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Total: 10647
Small molecule
Approved
OTHER
ORAL
Cardiovascular Diseases; Hypertension
Voltage-gated L-type calcium channel blocker
Small molecule
Approved
OTHER
ORAL
Angina, Stable; Arthritis, Rheumatoid; Glioblastoma; Vascular Diseases; Breast Neoplasms; Cardiomyopathies; Cocaine-Related Disorders; Epilepsy; Esophageal and Gastric Varices; Hypertension, Pulmonary; Hypoglycemia; Kidney Diseases; Neoplasms; Prostatic Neoplasms, Castration-Resistant; Stress Disorders, Post-Traumatic; Atherosclerosis; Atrial Fibrillation; Coronary Disease; Diabetes Mellitus, Type 2; Essential Hypertension; Hematologic Neoplasms; Hypercholesterolemia; Hypertension, Portal; Hypertrophy, Left Ventricular; Kidney Failure, Chronic; Leukemia, Lymphoid; Leukemia, Myeloid, Acute; Lymphoma; Multiple Myeloma; Renal Insufficiency, Chronic; Cardiovascular Diseases; Heart Failure; Hypertension; Myocardial Infarction; Ventricular Dysfunction, Left
Adrenergic receptor alpha-1 antagonist
Small molecule
Approved
DERMATOLOGY; OTHER
TOPICAL
Melanosis; Dermatitis, Perioral; Dermatitis, Seborrheic; Acne Vulgaris; Erythema; Rosacea
Unknown
Small molecule
Approved
CARDIOVASCULAR; OTHER
INJECTION
Unknown
HERG blocker
Small molecule
Approved
Unknown
Unknown
Pre-Eclampsia; Eosinophilic Esophagitis; Non-alcoholic Fatty Liver Disease; Essential Hypertension; Hypertrophy, Left Ventricular; Marfan Syndrome; Hypertension; Kidney Diseases; Kidney Failure, Chronic; Proteinuria; Stroke
Type-1 angiotensin II receptor antagonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Atherosclerosis; Coronary Disease; Hypercholesterolemia; Hypertension; Diabetes Mellitus; Diabetes Mellitus, Type 2
Sulfonylurea receptor 1, Kir6.2 blocker
Small molecule
Approved
DERMATOLOGY
ORAL
Osteomyelitis; Bacterial Infections
Bacterial 70S ribosome inhibitor
Small molecule
Approved
Unknown
Unknown
Alopecia Areata; Anemia, Sickle Cell; Anxiety Disorders; Barrett Esophagus; Breast Carcinoma In Situ; Cardiovascular Diseases; Colonic Neoplasms; Depressive Disorder, Major; Diabetes Insipidus; Diabetic Retinopathy; Glomerulosclerosis, Focal Segmental; Head and Neck Neoplasms; HIV Infections; Li-Fraumeni Syndrome; Liver Diseases; Malaria; Multiple Sclerosis, Chronic Progressive; Muscular Dystrophy, Duchenne; Neuralgia; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Sleep Apnea, Obstructive; Thoracic Neoplasms; Tuberculosis; Acne Vulgaris; Adenocarcinoma; Adenocarcinoma, Bronchiolo-Alveolar; Adenocarcinoma of Lung; Adenomatous Polyposis Coli; Aortic Aneurysm, Abdominal; Arthritis, Rheumatoid; Atrial Fibrillation; Bardet-Biedl Syndrome; Blindness; Breast Neoplasms; Burns; Carcinoma; Carcinoma, Hepatocellular; Carcinoma, Large Cell; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Cerebral Palsy; Colitis, Ulcerative; Diabetic Foot; Endocrine Gland Neoplasms; Esophageal Neoplasms; Fibromyalgia; Fragile X Syndrome; Frontotemporal Dementia; Geographic Atrophy; Glioblastoma; Heart Failure; Heart Failure, Systolic; Hemangiosarcoma; Hepatitis; HIV-Associated Lipodystrophy Syndrome; Hypertension, Pulmonary; Inflammatory Bowel Diseases; Intellectual Disability; Leprosy; Leukemia, Lymphocytic, Chronic, B-Cell; Leukoplakia, Oral; Low Back Pain; Lung Neoplasms; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Melanoma; Melanosis; Motor Activity; Multiple Myeloma; Multiple Sclerosis; Neoplasms; Neurobehavioral Manifestations; Neuroendocrine Tumors; Ovarian Neoplasms; Pancreatic Neoplasms; Parkinson Disease; Periodontitis; Peripheral Nervous System Diseases; Pregnancy; Prostatic Neoplasms; Pulmonary Disease, Chronic Obstructive; Rectal Neoplasms; Renal Insufficiency, Chronic; Sarcoidosis; Sex Chromosome Disorders of Sex Development; Small Cell Lung Carcinoma; Squamous Cell Carcinoma of Head and Neck; Triple Negative Breast Neoplasms; Urinary Bladder Neoplasms; Uterine Cervical Neoplasms; Weight Gain; Acute Coronary Syndrome; Aging; Atherosclerosis; Bipolar Disorder; Brain Neoplasms; Cognitive Dysfunction; Colorectal Neoplasms; Coronary Disease; Diabetes, Gestational; Diabetes Mellitus, Type 1; Diabetes Mellitus, Type 2; Endometrial Neoplasms; Epilepsy; Fatty Liver; Glaucoma; Glucose Intolerance; Hidradenitis Suppurativa; Huntington Disease; Hypercholesterolemia; Hypertension; Infertility; Insulin Resistance; Intermittent Claudication; Lipid Metabolism Disorders; Liver Neoplasms; Metabolic Diseases; Metabolic Syndrome; Migraine Disorders; Muscular Dystrophies; Non-alcoholic Fatty Liver Disease; Obesity; Osteoarthritis; Peripheral Arterial Disease; Polycystic Kidney, Autosomal Dominant; Polycystic Ovary Syndrome; Post-Acute COVID-19 Syndrome; Prediabetic State; Pre-Eclampsia; Prostatic Neoplasms, Castration-Resistant; Psoriasis; Psychotic Disorders; Reperfusion Injury; Schizophrenia; Sepsis; Severe Acute Respiratory Syndrome; Thyroid Neoplasms; Diabetes Mellitus
Unknown
Small molecule
Approved
IMMUNE SYSTEM
ORAL
Intestinal Diseases; Hookworm Infections; Onchocerciasis, Ocular; Severe Acute Respiratory Syndrome; Trichuriasis; Ectoparasitic Infestations; Elephantiasis, Filarial; Filariasis; HIV Infections; Malaria; Malnutrition; Onchocerciasis; Strongyloidiasis; Toxocariasis; Helminthiasis; Infections; Neurocysticercosis
Tubulin inhibitor
Small molecule
Approved
GASTROINTESTINAL; NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
INJECTION; INTRAVENOUS
Gram-Negative Bacterial Infections; Osteomyelitis; Pancreatitis; Respiratory Insufficiency; Appendicitis; Communicable Diseases; Hematologic Neoplasms; Tuberculosis; Tuberculosis, Pulmonary; Enterobacteriaceae Infections; Lung Diseases; Mental Disorders; Neonatal Sepsis; Pneumonia; Pneumonia, Bacterial; Pneumonia, Ventilator-Associated; Pyelonephritis; Sepsis; Shock, Septic; Urinary Bladder Neoplasms; Bacteremia; Bacterial Infections; Infections; Intraabdominal Infections; Meningitis; Meningitis, Bacterial; Urinary Tract Infections
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
Unknown
Unknown
Melanoma; Muscle Spasticity; Pain
Unknown
Small molecule
Approved
Unknown
Unknown
Tinea Pedis
Unknown
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Cardiovascular Diseases; Heart Failure; Hypertension; Myocardial Infarction; Ventricular Dysfunction, Left
Angiotensin-converting enzyme inhibitor
Small molecule
Approved
OTHER
INTRAMUSCULAR; ORAL
Dyskinesia, Drug-Induced; Lecithin Cholesterol Acyltransferase Deficiency; Mood Disorders; Weight Loss; Amyotrophic Lateral Sclerosis; Anorexia Nervosa; Autistic Disorder; Delirium; Opioid-Related Disorders; Vomiting; Alcoholism; Anorexia; Anxiety; Borderline Personality Disorder; Dementia; Depressive Disorder; Depressive Disorder, Treatment-Resistant; Developmental Disabilities; Feeding and Eating Disorders; Gambling; Genital Neoplasms, Female; Huntington Disease; Intellectual Disability; Nausea; Neoplasms; Postoperative Nausea and Vomiting; Testicular Neoplasms; Weight Gain; Bipolar Disorder; Depressive Disorder, Major; Mental Disorders; Psychomotor Agitation; Psychotic Disorders; Schizophrenia
D2-like dopamine receptor antagonist
Small molecule
Approved
OTHER
ORAL
Prostatic Neoplasms, Castration-Resistant; Neoplasms; Prostatic Neoplasms
Androgen Receptor antagonist
Small molecule
Approved
Unknown
Unknown
Fasciitis, Plantar; Hernia, Inguinal; Rib Fractures; Sinusitis; Appendicitis; Joint Diseases; Leiomyoma; Neoplasms; Osteoarthritis; Postoperative Nausea and Vomiting; Pregnancy; Rotator Cuff Injuries; Shoulder Pain; Stress Disorders, Post-Traumatic; Abdominal Pain; Analgesia; Breast Neoplasms; Chronic Pain; Fractures, Bone; Genital Neoplasms, Male; Hallux Valgus; Hypotension; Knee Injuries; Osteoarthritis, Knee; Ovarian Cysts; Ovarian Neoplasms; Pain; Paralysis; Stomach Neoplasms
Unknown
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER; PEDIATRICS
ORAL
Bulimia Nervosa; Cognitive Dysfunction; Feeding and Eating Disorders; Hernias, Diaphragmatic, Congenital; HIV Infections; Liver Diseases; Alcohol Drinking; Amphetamine-Related Disorders; Brain Ischemia; Deafness; Diabetes Mellitus; Hearing Loss, Sudden; Marijuana Abuse; Multiple Sclerosis; Parkinson Disease; Sciatica; Stress Disorders, Post-Traumatic; Alcoholism; Anxiety; Bipolar Disorder; Bulimia; Cocaine-Related Disorders; Dementia; Depressive Disorder; Diabetes Mellitus, Type 2; Epilepsies, Partial; Epilepsy, Tonic-Clonic; Essential Tremor; Gambling; Headache; Hyperlipidemias; Hypertension; Hypertriglyceridemia; Metabolic Syndrome; Mood Disorders; Obesity; Obsessive-Compulsive Disorder; Pain; Prader-Willi Syndrome; Schizophrenia; Smoking Cessation; Tobacco Use Disorder; Tourette Syndrome; Epilepsy; Lennox Gastaut Syndrome; Migraine Disorders; Seizures
Carbonic anhydrase II inhibitor
Small molecule
Approved
OTHER; RESPIRATORY
ORAL
Anemia, Sickle Cell; Inflammation; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Acne Vulgaris; Idiopathic Pulmonary Fibrosis; Lung Neoplasms; Tobacco Use Disorder; Pulmonary Disease, Chronic Obstructive; Asthma
Arachidonate 5-lipoxygenase inhibitor
Small molecule
Approved
IMMUNE SYSTEM; OTHER
DENTAL; TOPICAL
Stomatitis; Lung Diseases, Obstructive
Phosphodiesterase 4 inhibitor
Small molecule
Approved
OTHER
ORAL
HIV Infections; Alzheimer Disease; Dermatitis; Melanoma; Psoriasis
Retinoid receptor agonist
Small molecule
Approved
OTHER; RESPIRATORY
ORAL
Breast Neoplasms; Hypersensitivity; Ovarian Neoplasms; Asthma; Lung Diseases, Obstructive
Cysteinyl leukotriene receptor 1 antagonist
Unknown
Approved
OTHER
INJECTION
Acute Kidney Injury
Diagnostic agent
Enzyme
Approved
Unknown
Unknown
Hepatitis C; HIV Infections
Polypeptides hydrolytic enzyme
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Breast Neoplasms; Obesity; Substance-Related Disorders; Cocaine-Related Disorders; Endometriosis; Infertility; Paget Disease, Extramammary; Pituitary ACTH Hypersecretion; Polycystic Ovary Syndrome; Diabetes Mellitus; Ovarian Hyperstimulation Syndrome; Restless Legs Syndrome; Parkinson Disease; Pituitary Neoplasms
Dopamine D2 receptor agonist
Small molecule
Approved
Unknown
ORAL
Hepatitis C, Chronic; Infertility, Male; Hepatitis C; Hyperoxaluria, Primary; Non-alcoholic Fatty Liver Disease; Obesity; Syringomyelia; Xerostomia; Depressive Disorder; Homocystinuria
Betaine-homocysteine S-methyltransferase substrate
Small molecule
Approved
RESPIRATORY
ORAL
Osteomyelitis; Bacterial Infections
Bacterial DNA gyrase inhibitor
Small molecule
Approved
Unknown
Unknown
Amyotrophic Lateral Sclerosis; Cystic Fibrosis; Lymphoma; Muscular Atrophy, Spinal; Myelodysplastic-Myeloproliferative Diseases; Myelodysplastic Syndromes; Argininosuccinic Aciduria; HIV Infections; Huntington Disease; Leukemia; Machado-Joseph Disease; Pyruvate Dehydrogenase Complex Deficiency Disease; Tuberculosis, Pulmonary; Carbamoyl-Phosphate Synthase I Deficiency Disease; Citrullinemia; Hyperammonemia; Ornithine Carbamoyltransferase Deficiency Disease; Urea Cycle Disorders, Inborn
Glutamine sequestering agent
Small molecule
Approved
EYE; OTHER; UROLOGY AND KIDNEY
INJECTION; OPHTHALMIC; ORAL
Endophthalmitis; Escherichia coli Infections; HIV Infections; Kidney Diseases; Appendicitis; Cellulitis; Diabetic Foot; Lymphoma, Non-Hodgkin; Neoplasms; Sarcoidosis; Tuberculosis, Multidrug-Resistant; Bronchitis; Cataract; Dyspepsia; Endocarditis; Fever; Helicobacter Infections; Hot Flashes; Influenza, Human; Maxillary Sinusitis; Neutropenia; Otitis Media; Pelvic Inflammatory Disease; Pneumonia, Bacterial; Prostatic Hyperplasia; Prostatitis; Pulmonary Disease, Chronic Obstructive; Pyelonephritis; Severe Acute Respiratory Syndrome; Skin Diseases; Staphylococcal Infections; Tuberculosis; Tuberculosis, Pulmonary; Bacterial Infections; Bronchitis, Chronic; Conjunctivitis, Bacterial; Cystic Fibrosis; Eye Infections; Infections; Pneumonia; Respiratory Tract Infections; Sinusitis; Urinary Tract Infections
DNA gyrase inhibitor
Small molecule
Approved
Unknown
Unknown
Arthritis, Rheumatoid; Carcinoma, Non-Small-Cell Lung; Prostatic Neoplasms; Dermatitis, Atopic; Edema; Gastroesophageal Reflux; Rhinitis, Allergic, Perennial; Asthma; Diabetic Nephropathies; Pruritus; Rhinitis, Allergic, Seasonal; Hypersensitivity
Unknown
Small molecule
Approved
Unknown
Unknown
Status Epilepticus; Epilepsy
Unknown
Small molecule
Approved
Unknown
Unknown
Acquired Immunodeficiency Syndrome; Infections; Tuberculosis; HIV Infections; Virus Diseases
Human immunodeficiency virus type 1 reverse transcriptase inhibitor
Small molecule
Approved
Unknown
Unknown
Sarcoma, Kaposi; Acquired Immunodeficiency Syndrome; HIV Infections; Virus Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Hepatopulmonary Syndrome; Hypotension, Orthostatic; Ischemic Stroke; Ascites; Hypotension; Shock, Septic; Spinal Cord Injuries; Cardiovascular Diseases
Unknown
Enzyme
Approved
Unknown
Unknown
Diabetes Mellitus, Type 1; Hypoglycemia; Pancreatic Neoplasms; Pancreatitis; Cystic Fibrosis; Exocrine Pancreatic Insufficiency; Pancreatitis, Chronic
Fatty acids hydrolytic enzyme