
Unknown
Protein
Approved
OTHER
INJECTION
Glomerulonephritis; Glomerulonephritis, Membranous; Optic Neuritis; Polycystic Ovary Syndrome; Renal Insufficiency, Chronic; Vitreoretinopathy, Proliferative; Amyotrophic Lateral Sclerosis; Dermatomyositis; Diabetic Nephropathies; Epilepsy; Migraine Disorders; Multiple Sclerosis, Chronic Progressive; Sarcoidosis; Scleritis; Uveitis; Arthritis, Rheumatoid; Glomerulosclerosis, Focal Segmental; Kidney Diseases; Multiple Sclerosis, Relapsing-Remitting; Nephrotic Syndrome; Multiple Sclerosis; Spasms, Infantile
Melanocortin receptor 2 agonist
Small molecule
Approved
OTHER
ORAL
Adenocarcinoma of Lung; Adenomyosis; Aging; Anemia, Sickle Cell; Digestive System Diseases; Fatigue; Fractures, Bone; Head and Neck Neoplasms; Herpes Simplex; Hypertriglyceridemia; Inflammation; Leukemia, Hairy Cell; Leukoplakia, Oral; Liver Diseases, Alcoholic; Neuralgia, Postherpetic; Peripheral Vascular Diseases; Sleep Initiation and Maintenance Disorders; Ulcer; Acute Lung Injury; Adenoma; Barrett Esophagus; Blood Coagulation Disorders; Carotid Stenosis; Depressive Disorder; Depressive Disorder, Major; Depressive Disorder, Treatment-Resistant; Disseminated Intravascular Coagulation; Duodenal Ulcer; Endometrial Neoplasms; Glioblastoma; HIV Infections; Hypercholesterolemia; Hypertension, Pulmonary; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Lupus Erythematosus, Systemic; Melanoma; Metabolic Syndrome; Mouth Neoplasms; Nasopharyngeal Carcinoma; Neoplasms; Ovarian Neoplasms; Pancreatic Neoplasms; Periodontitis; Placental Insufficiency; Pneumonia, Viral; Pregnancy; Prostatic Neoplasms; Purpura, Thrombocytopenic, Idiopathic; Purpura, Thrombotic Thrombocytopenic; Rectal Neoplasms; Respiratory Distress Syndrome; Respiratory Insufficiency; Respiratory Tract Diseases; Sepsis; Tension-Type Headache; Tobacco Use Disorder; Tuberculosis; Uterine Cervical Neoplasms; Venous Thrombosis; Vitamin D Deficiency; Abortion, Habitual; Acute Chest Syndrome; Acute Coronary Syndrome; Adenomatous Polyposis Coli; Angina, Stable; Aortic Valve Stenosis; Asthma; Asthma, Aspirin-Induced; Atherosclerosis; Atrial Fibrillation; Bipolar Disorder; Blindness; Brain Infarction; Breast Neoplasms; Carcinoma, Hepatocellular; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Cardiomyopathy, Hypertrophic; Cardiovascular Diseases; Cataract; Cerebral Infarction; Cerebrovascular Disorders; Colitis, Ulcerative; Colonic Neoplasms; Colorectal Neoplasms; Colorectal Neoplasms, Hereditary Nonpolyposis; Diabetes Mellitus; Diabetes Mellitus, Type 2; Diabetic Retinopathy; Esophageal Neoplasms; Fetal Growth Retardation; Gastrointestinal Hemorrhage; Heart Diseases; Heart Failure; Hemorrhage; Hip Fractures; Hypertension; Infertility; Influenza, Human; Intracranial Aneurysm; Intracranial Arteriosclerosis; Ischemia; Ischemic Attack, Transient; Ischemic Stroke; Lipid Metabolism Disorders; Low Back Pain; Macular Degeneration; Meningitis; Mucocutaneous Lymph Node Syndrome; Multiple Myeloma; Multiple Sclerosis; Myocardial Ischemia; Non-ST Elevated Myocardial Infarction; Osteoarthritis; Osteonecrosis; Peptic Ulcer; Peripheral Arterial Disease; Pharyngitis; Pneumonia; Polycythemia Vera; Pre-Eclampsia; Prostatic Neoplasms, Castration-Resistant; Psychotic Disorders; Pulmonary Disease, Chronic Obstructive; Renal Insufficiency, Chronic; Retinal Artery Occlusion; Retinal Vein Occlusion; Rheumatic Heart Disease; Schizophrenia; Severe Acute Respiratory Syndrome; ST Elevation Myocardial Infarction; Stomach Neoplasms; Stomach Ulcer; Thrombocythemia, Essential; Thrombophilia; Varicose Ulcer; Vascular Diseases; Venous Thromboembolism; Wounds and Injuries; Arthritis; Back Pain; Common Cold; Coronary Artery Disease; Dysmenorrhea; Fever; Headache; Migraine Disorders; Muscle Cramp; Myalgia; Myocardial Infarction; Pain; Spasm; Stroke; Thrombosis; Toothache
Cyclooxygenase inhibitor
Small molecule
Approved
Unknown
Unknown
Atrial Fibrillation; Death, Sudden, Cardiac; Heart Failure; Myocardial Infarction; Ventricular Fibrillation; Arrhythmias, Cardiac
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Sunburn; Back Pain; Common Cold; Cough; Fever; Headache; Hypersensitivity; Nasal Obstruction; Pain; Pharyngitis; Rhinitis, Allergic, Seasonal; Sinusitis
Histamine H1 receptor antagonist
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Bacterial Infections; Eye Infections; Infections
Unknown
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER; RHEUMATOLOGY
ORAL
Glioblastoma; Hypertension, Pulmonary; Intestinal Obstruction; Leukemia, Myeloid, Acute; Nausea; Osteomyelitis; Paraganglioma; Cholangitis, Sclerosing; Peripheral Nervous System Diseases; Premature Birth; Spondylitis, Ankylosing; Arthritis, Psoriatic; Arthritis, Juvenile; Arthritis, Rheumatoid; Colitis, Ulcerative
Arachidonate 5-lipoxygenase inhibitor
Small molecule
Approved
OTHER
ORAL
Gliosarcoma; Dermatomyositis; Glioblastoma; Graves Disease; Polymyositis; Graves Ophthalmopathy; Hyperthyroidism; Thyroid Diseases
Thyroid peroxidase inhibitor
Small molecule
Approved
OTHER
ORAL
Osteomyelitis; Colitis, Ulcerative; Crohn Disease; Tuberculosis, Pulmonary; Tuberculosis
Dihydrofolate reductase inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Hepatitis B, Chronic; Rhinitis, Allergic, Seasonal; Sunburn; Influenza, Human; Hypersensitivity
Unknown
Small molecule
Approved
Unknown
Unknown
Colorectal Neoplasms; Depressive Disorder; Head and Neck Neoplasms; Intervertebral Disc Degeneration; Respiratory Insufficiency; Kidney Neoplasms; Neuralgia; Nutrition Disorders; Opioid-Related Disorders; Pre-Eclampsia; Sinusitis; Spinal Cord Injuries; Toothache; Back Pain; Cancer Pain; Diabetic Neuropathies; Genital Neoplasms, Female; Hypospadias; Joint Diseases; Kidney Calculi; Low Back Pain; Neck Pain; Neoplasms; Osteoarthritis; Osteoarthritis, Hip; Osteoarthritis, Knee; Parkinson Disease; Pruritus; Restless Legs Syndrome; Chronic Pain; Pain; Substance-Related Disorders
Mu opioid receptor agonist
Small molecule
Approved
Unknown
Unknown
Constipation; Hepatitis B, Chronic; Non-alcoholic Fatty Liver Disease; Respiratory Syncytial Virus Infections; Severe Acute Respiratory Syndrome; Depressive Disorder; Depressive Disorder, Major; Migraine Disorders; Amyotrophic Lateral Sclerosis; Atrial Fibrillation; Death, Sudden, Cardiac; Multiple Sclerosis; Myocardial Infarction; Ventricular Fibrillation; Arrhythmias, Cardiac
Unknown
Small molecule
Approved
Unknown
Unknown
Urinary Bladder, Neurogenic; Digestive System Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Crohn Disease; Gastroparesis; Motion Sickness; Anxiety; Dementia; Depressive Disorder; Hyperemesis Gravidarum; Migraine with Aura; Migraine without Aura; Nausea; Pain; Schizophrenia; Vertigo; Vomiting; Hypersensitivity; Pruritus
Unknown