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Total: 10647
Small molecule
Approved
Unknown
Unknown
Pain; Postoperative Nausea and Vomiting; Psychotic Disorders
D2-like dopamine receptor antagonist
Protein
Approved
Unknown
Unknown
Adrenal Gland Diseases; Hypertension; Glomerulonephritis, Membranous; Spasms, Infantile
Melanocortin receptor 2 agonist
Small molecule
Approved
Unknown
Unknown
Dermatitis, Atopic; Epidermolysis Bullosa Dystrophica; Muscular Dystrophy, Duchenne; Osteomyelitis; Pneumonia, Ventilator-Associated; Chorioamnionitis; Cystic Fibrosis; Diabetic Foot; Folliculitis; Leishmaniasis; Leishmaniasis, Cutaneous; Meniere Disease; Neoplasms; Urinary Tract Infections; Breast Neoplasms; Cat-Scratch Disease; Colonic Neoplasms; Eczema; Infections; Kidney Calculi; Pain; Plague; Premature Birth; Rectal Neoplasms; Sepsis; Bacterial Infections; Eye Infections
Unknown
Small molecule
Approved
OTHER
ORAL
Central Nervous System Neoplasms; Head and Neck Neoplasms; Arthritis, Rheumatoid; Cystinuria; Hepatolenticular Degeneration; Inflammation; Rheumatic Diseases; Spondylitis
Copper chelating agent
Small molecule
Approved
Unknown
Unknown
Polyuria; Urinary Incontinence
Unknown
Small molecule
Approved
Unknown
Unknown
Alcoholism; Autistic Disorder; Brain Injuries; Cerebral Amyloid Angiopathy; Cerebral Hemorrhage; Child Development Disorders, Pervasive; Cholangitis, Sclerosing; Fibromyalgia; Glioblastoma; Glioma; Hemorrhage; Macular Edema; Memory Disorders; Osteomyelitis; Paraganglioma; Periapical Periodontitis; Pneumonia; Retinal Vein Occlusion; Retinitis Pigmentosa; Skin Diseases; Angelman Syndrome; Asthma; Atrial Fibrillation; Autoimmune Diseases of the Nervous System; Carcinoma, Non-Small-Cell Lung; Carotid Stenosis; Chronic Pain; Colorectal Neoplasms; Cystic Fibrosis; Depressive Disorder, Major; Esophageal Neoplasms; Fragile X Syndrome; Head and Neck Neoplasms; HIV Infections; Huntington Disease; Impetigo; Inflammatory Bowel Diseases; Lung Neoplasms; Macular Degeneration; Multiple Myeloma; Multiple Sclerosis, Relapsing-Remitting; Mycobacterium avium-intracellulare Infection; Neuralgia; Obsessive-Compulsive Disorder; Oropharyngeal Neoplasms; Pancreatic Neoplasms; Parkinson Disease; Retinal Detachment; Stroke; Amyotrophic Lateral Sclerosis; Arthritis, Rheumatoid; Bipolar Disorder; Depressive Disorder; Depressive Disorder, Treatment-Resistant; Heroin Dependence; Hypertension; Idiopathic Pulmonary Fibrosis; Lichen Planus, Oral; Multiple Sclerosis; Neurobehavioral Manifestations; Peri-Implantitis; Periodontitis; Pneumothorax; Psychotic Disorders; Rosacea; Schizophrenia; Spinal Cord Injuries; Substance-Related Disorders; Acne Vulgaris; Bacterial Infections; Infections
Unknown
Small molecule
Approved
OTHER
ORAL
Adrenal Cortex Neoplasms; Carcinoma in Situ; Dementia; Head and Neck Neoplasms; HIV Wasting Syndrome; Pulmonary Disease, Chronic Obstructive; Uterine Neoplasms; Breast Neoplasms; Endometrial Neoplasms; Hot Flashes; Liver Neoplasms; Acquired Immunodeficiency Syndrome; Anorexia; Cachexia; Neoplasms; Primary Immunodeficiency Diseases
Progesterone receptor agonist
Small molecule
Approved
Unknown
Unknown
Infections; Bacteremia; Gram-Positive Bacterial Infections; Osteomyelitis; Bacterial Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Hyperemia; Neoplasms; Common Cold; Conjunctivitis, Allergic; Influenza, Human; Respiratory Tract Diseases; Eye Manifestations; Nasal Obstruction
Unknown
Protein
Approved
Unknown
Unknown
Osteomyelitis; Tuberculosis
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Leukemia, Myeloid, Acute; Urinary Bladder, Overactive; Breast Neoplasms; Cellulitis; Dermatitis; Eczema; Staphylococcal Infections; Tuberculosis; Urinary Tract Infections; Cystic Fibrosis; Nasal Obstruction; Skin Diseases; Urinary Bladder Neoplasms; Bacterial Infections; Infections; Otitis Media; Prostatitis; Respiratory Tract Infections; Sprains and Strains
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
OTHER
ORAL
Astrocytoma; Brain Neoplasms; Carcinoma, Hepatocellular; Colorectal Neoplasms; Digestive System Neoplasms; Glioblastoma; Gliosarcoma; Neoplasms; Oligodendroglioma; Intracranial Hypertension; Meningitis, Cryptococcal; Candidiasis; Infections; Meningitis
Thymidylate synthase inhibitor
Small molecule
Approved
OTHER
ORAL
HIV Infections; Osteomyelitis; Acquired Immunodeficiency Syndrome; Meningitis; Tuberculosis, Multidrug-Resistant; Tuberculosis; Tuberculosis, Pulmonary
70S ribosome inhibitor
Small molecule
Approved
DERMATOLOGY; OTHER
ORAL; TOPICAL
Amyotrophic Lateral Sclerosis; Autistic Disorder; Glioblastoma; Hematologic Neoplasms; Hypercholesterolemia; Myelodysplastic-Myeloproliferative Diseases; Neoplasms, Plasma Cell; Anemia; Anti-Neutrophil Cytoplasmic Antibody-Associated Vasculitis; Carcinoma, Adenoid Cystic; Cholangitis, Sclerosing; Colorectal Neoplasms; Emphysema; Keratosis, Actinic; Kidney Neoplasms; Lung Neoplasms; Lymphoma; Melanoma; Multiple Myeloma; Neuroblastoma; Pancreatic Neoplasms; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Severe Acute Respiratory Syndrome; Small Cell Lung Carcinoma; Striae Distensae; Breast Neoplasms; Carcinoma, Basal Cell; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Leukemia; Leukemia, Myeloid, Acute; Myelodysplastic Syndromes; Myeloproliferative Disorders; Purpura, Thrombocytopenic, Idiopathic; Rosacea; Skin Neoplasms; Acne Vulgaris; Hyperpigmentation; Leukemia, Promyelocytic, Acute; Melanosis; Neoplasms
Retinoic acid receptor agonist
Small molecule
Approved
Unknown
Unknown
Analgesia; Hepatitis C; Intestinal Obstruction; Paget Disease, Extramammary; Diabetes Mellitus, Type 1; Diabetic Neuropathies; Feeding and Eating Disorders; Hypogonadism; Irritable Bowel Syndrome; Neuralgia; Obesity; Pruritus; Chronic Pain; Epilepsy; Heroin Dependence; Low Back Pain; Morphine Dependence; Mycosis Fungoides; Opioid-Related Disorders; Osteoarthritis; Pain; Parkinson Disease; Restless Legs Syndrome; Sezary Syndrome; Substance-Related Disorders; Substance Withdrawal Syndrome; Constipation
Unknown
Small molecule
Approved
OTHER
TOPICAL
Psoriasis; Breast Neoplasms; Dermatitis, Atopic; Hemorrhoids; Skin Diseases
Glucocorticoid receptor agonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Anti-Neutrophil Cytoplasmic Antibody-Associated Vasculitis; Arthritis, Rheumatoid; Carcinoma, Non-Small-Cell Lung; Constipation; Coronary Disease; Diabetes Mellitus; Diabetes Mellitus, Type 2; Endometriosis; Erectile Dysfunction; Essential Hypertension; Hematologic Neoplasms; Hepatitis B, Chronic; HIV Infections; Hodgkin Disease; Hypercalcemia; Hypertension, Pulmonary; Leukemia, Lymphocytic, Chronic, B-Cell; Lymphoma; Lymphoma, Non-Hodgkin; Melanoma; Mycoses; Nausea; Neoplasms; Non-alcoholic Fatty Liver Disease; Osteomyelitis; Pain; Parkinson Disease; Primary Myelofibrosis; Renal Insufficiency; Renal Insufficiency, Chronic; Respiratory Syncytial Virus Infections; Rhinoscleroma; Sepsis; Severe Acute Respiratory Syndrome; Thrombosis; Acquired Immunodeficiency Syndrome; Buruli Ulcer; Cystic Fibrosis; Multiple Sclerosis; Mycobacterium avium-intracellulare Infection; Onchocerciasis; Sarcoidosis; Alzheimer Disease; Arthritis, Reactive; Diarrhea; Endocarditis; Enterocolitis, Pseudomembranous; Infections; Leprosy; Meningitis; Multiple System Atrophy; Tuberculosis; Tuberculosis, Pulmonary
Bacterial DNA-directed RNA polymerase inhibitor
Small molecule
Approved
OTHER
ORAL
Pain
Mu opioid receptor agonist
Small molecule
Approved
OTHER
ORAL
Osteomyelitis; Bacterial Infections; Eye Infections
Bacterial dihydropteroate synthase inhibitor
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Bacterial Infections
Unknown
Small molecule
Approved
OTHER
ORAL
Anxiety; Anxiety Disorders; Seizures
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
OTHER
INTRAOCULAR
Presbyopia; Cataract; Glaucoma; Miosis
Muscarinic acetylcholine receptor M3 agonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
EMERGENCY MEDICINE; NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
INJECTION
Aortic Coarctation; Brain Neoplasms; Hernia, Ventral; HIV Infections; Lung Diseases; Neuralgia; Obesity, Morbid; Prostatic Neoplasms, Castration-Resistant; Sarcoma; Sinusitis; Stress Disorders, Post-Traumatic; Subarachnoid Hemorrhage; Vasospasm, Intracranial; Abdominal Pain; Appendicitis; Atrial Fibrillation; Blepharoptosis; Blood Coagulation Disorders; Cleft Palate; Complex Regional Pain Syndromes; Dupuytren Contracture; Fasciitis, Plantar; Femoral Neck Fractures; Headache; Hemorrhage; Hernia, Umbilical; Hip Fractures; Hypospadias; Hypotension; Lacrimal Apparatus Diseases; Low Back Pain; Mucositis; Musculoskeletal Diseases; Osteoarthritis, Hip; Pregnancy; Pulpitis; Rib Fractures; Shoulder Pain; Spinal Stenosis; Analgesia; Ankle Fractures; Breast Neoplasms; Breech Presentation; Carcinoma, Non-Small-Cell Lung; Chronic Pain; Cough; Fractures, Bone; Genital Neoplasms, Female; Hallux Valgus; Hemorrhoids; Hernia, Inguinal; Ileus; Liver Diseases; Lung Neoplasms; Migraine Disorders; Neoplasms; Osteoarthritis; Osteoarthritis, Knee; Pancreatic Neoplasms; Pancreatitis, Chronic; Peritoneal Neoplasms; Postoperative Nausea and Vomiting; Radiculopathy; Radius Fractures; Rotator Cuff Injuries; Toothache; Urethral Stricture; Wounds and Injuries; Acute Pain; Hernia; Pain
Sodium channel protein type IV alpha subunit blocker
Small molecule
Approved
Unknown
Unknown
Aortic Valve Stenosis; Neoplasms; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant
Unknown
Small molecule
Approved
DERMATOLOGY; OTHER
TOPICAL
Dermatitis, Atopic; Eye Diseases; Skin Diseases
Glucocorticoid receptor agonist
Small molecule
Approved
OTHER
OPHTHALMIC; TOPICAL
Corneal Opacity; Dry Eye Syndromes; Acne Vulgaris; Eye Diseases; Hemorrhoids; Inflammation
Glucocorticoid receptor agonist
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Bacterial Infections
Unknown
Small molecule
Approved
CARDIOVASCULAR; DIABETES DRUGS & ENDOCRINOLOGY; OTHER
BUCCAL; IMPLANTATION; INJECTION; NASAL; TRANSDERMAL
Aging; Cerebral Arterial Diseases; Dyspareunia; Insulin Resistance; Kallmann Syndrome; Pain; Penile Induration; Polycystic Ovary Syndrome; Acquired Immunodeficiency Syndrome; Anorexia Nervosa; Carcinoma, Intraductal, Noninfiltrating; Dwarfism; Heart Failure; Hereditary Breast and Ovarian Cancer Syndrome; Multiple Sclerosis; Muscle Weakness; Obesity; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Sarcopenia; Spinal Cord Injuries; Testicular Neoplasms; Coronary Disease; Disorders of Sex Development; Erectile Dysfunction; Hip Fractures; Infertility; Kidney Failure, Chronic; Menopause; Metabolic Syndrome; Hypogonadism; Klinefelter Syndrome; Neoplasms; Orchitis; Sexual Dysfunctions, Psychological
Androgen Receptor agonist
Small molecule
Approved
OTHER
INHALATION
Unknown
GABA-A receptor; anion channel positive modulator
Small molecule
Approved
OTHER
ORAL
Unknown
Androgen Receptor agonist
Small molecule
Approved
OTHER
INJECTION
Unknown
Muscle-type nicotinic acetylcholine receptor antagonist