Display Options:
Total: 10647
Small molecule
Approved
OTHER
INJECTION; ORAL; SUBCUTANEOUS
Pregnancy; Alzheimer Disease; Breast Neoplasms; HIV Infections; Pain; Primary Ovarian Insufficiency; Sleep Apnea Syndromes; Bone Diseases; Cardiovascular Diseases; Coronary Disease; Diabetes Mellitus; Endometrial Neoplasms; Heart Diseases; Hot Flashes; Hypercholesterolemia; Hypertension; Infertility; Kidney Neoplasms; Lupus Erythematosus, Systemic; Menopause; Menorrhagia; Myocardial Ischemia; Osteoporosis; Prostatic Neoplasms; Thrombosis; Turner Syndrome; Carcinoma, Renal Cell; Endometriosis; Hyperplasia; Neoplasms; Uterine Hemorrhage
Progesterone receptor agonist
Small molecule
Approved
OTHER; PEDIATRICS; RESPIRATORY
DENTAL; INHALATION; INJECTION; INTRA-ARTICULAR; INTRAMUSCULAR; INTRAVITREAL; NASAL; SUSPENSION; TOPICAL
Fibroma; Hearing Loss; Mucositis; Neuroma, Acoustic; Papilledema; Rotator Cuff Injuries; Tendon Entrapment; Alopecia Areata; Breast Neoplasms; Cataract; Complex Regional Pain Syndromes; Dermatitis, Atopic; Glaucoma; Hand Dermatoses; Humeral Fractures; Keloid; Lichen Planus; Pemphigoid, Benign Mucous Membrane; Psoriasis; Shoulder Pain; Ulnar Neuropathies; Uveal Melanoma; Uveomeningoencephalitic Syndrome; Vitiligo; Wet Macular Degeneration; Chalazion; Choroidal Neovascularization; Cough; Cystitis, Interstitial; Diabetic Retinopathy; Dupuytren Contracture; Eye Injuries; Lichen Planus, Oral; Macular Degeneration; Macular Edema; Optic Neuropathy, Ischemic; Osteoarthritis, Hip; Osteoarthritis, Knee; Otitis Media with Effusion; Pemphigus; Radiculopathy; Retinal Vein Occlusion; Rhinitis; Tendinopathy; Uveitis; Vitreoretinopathy, Proliferative; Anemia; Arthritis, Gouty; Arthritis, Rheumatoid; Asthma; Bursitis; Dermatitis; Multiple Sclerosis; Mycoses; Nasal Obstruction; Osteoarthritis; Pain; Rhinitis, Allergic, Seasonal; Serum Sickness; Skin Diseases; Tennis Elbow; Tenosynovitis; Tuberculosis, Pulmonary; Wounds and Injuries
Glucocorticoid receptor agonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Depressive Disorder; Migraine Disorders; Complex Regional Pain Syndromes; Neuralgia; Epilepsy, Absence; Irritable Bowel Syndrome; Seizures; Epilepsy
Voltage-gated T-type calcium channel blocker
Small molecule
Approved
Unknown
Unknown
Pain
Sodium channel alpha subunit blocker
Small molecule
Approved
OTHER
INTRAMUSCULAR
Hypoglycemia; Hypotension, Orthostatic; Insulin Resistance; Orthostatic Intolerance; Postoperative Complications; Prediabetic State; Amyotrophic Lateral Sclerosis; Blood Coagulation Disorders; Bradycardia; Breast Neoplasms; Heart Arrest; Hemorrhage; Hypospadias; Organophosphate Poisoning; Pneumonia, Ventilator-Associated; Rhinitis, Allergic, Seasonal; Amblyopia; Anisometropia; Dwarfism, Pituitary; Headache; Myopia; Myopia, Degenerative; Pain; Strabismus; Digestive System Diseases; Mydriasis; Poisoning
Muscarinic acetylcholine receptor M1 antagonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Adrenergic receptor alpha-2 agonist
Small molecule
Approved
Unknown
Unknown
Compartment Syndromes; Osteoarthritis, Hip; Osteoarthritis, Knee; Pain
Unknown
Small molecule
Approved
OTHER
ORAL
Alcoholism; Chorioretinitis; Diabetes Mellitus; Diabetic Nephropathies; Dry Eye Syndromes; Leukemia; Leukemia, Myeloid, Acute; Melanosis; Non-alcoholic Fatty Liver Disease; Arrhythmogenic Right Ventricular Dysplasia; Cardiomyopathies; Cerebral Hemorrhage; Fatty Liver; Hypertension, Pulmonary; Macular Degeneration; Neoplasms; Neuroblastoma; Polycystic Ovary Syndrome; Puberty, Precocious; Severe Acute Respiratory Syndrome; Acne Vulgaris; Acute Kidney Injury; Aortic Valve Stenosis; Arthritis, Rheumatoid; Atrial Fibrillation; Heart Failure, Diastolic; Muscular Dystrophy, Duchenne; Non-ST Elevated Myocardial Infarction; Polycystic Kidney, Autosomal Dominant; Renal Insufficiency, Chronic; ST Elevation Myocardial Infarction; Ascites; Cardiovascular Diseases; Edema; Essential Hypertension; Fibrosis; Heart Failure; Hyperaldosteronism; Hypertension; Liver Cirrhosis; Myocardial Infarction; Nephrotic Syndrome; Toxemia
Mineralocorticoid receptor antagonist
Small molecule
Approved
OTHER
OPHTHALMIC
Unknown
Acetylcholinesterase inhibitor
Small molecule
Approved
Unknown
Unknown
Glaucoma
Acetylcholinesterase inhibitor
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Bacterial Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Diabetes Mellitus, Type 1; Kidney Calculi; Atherosclerosis; Cerebrovascular Disorders; Coronary Disease; Death, Sudden, Cardiac; Diabetes Mellitus; Diabetes Mellitus, Type 2; Essential Hypertension; Heart Diseases; Hypercholesterolemia; Myocardial Infarction; Myocardial Ischemia; Vascular Diseases; Angina Pectoris; Cardiovascular Diseases; Glomerulonephritis; Heart Failure; Hypertension; Kidney Failure, Chronic; Nephrotic Syndrome; Toxemia
Thiazide-sensitive sodium-chloride cotransporter inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Glaucoma; Hypertension
Unknown
Small molecule
Approved
OTHER
OPHTHALMIC
Ocular Hypertension; Parkinson Disease; Presbyopia; Sialorrhea; Eye Diseases; Mydriasis
Muscarinic acetylcholine receptor M3 antagonist
Small molecule
Approved
OTHER
ORAL
Depressive Disorder, Major; Substance Withdrawal Syndrome; Alcoholism; Anxiety; Anxiety Disorders
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
OTHER
ORAL
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Cardiovascular Diseases
Thiazide-sensitive sodium-chloride cotransporter inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Cardiovascular Diseases
Thiazide-sensitive sodium-chloride cotransporter inhibitor
Small molecule
Approved
OTHER
ORAL
Unknown
Thiazide-sensitive sodium-chloride cotransporter inhibitor
Small molecule
Approved
OTHER
INJECTION; ORAL
Amphetamine-Related Disorders; Hypertension, Pulmonary; Cocaine-Related Disorders; Substance-Related Disorders; Vascular Diseases; Atherosclerosis; Cardiovascular Diseases; Cerebrovascular Disorders; Coronary Disease; Diabetes Mellitus, Type 2; Heart Diseases; Hypercholesterolemia; Hypertension
Synaptic vesicular amine transporter inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Mu opioid receptor agonist
Small molecule
Approved
Unknown
Unknown
Stroke; Abdominal Pain; Alcoholism; Mitral Valve Insufficiency; Severe Acute Respiratory Syndrome; Hypersensitivity
Unknown
Small molecule
Approved
Unknown
Unknown
Alzheimer Disease; Hernia, Inguinal; Hypersensitivity
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Unknown
GABA-A receptor; anion channel positive modulator
Small molecule
Approved
Unknown
Unknown
Unknown
Progesterone receptor agonist
Small molecule
Approved
Unknown
Unknown
Cough
Unknown
Small molecule
Approved
OTHER; PEDIATRICS
INHALATION; INJECTION; INTRAMUSCULAR; INTRAVENOUS; ORAL
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Psychotic Disorders
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
HIV Infections; Hypertension; IgA Vasculitis; Anemia, Sickle Cell; Arthritis, Rheumatoid; Carotid Stenosis; Ovarian Neoplasms; Pancreatic Neoplasms; Angina, Stable; Cardiovascular Diseases; Heart Diseases; Myocardial Ischemia; Severe Acute Respiratory Syndrome; Coronary Artery Disease; Stroke; Thrombosis
3',5'-cyclic phosphodiesterase inhibitor