Display Options:
Total: 10647
Small molecule
Approved
OTHER
OPHTHALMIC; ORAL
Optic Neuropathy, Ischemic; Corneal Edema; Hemangioma; Hypertension, Portal; Glaucoma; Glaucoma, Open-Angle; Ocular Hypertension
Beta-1 adrenergic receptor antagonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
INJECTION
Rhabdomyosarcoma; Carcinoma, Basal Cell; Carcinoma, Endometrioid; Carcinoma, Merkel Cell; Cystadenoma, Serous; Digestive System Neoplasms; Genital Neoplasms, Female; Kidney Diseases; Klatskin Tumor; Liver Diseases; Xerostomia; Carcinoid Tumor; Carcinoma, Islet Cell; Carcinoma, Neuroendocrine; Carcinoma, Pancreatic Ductal; Carcinoma, Renal Cell; Digestive System Diseases; Ganglioneuroblastoma; Gastrointestinal Stromal Tumors; Glioma; Granuloma, Lethal Midline; Immunoblastic Lymphadenopathy; Kidney Neoplasms; Leukemia; Leukemia-Lymphoma, Adult T-Cell; Lymphoma, AIDS-Related; Lymphoma, Follicular; Lymphoma, Large-Cell, Anaplastic; Myelodysplastic Syndromes; Nausea; Neoplasm Metastasis; Penile Neoplasms; Prostatic Neoplasms, Castration-Resistant; Salivary Gland Neoplasms; Thymoma; Thyroid Neoplasms; Tongue Neoplasms; Triple Negative Breast Neoplasms; Adenocarcinoma; Adenocarcinoma of Lung; Adrenal Cortex Neoplasms; Anemia; Anus Neoplasms; Biliary Tract Neoplasms; Brain Neoplasms; Breast Neoplasms; Carcinoma; Carcinoma, Embryonal; Carcinoma, Hepatocellular; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Central Nervous System Neoplasms; Cholangiocarcinoma; Choriocarcinoma; Choroid Plexus Neoplasms; Colorectal Neoplasms; Endodermal Sinus Tumor; Endometrial Neoplasms; Ependymoma; Esophageal Neoplasms; Fallopian Tube Neoplasms; Gallbladder Neoplasms; Gestational Trophoblastic Disease; Head and Neck Neoplasms; Hepatoblastoma; Hodgkin Disease; Hypopharyngeal Neoplasms; Inflammatory Breast Neoplasms; Laryngeal Neoplasms; Liver Neoplasms; Lung Neoplasms; Lymphoma; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Lymphoma, Non-Hodgkin; Lymphoma, T-Cell, Peripheral; Malaria; Mediastinal Neoplasms; Medulloblastoma; Melanoma; Mesothelioma; Mouth Neoplasms; Mucositis; Multiple Myeloma; Nasopharyngeal Neoplasms; Neoplasms, Germ Cell and Embryonal; Neuroblastoma; Neuroectodermal Tumors, Primitive; Oropharyngeal Neoplasms; Osteosarcoma; Ovarian Neoplasms; Pancreatic Neoplasms; Paranasal Sinus Neoplasms; Peritoneal Neoplasms; Pharyngeal Neoplasms; Pleural Effusion; Postoperative Nausea and Vomiting; Retinoblastoma; Sarcoma; Seminoma; Sex Cord-Gonadal Stromal Tumors; Skin Neoplasms; Small Cell Lung Carcinoma; Squamous Cell Carcinoma of Head and Neck; Stomach Neoplasms; Stomatitis; Teratoma; Testicular Neoplasms; Thymus Neoplasms; Urethral Neoplasms; Urinary Bladder Neoplasms; Urogenital Neoplasms; Uterine Cervical Neoplasms; Uterine Neoplasms; Vulvar Neoplasms; Neoplasms
DNA inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
ORAL
Alzheimer Disease; Urinary Bladder Neoplasms; Astrocytoma; Burkitt Lymphoma; Carcinoma, Non-Small-Cell Lung; Central Nervous System Neoplasms; Colorectal Neoplasms; Lung Neoplasms; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Medulloblastoma; Nasopharyngeal Neoplasms; Neoplasms; Ovarian Neoplasms; Sarcoma; Shock; Wounds and Injuries; Alopecia; Brain Neoplasms; Breast Neoplasms; Carcinoma, Squamous Cell; Glioblastoma; Glioma; Head and Neck Neoplasms; HIV Infections; Leukemia; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Lymphoma; Melanoma; Muscular Atrophy, Spinal; Myelodysplastic Syndromes; Neuralgia; Pancreatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Retinitis Pigmentosa; Small Cell Lung Carcinoma; Supranuclear Palsy, Progressive; Thyroid Neoplasms; Anxiety; Dementia; Depressive Disorder; Paraparesis, Tropical Spastic; Schizophrenia; Status Epilepticus; Anorexia; Bipolar Disorder; Epilepsy; Epilepsy, Absence; Epilepsy, Complex Partial; Migraine Disorders; Mitochondrial Diseases; Seizures; Vomiting
Succinate semialdehyde dehydrogenase inhibitor
Small molecule
Approved
OTHER
INTRAVESICAL
HIV Infections; Melanoma; Neoplasms; Osteoarthritis; Contracture; Cystitis, Interstitial; Reflex, Abnormal; Urinary Bladder, Overactive; Urinary Incontinence, Urge; Arthralgia; Cystitis; Infections; Myalgia
Unknown
Small molecule
Approved
Unknown
Unknown
Dermatitis, Atopic; HIV Infections; Malaria; Neoplasms; Psoriasis; Arrhythmias, Cardiac; beta-Thalassemia; Death, Sudden, Cardiac; Heart Diseases; Hypotension, Orthostatic; Obesity; Prader-Willi Syndrome; Premature Birth; Tachycardia, Ventricular; Ventricular Fibrillation; Atherosclerosis; Atrial Fibrillation; Breast Neoplasms; Coronary Disease; Diabetes Mellitus, Type 2; Heart Failure; Hypercholesterolemia; Hypertension; Myocardial Infarction; Non-ST Elevated Myocardial Infarction; ST Elevation Myocardial Infarction; Cardiovascular Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Protein
Approved
Unknown
Unknown
Prostatic Neoplasms, Castration-Resistant; Hypertension; Breast Neoplasms; Leptospirosis; Urinary Bladder, Overactive; Diabetes Insipidus; Enuresis; Renal Colic
Unknown
Small molecule
Approved
OTHER
INJECTION
Unknown
Diagnostic agent
Small molecule
Approved
Unknown
Unknown
Unknown
Cyclooxygenase inhibitor
Small molecule
Approved
Unknown
Unknown
Tuberculosis, Pulmonary; Bacterial Infections; Infections; Pharyngitis
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
OTHER
ORAL
Substance-Related Disorders; Anxiety; Dementia; Depressive Disorder; Schizophrenia; Sleep Initiation and Maintenance Disorders
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
OTHER
OPHTHALMIC
Mycoses; Keratitis; Eye Infections; Infections
Ergosterol sequestering agent
Small molecule
Approved
Unknown
Unknown
Acute Lung Injury; Brain Injuries; Shock; Shock, Septic; Heart Failure; Cardiovascular Diseases
Unknown
Protein
Approved
MUSCULOSKELETAL; OTHER; PREGNANCY AND GYNECOLOGY
INJECTION; NASAL
Menopause; Osteoporosis; Hypercalcemia; Osteitis Deformans; Osteoporosis, Postmenopausal
Calcitonin receptor agonist
Small molecule
Approved
Unknown
Unknown
Anorexia Nervosa; Adenomyosis; Alzheimer Disease; Diabetes Mellitus, Type 1; Intellectual Disability; Obesity; Ovarian Hyperstimulation Syndrome; Parkinson Disease
Unknown
Small molecule
Approved
Unknown
Unknown
Anxiety; Pain
Unknown
Small molecule
Approved
OTHER
ORAL
Psychotic Disorders; Hypertension; Pheochromocytoma
Tyrosine 3-hydroxylase inhibitor
Small molecule
Approved
Unknown
Unknown
Hematologic Neoplasms; Leukemia, Biphenotypic, Acute; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Polycythemia Vera; Primary Myelofibrosis; Thrombocythemia, Essential; Anemia, Refractory; Leukemia, Myeloid; Myelodysplastic Syndromes; Hepatitis B, Chronic; Leukemia; Lymphoma, Non-Hodgkin; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Renal Insufficiency, Chronic; Sarcoma, Kaposi; Leukemia, Lymphoid; Leukemia, Myeloid, Acute; Neoplasms
DNA inhibitor
Small molecule
Approved
Unknown
Unknown
Dry Eye Syndromes; Eye Manifestations; Nasal Obstruction
Unknown
Small molecule
Approved
Unknown
Unknown
Lung Diseases, Obstructive
Unknown
Small molecule
Approved
OTHER
ORAL
Osteomyelitis; Bacterial Infections; Bronchitis, Chronic; Infections; Otitis Media; Pharyngitis; Pneumonia; Sprains and Strains; Tonsillitis; Urinary Tract Infections
Bacterial penicillin-binding protein inhibitor
Small molecule
Unknown
Unknown
Unknown
Alzheimer Disease; Dementia; Depressive Disorder, Major; Phobia, Social; Renal Colic; Amyotrophic Lateral Sclerosis; Bipolar Disorder; Depressive Disorder; Pain; Motion Sickness; Nausea; Postoperative Nausea and Vomiting
Muscarinic acetylcholine receptor M1 antagonist
Small molecule
Approved
OTHER
ORAL
Unknown
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
OTHER
TOPICAL
Unknown
Glucocorticoid receptor agonist
Small molecule
Approved
OTHER
ORAL; TOPICAL
Carcinoma, Non-Small-Cell Lung; Pemphigoid, Benign Mucous Membrane; Pemphigus; Pulmonary Fibrosis; Rosacea; Sarcoidosis; Stroke; Fever; HIV Infections; Malaria; Malaria, Falciparum; Malaria, Vivax; Pneumonia, Pneumocystis; Severe Acute Respiratory Syndrome; Acne Vulgaris; Dermatitis Herpetiformis; Leprosy
Dihydropteroate synthase 1 inhibitor
Small molecule
Approved
Unknown
Unknown
Rheumatic Diseases
Cyclooxygenase inhibitor
Small molecule
Approved
Unknown
Unknown
Cardiovascular Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
INHALATION
Heart Diseases; Opioid-Related Disorders; Hernia, Inguinal; Respiratory Insufficiency; Severe Acute Respiratory Syndrome
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
Unknown
Unknown
Hypotension, Orthostatic; Orthostatic Intolerance; Gastrointestinal Hemorrhage; Hyperemesis Gravidarum; Hypoglycemia; Intestinal Obstruction; Myelodysplastic Syndromes; Pain; Wounds and Injuries; Gastroenteritis; Gastroparesis; Gastroschisis; Headache; HIV Infections; Migraine Disorders; Nausea; Neoplasms; Sepsis; Vomiting; Digestive System Diseases
Unknown
Protein
Approved
OTHER
INJECTION
Unknown
Insulin receptor agonist
Protein
Approved
OTHER
INJECTION
Unknown
Insulin receptor agonist
Small molecule
Approved
Unknown
Unknown
Anxiety; Dementia; Schizophrenia; Depressive Disorder
Unknown