Display Options:
Total: 10647
Small molecule
Approved
Unknown
Unknown
Pain
Unknown
Small molecule
Approved
OTHER
INJECTION
HIV Wasting Syndrome; Hip Fractures; Malnutrition; Eye Diseases
Androgen Receptor agonist
Small molecule
Approved
OTHER
INJECTION; ORAL
Neoplasms, Neuroepithelial; Fallopian Tube Neoplasms; Graft vs Host Disease; Hematologic Neoplasms; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Plasma Cell; Lymphoma, B-Cell; Myelodysplastic-Myeloproliferative Diseases; Peritoneal Neoplasms; Sarcoma, Kaposi; Acquired Immunodeficiency Syndrome; Astrocytoma; Carcinoid Tumor; Carcinoma, Hepatocellular; Carcinoma, Islet Cell; Carcinoma, Merkel Cell; Carcinoma, Neuroendocrine; Castleman Disease; Glioblastoma; Glioma; Gliosarcoma; Hematologic Diseases; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Lymphoid; Lymphoma, AIDS-Related; Lymphoma, Large-Cell, Anaplastic; Lymphoma, T-Cell; Multiple Sclerosis, Relapsing-Remitting; Myasthenia Gravis; Neuromyelitis Optica; Neutropenia; Oligodendroglioma; Opsoclonus-Myoclonus Syndrome; Optic Nerve Glioma; Oropharyngeal Neoplasms; Pancreatic Neoplasms; Polyradiculoneuropathy, Chronic Inflammatory Demyelinating; Precursor T-Cell Lymphoblastic Leukemia-Lymphoma; Rhabdomyosarcoma, Alveolar; Rhabdomyosarcoma, Embryonal; Severe Acute Respiratory Syndrome; Stiff-Person Syndrome; Thymoma; Waldenstrom Macroglobulinemia; Adenocarcinoma of Lung; Adrenal Cortex Neoplasms; Anemia, Refractory; Anemia, Refractory, with Excess of Blasts; Brain Neoplasms; Breast Neoplasms; Burkitt Lymphoma; Carcinoma; Carcinoma, Embryonal; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Central Nervous System Neoplasms; Choriocarcinoma; Choroid Plexus Neoplasms; Colorectal Neoplasms; Endodermal Sinus Tumor; Ependymoma; Ganglioneuroblastoma; Gestational Trophoblastic Disease; Granuloma, Lethal Midline; Hepatoblastoma; HIV Infections; Hodgkin Disease; Kidney Neoplasms; Leukemia; Leukemia, Basophilic, Acute; Leukemia, Biphenotypic, Acute; Leukemia, Erythroblastic, Acute; Leukemia-Lymphoma, Adult T-Cell; Leukemia, Megakaryoblastic, Acute; Leukemia, Monocytic, Acute; Leukemia, Myeloid, Acute; Leukemia, Myelomonocytic, Acute; Leukemia, Myelomonocytic, Chronic; Lung Neoplasms; Lymphohistiocytosis, Hemophagocytic; Lymphoma; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Lymphoma, Non-Hodgkin; Lymphoma, T-Cell, Peripheral; Mediastinal Neoplasms; Medulloblastoma; Multiple Myeloma; Myelodysplastic Syndromes; Myeloproliferative Disorders; Neoplasms, Germ Cell and Embryonal; Neuroblastoma; Neuroectodermal Tumors, Primitive; Osteosarcoma; Ovarian Neoplasms; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Prostatic Neoplasms, Castration-Resistant; Retinoblastoma; Rhabdomyosarcoma; Sarcoma; Sarcoma, Ewing; Sarcoma, Myeloid; Seminoma; Sex Cord-Gonadal Stromal Tumors; Small Cell Lung Carcinoma; Stomach Neoplasms; Teratoma; Testicular Neoplasms; Thymus Neoplasms; Wilms Tumor; Neoplasms
DNA topoisomerase II inhibitor
Small molecule
Approved
Unknown
Unknown
Pain
Mu opioid receptor agonist
Small molecule
Approved
Unknown
Unknown
Cardiovascular Diseases
Unknown
Protein
Approved
Unknown
Unknown
Unknown
Diagnostic agent
Small molecule
Approved
OTHER
INHALATION
Unknown
Beta-2 adrenergic receptor agonist
Small molecule
Unknown
Unknown
Unknown
Depressive Disorder; Tobacco Use Disorder
Neuronal acetylcholine receptor; alpha4/beta2 agonist
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Atherosclerosis; Renal Insufficiency, Chronic; Diabetes Mellitus; Diabetes Mellitus, Type 2
Sulfonylurea receptor 1, Kir6.2 blocker
Small molecule
Approved
OTHER
INJECTION
Bacterial Infections
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Bacterial Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Heart Diseases; Hypertension; Hemangioma; Cardiovascular Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Acute Coronary Syndrome; Hypotension; Pain; Cerebral Hemorrhage; Cocaine-Related Disorders; Pre-Eclampsia; Sinusitis; Stroke; Tobacco Use Disorder; Hypertension; Cardiovascular Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Carcinoma, Hepatocellular; Hodgkin Disease; Kidney Diseases; Pancreatic Neoplasms; Colorectal Neoplasms; Diabetes Mellitus, Type 1; Leishmaniasis; Lymphoma, AIDS-Related; Melanoma; Trypanosomiasis; Infections
Unknown
Small molecule
Approved
OTHER
INJECTION
Unknown
Phosphodiesterase 3A inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Arthralgia; Eye Diseases; Myalgia
Xanthine dehydrogenase inhibitor
Small molecule
Approved
Unknown
Unknown
Arrhythmias, Cardiac
Unknown
Small molecule
Approved
Unknown
Unknown
Delirium; Chronic Pain; Pulpitis; Wounds and Injuries; Back Pain; Pain; Pregnancy
Unknown
Small molecule
Approved
Unknown
Unknown
Constipation; Heart Arrest; Heroin Dependence; Restless Legs Syndrome; Rheumatic Diseases; Blood Coagulation Disorders; Chronic Pain; Fractures, Multiple; Hemorrhage; Mucositis; Neuralgia; Postoperative Complications; Premature Birth; Respiratory Insufficiency; Rotator Cuff Injuries; Stomatitis; Tonsillitis; Anemia, Sickle Cell; Back Pain; Dyspnea; Fractures, Bone; Kidney Calculi; Leukemia, Myeloid, Acute; Myocardial Infarction; Neonatal Abstinence Syndrome; Neoplasms; Obesity; Opioid-Related Disorders; Pregnancy; Prostatic Neoplasms, Castration-Resistant; Pruritus; Pulmonary Disease, Chronic Obstructive; Renal Colic; Scoliosis; Sleep Apnea, Obstructive; Wounds and Injuries; Pain
Unknown
Small molecule
Approved
OTHER
INHALATION
Unknown
Beta-2 adrenergic receptor agonist
Small molecule
Approved
OTHER
ORAL
Amyotrophic Lateral Sclerosis; Anxiety; Dementia; Depressive Disorder; Schizophrenia; Psychotic Disorders; Tics; Tourette Syndrome
Dopamine receptor antagonist
Small molecule
Approved
Unknown
Unknown
Unknown
Monoamine transporter inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Alpha-1a adrenergic receptor agonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Diarrhea; Osteomyelitis; Astrocytoma; Brain Neoplasms; Cocaine-Related Disorders; Glioblastoma; Obesity; Respiratory Tract Infections; Sepsis; Asthma; Depressive Disorder, Major; Erectile Dysfunction; Head and Neck Neoplasms; Mastitis; Periapical Periodontitis; Pneumonia, Bacterial; Tobacco Use Disorder; Tuberculosis; Tuberculosis, Pulmonary; Abscess; Bronchitis, Chronic; Cholecystitis; Enterobacteriaceae Infections; Helicobacter Infections; Infections; Otitis Media; Otitis Media, Suppurative; Pneumonia; Severe Acute Respiratory Syndrome; Sinusitis; Urinary Tract Infections
Unknown
Small molecule
Approved
CARDIOVASCULAR; OTHER
ORAL
Anemia; Bipolar Disorder; Crohn Disease; Infertility; Pancreatitis; Central Nervous System Neoplasms; Hepatopulmonary Syndrome; HIV Infections; Muscular Dystrophy, Duchenne; Schizophrenia; Severe Acute Respiratory Syndrome; Acute Coronary Syndrome; Acute Kidney Injury; Behcet Syndrome; Biliary Atresia; Brain Diseases; Breast Neoplasms; Carcinoma, Non-Small-Cell Lung; Coronary Disease; Depressive Disorder, Major; Diabetic Nephropathies; Ductus Arteriosus, Patent; Enterocolitis, Necrotizing; Fatty Liver; Fibrosis; Head and Neck Neoplasms; Leishmaniasis; Leishmaniasis, Cutaneous; Liver Cirrhosis, Biliary; Malaria, Falciparum; Neoplasms; Non-alcoholic Fatty Liver Disease; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Sarcoidosis, Pulmonary; Wounds and Injuries; Brachial Plexus Neuropathies; Endometriosis; Glomerulonephritis; Hepatitis, Alcoholic; Liver Cirrhosis; Liver Failure; Neonatal Sepsis; Nephrotic Syndrome; Osteonecrosis; Renal Insufficiency, Chronic; Cardiovascular Diseases
3',5'-cyclic phosphodiesterase inhibitor
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM
INTRAMUSCULAR
Bulimia; Alcohol Drinking; Child Development Disorders, Pervasive; Dermatitis, Atopic; Psoriasis; Schizophrenia; Alcohol-Related Disorders; Amphetamine-Related Disorders; Breast Neoplasms; Colitis, Ulcerative; Coronavirus Infections; Crohn Disease; Cystitis, Interstitial; Depressive Disorder, Major; Diabetic Neuropathies; Dry Eye Syndromes; Fibromyalgia; Low Back Pain; Marijuana Abuse; Migraine Disorders; Obsessive-Compulsive Disorder; Respiratory Distress Syndrome; Severe Acute Respiratory Syndrome; Trichotillomania; Borderline Personality Disorder; Chronic Pain; Cocaine-Related Disorders; Depressive Disorder; Endometriosis; Gambling; Heroin Dependence; HIV Infections; Multiple Sclerosis; Obesity; Opioid-Related Disorders; Pain; Stress Disorders, Post-Traumatic; Substance-Related Disorders; Tobacco Use Disorder; Alcoholism
Opioid receptors; mu/kappa/delta antagonist
Small molecule
Approved
OTHER
NASAL; ORAL; TRANSDERMAL
Aging; Attention Deficit Disorder with Hyperactivity; Cocaine-Related Disorders; Memory Disorders; Sarcoidosis; Schizophrenia; Alcohol Drinking; Carcinoma in Situ; Cognitive Dysfunction; Depressive Disorder; Parkinson Disease; Postoperative Nausea and Vomiting; Sarcoma; Substance-Related Disorders; Wounds and Injuries; Heart Failure; Lung Neoplasms; Marijuana Abuse; Pulmonary Disease, Chronic Obstructive; Severe Acute Respiratory Syndrome; Smoking Cessation; Tuberculosis; Uterine Cervical Neoplasms; Tobacco Use Disorder
Neuronal acetylcholine receptor; alpha4/beta2 agonist
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; HEMATOLOGY; OTHER
ORAL
Angina, Stable; Ischemic Stroke; Spinal Cord Injuries; Brain Injuries; Diabetes Mellitus, Type 1; Stroke; Diabetes, Gestational; Diabetes Mellitus; Diabetes Mellitus, Type 2
Sulfonylurea receptor 1, Kir6.2 blocker
Small molecule
Approved
Unknown
Unknown
Sepsis; Mastitis; Periapical Periodontitis; Tuberculosis; Enterobacteriaceae Infections; Pyelonephritis; Infections; Otitis Media; Pneumonia; Respiratory Tract Infections; Sinusitis; Soft Tissue Infections; Urinary Tract Infections
Bacterial beta-lactamase TEM inhibitor
Small molecule
Approved
Unknown
Unknown
Cardiovascular Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Depressive Disorder
Unknown
Small molecule
Approved
Unknown
Unknown
Keratosis, Actinic; Infections; Acne Vulgaris
Releases active oxygen