Display Options:
Total: 10647
Small molecule
Approved
OTHER
INJECTION
Unknown
Unknown
Small molecule
Approved
OTHER
INTRAVENOUS; ORAL
Acute Kidney Injury; Alzheimer Disease; Ankle Fractures; Bipolar Disorder; Glycogen Storage Disease Type III; Hypotension, Orthostatic; Malaria; Muscular Dystrophy, Duchenne; Osteoarthritis, Knee; Premature Birth; Rhinitis, Allergic, Seasonal; Uveal Melanoma; Brachial Plexus Neuritis; Bronchopulmonary Dysplasia; Cognitive Dysfunction; Depressive Disorder, Major; Diabetes Mellitus, Type 1; Emphysema; Enuresis; Epilepsies, Partial; Epilepsy; Glioma; Granulomatous Disease, Chronic; Hemorrhage; Hypertension; Kidney Neoplasms; Muscular Diseases; Pancreatitis; Periodontitis; Pre-Eclampsia; Retinopathy of Prematurity; Sinusitis; Spondylarthropathies; Spondylosis; Stomatitis, Aphthous; Sunburn; Temporomandibular Joint Disorders; Tension-Type Headache; Tooth Diseases; Tuberculosis; Wounds and Injuries; Altitude Sickness; Breast Neoplasms; Burns; Causalgia; Cerebral Palsy; Chronic Pain; Fractures, Bone; HIV Infections; Hypospadias; Infections; Low Back Pain; Mucopolysaccharidosis I; Multiple Sclerosis; Neck Pain; Peptic Ulcer; Pulpitis; Respiratory Distress Syndrome; Shock, Septic; Sleep Apnea, Obstructive; Sprains and Strains; Tibial Fractures; Vasculitis; Acute Pain; Arthralgia; Arthritis; Arthritis, Juvenile; Arthritis, Rheumatoid; Back Pain; Cardiovascular Diseases; Common Cold; Ductus Arteriosus, Patent; Dysmenorrhea; Fever; Headache; Influenza, Human; Migraine Disorders; Muscle Cramp; Myalgia; Osteoarthritis; Pain; Pharyngitis; Rheumatic Diseases; Toothache; Vaginitis
Cyclooxygenase inhibitor
Small molecule
Approved
Unknown
Unknown
Hypersensitivity
Unknown
Small molecule
Approved
OTHER
TOPICAL
Lice Infestations; Ectoparasitic Infestations
GABA-A receptor negative allosteric modulator
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Bacterial Infections
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
Unknown
Unknown
Attention Deficit Disorder with Hyperactivity; Psychotic Disorders
Unknown
Small molecule
Approved
OTHER
ORAL
Neoplasms; Prostatic Neoplasms, Castration-Resistant; Small Cell Lung Carcinoma; Carcinoma, Squamous Cell; Hypertension; Laryngeal Neoplasms; Leukemia, Lymphocytic, Chronic, B-Cell; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Prostatic Neoplasms; Angina, Stable
Osmotic agent
Small molecule
Approved
Unknown
Unknown
Bacterial Infections
Unknown
Small molecule
Approved
OTHER
TOPICAL
Skin Diseases
Glucocorticoid receptor agonist
Small molecule
Approved
Unknown
Unknown
Breast Carcinoma In Situ; Breast Neoplasms, Male; Carcinoma, Pancreatic Ductal; Castleman Disease; Hematologic Diseases; Immunoglobulin Light-chain Amyloidosis; Lymphoma, B-Cell; Lymphoma, Primary Effusion; Lymphoma, T-Cell, Cutaneous; Melanoma; Thymoma; Urethral Neoplasms; Adrenal Cortex Neoplasms; Astrocytoma; Blast Crisis; Blastic Plasmacytoid Dendritic Cell Neoplasm; Bone Neoplasms; Burkitt Lymphoma; Carcinoma, Adenoid Cystic; Carcinoma, Intraductal, Noninfiltrating; Carcinoma, Non-Small-Cell Lung; Carcinoma, Ovarian Epithelial; Carcinoma, Renal Cell; Carcinosarcoma; Cholangiocarcinoma; Glioblastoma; Glioma; Hemangiosarcoma; Hematologic Neoplasms; Hereditary Breast and Ovarian Cancer Syndrome; Leukemia, Lymphoid; Leukemia, Myeloid, Acute; Leukemia, Plasma Cell; Liposarcoma; Lung Neoplasms; Lymphoma, AIDS-Related; Lymphoma, Large-Cell, Anaplastic; Lymphoma, T-Cell; Mesothelioma; Mouth Neoplasms; Myelodysplastic Syndromes; Nasopharyngeal Neoplasms; Neoplasm Metastasis; Neoplasms, Plasma Cell; Neuroendocrine Tumors; Oligodendroglioma; Optic Nerve Glioma; Pancreatic Neoplasms; Paraganglioma; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Rhabdomyosarcoma; Salivary Gland Neoplasms; Stomach Neoplasms; Thyroid Neoplasms; Uterine Cervical Neoplasms; Wilms Tumor; Brain Neoplasms; Breast Neoplasms; Carcinoma; Carcinoma, Hepatocellular; Choroid Plexus Neoplasms; Desmoid Tumors; Endometrial Neoplasms; Fallopian Tube Neoplasms; Ganglioneuroblastoma; Granuloma, Lethal Midline; Hepatoblastoma; Hodgkin Disease; Immunoblastic Lymphadenopathy; Inflammatory Breast Neoplasms; Kidney Neoplasms; Leiomyosarcoma; Leukemia; Leukemia, Biphenotypic, Acute; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia-Lymphoma, Adult T-Cell; Liver Neoplasms; Lymphohistiocytosis, Hemophagocytic; Lymphoma; Lymphoma, B-Cell, Marginal Zone; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Lymphoma, Non-Hodgkin; Lymphoma, T-Cell, Peripheral; Multiple Myeloma; Neuroblastoma; Neutropenia; Osteosarcoma; Ovarian Neoplasms; Peritoneal Neoplasms; Postoperative Nausea and Vomiting; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Precursor T-Cell Lymphoblastic Leukemia-Lymphoma; Retinoblastoma; Sarcoma; Sarcoma, Ewing; Sarcoma, Kaposi; Small Cell Lung Carcinoma; Triple Negative Breast Neoplasms; Urinary Bladder Neoplasms; Waldenstrom Macroglobulinemia; Neoplasms
Unknown
Small molecule
Approved
OTHER
INJECTION
Atrophic Vaginitis
Androgen Receptor agonist
Small molecule
Approved
OTHER
OPHTHALMIC
Myopia; Urinary Incontinence; Dry Eye Syndromes; Presbyopia; Glaucoma; Glaucoma, Angle-Closure; Glaucoma, Open-Angle; Miosis; Ocular Hypertension; Sjogren's Syndrome; Xerostomia
Muscarinic acetylcholine receptor M1 agonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Glioma; Hookworm Infections; Pruritus; Anemia; Colorectal Neoplasms; Necatoriasis; Helminthiasis
Tubulin inhibitor
Small molecule
Approved
Unknown
Unknown
Diabetes Mellitus, Type 1; Neuralgia; Purpura, Thrombocytopenic, Idiopathic; Asthma; Pulmonary Disease, Chronic Obstructive; Lung Diseases, Obstructive
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Carnitine O-palmitoyltransferase 1, muscle isoform inhibitor
Small molecule
Approved
IMMUNE SYSTEM; PREGNANCY AND GYNECOLOGY
BUCCAL; INJECTION
Intertrigo; Stomatitis; HIV Infections; Otomycosis; Infections; Mycoses; Pruritus; Tinea; Tinea Pedis
Cytochrome P450 51 inhibitor
Small molecule
Approved
Unknown
Unknown
Bacterial Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Depressive Disorder; Diabetes Mellitus; Cognitive Dysfunction; Heart Failure; Premature Birth; Hernias, Diaphragmatic, Congenital; Parkinson Disease; Shock; Shock, Septic; Cardiovascular Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Bile acids sequestering agent
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Gram-Positive Bacterial Infections; Mastitis; Enterobacteriaceae Infections; Staphylococcal Infections; Bacterial Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Diabetic Cardiomyopathies; Heart Failure; Heart Failure, Diastolic; Cardiomyopathy, Hypertrophic; Cardiovascular Diseases
Unknown
Small molecule
Approved
OTHER
ORAL
Amyotrophic Lateral Sclerosis; Angelman Syndrome; Asthma; Diabetic Retinopathy; Hypertension; Hypotension, Orthostatic; Tobacco Use Disorder; Albinism; Albinism, Oculocutaneous; Aphasia; Attention Deficit Disorder with Hyperactivity; Back Pain; Chronic Pain; Cocaine-Related Disorders; Fibromyalgia; Macular Degeneration; Multiple Sclerosis; Pain; Retinitis Pigmentosa; Schizophrenia; Spinal Cord Injuries; Amblyopia; Dysautonomia, Familial; Stroke; Parkinson Disease; Parkinson Disease, Postencephalitic; Parkinson Disease, Secondary; Wounds and Injuries
DOPA decarboxylase inhibitor
Small molecule
Approved
OTHER
TOPICAL
Dermatitis, Atopic; Oral Submucous Fibrosis; Lichen Planus, Oral; Sinusitis; Gout; Periarthritis; Infections; Psoriasis; Skin Diseases
Glucocorticoid receptor agonist
Small molecule
Approved
Unknown
Unknown
Unknown
Dopamine transporter releasing agent
Small molecule
Approved
OTHER
ORAL
Unknown
Dihydropteroate synthetase inhibitor
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; MUSCULOSKELETAL; OTHER; PREGNANCY AND GYNECOLOGY; RHEUMATOLOGY
ORAL; TOPICAL; TRANSDERMAL; VAGINAL
Blood Coagulation Disorders; Cerebral Arterial Diseases; Diabetes Mellitus; Diabetes Mellitus, Type 1; Diabetes Mellitus, Type 2; Polycystic Ovary Syndrome; Aging; Alzheimer Disease; Atherosclerosis; Bulimia Nervosa; Carcinoid Tumor; Depression, Postpartum; Depressive Disorder; Dry Eye Syndromes; Hereditary Breast and Ovarian Cancer Syndrome; HIV Infections; Migraine Disorders; Prostatic Neoplasms; Psychotic Disorders; Schizophrenia; Severe Acute Respiratory Syndrome; Triple Negative Breast Neoplasms; Urinary Tract Infections; Amenorrhea; Anorexia Nervosa; Bone Diseases, Metabolic; Coronary Disease; Dysmenorrhea; Endometriosis; Heart Diseases; Hot Flashes; Infertility; Multiple Sclerosis; Myocardial Ischemia; Non-alcoholic Fatty Liver Disease; Obesity; Pain; Prostatic Neoplasms, Castration-Resistant; Sexual Dysfunction, Physiological; Stress Disorders, Post-Traumatic; Turner Syndrome; Atrophic Vaginitis; Atrophy; Breast Neoplasms; Dyspareunia; Hypogonadism; Menopause; Osteoporosis; Osteoporosis, Postmenopausal; Primary Ovarian Insufficiency
Estrogen receptor alpha agonist
Small molecule
Approved
OTHER
INJECTION; ORAL
Angioedemas, Hereditary; Cytomegalovirus Infections; Depressive Disorder; Depressive Disorder, Major; Diabetes Mellitus; Diabetes Mellitus, Type 2; Epilepsy; Essential Hypertension; Head and Neck Neoplasms; Hepatitis B, Chronic; Hepatitis C; HIV Infections; Infections; Inflammation; Influenza, Human; Leukemia, Myeloid, Acute; Melanoma; Myelodysplastic Syndromes; Nausea; Neoplasms; Obesity; Pain; Pulmonary Disease, Chronic Obstructive; Substance-Related Disorders; von Hippel-Lindau Disease; Arthritis, Rheumatoid; Breast Neoplasms; Carcinoma, Non-Small-Cell Lung; Keratosis, Actinic; Non-alcoholic Fatty Liver Disease; Pancreatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Sarcoma, Kaposi; Arrhythmias, Cardiac; Tachycardia, Supraventricular; Atrial Fibrillation; Cardiovascular Diseases; Heart Failure
Sodium/potassium-transporting ATPase inhibitor
Protein
Approved
Unknown
Unknown
Infertility
Luteinizing hormone/Choriogonadotropin receptor agonist
Small molecule
Approved
OTHER; UROLOGY AND KIDNEY
TRANSDERMAL
Paget Disease, Extramammary; Rhinitis, Allergic, Seasonal; Sialorrhea; Sleep Apnea, Obstructive; Sleep Apnea Syndromes; Breast Neoplasms; Enuresis; Hyperhidrosis; Polyneuropathies; Urinary Bladder, Neurogenic; Polyuria; Urinary Bladder, Overactive; Urinary Incontinence; Urinary Incontinence, Urge
Muscarinic acetylcholine receptor M2 antagonist
Small molecule
Approved
Unknown
Unknown
Asthma; Pulmonary Disease, Chronic Obstructive; Tobacco Use Disorder; Migraine Disorders; Neuralgia; Anxiety; Delirium; Bipolar Disorder; Mental Disorders; Psychomotor Agitation; Psychotic Disorders; Schizophrenia
D2-like dopamine receptor antagonist
Small molecule
Approved
OTHER; RESPIRATORY
INHALATION; OPHTHALMIC
Bronchopulmonary Dysplasia; Diabetic Foot; Dry Eye Syndromes; Osteomyelitis; Renal Insufficiency, Chronic; Sinusitis; Bronchiectasis; Pneumonia, Bacterial; Blepharitis; Cataract; Conjunctivitis, Bacterial; Fractures, Bone; Pneumonia; Pseudomonas Infections; Bacterial Infections; Conjunctivitis, Allergic; Cystic Fibrosis; Eye Infections; Infections; Inflammation; Respiratory Tract Infections
70S ribosome inhibitor
Small molecule
Approved
Unknown
Unknown
Cocaine-Related Disorders; Attention Deficit Disorder with Hyperactivity
Unknown