Display Options:
Total: 139
Small molecule
Approved
OTHER; PEDIATRICS; RESPIRATORY
INHALATION; NASAL
Pulmonary Disease, Chronic Obstructive; Chronic Disease; Hypersensitivity; Respiratory Tract Diseases; Severe Acute Respiratory Syndrome; Asthma; Lung Diseases, Obstructive; Nasal Obstruction; Rhinitis, Allergic, Perennial; Rhinitis, Allergic, Seasonal
Glucocorticoid receptor agonist
Small molecule
Approved
HEMATOLOGY; OTHER
INTRAVENOUS
Burkitt Lymphoma; Carcinoma, Squamous Cell; Head and Neck Neoplasms; Hematologic Neoplasms; HIV Infections; Leukemia, Promyelocytic, Acute; Lymphoma, Follicular; Lymphoma, Mantle-Cell; Lymphoma, Non-Hodgkin; Lymphoma, T-Cell, Cutaneous; Mastocytosis, Systemic; Medulloblastoma; Multiple Myeloma; Neuroblastoma; Paraganglioma; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Precursor T-Cell Lymphoblastic Leukemia-Lymphoma; Prostatic Neoplasms; Sarcoma, Synovial; Triple Negative Breast Neoplasms; Adenocarcinoma, Follicular; Anemia, Aplastic; Anemia, Sickle Cell; Breast Neoplasms; Carcinoma, Non-Small-Cell Lung; Carcinoma, Renal Cell; Esophageal Neoplasms; Fallopian Tube Neoplasms; Granuloma, Lethal Midline; Hodgkin Disease; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Lung Neoplasms; Lymphoma; Melanoma; Ovarian Neoplasms; Peritoneal Neoplasms; Primary Myelofibrosis; Severe Acute Respiratory Syndrome; Thalassemia; Thyroid Neoplasms; Graft vs Host Disease; Hematologic Diseases; Leukemia; Leukemia, Myeloid, Acute; Lymphoma, Large B-Cell, Diffuse; Lymphoma, T-Cell, Peripheral; Myeloproliferative Disorders; Purpura, Thrombocytopenic, Idiopathic; Thrombocytopenia; Anemia; Anemia, Refractory, with Excess of Blasts; Leukemia, Myeloid; Leukemia, Myelomonocytic, Chronic; Myelodysplastic Syndromes; Neoplasms
DNA (cytosine-5)-methyltransferase 1 inhibitor
Small molecule
Approved
Unknown
Unknown
Amphetamine-Related Disorders; Cocaine-Related Disorders; Multiple Sclerosis; Substance-Related Disorders; Bipolar Disorder; Depressive Disorder; Feeding and Eating Disorders; Attention Deficit Disorder with Hyperactivity
Unknown
Small molecule
Approved
Unknown
Unknown
Amnesia; Colorectal Neoplasms; Depressive Disorder; Inflammation; Neural Tube Defects; Obesity, Morbid; Premature Birth; Psychomotor Agitation; Renal Insufficiency; Renal Insufficiency, Chronic; Coronary Disease; Depressive Disorder, Treatment-Resistant; Hypotension; Leukemia; Migraine Disorders; Neoplasms; Postoperative Nausea and Vomiting; Pulmonary Disease, Chronic Obstructive; Tonsillitis; Wounds and Injuries; Atrial Fibrillation; Back Pain; Brain Injuries; Delirium; Genital Neoplasms, Male; Heart Diseases; Hypertension; Liver Cirrhosis; Obesity; Pain; Pruritus; Reperfusion Injury; Respiratory Distress Syndrome; Respiratory Insufficiency; Severe Acute Respiratory Syndrome; Status Epilepticus; Stroke; Subarachnoid Hemorrhage
Unknown
Small molecule
Approved
Unknown
Unknown
Brain Injuries; Multiple Myeloma; Nasopharyngeal Carcinoma; Vomiting; Genital Neoplasms, Female; Nausea; Neoplasms; Postoperative Nausea and Vomiting
Unknown
Small molecule
Approved
EYE
OPHTHALMIC
Dry Eye Syndromes; Cataract; Keratitis; Panuveitis; Uveitis; Eye Diseases; Inflammation; Uveitis, Anterior
Glucocorticoid receptor agonist
Small molecule
Approved
Unknown
Unknown
HIV Infections; Asthma; Cardiovascular Diseases; Heart Diseases; Acute Coronary Syndrome; Anemia, Sickle Cell; Atrial Fibrillation; Coronary Disease; Influenza, Human; Kidney Failure, Chronic; Myocardial Infarction; Pneumonia; Severe Acute Respiratory Syndrome; ST Elevation Myocardial Infarction; Thrombosis
Unknown
Small molecule
Approved
Unknown
Unknown
HIV Infections; Neoplasms; Schistosomiasis haematobia; Fever; Malaria, Falciparum; Malaria, Vivax; Malaria
Ferriprotoporphyrin IX inhibitor
Protein
Approved
HEMATOLOGY
INTRAVENOUS
Astrocytoma; Brain Neoplasms; Carcinoma, Pancreatic Ductal; Glioblastoma; Gliosarcoma; Hematologic Neoplasms; Hodgkin Disease; Inflammatory Breast Neoplasms; Leukemia; Liposarcoma; Lymphoma, Non-Hodgkin; Mycosis Fungoides; Oligodendroglioma; Pancreatic Neoplasms; Sezary Syndrome; Triple Negative Breast Neoplasms; Adenocarcinoma, Follicular; Breast Neoplasms; Breast Neoplasms, Male; Carcinoma, Non-Small-Cell Lung; Colorectal Neoplasms; HIV Infections; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Promyelocytic, Acute; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Large-Cell, Anaplastic; Lymphoma, Mantle-Cell; Melanoma; Multiple Myeloma; Ovarian Neoplasms; Prostatic Neoplasms, Castration-Resistant; Small Cell Lung Carcinoma; Stomach Neoplasms; Thyroid Neoplasms; Urethral Neoplasms; Urinary Bladder Neoplasms; Immunoblastic Lymphadenopathy; Lymphoma; Lymphoma, T-Cell; Lymphoma, T-Cell, Cutaneous; Lymphoma, T-Cell, Peripheral; Neoplasms
Histone deacetylase inhibitor
Small molecule
Approved
Unknown
ORAL
Carcinoma, Non-Small-Cell Lung; Hematologic Diseases; Non-alcoholic Fatty Liver Disease; Prostatic Neoplasms; Renal Insufficiency; Renal Insufficiency, Chronic; Coronary Disease; Atrial Fibrillation; Stroke; Thromboembolism; Venous Thromboembolism; Venous Thrombosis; Thrombosis
Unknown
Small molecule
Approved
OTHER; RESPIRATORY
INTRAVENOUS
Kidney Diseases; Systemic Inflammatory Response Syndrome; Sepsis; Urinary Tract Infections; Infections; Pneumonia, Bacterial; Bacterial Infections
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
MUSCULOSKELETAL
ORAL
Astrocytoma; Breast Neoplasms; Cerebral Hemorrhage; Glioblastoma; Renal Insufficiency; Rett Syndrome; Asthma; Optic Neuritis; Schizophrenia; Severe Acute Respiratory Syndrome; Stroke; Uveitis; Multiple Sclerosis; Multiple Sclerosis, Chronic Progressive; Multiple Sclerosis, Relapsing-Remitting; Polyradiculoneuropathy, Chronic Inflammatory Demyelinating
Unknown
Small molecule
Approved
Unknown
Unknown
Cardiovascular Diseases; Essential Hypertension; Hypertension
Unknown
Small molecule
Approved
CARDIOVASCULAR; OTHER
ORAL
Hypertension; Stroke
Type-1 angiotensin II receptor antagonist
Antibody
Approved
CANCER; OTHER
INJECTION
Hematologic Neoplasms; HIV Infections; Leukemia; Leukemia, Myeloid, Acute; Enteropathy-Associated T-Cell Lymphoma; Graft vs Host Disease; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia-Lymphoma, Adult T-Cell; Leukemia, Mast-Cell; Lupus Erythematosus, Systemic; Lymphoma, Follicular; Lymphoma, T-Cell, Peripheral; Mastocytosis, Systemic; Mesothelioma, Malignant; Neoplasms, Germ Cell and Embryonal; Scleroderma, Diffuse; Sezary Syndrome; Lymphoma; Lymphoma, Large B-Cell, Diffuse; Lymphoma, T-Cell, Cutaneous; Mycosis Fungoides; Hodgkin Disease; Lymphoma, Large-Cell, Anaplastic; Lymphoma, Non-Hodgkin; Neoplasms
Tubulin inhibitor
Small molecule
Approved
DERMATOLOGY; NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
ORAL
Kidney Diseases; Alcoholism; Diabetic Neuropathies; Migraine Disorders; Neuralgia, Postherpetic; Restless Legs Syndrome
Voltage-gated calcium channel modulator
Small molecule
Approved
EYE
OPHTHALMIC
Glaucoma; Glaucoma, Open-Angle; Ocular Hypertension
Prostanoid FP receptor agonist
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY
INTRAMUSCULAR; ORAL
Carcinoma, Renal Cell; Coronary Disease; Prostatic Neoplasms, Castration-Resistant; Sexual Dysfunction, Physiological; Spinal Cord Injuries; Aging; Malnutrition; Respiratory Insufficiency; Hypogonadism; Klinefelter Syndrome; Neoplasms; Orchitis
Androgen Receptor agonist
Small molecule
Approved
Unknown
Unknown
Amyotrophic Lateral Sclerosis; Insulin Resistance; Hepatitis D; Leukemia, Lymphocytic, Chronic, B-Cell; Weight Gain; Acquired Immunodeficiency Syndrome; Hepatitis B, Chronic; HIV Infections; Severe Acute Respiratory Syndrome; Virus Diseases
Human immunodeficiency virus type 1 reverse transcriptase inhibitor
Small molecule
Approved
Unknown
ORAL
Acquired Immunodeficiency Syndrome; Hepatitis B; Hepatitis B, Chronic; HIV Infections
Human immunodeficiency virus type 1 reverse transcriptase inhibitor
Small molecule
Approved
Unknown
INTRAMUSCULAR
Psychotic Disorders; Schizophrenia
Dopamine D2 receptor partial agonist
Small molecule
Approved
Unknown
Unknown
Liver Diseases; Biliary Tract Neoplasms; Malignant Carcinoid Syndrome; Neuroendocrine Tumors; Pancreatic Neoplasms; Carcinoid Heart Disease
Tryptophan 5-hydroxylase inhibitor
Small molecule
Approved
Unknown
ORAL
Kidney Diseases; Liver Diseases; Aspergillosis, Allergic Bronchopulmonary; Muscular Dystrophies, Limb-Girdle; Muscular Dystrophies; Muscular Dystrophy, Duchenne
Glucocorticoid receptor agonist
Small molecule
Approved
Unknown
ORAL
Pneumonia; Severe Acute Respiratory Syndrome; Influenza, Human; Virus Diseases
Polymerase acidic protein inhibitor
Small molecule
Approved
Unknown
Unknown
Bronchiolitis Obliterans Syndrome; Hematologic Neoplasms; Lymphoma; Ovarian Neoplasms; Pneumonia; Anemia, Hemolytic, Autoimmune; Glomerulonephritis, IGA; Hidradenitis Suppurativa; Lymphoma, Large B-Cell, Diffuse; Primary Myelofibrosis; Severe Acute Respiratory Syndrome; Arthritis, Rheumatoid; Purpura, Thrombocytopenic, Idiopathic; Hemorrhage
Tyrosine-protein kinase SYK inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Pneumonia, Viral; Hemorrhagic Fever, Ebola; Respiratory Distress Syndrome; Influenza, Human; Pneumonia; Coronavirus Infections; COVID-19; Severe Acute Respiratory Syndrome; Virus Diseases
Replicase polyprotein 1ab inhibitor
Small molecule
Approved
Unknown
Unknown
Breast Neoplasms; Carcinoma, Hepatocellular; Friedreich Ataxia; Idiopathic Pulmonary Fibrosis; Neoplasms; Colorectal Neoplasms; Conjunctivitis, Allergic; Crohn Disease; Intestinal Neoplasms; Cytomegalovirus Infections; Fever; Malaria, Falciparum; Malaria, Vivax; Schistosomiasis; Schistosomiasis haematobia; Severe Acute Respiratory Syndrome; Malaria
Unknown
Small molecule
Investigational
Unknown
Unknown
Fever; Marburg Virus Disease; Severe Acute Respiratory Syndrome
Genome polyprotein inhibitor
Small molecule
Investigational
Unknown
Unknown
Hypercholesterolemia; Hyperlipidemias; Non-alcoholic Fatty Liver Disease
Thyroid hormone receptor beta-1 agonist
Small molecule
Investigational
Unknown
Unknown
Lymphoma; Neoplasms
Unknown
Small molecule
Investigational
Unknown
Unknown
Infections
Bacterial 70S ribosome inhibitor
Small molecule
Investigational
Unknown
Unknown
Neuralgia; Depressive Disorder; Depressive Disorder, Major; Hypertension, Pulmonary
Glutamate [NMDA] receptor antagonist
Small molecule
Approved
Unknown
Unknown
Severe Acute Respiratory Syndrome; Schizophrenia; Malaria
Unknown