Display Options:
Total: 10647
Small molecule
Approved
MUSCULOSKELETAL; OTHER; RHEUMATOLOGY
ORAL
Kidney Calculi; Renal Colic; Multiple Sclerosis; Paget Disease, Extramammary; Periodontitis; Bursitis; Inflammation; Low Back Pain; Migraine Disorders; Osteoarthritis, Knee; Postoperative Nausea and Vomiting; Sprains and Strains; Tendinopathy; Wounds and Injuries; Acute Pain; Arthralgia; Arthritis, Rheumatoid; Dysmenorrhea; Myalgia; Osteoarthritis; Rheumatic Diseases
Cyclooxygenase inhibitor
Small molecule
Approved
OTHER
TOPICAL
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER; RESPIRATORY
INHALATION; INJECTION
Carcinoma, Non-Small-Cell Lung; Osteomyelitis; Renal Insufficiency; Gonorrhea; Gram-Negative Bacterial Infections; Enterobacteriaceae Infections; Skin Diseases; Bacterial Infections; Cystic Fibrosis; Infections; Intraabdominal Infections; Pneumonia; Pyelonephritis; Sepsis; Urinary Tract Infections
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
OTHER
OPHTHALMIC; ORAL
Osteomyelitis; Hermanski-Pudlak Syndrome; Cystitis, Hemorrhagic; Esophageal and Gastric Varices; Liver Cirrhosis; Peritonitis; Bacterial Infections; Eye Infections
Bacterial DNA gyrase inhibitor
Small molecule
Approved
Unknown
Unknown
Polyuria; Urinary Incontinence
Unknown
Small molecule
Approved
Unknown
Unknown
Dyspepsia; Scleroderma, Systemic; Attention Deficit Disorder with Hyperactivity; Autistic Disorder; Child Development Disorders, Pervasive; Cocaine-Related Disorders; Depressive Disorder, Major; Gastroparesis; Marijuana Abuse; Sexual Dysfunction, Physiological; Spinal Cord Injuries; Anxiety Disorders; Apnea; Dementia; Depressive Disorder; Ischemic Stroke; Parkinson Disease; Schizophrenia; Anxiety
Unknown
Antibody
Approved
Unknown
Unknown
Colitis, Ulcerative; Neoplasms; Central Nervous System Neoplasms; Kidney Neoplasms; Melanoma; Non-alcoholic Fatty Liver Disease
T cell surface glycoprotein CD3 inhibitor
Unknown
Approved
Unknown
Unknown
Infertility, Female; Anovulation; Azoospermia; Infertility; Infertility, Male
Follicle stimulating hormone receptor agonist
Small molecule
Approved
OTHER; PREGNANCY AND GYNECOLOGY
INJECTION; INTRAVENOUS; ORAL
Back Pain; Hypotension; Liver Cirrhosis; Skin Neoplasms; Spinal Cord Neoplasms; Cerebral Hemorrhage; Epistaxis; Intervertebral Disc Degeneration; Osteoarthritis, Knee; Shock, Septic; Subarachnoid Hemorrhage; Urinary Bladder Neoplasms; Anemia; Angioedemas, Hereditary; Aortic Aneurysm, Abdominal; Astrocytoma; Blood Coagulation Disorders; Bone Neoplasms; Brain Injuries; Brain Neoplasms; Burns; Coronary Disease; Femoral Neck Fractures; Fractures, Bone; Gastrointestinal Hemorrhage; Genital Neoplasms, Female; Head and Neck Neoplasms; Hematologic Neoplasms; Hematoma; Hematoma, Subdural, Intracranial; Hemoptysis; Hip Fractures; Ileus; Inflammation; Joint Diseases; Leiomyoma; Melanoma; Melanosis; Meningioma; Nasal Polyps; Neoplasms; Osteoarthritis; Pain; Paraganglioma; Pelvic Organ Prolapse; Placenta Accreta; Placenta Previa; Postpartum Hemorrhage; Prostatic Neoplasms, Castration-Resistant; Scoliosis; Sepsis; Severe Acute Respiratory Syndrome; Shock; Shoulder Impingement Syndrome; Telangiectasia, Hereditary Hemorrhagic; Thrombocytopenia; von Willebrand Diseases; Wounds and Injuries; Hemophilia A; Hemorrhage; Menorrhagia
Plasminogen inhibitor
Protein
Approved
OTHER
UNKNOWN
Breast Carcinoma In Situ; Breast Neoplasms; Hematologic Neoplasms; Leukemia; Ovarian Neoplasms; Carcinoma, Renal Cell; Kidney Neoplasms; Leukemia-Lymphoma, Adult T-Cell; Liver Neoplasms; Pancreatic Neoplasms; Papillomavirus Infections; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Severe Acute Respiratory Syndrome; Uveal Melanoma; Carcinoma, Hepatocellular; Hepatitis C; HIV Infections; Liver Cirrhosis; Neoplasm Metastasis; Carcinoid Tumor; Condylomata Acuminata; Hepatitis B, Chronic; Hepatitis C, Chronic; Leukemia, Hairy Cell; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Lymphoma, Follicular; Melanoma; Multiple Myeloma; Neoplasms; Sarcoma, Kaposi
Interferon alpha/beta receptor agonist
Small molecule
Approved
Unknown
Unknown
Status Asthmaticus; Pulmonary Disease, Chronic Obstructive
Unknown
Small molecule
Approved
Unknown
Unknown
Aging; Brain Neoplasms; Ovarian Cysts; Reperfusion Injury; Atrial Fibrillation; Pain; Sinusitis; Cerebral Arterial Diseases; Coronary Disease; Intracranial Aneurysm; Respiratory Distress Syndrome; Shock, Septic; Cardiovascular Diseases
Unknown
Small molecule
Approved
OTHER
ORAL
Psoriasis
Retinoid receptor agonist
Small molecule
Approved
Unknown
Unknown
Carcinoma, Non-Small-Cell Lung; Colorectal Neoplasms; Fibrosis; Glycogen Storage Disease Type III; HIV Infections; Leukemia, Hairy Cell; Lupus Erythematosus, Systemic; Melanoma; Mesothelioma; Neoplasms; Psoriasis; Thyroid Neoplasms; Anemia, Sickle Cell; Breast Carcinoma In Situ; Breast Neoplasms; Eosinophilic Esophagitis; Immunoglobulin G4-Related Disease; Movement Disorders; Schizophrenia; Stomach Neoplasms; Gastrointestinal Hemorrhage; Severe Acute Respiratory Syndrome; Arthritis, Rheumatoid; Chest Pain; Duodenal Ulcer; Esophagitis; Gastroesophageal Reflux; Heartburn; Osteoarthritis; Peptic Ulcer; Stomach Ulcer; Ulcer
Histamine H2 receptor antagonist
Small molecule
Approved
OTHER
INJECTION
Arrhythmias, Cardiac; Ventricular Fibrillation
Norepinephrine transporter substrate
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Common Cold; Fecal Incontinence; Hypotension, Orthostatic; Presbyopia; Rhinitis, Allergic, Seasonal; Erythema; Rosacea; Eye Manifestations; Nasal Obstruction
Unknown
Protein
Approved
Unknown
Unknown
Psoriasis; Hepatitis C, Chronic; HIV Infections; Leukemia, Hairy Cell; Multiple Myeloma; Behcet Syndrome; Carcinoma, Renal Cell; Hepatitis C; Kidney Neoplasms; Lymphoma; Melanoma; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Retinal Vasculitis; Neoplasms
Interferon alpha/beta receptor agonist
Small molecule
Approved
Unknown
Unknown
Vitamin D Deficiency; Uremia
Unknown
Small molecule
Approved
OTHER
ORAL
Bacterial Infections; Cryptosporidiosis; Lung Diseases; Tuberculosis, Multidrug-Resistant; Crohn Disease; Mycobacterium avium-intracellulare Infection; Tuberculosis; Tuberculosis, Pulmonary; Leprosy
DNA inhibitor
Small molecule
Approved
Unknown
Unknown
Asthma
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Lung Diseases, Obstructive
Unknown
Small molecule
Approved
Unknown
Unknown
Cognitive Dysfunction; Ovarian Cysts; Shock, Septic; Diabetic Foot; Hypertension
Beta-1 adrenergic receptor antagonist
Small molecule
Approved
OTHER
TOPICAL
Lice Infestations; Lyme Disease; Ectoparasitic Infestations
Voltage-sensitive sodium channel blocker
Small molecule
Approved
Unknown
Unknown
Stress Disorders, Post-Traumatic; Alcohol Drinking; Alcoholism; Attention Deficit Disorder with Hyperactivity; Cocaine-Related Disorders; Depressive Disorder; Marijuana Abuse; Schizotypal Personality Disorder; Smoking Cessation; Stroke; Substance-Related Disorders; Tobacco Use Disorder; Trigeminal Neuralgia; Alzheimer Disease; Delirium; Tourette Syndrome; Hypertension
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Rheumatic Diseases
Cyclooxygenase inhibitor
Small molecule
Approved
CARDIOVASCULAR; OTHER
ORAL
Asthma; Inflammation; Leukemia, Myeloid, Acute; Metabolic Diseases; Porokeratosis; Stroke; Arthritis, Rheumatoid; Breast Neoplasms; Carotid Stenosis; Cerebrovascular Disorders; Cognitive Dysfunction; Fragile X Syndrome; HIV Infections; Intracranial Arteriosclerosis; Intracranial Arteriovenous Malformations; Learning Disabilities; Melanoma; Neurofibromatosis 1; Ovarian Neoplasms; Parkinson Disease; Prostatic Neoplasms, Castration-Resistant; Pulmonary Disease, Chronic Obstructive; Rett Syndrome; Xanthomatosis, Cerebrotendinous; Heart Diseases; Intermittent Claudication; Lipid Metabolism Disorders; Myocardial Ischemia; Peripheral Vascular Diseases; Atherosclerosis; Cardiovascular Diseases; Coronary Artery Disease; Coronary Disease; Hypercholesterolemia
HMG-CoA reductase inhibitor
Protein
Approved
OTHER
INJECTION
Unknown
Unknown
Small molecule
Approved
GASTROINTESTINAL; OTHER; RESPIRATORY
INJECTION; ORAL; OTIC
Arthritis, Rheumatoid; Carcinoma, Pancreatic Ductal; Diabetic Foot; Dysentery, Bacillary; Erectile Dysfunction; Gastroenteritis; Hearing Loss; Hepatitis, Alcoholic; Hepatitis C; Leukemia, Myeloid, Acute; Liver Cirrhosis, Alcoholic; Lung Diseases; Lymphoma; Neoplasms; Osteomyelitis; Periapical Periodontitis; Pseudomonas Infections; Purpura, Thrombocytopenic, Idiopathic; Rhinoscleroma; Amyotrophic Lateral Sclerosis; Anthrax; Cataract; Corneal Ulcer; Crohn Disease; Cystic Fibrosis; Endophthalmitis; Leukemia, Lymphocytic, Chronic, B-Cell; Pancreatic Neoplasms; Breast Neoplasms; Bronchiectasis; Communicable Diseases; Diarrhea; Digestive System Diseases; Fever; Hypertriglyceridemia; Kidney Calculi; Lipid Metabolism Disorders; Liver Abscess; Neutropenia; Otitis Media; Peritonitis; Plague; Pneumonia; Prostatic Neoplasms, Castration-Resistant; Pulmonary Disease, Chronic Obstructive; Sepsis; Urinary Bladder Neoplasms; Urolithiasis; Bacterial Infections; Bronchitis, Chronic; Cystitis; Eye Infections; Gonorrhea; Infections; Intraabdominal Infections; Otitis Externa; Prostatitis; Pyelonephritis; Sinusitis; Typhoid Fever; Urinary Tract Infections
Bacterial DNA gyrase inhibitor
Small molecule
Approved
Unknown
Unknown
Cardiovascular Diseases; Diabetes Mellitus; Heart Failure; Hypertension; Myocardial Infarction; Stroke
Angiotensin-converting enzyme inhibitor
Small molecule
Approved
Unknown
Unknown
Brain Neoplasms; Cognitive Dysfunction; Colorectal Neoplasms; Diabetes Mellitus, Type 1; Dysthymic Disorder; Wounds and Injuries; Cocaine-Related Disorders; Epilepsy; Gastroesophageal Reflux; Hypertension, Pulmonary; Ischemic Stroke; Marijuana Abuse; Multiple Sclerosis, Chronic Progressive; Multiple System Atrophy; Obesity; Panic Disorder; Sciatica; Anxiety; Autistic Disorder; Bipolar Disorder; Cerebral Hemorrhage; Dementia; Depressive Disorder; Depressive Disorder, Major; Depressive Disorder, Treatment-Resistant; Enuresis; Fibromyalgia; Influenza, Human; Obsessive-Compulsive Disorder; Phobia, Social; Schizophrenia; Severe Acute Respiratory Syndrome; Stress Disorders, Post-Traumatic; Stroke; Tobacco Use Disorder
Unknown