Display Options:
Total: 10647
Small molecule
Approved
OTHER
INHALATION
Unknown
GABA-A receptor; anion channel positive modulator
Small molecule
Approved
OTHER
INJECTION
Psoriasis
Dopamine D2 receptor antagonist
Small molecule
Approved
OTHER
INJECTION; ORAL; VAGINAL
Prostatic Neoplasms, Castration-Resistant; Neoplasms
Estrogen receptor alpha agonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Melanoma; Obesity; Fractures, Bone; Wounds and Injuries; Arrhythmias, Cardiac; Bacteremia; Cellulitis; Clostridium Infections; Gram-Positive Bacterial Infections; Infections; Laryngeal Neoplasms; Osteomyelitis; Prostatic Neoplasms, Castration-Resistant; Skin Diseases; Staphylococcal Infections; Bacterial Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Heart Diseases; Substance-Related Disorders; Brain Injuries; Status Epilepticus; Sleep Initiation and Maintenance Disorders
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
Unknown
Unknown
Common Cold; Cough; Headache; Nasal Obstruction
Adrenergic receptor alpha-1 agonist
Small molecule
Approved
OTHER
ORAL
Kidney Diseases; Smoldering Multiple Myeloma; Coronary Disease; Graves Disease; Heart Diseases; Hyperlipoproteinemia Type II; Hyperthyroidism; Lipid Metabolism Disorders; Multiple Sclerosis; Myocardial Infarction; Myocardial Ischemia; Cardiovascular Diseases; Hypercholesterolemia; Hypothyroidism; Nephrotic Syndrome
Bile acids sequestering agent
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Tuberculosis, Multidrug-Resistant; Tuberculosis; Bacterial Infections; Eye Infections
Unknown
Small molecule
Approved
OTHER
ORAL
Renal Insufficiency, Chronic; Cardiovascular Diseases; Heart Failure; Hypertension; Toxemia
Thiazide-sensitive sodium-chloride cotransporter inhibitor
Small molecule
Approved
OTHER
BUCCAL; ORAL; SUBLINGUAL
Menopause; Breast Neoplasms; Hypogonadism; Orchitis
Androgen Receptor agonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Protein
Approved
OTHER
INJECTION
Gonadal Disorders; Graft vs Host Disease; Anovulation; Azoospermia; Breast Neoplasms; Hypogonadism; Infertility; Klinefelter Syndrome; Polycystic Ovary Syndrome; Pregnancy
Luteinizing hormone/Choriogonadotropin receptor agonist
Small molecule
Approved
Unknown
Unknown
Infections; Osteomyelitis; Burns
Bacterial dihydropteroate synthase inhibitor
Small molecule
Approved
Unknown
Unknown
Lung Diseases, Obstructive
Unknown
Small molecule
Approved
OTHER
ORAL
Astrocytoma; Brain Neoplasms; Glioblastoma; Granulomatosis with Polyangiitis; Kidney Diseases; Leukemia; Leukemia, Biphenotypic, Acute; Macular Degeneration; Neoplasms; Osteomyelitis; Pulmonary Disease, Chronic Obstructive; Cystic Fibrosis; Dermatitis; Diabetes Mellitus, Type 1; Eczema; Lymphoma, AIDS-Related; Skin Diseases; Abscess; HIV Infections; Idiopathic Pulmonary Fibrosis; Malaria; Measles; Pneumonia; Pyelonephritis; Sepsis; Staphylococcal Infections; Toxoplasmosis, Ocular; Tuberculosis; Bacterial Infections; Infections; Pneumonia, Pneumocystis; Urinary Tract Infections
Bacterial dihydropteroate synthase inhibitor
Small molecule
Approved
Unknown
Unknown
Liver Neoplasms; Stomach Neoplasms; Carcinoma, Squamous Cell; Central Nervous System Neoplasms; Head and Neck Neoplasms; Lymphedema; Lymphoma, T-Cell, Peripheral; Neoplasms, Germ Cell and Embryonal; Rectal Neoplasms; Vulvar Neoplasms; HIV Infections; Hodgkin Disease; Lymphoma; Lymphoma, Large B-Cell, Diffuse; Ovarian Neoplasms; Pericardial Effusion; Seminoma; Sex Cord-Gonadal Stromal Tumors; Testicular Neoplasms; Neoplasms
Unknown
Small molecule
Approved
Unknown
Unknown
Coronary Disease; HIV Infections; Inflammation; Ischemia; Anemia; Anemia, Sickle Cell; Diabetes Mellitus, Type 2; Glaucoma
Unknown
Small molecule
Approved
Unknown
Unknown
Hypersensitivity; Pruritus
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Depressive Disorder; Diabetes Mellitus, Type 2; Obesity; Adenoma, Islet Cell; Hyperinsulinism; Hypertension; Hypoglycemia
Potassium channel, inwardly rectifying, subfamily J, member 11 opener
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Attention Deficit Disorder with Hyperactivity; Cocaine-Related Disorders; Narcolepsy; Obesity
Monoamine transporter inhibitor
Small molecule
Approved
Unknown
Unknown
Keratitis, Herpetic
Unknown
Small molecule
Approved
Unknown
Unknown
Substance-Related Disorders; Asthma
Beta-2 adrenergic receptor agonist
Small molecule
Approved
OTHER
ORAL
Anemia; Astrocytoma; Brain Neoplasms; Glioblastoma; Granulomatosis with Polyangiitis; Kidney Diseases; Leukemia; Leukemia, Biphenotypic, Acute; Macular Degeneration; Neoplasms; Osteomyelitis; Pulmonary Disease, Chronic Obstructive; Cystic Fibrosis; Dermatitis; Diabetes Mellitus, Type 1; Eczema; Epidermolysis Bullosa; Lymphoma, AIDS-Related; Skin Diseases; Abscess; HIV Infections; Idiopathic Pulmonary Fibrosis; Malaria; Measles; Pneumonia; Pyelonephritis; Sepsis; Staphylococcal Infections; Toxoplasmosis, Ocular; Tuberculosis; Bacterial Infections; Infections; Otitis Media; Pneumonia, Pneumocystis; Urinary Tract Infections
Bacterial dihydrofolate reductase inhibitor
Small molecule
Approved
OTHER
ORAL
Rhinitis, Allergic, Seasonal
Histamine H1 receptor antagonist
Small molecule
Approved
Unknown
Unknown
Adenoma; Carcinoma, Renal Cell; Colorectal Neoplasms; Hashimoto Disease; Lung Neoplasms; Lymphoma, Follicular; Prostatic Neoplasms, Castration-Resistant
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
INTRAVENOUS; ORAL
Acute Kidney Injury; Alzheimer Disease; Ankle Fractures; Bipolar Disorder; Glycogen Storage Disease Type III; Hypotension, Orthostatic; Malaria; Muscular Dystrophy, Duchenne; Osteoarthritis, Knee; Premature Birth; Rhinitis, Allergic, Seasonal; Uveal Melanoma; Brachial Plexus Neuritis; Bronchopulmonary Dysplasia; Cognitive Dysfunction; Depressive Disorder, Major; Diabetes Mellitus, Type 1; Emphysema; Enuresis; Epilepsies, Partial; Epilepsy; Glioma; Granulomatous Disease, Chronic; Hemorrhage; Hypertension; Kidney Neoplasms; Muscular Diseases; Pancreatitis; Periodontitis; Pre-Eclampsia; Retinopathy of Prematurity; Sinusitis; Spondylarthropathies; Spondylosis; Stomatitis, Aphthous; Sunburn; Temporomandibular Joint Disorders; Tension-Type Headache; Tooth Diseases; Tuberculosis; Wounds and Injuries; Altitude Sickness; Breast Neoplasms; Burns; Causalgia; Cerebral Palsy; Chronic Pain; Fractures, Bone; HIV Infections; Hypospadias; Infections; Low Back Pain; Mucopolysaccharidosis I; Multiple Sclerosis; Neck Pain; Peptic Ulcer; Pulpitis; Respiratory Distress Syndrome; Shock, Septic; Sleep Apnea, Obstructive; Sprains and Strains; Tibial Fractures; Vasculitis; Acute Pain; Arthralgia; Arthritis; Arthritis, Juvenile; Arthritis, Rheumatoid; Back Pain; Cardiovascular Diseases; Common Cold; Ductus Arteriosus, Patent; Dysmenorrhea; Fever; Headache; Influenza, Human; Migraine Disorders; Muscle Cramp; Myalgia; Osteoarthritis; Pain; Pharyngitis; Rheumatic Diseases; Toothache; Vaginitis
Cyclooxygenase inhibitor
Small molecule
Approved
Unknown
Unknown
Diabetic Cardiomyopathies; Heart Failure; Heart Failure, Diastolic; Cardiomyopathy, Hypertrophic; Cardiovascular Diseases
Unknown
Small molecule
Approved
IMMUNE SYSTEM; PREGNANCY AND GYNECOLOGY
BUCCAL; INJECTION
Intertrigo; Stomatitis; HIV Infections; Otomycosis; Infections; Mycoses; Pruritus; Tinea; Tinea Pedis
Cytochrome P450 51 inhibitor
Small molecule
Approved
Unknown
Unknown
Diabetes Mellitus, Type 1; Neuralgia; Purpura, Thrombocytopenic, Idiopathic; Asthma; Pulmonary Disease, Chronic Obstructive; Lung Diseases, Obstructive
Unknown
Small molecule
Approved
Unknown
Unknown
Diabetes Mellitus, Type 2; Diabetes Mellitus
Acyl coenzyme A:cholesterol acyltransferase 1 inhibitor
Small molecule
Approved
OTHER
OPHTHALMIC
Myopia; Urinary Incontinence; Dry Eye Syndromes; Presbyopia; Glaucoma; Glaucoma, Angle-Closure; Glaucoma, Open-Angle; Miosis; Ocular Hypertension; Sjogren's Syndrome; Xerostomia
Muscarinic acetylcholine receptor M1 agonist