Display Options:
Total: 10647
Small molecule
Approved
Unknown
Unknown
Pain; Neoplasm Metastasis
Unknown
Small molecule
Approved
Unknown
Unknown
Amphetamine-Related Disorders; Stress Disorders, Post-Traumatic; Substance-Related Disorders; Alzheimer Disease; Aortic Aneurysm, Abdominal; Breast Neoplasms; Neoplasms; Cardiomyopathy, Dilated; Diabetes Mellitus, Type 2; Hypertension; Marfan Syndrome; Cardiovascular Diseases
Unknown
Unknown
Approved
OTHER
INJECTION
Breast Neoplasms; Pancreatitis; Hemorrhage
Plasma kallikrein inhibitor
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Kidney Diseases; Otitis Media; Communicable Diseases; Graft vs Host Disease; Abscess; Cholecystitis, Acute; Diabetic Foot; Enterobacteriaceae Infections; Hematologic Neoplasms; Infections; Pancreatic Neoplasms; Pneumonia; Pneumonia, Bacterial; Pneumonia, Ventilator-Associated; Pseudomonas Infections; Pyelonephritis; Sepsis; Shock, Septic; Urinary Tract Infections; Bacterial Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Opioid-Related Disorders; Substance-Related Disorders
Unknown
Small molecule
Unknown
Unknown
Unknown
Lymphoma; Multiple Myeloma; Arthritis, Rheumatoid; Dermatitis, Atopic; Multiple Sclerosis; Back Pain; Breast Neoplasms; Eosinophilic Esophagitis; Asthma; Hypersensitivity; Pruritus; Rhinitis, Allergic, Perennial; Rhinitis, Allergic, Seasonal; Urticaria
Histamine H1 receptor antagonist
Small molecule
Approved
CANCER
SUBCUTANEOUS; TRANSDERMAL
Gastroparesis; Glioma; Leukemia, Mast-Cell; Lymphoma; Pruritus; Uterine Cervical Neoplasms; Vomiting; Nausea; Neoplasms; Postoperative Nausea and Vomiting
Serotonin 3a (5-HT3a) receptor antagonist
Small molecule
Approved
OTHER
INJECTION
Unknown
Diagnostic agent
Small molecule
Approved
OTHER
INJECTION; ORAL
Diabetes Mellitus, Type 2; Pre-Eclampsia; Cardiovascular Diseases; Heart Failure; Hypertension; Myocardial Infarction; Stroke
Sodium-(potassium)-chloride cotransporter 2 inhibitor
Small molecule
Approved
Unknown
Unknown
Digestive System Diseases
Serotonin 4 (5-HT4) receptor agonist
Protein
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
SUBCUTANEOUS
Cardiomyopathies; Coronavirus Infections; Severe Acute Respiratory Syndrome; HIV Infections; Multiple Sclerosis, Relapsing-Remitting; Multiple Sclerosis
Interferon alpha/beta receptor agonist
Small molecule
Approved
Unknown
Unknown
Common Cold; Hypersensitivity; Pruritus
Unknown
Small molecule
Approved
Unknown
Unknown
Heart Arrest; Kidney Diseases; Lung Neoplasms; Organophosphate Poisoning; Pain; Prostatic Neoplasms, Castration-Resistant; Myalgia; Pancreatic Neoplasms
Unknown
Small molecule
Approved
GASTROINTESTINAL; OTHER; RESPIRATORY
INHALATION; NASAL; ORAL; RECTAL
Cholangitis, Sclerosing; Snoring; Aspergillosis, Allergic Bronchopulmonary; Breast Neoplasms; Bronchiolitis Obliterans; Diarrhea; Esophageal Stenosis; Glomerulonephritis, IGA; Hepatitis, Autoimmune; Hypersensitivity; Lung Neoplasms; Malnutrition; Melanoma; Nasal Polyps; Radiation Pneumonitis; Respiratory Distress Syndrome; Status Asthmaticus; Altitude Sickness; Bronchopulmonary Dysplasia; Colitis, Collagenous; Colitis, Lymphocytic; Colitis, Microscopic; Eosinophilic Esophagitis; Graft vs Host Disease; Liver Cirrhosis, Biliary; Proctitis; Proctocolitis; Respiratory Tract Diseases; Severe Acute Respiratory Syndrome; Sinusitis; Sleep Apnea, Obstructive; Asthma; Bronchitis, Chronic; Colitis, Ulcerative; Crohn Disease; Emphysema; Lung Diseases, Obstructive; Nasal Obstruction; Pulmonary Disease, Chronic Obstructive; Rhinitis, Allergic, Perennial; Rhinitis, Allergic, Seasonal
Glucocorticoid receptor agonist
Enzyme
Approved
OTHER
UNKNOWN
Granuloma, Lethal Midline; Leukemia; Leukemia, Biphenotypic, Acute; Lymphohistiocytosis, Hemophagocytic; Lymphoma; Precursor T-Cell Lymphoblastic Leukemia-Lymphoma; Neoplasms; Precursor Cell Lymphoblastic Leukemia-Lymphoma
Asparagine hydrolytic enzyme
Enzyme
Approved
OTHER
INJECTION
Anemia; Gaucher Disease; Thrombocytopenia
Glucocerebroside hydrolytic enzyme
Small molecule
Approved
Unknown
Unknown
Common Cold; Influenza, Human; Respiratory Tract Infections
Histamine H1 receptor antagonist
Small molecule
Approved
Unknown
Unknown
Cardiovascular Diseases
Unknown
Small molecule
Approved
OTHER
OPHTHALMIC
Dry Eye Syndromes; Eye Diseases
Glucocorticoid receptor agonist
Small molecule
Unknown
Unknown
Unknown
Obesity; Bronchiolitis Obliterans; Asthma; Asthma, Exercise-Induced; Bronchial Spasm; Bronchitis, Chronic; Emphysema; Pulmonary Disease, Chronic Obstructive
Beta-2 adrenergic receptor agonist
Small molecule
Unknown
Unknown
Unknown
Neuroendocrine Tumors; Neuroblastoma; Heart Failure
Unknown
Small molecule
Approved
Unknown
Unknown
Breast Neoplasms; Alzheimer Disease; Arthritis, Rheumatoid; Carcinoma, Renal Cell; Gliosarcoma; Head and Neck Neoplasms; Hematologic Neoplasms; Melanoma; Mycosis Fungoides; Adenocarcinoma, Follicular; Carcinoma, Non-Small-Cell Lung; Glioblastoma; Hemangiosarcoma; Hodgkin Disease; Kidney Neoplasms; Lung Neoplasms; Lymphoma, Follicular; Neoplasms; Pancreatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Sarcoma; Stomach Neoplasms; Thyroid Neoplasms; Urethral Neoplasms; Urinary Bladder Neoplasms; Uterine Cervical Neoplasms; von Hippel-Lindau Disease; Lymphoma
Diagnostic agent
Small molecule
Approved
Unknown
Unknown
Neoplasms; Panic Disorder; Anxiety; Anxiety Disorders; Anxiety, Separation; Autistic Disorder; Dementia; Obsessive-Compulsive Disorder; Phobia, Social; Schizophrenia; Severe Acute Respiratory Syndrome; Depressive Disorder
Unknown
Small molecule
Approved
DERMATOLOGY; DIABETES DRUGS & ENDOCRINOLOGY; OTHER; UROLOGY AND KIDNEY
INJECTION; ORAL; TOPICAL
Neoplasms, Neuroepithelial; Alopecia; Aspergillosis; beta-Thalassemia; Blast Crisis; DiGeorge Syndrome; Hematologic Diseases; Hypercholesterolemia; Kidney Tubular Necrosis, Acute; Leukemia, Plasma Cell; Lymphedema; Lymphoma, T-Cell; Paget Disease, Extramammary; Peripheral Nerve Injuries; Respiratory Syncytial Virus Infections; Scleroderma, Localized; Vasculitis; Venous Thromboembolism; Amyotrophic Lateral Sclerosis; Anemia, Aplastic; Anemia, Sickle Cell; Asthma; Burkitt Lymphoma; Chemical and Drug Induced Liver Injury; Colitis; Crohn Disease; Diabetes Mellitus; Edema; Encephalomyelitis; Epidermolysis Bullosa; Glomerulonephritis, IGA; Glomerulosclerosis, Focal Segmental; Granuloma, Lethal Midline; Hematologic Neoplasms; Hemoglobinuria, Paroxysmal; Hepatitis, Autoimmune; Hepatitis C; Hepatitis C, Chronic; Histiocytosis, Langerhans-Cell; Hypertension, Pulmonary; Immunoblastic Lymphadenopathy; Kidney Neoplasms; Leukemia; Leukemia, Hairy Cell; Leukemia, Large Granular Lymphocytic; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia-Lymphoma, Adult T-Cell; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Leukemia, Myelomonocytic, Chronic; Leukemia, Myelomonocytic, Juvenile; Lichen Planus, Oral; Liver Diseases; Liver Failure; Lung Diseases; Lupus Erythematosus, Cutaneous; Lymphoma; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Large-Cell, Anaplastic; Lymphoma, Mantle-Cell; Lymphoma, T-Cell, Peripheral; Macular Degeneration; Multiple Myeloma; Multiple Sclerosis; Mycosis Fungoides; Myelodysplastic-Myeloproliferative Diseases; Myeloproliferative Disorders; Neoplasms; Nephrosis, Lipoid; Neuroblastoma; Polycythemia Vera; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Primary Myelofibrosis; Prostatic Neoplasms, Castration-Resistant; Purpura, Thrombocytopenic, Idiopathic; Sarcoma; Scleroderma, Systemic; Severe Combined Immunodeficiency; Sezary Syndrome; Shwachman-Diamond Syndrome; Thalassemia; Vulvar Lichen Sclerosus; Waldenstrom Macroglobulinemia; Wiskott-Aldrich Syndrome; Wounds and Injuries; Arthritis, Rheumatoid; Bronchiolitis Obliterans; Carcinoma, Hepatocellular; Colitis, Ulcerative; Conjunctivitis, Allergic; Dermatitis, Atopic; Dermatitis, Seborrheic; Diabetes Mellitus, Type 1; Glomerulonephritis, Membranous; Graft vs Host Disease; Heart Diseases; Hodgkin Disease; Infertility; Keratoconjunctivitis; Kidney Diseases; Lupus Nephritis; Lymphoma, Non-Hodgkin; Myasthenia Gravis; Myelodysplastic Syndromes; Nephrotic Syndrome; Psoriasis; Renal Insufficiency; Renal Insufficiency, Chronic; Severe Acute Respiratory Syndrome; Skin Neoplasms; Vitiligo; Eczema; Immune System Diseases
FK506-binding protein 1A inhibitor
Protein
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Carcinoma, Non-Small-Cell Lung; Colorectal Neoplasms
Unknown
Small molecule
Approved
OTHER
ORAL
Panic Disorder; Severe Acute Respiratory Syndrome; Obsessive-Compulsive Disorder
Serotonin transporter inhibitor
Small molecule
Approved
Unknown
Unknown
Desmoplastic Small Round Cell Tumor; Prostatic Neoplasms, Castration-Resistant; Small Cell Lung Carcinoma; Adenocarcinoma of Lung; Carcinoma, Large Cell; Diffuse Intrinsic Pontine Glioma; Fallopian Tube Neoplasms; Head and Neck Neoplasms; Hodgkin Disease; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Large-Cell, Anaplastic; Melanoma; Multiple Myeloma; Ovarian Neoplasms; Rhabdomyosarcoma; Sarcoma; Triple Negative Breast Neoplasms; Breast Neoplasms; Carcinoma; Carcinoma, Non-Small-Cell Lung; Esophageal Neoplasms; Lung Neoplasms; Lymphoma, Non-Hodgkin; Mesothelioma; Rhabdomyosarcoma, Alveolar; Rhabdomyosarcoma, Embryonal; Uterine Cervical Neoplasms; Neoplasms
Unknown
Small molecule
Approved
Unknown
Unknown
Hypersensitivity
Histamine H1 receptor antagonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Wet Macular Degeneration; Glaucoma, Open-Angle; Ocular Hypertension; Glaucoma
Unknown
Small molecule
Approved
IMMUNE SYSTEM; OTHER
ORAL
Herpes Simplex; Meniere Disease; Autoimmune Diseases; Eye Infections; Herpes Genitalis; Herpes Labialis; Herpes Zoster; Virus Diseases
Human herpesvirus 1 DNA polymerase inhibitor
Small molecule
Approved
Unknown
Unknown
Hypersensitivity; Nasal Obstruction
Unknown