Display Options:
Total: 10647
Small molecule
Approved
OTHER
ORAL
Hypertension
Unknown
Small molecule
Approved
CARDIOVASCULAR; DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Depressive Disorder; Depressive Disorder, Major; Cardiovascular Diseases
Beta-1 adrenergic receptor partial agonist
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Bacterial Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
INJECTION
Unknown
Acetylcholinesterase inhibitor
Protein
Approved
OTHER
NASAL
Unknown
Vasopressin receptor agonist
Small molecule
Approved
Unknown
Unknown
Digestive System Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Diagnostic agent
Protein
Approved
OTHER
INJECTION
Unknown
Unknown
Small molecule
Approved
OTHER
INJECTION
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Epilepsy
Voltage-gated T-type calcium channel blocker
Small molecule
Approved
OTHER
ORAL
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Bacterial Infections
Unknown
Small molecule
Approved
OTHER
INJECTION
Unknown
Mineralocorticoid receptor agonist
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Bacterial Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Pain
Unknown
Small molecule
Approved
OTHER
INJECTION
Endophthalmitis; Osteomyelitis; Appendicitis; Pneumonia; Bacterial Infections; Eye Infections
Unknown
Small molecule
Approved
OTHER
TOPICAL; VAGINAL
Unknown
Cytochrome P450 51 inhibitor
Small molecule
Approved
Unknown
Unknown
Constipation; Urinary Tract Infections
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Fallopian Tube Neoplasms; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Plasma Cell; Lymphoma, Primary Effusion; Myelodysplastic-Myeloproliferative Diseases; Neoplasms, Neuroepithelial; Neuroendocrine Tumors; Peritoneal Neoplasms; Sarcoma, Kaposi; Acquired Immunodeficiency Syndrome; Astrocytoma; Carcinoid Tumor; Carcinoma, Hepatocellular; Carcinoma, Islet Cell; Carcinoma, Large Cell; Carcinoma, Merkel Cell; Carcinoma, Neuroendocrine; Castleman Disease; Esthesioneuroblastoma, Olfactory; Glioblastoma; Glioma; Gliosarcoma; Graft vs Host Disease; Hematologic Diseases; Hematologic Neoplasms; Leukemia, Lymphocytic, Chronic, B-Cell; Lymphoma, AIDS-Related; Lymphoma, B-Cell, Marginal Zone; Lymphoma, Large-Cell, Anaplastic; Lymphoma, T-Cell; Multiple Sclerosis, Relapsing-Remitting; Myasthenia Gravis; Neoplasms, Plasma Cell; Neuromyelitis Optica; Neutropenia; Oligodendroglioma; Opsoclonus-Myoclonus Syndrome; Optic Nerve Glioma; Oropharyngeal Neoplasms; Pancreatic Neoplasms; Paraganglioma; Polyradiculoneuropathy, Chronic Inflammatory Demyelinating; Prostatic Neoplasms; Rhabdomyosarcoma, Alveolar; Rhabdomyosarcoma, Embryonal; Severe Acute Respiratory Syndrome; Stiff-Person Syndrome; Thymoma; Waldenstrom Macroglobulinemia; Adenocarcinoma of Lung; Adrenal Cortex Neoplasms; Anemia, Refractory; Anemia, Refractory, with Excess of Blasts; Brain Neoplasms; Breast Neoplasms; Burkitt Lymphoma; Carcinoma; Carcinoma, Embryonal; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Central Nervous System Neoplasms; Choriocarcinoma; Choroid Plexus Neoplasms; Colorectal Neoplasms; Endodermal Sinus Tumor; Ependymoma; Ganglioneuroblastoma; Gestational Trophoblastic Disease; Granuloma, Lethal Midline; Hepatoblastoma; HIV Infections; Hodgkin Disease; Kidney Neoplasms; Leukemia; Leukemia, Basophilic, Acute; Leukemia, Biphenotypic, Acute; Leukemia, Erythroblastic, Acute; Leukemia, Lymphoid; Leukemia-Lymphoma, Adult T-Cell; Leukemia, Megakaryoblastic, Acute; Leukemia, Monocytic, Acute; Leukemia, Myeloid, Acute; Leukemia, Myelomonocytic, Acute; Leukemia, Myelomonocytic, Chronic; Lymphohistiocytosis, Hemophagocytic; Lymphoma; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Lymphoma, Non-Hodgkin; Lymphoma, T-Cell, Peripheral; Mediastinal Neoplasms; Medulloblastoma; Multiple Myeloma; Myelodysplastic Syndromes; Myeloproliferative Disorders; Neoplasms, Germ Cell and Embryonal; Neuroblastoma; Neuroectodermal Tumors, Primitive; Osteosarcoma; Ovarian Neoplasms; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Precursor T-Cell Lymphoblastic Leukemia-Lymphoma; Prostatic Neoplasms, Castration-Resistant; Retinoblastoma; Rhabdomyosarcoma; Sarcoma; Sarcoma, Ewing; Sarcoma, Myeloid; Seminoma; Sex Cord-Gonadal Stromal Tumors; Stomach Neoplasms; Teratoma; Testicular Neoplasms; Thymus Neoplasms; Wilms Tumor; Carcinoma, Small Cell; Lung Neoplasms; Neoplasms; Small Cell Lung Carcinoma
DNA topoisomerase II inhibitor
Small molecule
Approved
Unknown
Unknown
Pain
Mu opioid receptor agonist
Small molecule
Approved
Unknown
Unknown
Dengue; HIV Infections; Infections; Influenza, Human; Leishmaniasis, Cutaneous; Malaria; Malaria, Falciparum; Plague; Respiratory Syncytial Virus Infections; Schistosomiasis; Severe Acute Respiratory Syndrome; Shock; Staphylococcal Infections; Anthrax; Diabetes Mellitus, Type 1; Hookworm Infections; Influenza in Birds; Pneumonia, Pneumococcal; Stomatitis; Tobacco Use Disorder; Heartburn
Antacid
Small molecule
Approved
Unknown
Unknown
Unknown
Neutralises acid
Small molecule
Approved
Unknown
Unknown
Hypersensitivity
Unknown
Small molecule
Approved
Unknown
Unknown
Cardiovascular Diseases
Unknown
Small molecule
Approved
GASTROINTESTINAL
ORAL
Carcinoma, Medullary; Esophagitis, Peptic; Hypotension, Orthostatic; Immune System Diseases; Neoplasms; Breast Carcinoma In Situ; Breast Neoplasms; Carcinoma, Renal Cell; Helicobacter Infections; Job Syndrome; Leukemia, T-Cell; Postpartum Hemorrhage; Precursor T-Cell Lymphoblastic Leukemia-Lymphoma; Barrett Esophagus; Cough; Multiple Sclerosis; Stomach Ulcer; Gastroesophageal Reflux; Peptic Ulcer
Histamine H2 receptor antagonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Irritable Bowel Syndrome; Paraplegia; Metabolism, Inborn Errors; Xanthomatosis, Cerebrotendinous
Bile acid receptor FXR agonist
Protein
Approved
Unknown
Unknown
Unknown
Unknown
Protein
Approved
Unknown
Unknown
Anemia, Sickle Cell; Angioedemas, Hereditary; Aspergillosis; beta-Thalassemia; Brain Neoplasms; Carcinoma, Renal Cell; Diabetes Mellitus, Type 2; DiGeorge Syndrome; Fanconi Anemia; Mucopolysaccharidoses; Mycosis Fungoides; Myeloproliferative Disorders; Neoplasms, Neuroepithelial; Neutropenia; Osteogenesis Imperfecta; Pulmonary Disease, Chronic Obstructive; Respiratory Syncytial Virus Infections; Sezary Syndrome; Urticaria; Uveitis; Venous Thromboembolism; Acute Kidney Injury; Aortic Aneurysm, Abdominal; Brain Injuries; Bronchiolitis Obliterans Syndrome; Burkitt Lymphoma; Cystitis, Interstitial; Diabetes Mellitus; Fallopian Tube Neoplasms; Glaucoma; Granulomatous Disease, Chronic; Hematologic Neoplasms; Hepatitis C; HIV Infections; Hyperlipoproteinemia Type I; Kidney Neoplasms; Lacrimal Apparatus Diseases; Leprosy; Leukemia, Large Granular Lymphocytic; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Mast-Cell; Leukemia, Prolymphocytic, B-Cell; Leukemia, Prolymphocytic, T-Cell; Liver Diseases; Lung Diseases; Lymphoma, AIDS-Related; Lymphoma, Follicular; Melanoma; Myelodysplastic-Myeloproliferative Diseases; Myocarditis; Myositis; Neoplasm Metastasis; Neoplasms; Neoplasms, Plasma Cell; Neuroblastoma; Optic Atrophy, Hereditary, Leber; Ovarian Neoplasms; Paraparesis, Tropical Spastic; Periodontitis; Prostatic Neoplasms, Castration-Resistant; Pterygium; Renal Artery Obstruction; Reperfusion Injury; Retinoblastoma; Sarcoma; Severe Acute Respiratory Syndrome; Systemic Inflammatory Response Syndrome; Takotsubo Cardiomyopathy; Anemia, Aplastic; Anemia, Hemolytic, Autoimmune; Behcet Syndrome; Breast Neoplasms; Bronchiolitis Obliterans; Carcinoma, Hepatocellular; Colorectal Neoplasms; Conjunctivitis, Allergic; Dermatitis, Atopic; Dermatomyositis; Diabetes Mellitus, Type 1; Dry Eye Syndromes; Eczema; Endocardial Cushion Defects; Glomerulonephritis, Membranoproliferative; Glomerulonephritis, Membranous; Glomerulosclerosis, Focal Segmental; Graft vs Host Disease; Heart Arrest; Heart Diseases; Hepatitis, Autoimmune; Hepatitis C, Chronic; Hodgkin Disease; Infections; Kidney Diseases; Kidney Failure, Chronic; Leukemia; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Lupus Nephritis; Lymphohistiocytosis, Hemophagocytic; Lymphoma; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Lymphoma, Non-Hodgkin; Multiple Myeloma; Myelodysplastic Syndromes; Myocardial Infarction; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Purpura, Thrombocytopenic, Idiopathic; Purpura, Thrombotic Thrombocytopenic; Red-Cell Aplasia, Pure; Renal Insufficiency; Renal Insufficiency, Chronic; Retinal Vasculitis; Skin Neoplasms; Stevens-Johnson Syndrome; Waldenstrom Macroglobulinemia; Arthritis, Rheumatoid; Conjunctivitis; Corneal Diseases; Eye Diseases; Immune System Diseases; Inflammation; Keratitis; Keratoconjunctivitis; Psoriasis
Cyclophilin A modulator
Protein
Approved
OTHER
INJECTION
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Migraine Disorders
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown