Display Options:
Total: 10647
Small molecule
Approved
OTHER
ORAL
HIV Infections; Tobacco Use Disorder; Dementia; Depressive Disorder; Schizophrenia; Anxiety; Anxiety Disorders; Mental Disorders
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
Unknown
Unknown
Low Back Pain; Osteoarthritis; Tendinopathy; Anemia; Asthma; Colitis, Ulcerative; Dermatitis; Eye Diseases; Hemorrhoids; Lung Diseases, Obstructive; Nasal Obstruction; Nephrotic Syndrome; Serum Sickness
Glucocorticoid receptor agonist
Small molecule
Approved
Unknown
Unknown
Bacteremia; Gram-Positive Bacterial Infections; Infections; Osteomyelitis; Bacterial Infections
Unknown
Small molecule
Approved
OTHER
ORAL
Unknown
Unknown
Small molecule
Approved
OTHER
INJECTION
Cystic Fibrosis; Neoplasms; Pain; Cataract; Malaria; Urinary Tract Infections; Acidosis
Unknown
Small molecule
Approved
Unknown
Unknown
Central Nervous System Neoplasms; Carcinoma, Renal Cell; Constriction, Pathologic; Glioma; Neurofibromatosis 1; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Histiocytosis, Langerhans-Cell; Hodgkin Disease; Leukemia; Lung Neoplasms; Lymphoma; Lymphoma, Large B-Cell, Diffuse; Lymphoma, T-Cell, Peripheral; Melanoma; Prostatic Neoplasms, Castration-Resistant; Skin Neoplasms; Testicular Neoplasms; Urethral Neoplasms; Urinary Bladder Neoplasms; Neoplasms
Unknown
Small molecule
Unknown
Unknown
Unknown
Asthma; Breast Neoplasms; Hypotension, Orthostatic; Lecithin Cholesterol Acyltransferase Deficiency; Prostatic Neoplasms, Castration-Resistant; Severe Acute Respiratory Syndrome; Carcinoma, Squamous Cell; Histiocytosis, Langerhans-Cell; Melanoma; Pancreatitis, Chronic; Prostatic Neoplasms; Squamous Intraepithelial Lesions; Toothache; Alzheimer Disease; Hemorrhage; Inflammation; Pancreatitis; Premature Birth; Renal Colic; Squamous Cell Carcinoma of Head and Neck; Acute Pain; Arthralgia; Arthritis, Gouty; Arthritis, Rheumatoid; Cardiovascular Diseases; Ductus Arteriosus, Patent; Eye Diseases; Gout; Myalgia; Osteoarthritis; Pain; Rheumatic Diseases; Spondylitis; Spondylitis, Ankylosing
Cyclooxygenase inhibitor
Protein
Approved
OTHER
INJECTION
Unknown
Insulin receptor agonist
Small molecule
Approved
OTHER
ORAL
Diabetes Mellitus; Diabetes Mellitus, Type 2
Sulfonylurea receptor 1, Kir6.2 blocker
Protein
Approved
OTHER
INJECTION
Unknown
Insulin receptor agonist
Small molecule
Approved
OTHER
ORAL
Polycythemia Vera; Neoplasms
DNA inhibitor
Small molecule
Approved
OTHER
ORAL
Inflammatory Bowel Diseases; Leukemia, Biphenotypic, Acute; Osteoarthritis; Tuberculosis; Angina, Stable; Diabetes Mellitus; Essential Hypertension; Fallopian Tube Neoplasms; Hand-Foot Syndrome; Heart Failure; Kidney Calculi; Leishmaniasis; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Myeloid, Acute; Metabolic Syndrome; Multiple Myeloma; Myelodysplastic Syndromes; Myeloproliferative Disorders; Ovarian Neoplasms; Peritoneal Neoplasms; Renal Insufficiency, Chronic; Bipolar Disorder; Cardiovascular Diseases; Colitis, Ulcerative; Diabetes Mellitus, Type 2; Heart Diseases; Hernias, Diaphragmatic, Congenital; Hypertension; Hyperuricemia; Lymphoma, Non-Hodgkin; Obesity; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Sprains and Strains; Tumor Lysis Syndrome; Gout; Leukemia; Lymphoma; Neoplasms; Response Evaluation Criteria in Solid Tumors
Xanthine dehydrogenase inhibitor
Protein
Unknown
Unknown
Unknown
Coronary Disease; Diabetes Mellitus; Diabetes Mellitus, Type 1; Diabetes Mellitus, Type 2; Insulin Resistance
Insulin receptor agonist
Small molecule
Approved
OTHER
INJECTION; ORAL
Premature Birth; Diabetes Mellitus; Dyspnea; Edema; Leukemia; Leukemia, Myeloid, Acute; Schizophrenia; Acute Kidney Injury; Acute Lung Injury; Bronchopulmonary Dysplasia; Hypertension, Pregnancy-Induced; Keratosis, Actinic; Nasal Polyps; Neoplasms; Renal Insufficiency, Chronic; Atherosclerosis; Bronchiolitis; Coronary Disease; Diabetes Mellitus, Type 2; Essential Hypertension; Hypercholesterolemia; Kidney Diseases; Lung Diseases; Myocardial Infarction; Pre-Eclampsia; Pulmonary Embolism; Renal Insufficiency; Tachypnea; Warts; Cardiovascular Diseases; Fibrosis; Heart Failure; Hypertension; Liver Cirrhosis; Nephrotic Syndrome; Pulmonary Edema; Syndrome
Sodium-(potassium)-chloride cotransporter 2 inhibitor
Small molecule
Approved
OTHER
ORAL
Lymphoma, Non-Hodgkin; Glioblastoma; Histiocytosis, Langerhans-Cell; Hodgkin Disease; Leukemia, Lymphoid; Anemia, Refractory; Anemia, Refractory, with Excess of Blasts; Brain Neoplasms; Leukemia; Leukemia, Basophilic, Acute; Leukemia, Biphenotypic, Acute; Leukemia, Erythroblastic, Acute; Leukemia, Megakaryoblastic, Acute; Leukemia, Monocytic, Acute; Leukemia, Myeloid, Acute; Leukemia, Myelomonocytic, Acute; Leukemia, Myelomonocytic, Chronic; Lymphoma; Myelodysplastic Syndromes; Myeloproliferative Disorders; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Precursor T-Cell Lymphoblastic Leukemia-Lymphoma; Neoplasms
DNA inhibitor
Small molecule
Unknown
Unknown
Unknown
Unknown
Progesterone receptor agonist
Small molecule
Approved
OTHER
ORAL
Bacterial Infections
Bacterial dihydropteroate synthase inhibitor
Small molecule
Approved
OTHER
INJECTION; ORAL
Anxiety; Dementia; Depressive Disorder; Schizophrenia; Psychotic Disorders
Dopamine D2 receptor antagonist
Small molecule
Unknown
Unknown
Unknown
Down Syndrome; Cardiovascular Diseases
Thyroid hormone receptor agonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Unknown
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
DENTISTRY; OTHER
INJECTION; ORAL; PERIODONTAL
Pelvic Inflammatory Disease; Tennis Elbow; Macular Degeneration; Mucositis; Sexually Transmitted Diseases, Bacterial; Telangiectasia, Hereditary Hemorrhagic; Chlamydia Infections; Periodontitis; Rosacea; Acne Vulgaris
Bacterial 70S ribosome inhibitor
Small molecule
Approved
Unknown
Unknown
Leiomyoma; Acromegaly; Anovulation; Hypogonadism; Infertility, Female; Obesity; Paget Disease, Extramammary; Azoospermia; Infertility; Polycystic Ovary Syndrome
Unknown
Small molecule
Approved
OTHER
ORAL
Helminthiasis
Tubulin inhibitor
Small molecule
Approved
Unknown
Unknown
Depressive Disorder
Unknown
Small molecule
Approved
HEMATOLOGY; OTHER
ORAL
Hypertension, Pulmonary; Lung Neoplasms; beta-Thalassemia; Central Nervous System Neoplasms; Esophageal Neoplasms; Fibromatosis, Aggressive; Gliosarcoma; Head and Neck Neoplasms; Hemoglobin SC Disease; Leukemia, Myeloid, Acute; Lymphoma; Meningioma; Multiple Sclerosis; Muscular Atrophy, Spinal; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Stomach Neoplasms; Carcinoma; Glioblastoma; Hematologic Diseases; Hemochromatosis; HIV Infections; Laryngeal Neoplasms; Leukemia; Leukemia, Promyelocytic, Acute; Mouth Neoplasms; Myelodysplastic Syndromes; Myeloproliferative Disorders; Paranasal Sinus Neoplasms; Pharyngeal Neoplasms; Polycythemia Vera; Primary Myelofibrosis; Stroke; Thrombocythemia, Essential; Anemia, Sickle Cell; Carcinoma, Squamous Cell; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Melanoma; Neoplasms
Ribonucleoside-diphosphate reductase RR1 inhibitor
Small molecule
Approved
OTHER
ORAL
Glaucoma; Urinary Bladder Neoplasms; Cardiovascular Diseases; Fibrosis; Heart Failure; Kidney Diseases; Nephrotic Syndrome; Pulmonary Edema
Sodium-(potassium)-chloride cotransporter 2 inhibitor
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Dysuria; Bacterial Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Child Development Disorders, Pervasive; Hypoglycemia; Osteoporosis; Depressive Disorder, Major; Fibromyalgia; Hemangioma, Cavernous, Central Nervous System; Kidney Diseases; Memory Disorders; Orthostatic Intolerance; Pulmonary Disease, Chronic Obstructive; Alcohol Drinking; Anemia, Sickle Cell; Asthma; Brain Injuries; Breast Neoplasms; Burns; Carcinoma, Hepatocellular; Carcinoma, Renal Cell; Cocaine-Related Disorders; Diabetes Mellitus, Type 1; Dystocia; Hemangiosarcoma; Hypertension; Hypotension; Hypotension, Orthostatic; Low Back Pain; Lymphedema; Marfan Syndrome; Melanoma; Migraine with Aura; Migraine without Aura; Multiple Myeloma; Pain; Pancreatic Neoplasms; Panic Disorder; Papilloma; Retinopathy of Prematurity; Shoulder Pain; Sleep Apnea, Obstructive; Stomach Neoplasms; Stress Disorders, Post-Traumatic; Stroke; Substance-Related Disorders; Syncope; Wounds and Injuries; Anxiety; Ascites; Colorectal Neoplasms; Death, Sudden, Cardiac; Esophageal and Gastric Varices; Headache; Hemangioma; Hypertension, Portal; Liver Cirrhosis; Migraine Disorders; Myocardial Infarction; Myocardial Ischemia; Smoking Cessation; Tachycardia, Supraventricular; Telangiectasia, Hereditary Hemorrhagic; Ventricular Fibrillation; Cardiovascular Diseases
Unknown
Small molecule
Approved
OTHER
ORAL
Lymphoma, T-Cell, Cutaneous; Osteomyelitis; Melanoma; Adenomatous Polyposis Coli; Amyloidosis; Amyloidosis, Familial; Aneurysm; Aortic Aneurysm, Abdominal; Blepharitis; Carcinoma, Non-Small-Cell Lung; Colitis, Ulcerative; Colorectal Neoplasms; Crohn Disease; Cystic Fibrosis; Dermatitis, Atopic; Diabetic Foot; Diabetic Retinopathy; Dry Eye Syndromes; Eczema; Eye Burns; Graves Ophthalmopathy; Lichen Planus, Oral; Lymphoma, Follicular; Lymphoma, Non-Hodgkin; Mansonelliasis; Marfan Syndrome; Mycosis Fungoides; Myocardial Infarction; Neoplasms; Pain; Pancreatic Neoplasms; Pelvic Inflammatory Disease; Plague; Reperfusion Injury; Seizures; Sezary Syndrome; Squamous Cell Carcinoma of Head and Neck; Tuberculosis; Alzheimer Disease; Arthritis, Reactive; Chlamydia Infections; Elephantiasis, Filarial; Hemorrhage; Idiopathic Pulmonary Fibrosis; Lyme Disease; Lymphoma; Osteoarthritis; Persian Gulf Syndrome; Pleural Effusion; Pulmonary Disease, Chronic Obstructive; Scrub Typhus; Severe Acute Respiratory Syndrome; Syphilis; Urethritis; Acne Vulgaris; Anthrax; Bacterial Infections; Brucellosis; Cholera; Gonorrhea; Infections; Malaria; Periodontitis; Pneumonia; Psittacosis; Rocky Mountain Spotted Fever; Rosacea; Spotted Fever Group Rickettsiosis; Tularemia; Typhus, Epidemic Louse-Borne
Bacterial 70S ribosome inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Osteomyelitis; Infections; Urinary Tract Infections
DNA inhibitor
Small molecule
Approved
OTHER
ORAL
Diabetes Mellitus; Pain; Hemorrhage; Dysmenorrhea; Rheumatic Diseases
Cyclooxygenase inhibitor
Small molecule
Approved
Unknown
Unknown
Bipolar Disorder; Pain
Unknown
Small molecule
Approved
OTHER
ORAL
Psychotic Disorders; Schizophrenia
Dopamine D2 receptor antagonist