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Total: 10647
Small molecule
Approved
Unknown
Unknown
Unknown
Diagnostic
Small molecule
Approved
Unknown
INTRAVENOUS
Acne Vulgaris; Ascorbic Acid Deficiency; Asthma; Astrocytoma; Autistic Disorder; Breast Neoplasms; Burns; Carcinoma, Basal Cell; Carcinoma, Pancreatic Ductal; Colonic Neoplasms; Diabetes Mellitus, Type 1; Diabetic Neuropathies; Glioma; Gliosarcoma; Hereditary Breast and Ovarian Cancer Syndrome; Hypertension; Hypoxia; Neoplasms; Oligodendroglioma; Osteoarthritis; Polycythemia Vera; Postpartum Hemorrhage; Primary Myelofibrosis; Pulmonary Alveolar Proteinosis; Sarcoma; Temporomandibular Joint Disorders; Thrombocythemia, Essential; Urinary Bladder Neoplasms; Acute Lung Injury; Atherosclerosis; beta-Thalassemia; Carcinoma, Non-Small-Cell Lung; Carcinoma, Renal Cell; Carotid Artery Diseases; Charcot-Marie-Tooth Disease; Depressive Disorder; Diabetes Mellitus, Type 2; Epilepsy; Fatigue; Glioblastoma; Heart Arrest; Heart Diseases; Hodgkin Disease; Inflammation; Intracranial Arteriosclerosis; Leukemia, Myeloid, Acute; Leukemia, Promyelocytic, Acute; Lung Neoplasms; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Non-Hodgkin; Multiple Myeloma; Muscular Diseases; Myelodysplastic Syndromes; Myocardial Infarction; Neoplasms, Plasma Cell; Neuralgia; Ovarian Neoplasms; Pancreatic Neoplasms; Pre-Eclampsia; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Rectal Neoplasms; Renal Insufficiency, Chronic; Shock; Stomatitis; Tobacco Use Disorder; Urinary Tract Infections; Uterine Cervical Neoplasms; Vascular Diseases; Virus Diseases; Wounds and Injuries; Anorexia; Atrial Fibrillation; Atrial Flutter; Cataract; Colorectal Neoplasms; Complex Regional Pain Syndromes; Coronary Disease; Diabetes Mellitus; Heart Failure; Influenza, Human; Leiomyoma; Macular Degeneration; Menopause; Myocardial Ischemia; Pain; Paraganglioma; Respiratory Tract Infections; Schizophrenia; Sepsis; Severe Acute Respiratory Syndrome; Shock, Septic; Stomach Neoplasms; Anemia; Anemia, Iron-Deficiency; Eye Diseases; Kidney Failure, Chronic; Pneumonia; Scurvy
Supplement
Protein
Approved
OTHER
INJECTION
Unknown
Growth hormone receptor agonist
Small molecule
Approved
Unknown
Unknown
Anemia, Sickle Cell; Amyotrophic Lateral Sclerosis; Anemia, Neonatal; Heart Failure; Huntington Disease; Asthma; Multiple Sclerosis; Anemia; Anemia, Iron-Deficiency; Diabetes Mellitus, Type 2; Kidney Failure, Chronic
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Diagnostic agent
Small molecule
Approved
Unknown
Unknown
Endocarditis; Infections; Intraabdominal Infections; Pneumonia; Sepsis; Urinary Tract Infections
Renal dipeptidase inhibitor
Small molecule
Approved
Unknown
Unknown
Anemia; Arthritis, Rheumatoid; Asthma; Infertility; Ovarian Neoplasms; Pancreatic Neoplasms; Penile Induration; Acute Kidney Injury; Adrenoleukodystrophy; Asthenozoospermia; Atherosclerosis; Brain Diseases; Burns; Cardiovascular Diseases; Carotid Artery Diseases; Diabetes Mellitus, Type 2; Endometriosis; Fibrosis; Friedreich Ataxia; Heart Diseases; Heart Failure; Heavy Metal Poisoning; Infertility, Male; Intracranial Arteriosclerosis; Lung Neoplasms; Mastodynia; Neoplasms; Neuromuscular Diseases; Peripheral Nervous System Diseases; Polycystic Ovary Syndrome; Renal Insufficiency, Chronic; Reperfusion Injury; Stomatitis; Tobacco Use Disorder; Wounds and Injuries; Alzheimer Disease; Amyotrophic Lateral Sclerosis; Breast Neoplasms; Cataract; Cerebrovascular Disorders; Colorectal Neoplasms; Coronary Disease; Delirium; Depressive Disorder; Fatty Liver; Gaucher Disease; Glaucoma; Head and Neck Neoplasms; Hypobetalipoproteinemias; Infections; Kidney Diseases; Liver Cirrhosis; Liver Diseases; Macular Degeneration; Menopause; Migraine Disorders; Myocardial Infarction; Myocardial Ischemia; Non-alcoholic Fatty Liver Disease; Osteonecrosis; Pain; Parkinson Disease; Prostatic Neoplasms, Castration-Resistant; Psoriasis; Pulmonary Disease, Chronic Obstructive; Rectal Neoplasms; Retinitis Pigmentosa; Schizophrenia; Urinary Bladder Neoplasms; Vascular Diseases
Unknown
Protein
Approved
Unknown
Unknown
HIV Infections; Menopause; Obesity; Hyperandrogenism; Hypogonadism; Liver Neoplasms; Melanoma; Salivary Gland Neoplasms; Breast Neoplasms; Endometriosis; Infertility; Leiomyoma; Myoma; Pain; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Neoplasms
Unknown
Small molecule
Approved
Unknown
Unknown
Alzheimer Disease; Anemia, Sickle Cell; Bipolar Disorder; Carcinoma, Non-Small-Cell Lung; Diabetes Mellitus, Type 2; Head and Neck Neoplasms; Leukemia, Lymphocytic, Chronic, B-Cell; Melanoma; Mitochondrial Diseases; Neoplasms; Prostatic Neoplasms, Castration-Resistant; Sexual Dysfunction, Physiological; Alcoholism; Amphetamine-Related Disorders; Cocaine-Related Disorders; Crohn Disease; Huntington Disease; Marijuana Abuse; Restless Legs Syndrome; Substance-Related Disorders; Anxiety; Attention Deficit Disorder with Hyperactivity; Dementia; Depressive Disorder, Treatment-Resistant; Obesity; Schizophrenia; Smoking Cessation; Tobacco Use Disorder; Depressive Disorder; Depressive Disorder, Major
Unknown
Protein
Approved
OTHER
INJECTION
Diabetes Mellitus
Insulin receptor agonist
Small molecule
Approved
Unknown
Unknown
Cheilitis; Erythema; Stomatitis; Skin Diseases; Eye Diseases; Skin Ulcer
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Opioid receptors; mu/kappa/delta agonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Multiple Sclerosis; Acidosis, Lactic; Heart Arrest; Huntington Disease; Respiratory Insufficiency; Heart Failure; Hyperemesis Gravidarum; Sepsis; Shock, Septic; Anemia; Brain Diseases; Kidney Failure, Chronic; Thiamine Deficiency
Unknown
Small molecule
Approved
OTHER
ORAL
Adenocarcinoma of Lung; Amebiasis; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Glioblastoma; HIV Infections; Small Cell Lung Carcinoma; Leukemia; Leukemia, Lymphocytic, Chronic, B-Cell; Ovarian Neoplasms; Pain; Tuberculosis; Arthritis, Rheumatoid; Rheumatic Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Irritable Bowel Syndrome; Blepharospasm; Charcot-Marie-Tooth Disease; Chronic Pain; Dystonic Disorders; Death, Sudden, Cardiac; Myocardial Infarction; Myotonic Dystrophy; Ventricular Fibrillation; Arrhythmias, Cardiac
Unknown
Unknown
Approved
Unknown
Unknown
Bacterial Infections; Osteoarthritis; Otomycosis; Sinusitis; Thymoma; Acanthamoeba Keratitis; Acne Vulgaris; Appendicitis; Empyema; Stomatitis; Conjunctivitis, Viral; Dental Caries; Pneumonia; Retinal Diseases; Severe Acute Respiratory Syndrome; Wounds and Injuries; Burns; Eczema; Eye Infections; Infections
Unknown
Small molecule
Approved
GASTROINTESTINAL; IMMUNE SYSTEM; OTHER
INHALATION; ORAL
Breast Neoplasms; Neoplasms; Diabetes Mellitus, Type 1; Encephalitis, Japanese; Hemorrhagic Fever with Renal Syndrome; Hepatitis D; Influenza, Human; Lassa Fever; Leukemia, Myeloid, Acute; Thrombocytopenia; Depressive Disorder; Hepatitis; Hepatitis B, Chronic; Hepatitis C; HIV Infections; Infections; Respiratory Syncytial Virus Infections; Severe Acute Respiratory Syndrome; Fibrosis; Hepatitis C, Chronic; Liver Cirrhosis; Virus Diseases
Inosine-5'-monophosphate dehydrogenase 1 inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Hepatolenticular Degeneration; Alcoholism; Feeding and Eating Disorders; Obesity; Bipolar Disorder; Lung Neoplasms; Neoplasms; Smoking; Smoking Cessation; Tobacco Use Disorder; Depressive Disorder; Depressive Disorder, Major; Mood Disorders; Seasonal Affective Disorder
Dopamine transporter inhibitor
Small molecule
Approved
Unknown
Unknown
Cholecystitis; Osteomyelitis; Bacterial Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Breast Neoplasms; Esophageal Neoplasms; Urinary Bladder Neoplasms; Asthma; Hepatitis B, Chronic; Hepatitis D; Lymphoma, Large B-Cell, Diffuse; Peanut Hypersensitivity; Mucopolysaccharidosis I; Multiple Sclerosis; Multiple Sclerosis, Chronic Progressive; Hypersensitivity
Histamine H1 receptor antagonist
Small molecule
Approved
OTHER
BILIARY; PERFUSION
Unknown
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Azoospermia; Endocardial Cushion Defects; Heart Septal Defects, Ventricular; Infertility; Acquired Immunodeficiency Syndrome; beta-Thalassemia; Carbon Monoxide Poisoning; Diabetes Mellitus, Type 2; Heart Failure; Muscle Cramp; Neoplasms; Non-alcoholic Fatty Liver Disease; Poisoning; Polycystic Ovary Syndrome; Renal Insufficiency, Chronic; Shock, Septic; Spinal Cord Injuries; Acute Kidney Injury; Arthritis, Rheumatoid; Asthma; Atrial Fibrillation; Cytomegalovirus Infections; Gastrointestinal Stromal Tumors; HIV Infections; Hyperthyroidism; Hypotension; Lipid Metabolism Disorders; Multiple Sclerosis; Muscular Atrophy, Spinal; Pancreatic Neoplasms; Postpoliomyelitis Syndrome; Pyelonephritis; Brain Diseases; Kidney Failure, Chronic; Muscle Weakness
Unknown
Protein
Approved
OTHER
INJECTION
Hyperglycemia; Atherosclerosis; Coronary Disease; Diabetes Mellitus, Type 2; Hypercholesterolemia; Hypertension
Insulin receptor agonist
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Hematologic Neoplasms; Lung Diseases; Bacterial Infections; Enterobacteriaceae Infections; Pneumonia, Bacterial; Pneumonia, Ventilator-Associated; Pyelonephritis; Endocarditis; Infections; Intraabdominal Infections; Pneumonia; Sepsis; Urinary Tract Infections
Bacterial penicillin-binding protein inhibitor
Protein
Approved
Unknown
Unknown
Psoriasis; Hepatitis C, Chronic; HIV Infections; Leukemia, Hairy Cell; Multiple Myeloma; Behcet Syndrome; Carcinoma, Renal Cell; Hepatitis C; Kidney Neoplasms; Lymphoma; Melanoma; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Retinal Vasculitis; Neoplasms
Interferon alpha/beta receptor agonist
Protein
Approved
OTHER
INJECTION
Parathyroid Diseases
Calcitonin receptor agonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Asthma
Unknown
Small molecule
Approved
OTHER
INJECTION
Delirium; Schizophrenia
D2-like dopamine receptor inverse agonist
Small molecule
Approved
OTHER
OPHTHALMIC; ORAL
Osteomyelitis; Hermanski-Pudlak Syndrome; Cystitis, Hemorrhagic; Esophageal and Gastric Varices; Liver Cirrhosis; Peritonitis; Bacterial Infections; Eye Infections
Bacterial DNA gyrase inhibitor
Small molecule
Approved
Unknown
Unknown
Stress Disorders, Post-Traumatic; Alcohol Drinking; Alcoholism; Attention Deficit Disorder with Hyperactivity; Cocaine-Related Disorders; Depressive Disorder; Marijuana Abuse; Schizotypal Personality Disorder; Smoking Cessation; Stroke; Substance-Related Disorders; Tobacco Use Disorder; Trigeminal Neuralgia; Alzheimer Disease; Delirium; Tourette Syndrome; Hypertension
Unknown
Small molecule
Approved
MUSCULOSKELETAL; OTHER; RHEUMATOLOGY
ORAL
Kidney Calculi; Renal Colic; Multiple Sclerosis; Paget Disease, Extramammary; Periodontitis; Bursitis; Inflammation; Low Back Pain; Migraine Disorders; Osteoarthritis, Knee; Postoperative Nausea and Vomiting; Sprains and Strains; Tendinopathy; Wounds and Injuries; Acute Pain; Arthralgia; Arthritis, Rheumatoid; Dysmenorrhea; Myalgia; Osteoarthritis; Rheumatic Diseases
Cyclooxygenase inhibitor
Small molecule
Approved
OTHER; RESPIRATORY
INHALATION; INJECTION
Carcinoma, Non-Small-Cell Lung; Osteomyelitis; Renal Insufficiency; Gonorrhea; Gram-Negative Bacterial Infections; Enterobacteriaceae Infections; Skin Diseases; Bacterial Infections; Cystic Fibrosis; Infections; Intraabdominal Infections; Pneumonia; Pyelonephritis; Sepsis; Urinary Tract Infections
Bacterial penicillin-binding protein inhibitor