Display Options:
Total: 10647
Small molecule
Approved
Unknown
Unknown
Sepsis; Mastitis; Periapical Periodontitis; Tuberculosis; Enterobacteriaceae Infections; Pyelonephritis; Infections; Otitis Media; Pneumonia; Respiratory Tract Infections; Sinusitis; Soft Tissue Infections; Urinary Tract Infections
Bacterial beta-lactamase TEM inhibitor
Small molecule
Approved
Unknown
Unknown
Depressive Disorder
Unknown
Small molecule
Approved
Unknown
Unknown
Constipation; Kidney Neoplasms; Opioid-Related Disorders; Wounds and Injuries; Anemia, Sickle Cell; Cancer Pain; Chronic Pain; Heroin Dependence; Ileus; Low Back Pain; Mucositis; Osteoarthritis, Hip; Osteoarthritis, Knee; Pain
Unknown
Small molecule
Approved
Unknown
Unknown
Depressive Disorder; Smoking; Tobacco Use Disorder
Neuronal acetylcholine receptor; alpha4/beta2 agonist
Small molecule
Approved
OTHER
INJECTION
Unknown
Phosphodiesterase 3A inhibitor
Small molecule
Approved
Unknown
Unknown
Lung Diseases, Obstructive
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Constipation; Fractures, Bone; Heart Arrest; Heroin Dependence; Restless Legs Syndrome; Rheumatic Diseases; Blood Coagulation Disorders; Fractures, Multiple; Hemorrhage; Mucositis; Neuralgia; Postoperative Complications; Premature Birth; Respiratory Insufficiency; Rotator Cuff Injuries; Stomatitis; Tonsillitis; Anemia, Sickle Cell; Back Pain; Cancer Pain; Chronic Pain; Dyspnea; Kidney Calculi; Leukemia; Leukemia, Myeloid, Acute; Myocardial Infarction; Neonatal Abstinence Syndrome; Neoplasms; Obesity; Opioid-Related Disorders; Pregnancy; Prostatic Neoplasms, Castration-Resistant; Pruritus; Pulmonary Disease, Chronic Obstructive; Renal Colic; Rib Fractures; Scoliosis; Sleep Apnea, Obstructive; Wounds and Injuries; Pain
Unknown
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Sepsis; Hematologic Neoplasms; Infections; Bacterial Infections; Pneumonia, Bacterial; Pneumonia, Ventilator-Associated; Pyelonephritis; Urinary Tract Infections
Renal dipeptidase inhibitor
Small molecule
Approved
Unknown
Unknown
Cheilitis; Erythema; Stomatitis; Skin Diseases; Eye Diseases; Skin Ulcer
Unknown
Small molecule
Approved
Unknown
Unknown
Glaucoma
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Multiple Sclerosis; Acidosis, Lactic; Heart Arrest; Huntington Disease; Respiratory Insufficiency; Heart Failure; Hyperemesis Gravidarum; Sepsis; Shock, Septic; Anemia; Brain Diseases; Kidney Failure, Chronic; Thiamine Deficiency
Unknown
Small molecule
Approved
OTHER
ORAL
Sleep Initiation and Maintenance Disorders
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
Unknown
Unknown
Nausea; Neoplasms; Pulmonary Alveolar Proteinosis; Atherosclerosis; Attention Deficit Disorder with Hyperactivity; Colorectal Neoplasms; Epilepsy; Fatty Liver, Alcoholic; Heart Diseases; Heart Failure; Hepatitis, Alcoholic; HIV Infections; Lymphoma; Multiple Myeloma; Myocardial Infarction; Myocardial Ischemia; Psychotic Disorders; Tuberculosis, Pulmonary; Vomiting; Alzheimer Disease; Hand-Foot Syndrome; Movement Disorders; Non-alcoholic Fatty Liver Disease; Spasms, Infantile; Tuberculosis; Anemia; Diabetes Mellitus, Type 2; Kidney Failure, Chronic; Osteoporosis; Postoperative Nausea and Vomiting
Unknown
Small molecule
Approved
Unknown
Unknown
Cholecystitis; Osteomyelitis; Bacterial Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Melanoma; Neoplasms; Cardiomyopathy, Hypertrophic; Hepatolenticular Degeneration
Unknown
Small molecule
Approved
Unknown
Unknown
Endocarditis; Infections; Intraabdominal Infections; Pneumonia; Sepsis; Urinary Tract Infections
Renal dipeptidase inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Diagnostic
Small molecule
Approved
Unknown
Unknown
Coronary Disease; Amyloidosis, Familial; Hemorrhagic Fever, Ebola; Severe Acute Respiratory Syndrome; Tachycardia, Supraventricular; Atrial Fibrillation; Atrial Flutter; Cardiomyopathies; Death, Sudden, Cardiac; Heart Arrest; Heart Diseases; Heart Failure; Myocardial Infarction; Tachycardia, Ventricular; Ventricular Fibrillation; Arrhythmias, Cardiac
Unknown
Small molecule
Approved
OTHER
ORAL
Alcoholism; Bipolar Disorder; Cognitive Dysfunction; Diabetes Mellitus, Type 2; Essential Tremor; Joint Diseases; Mental Disorders; Schizophrenia; Substance-Related Disorders; Alcohol Drinking; Amyotrophic Lateral Sclerosis; Anemia, Sickle Cell; Arthritis, Psoriatic; Arthritis, Rheumatoid; Child Development Disorders, Pervasive; Chronic Pain; Dementia; HIV Infections; Irritable Bowel Syndrome; Marijuana Abuse; Migraine with Aura; Migraine without Aura; Multiple Sclerosis; Neuralgia; Opioid-Related Disorders; Pain; Sleep Apnea, Obstructive; Stress Disorders, Post-Traumatic; Torticollis; Tourette Syndrome; Trichotillomania; Anorexia Nervosa; Osteoarthritis, Knee; Anorexia; Nausea; Neoplasms; Vomiting
Cannabinoid CB1 receptor agonist
Small molecule
Approved
OTHER
BILIARY; PERFUSION
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Glaucoma, Open-Angle; Ocular Hypertension; Cardiovascular Diseases; Glaucoma
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Azoospermia; Endocardial Cushion Defects; Heart Septal Defects, Ventricular; Infertility; Acquired Immunodeficiency Syndrome; beta-Thalassemia; Carbon Monoxide Poisoning; Diabetes Mellitus, Type 2; Heart Failure; Muscle Cramp; Neoplasms; Non-alcoholic Fatty Liver Disease; Poisoning; Polycystic Ovary Syndrome; Renal Insufficiency, Chronic; Shock, Septic; Spinal Cord Injuries; Acute Kidney Injury; Arthritis, Rheumatoid; Asthma; Atrial Fibrillation; Cytomegalovirus Infections; Gastrointestinal Stromal Tumors; HIV Infections; Hyperthyroidism; Hypotension; Lipid Metabolism Disorders; Multiple Sclerosis; Muscular Atrophy, Spinal; Pancreatic Neoplasms; Postpoliomyelitis Syndrome; Pyelonephritis; Brain Diseases; Kidney Failure, Chronic; Muscle Weakness
Unknown
Small molecule
Approved
Unknown
Unknown
Barrett Esophagus; Erectile Dysfunction; Ischemia; Renal Insufficiency, Chronic; Cerebral Hemorrhage; Diabetes Mellitus, Type 1; Essential Hypertension; Glomerulonephritis, IGA; Heart Diseases; Melanoma; Pseudohypoaldosteronism; Stroke; Vascular Diseases; Cardiomyopathies; Cardiotoxicity; Chagas Cardiomyopathy; Coronary Disease; Heart Failure; Hematologic Neoplasms; Hypertension; Influenza, Human; Leukemia, Lymphoid; Leukemia, Myeloid, Acute; Lymphoma; Multiple Myeloma; Myocardial Ischemia; Neoplasms; Pneumonia; Severe Acute Respiratory Syndrome; ST Elevation Myocardial Infarction; Cardiovascular Diseases
Unknown
Small molecule
Approved
OTHER
TOPICAL
Tinea Pedis
Cytochrome P450 51 inhibitor
Small molecule
Approved
Unknown
Unknown
Amyloidosis, Familial; Atrial Fibrillation; Chagas Cardiomyopathy; Heart Failure; Arrhythmias, Cardiac; Tachycardia, Ventricular; Ventricular Fibrillation
HERG blocker
Small molecule
Approved
Unknown
Unknown
Irritable Bowel Syndrome; Blepharospasm; Charcot-Marie-Tooth Disease; Chronic Pain; Dystonic Disorders; Death, Sudden, Cardiac; Myocardial Infarction; Myotonic Dystrophy; Ventricular Fibrillation; Arrhythmias, Cardiac
Unknown
Small molecule
Approved
OTHER
INJECTION
Cystic Fibrosis; Osteomyelitis; Esophageal Achalasia; Meningitis, Bacterial; Enterobacteriaceae Infections; Skin Diseases; Staphylococcal Skin Infections; Bacterial Infections; Infections; Intraabdominal Infections; Parametritis; Peritonitis; Pneumonia; Pyelonephritis; Urinary Tract Infections
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
Unknown
Unknown
Arrhythmogenic Right Ventricular Dysplasia; Atrial Fibrillation; Arrhythmias, Cardiac
Unknown
Protein
Approved
OTHER
INJECTION
Hyperglycemia; Atherosclerosis; Coronary Disease; Diabetes Mellitus, Type 2; Hypercholesterolemia; Hypertension
Insulin receptor agonist
Small molecule
Approved
Unknown
Unknown
Anemia, Sickle Cell; Amyotrophic Lateral Sclerosis; Anemia, Neonatal; Heart Failure; Huntington Disease; Asthma; Multiple Sclerosis; Anemia; Anemia, Iron-Deficiency; Diabetes Mellitus, Type 2; Kidney Failure, Chronic
Unknown
Small molecule
Approved
Unknown
Unknown
Breast Neoplasms; Esophageal Neoplasms; Urinary Bladder Neoplasms; Asthma; Hepatitis B, Chronic; Hepatitis D; Lymphoma, Large B-Cell, Diffuse; Peanut Hypersensitivity; Mucopolysaccharidosis I; Multiple Sclerosis; Multiple Sclerosis, Chronic Progressive; Hypersensitivity
Histamine H1 receptor antagonist
Small molecule
Approved
OTHER
OPHTHALMIC
Rheumatic Diseases
Cyclooxygenase inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown