Display Options:
Total: 10647
Small molecule
Approved
Unknown
Unknown
Pain; Neoplasm Metastasis
Unknown
Small molecule
Approved
Unknown
Unknown
Amphetamine-Related Disorders; Stress Disorders, Post-Traumatic; Substance-Related Disorders; Alzheimer Disease; Aortic Aneurysm, Abdominal; Breast Neoplasms; Neoplasms; Cardiomyopathy, Dilated; Diabetes Mellitus, Type 2; Hypertension; Marfan Syndrome; Cardiovascular Diseases
Unknown
Unknown
Approved
OTHER
INJECTION
Breast Neoplasms; Pancreatitis; Hemorrhage
Plasma kallikrein inhibitor
Small molecule
Approved
Unknown
Unknown
Kidney Diseases; Osteomyelitis; Otitis Media; Appendicitis; Communicable Diseases; Graft vs Host Disease; Abscess; Cholecystitis, Acute; Diabetic Foot; Enterobacteriaceae Infections; Hematologic Neoplasms; Infections; Influenza, Human; Lung Diseases; Pneumonia; Pneumonia, Bacterial; Pneumonia, Ventilator-Associated; Pseudomonas Infections; Pyelonephritis; Sepsis; Severe Acute Respiratory Syndrome; Shock, Septic; Urinary Tract Infections; Bacterial Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Opioid-Related Disorders; Substance-Related Disorders
Mu opioid receptor agonist
Small molecule
Approved
Unknown
Unknown
Arthritis, Rheumatoid; Dermatitis, Atopic; Lymphoma; Multiple Myeloma; Multiple Sclerosis; Back Pain; Breast Neoplasms; Eosinophilic Esophagitis; Lymphangioleiomyomatosis; Severe Acute Respiratory Syndrome; Asthma; Hypersensitivity; Pruritus; Rhinitis, Allergic, Perennial; Rhinitis, Allergic, Seasonal; Urticaria
Histamine H1 receptor antagonist
Small molecule
Approved
CANCER
SUBCUTANEOUS; TRANSDERMAL
Gastroparesis; Glioma; Leukemia, Mast-Cell; Lymphoma; Pruritus; Carcinoma, Hepatocellular; Pain; Uterine Cervical Neoplasms; Nausea; Neoplasms; Postoperative Nausea and Vomiting; Vomiting
Serotonin 3a (5-HT3a) receptor antagonist
Small molecule
Approved
Unknown
Unknown
Digestive System Diseases
Unknown
Small molecule
Approved
OTHER
INJECTION
Unknown
Diagnostic agent
Small molecule
Approved
OTHER
INJECTION; ORAL
Diabetes Mellitus, Type 2; Pre-Eclampsia; Cardiovascular Diseases; Heart Failure; Hypertension; Myocardial Infarction; Stroke
Sodium-(potassium)-chloride cotransporter 2 inhibitor
Protein
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
SUBCUTANEOUS
Cardiomyopathies; Coronavirus Infections; Severe Acute Respiratory Syndrome; HIV Infections; Multiple Sclerosis, Relapsing-Remitting; Multiple Sclerosis; Neoplasms
Interferon alpha/beta receptor agonist
Small molecule
Approved
Unknown
Unknown
Common Cold; Hypersensitivity; Pruritus
Unknown
Small molecule
Approved
Unknown
Unknown
Fractures, Bone; Heart Arrest; Kidney Diseases; Lung Neoplasms; Organophosphate Poisoning; Pain; Prostatic Neoplasms, Castration-Resistant; Myalgia; Pancreatic Neoplasms
Unknown
Small molecule
Approved
GASTROINTESTINAL; OTHER; RESPIRATORY
INHALATION; NASAL; ORAL; RECTAL
Cholangitis, Sclerosing; Anosmia; Aspergillosis, Allergic Bronchopulmonary; Breast Neoplasms; Bronchiolitis Obliterans; Diarrhea; Esophageal Stenosis; Hepatitis, Autoimmune; Hypersensitivity; Inflammatory Bowel Diseases; Lung Neoplasms; Malnutrition; Melanoma; Multiple Myeloma; Nasal Polyps; Proctitis; Radiation Pneumonitis; Respiratory Distress Syndrome; Status Asthmaticus; Altitude Sickness; Bronchiolitis Obliterans Syndrome; Bronchopulmonary Dysplasia; Colitis, Collagenous; Colitis, Lymphocytic; Colitis, Microscopic; Eosinophilic Esophagitis; Graft vs Host Disease; Liver Cirrhosis, Biliary; Proctocolitis; Respiratory Tract Diseases; Severe Acute Respiratory Syndrome; Sinusitis; Sleep Apnea, Obstructive; Snoring; Asthma; Bronchitis, Chronic; Colitis, Ulcerative; Crohn Disease; Emphysema; Esophageal Diseases; Glomerulonephritis, IGA; Lung Diseases, Obstructive; Nasal Obstruction; Pulmonary Disease, Chronic Obstructive; Rhinitis, Allergic, Perennial; Rhinitis, Allergic, Seasonal
Glucocorticoid receptor agonist
Enzyme
Approved
OTHER
UNKNOWN
Leukemia, Myeloid, Acute; Granuloma, Lethal Midline; Leukemia; Leukemia, Biphenotypic, Acute; Leukemia, Lymphoid; Lymphohistiocytosis, Hemophagocytic; Lymphoma; Precursor T-Cell Lymphoblastic Leukemia-Lymphoma; Neoplasms; Precursor Cell Lymphoblastic Leukemia-Lymphoma
Asparagine hydrolytic enzyme
Small molecule
Approved
Unknown
Unknown
Common Cold; Influenza, Human; Respiratory Tract Diseases; Respiratory Tract Infections
Histamine H1 receptor antagonist
Enzyme
Approved
OTHER
INJECTION
Anemia; Gaucher Disease; Thrombocytopenia
Glucocerebroside hydrolytic enzyme
Small molecule
Approved
Unknown
Unknown
Cardiovascular Diseases
Unknown
Small molecule
Approved
OTHER
OPHTHALMIC
Dry Eye Syndromes; Eye Diseases
Glucocorticoid receptor agonist
Small molecule
Approved
Unknown
Unknown
Obesity; Asthma; Asthma, Exercise-Induced; Bronchial Spasm; Bronchitis, Chronic; Emphysema; Pulmonary Disease, Chronic Obstructive
Beta-2 adrenergic receptor agonist
Small molecule
Approved
Unknown
Unknown
Neuroendocrine Tumors; Neuroblastoma; Paraganglioma; Pheochromocytoma; Heart Failure
Unknown
Small molecule
Approved
Unknown
Unknown
Alzheimer Disease; Arthritis, Rheumatoid; Brain Neoplasms; Carcinoma, Renal Cell; Cardiovascular Diseases; Gliosarcoma; Head and Neck Neoplasms; Hematologic Neoplasms; Idiopathic Pulmonary Fibrosis; Leukemia, Promyelocytic, Acute; Lymphoma, Non-Hodgkin; Lymphoma, T-Cell, Cutaneous; Melanoma; Mesothelioma; Multiple Myeloma; Mycosis Fungoides; Adenocarcinoma, Follicular; Breast Neoplasms; Carcinoid Tumor; Carcinoma, Hepatocellular; Carcinoma, Neuroendocrine; Glioblastoma; Hemangiosarcoma; Hodgkin Disease; Kidney Neoplasms; Lung Neoplasms; Lymphoma, Follicular; Neoplasms; Neuroendocrine Tumors; Pancreatic Neoplasms; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Sarcoma; Stomach Neoplasms; Thyroid Neoplasms; Urethral Neoplasms; Urinary Bladder Neoplasms; Uterine Cervical Neoplasms; von Hippel-Lindau Disease; Carcinoma, Non-Small-Cell Lung; Histiocytosis; Leukemia, Myeloid, Acute; Lymphoma; Lymphoma, Mantle-Cell
Diagnostic agent
Small molecule
Approved
Unknown
Unknown
Neoplasms; Panic Disorder; Post-Acute COVID-19 Syndrome; Anxiety; Anxiety Disorders; Anxiety, Separation; Autistic Disorder; Dementia; Obsessive-Compulsive Disorder; Phobia, Social; Schizophrenia; Severe Acute Respiratory Syndrome; Depressive Disorder
Unknown
Small molecule
Approved
DERMATOLOGY; DIABETES DRUGS & ENDOCRINOLOGY; OTHER; UROLOGY AND KIDNEY
INJECTION; ORAL; TOPICAL
Hematologic Neoplasms; Anemia, Aplastic; Anemia, Sickle Cell; Graft vs Host Disease; Lichen Planus, Oral; Thalassemia; Conjunctivitis, Allergic; Keratoconjunctivitis; Delayed Graft Function; Dermatitis, Atopic; Eczema; Immune System Diseases; Kidney Transplantation; Liver Transplantation
FK506-binding protein 1A inhibitor
Protein
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Carcinoma, Non-Small-Cell Lung; Colorectal Neoplasms
Unknown
Small molecule
Approved
OTHER
ORAL
Panic Disorder; Obsessive-Compulsive Disorder
Serotonin transporter inhibitor
Small molecule
Approved
Unknown
Unknown
Desmoplastic Small Round Cell Tumor; Prostatic Neoplasms, Castration-Resistant; Small Cell Lung Carcinoma; Adenocarcinoma of Lung; Carcinoma, Large Cell; Diffuse Intrinsic Pontine Glioma; Fallopian Tube Neoplasms; Glioma; Head and Neck Neoplasms; Lymphoma; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Large-Cell, Anaplastic; Melanoma; Multiple Myeloma; Ovarian Neoplasms; Rhabdomyosarcoma; Sarcoma; Breast Neoplasms; Carcinoma; Carcinoma, Non-Small-Cell Lung; Esophageal Neoplasms; Hodgkin Disease; Lung Neoplasms; Lymphoma, Non-Hodgkin; Mesothelioma; Rhabdomyosarcoma, Alveolar; Rhabdomyosarcoma, Embryonal; Triple Negative Breast Neoplasms; Uterine Cervical Neoplasms; Neoplasms
Unknown
Small molecule
Approved
Unknown
Unknown
Hypersensitivity
Histamine H1 receptor antagonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Macular Degeneration; Wet Macular Degeneration; Glaucoma, Open-Angle; Ocular Hypertension; Glaucoma
Unknown
Small molecule
Approved
IMMUNE SYSTEM; OTHER
ORAL
Multiple Sclerosis; Herpes Simplex; Meniere Disease; Autoimmune Diseases; Eye Infections; Herpes Genitalis; Herpes Labialis; Herpes Zoster; Virus Diseases
Human herpesvirus 1 DNA polymerase inhibitor
Small molecule
Approved
Unknown
Unknown
Hypersensitivity; Nasal Obstruction
Unknown