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Total: 10647
Small molecule
Approved
Unknown
Unknown
Esophagitis, Peptic; Laryngopharyngeal Reflux; Cerebrovascular Disorders; Helicobacter Infections; Duodenal Ulcer; Gastroesophageal Reflux; Zollinger-Ellison Syndrome
Potassium-transporting ATPase inhibitor
Small molecule
Approved
OTHER
ORAL
CADASIL; Fatty Liver; Osteoarthritis; Pain; Cerebral Small Vessel Diseases; Cognitive Dysfunction; Heart Failure; Intermittent Claudication; Stroke; Urticaria; Wounds and Injuries; Arthritis, Rheumatoid; Atherosclerosis; Cardiovascular Diseases; Cerebral Infarction; Cerebrovascular Disorders; Coronary Disease; Ischemic Stroke; Peripheral Arterial Disease; Peripheral Vascular Diseases; Thrombosis
Phosphodiesterase 3A inhibitor
Small molecule
Approved
Unknown
Unknown
Anemia; Breast Neoplasms; Erectile Dysfunction; Glomerulosclerosis, Focal Segmental; Malaria; Malaria, Falciparum; Nausea; Neoplasms; Arthritis, Rheumatoid; Asthma; Cognitive Dysfunction; Colitis, Ulcerative; Endometriosis; HIV Infections; Inflammatory Bowel Diseases; Insulin Resistance; Mycosis Fungoides; Non-alcoholic Fatty Liver Disease; Prediabetic State; Sezary Syndrome; Alzheimer Disease; Atherosclerosis; Cardiovascular Diseases; Coronary Disease; Diabetic Neuropathies; Glucose Intolerance; Hypercholesterolemia; Hypertension; Lipid Metabolism Disorders; Metabolic Diseases; Metabolic Syndrome; Multiple Organ Failure; Prostatic Neoplasms; Diabetes Mellitus; Diabetes Mellitus, Type 2
Peroxisome proliferator-activated receptor gamma agonist
Small molecule
Approved
IMMUNE SYSTEM; OTHER
ORAL
Acquired Immunodeficiency Syndrome; HIV Infections; Virus Diseases
Human immunodeficiency virus type 1 protease inhibitor
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
ORAL
Amphetamine-Related Disorders; Epilepsy; Gastrointestinal Stromal Tumors; Obesity; Cocaine-Related Disorders; Parkinson Disease
Catechol O-methyltransferase inhibitor
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
HIV Infections; Central Nervous System Neoplasms; Head and Neck Neoplasms; Heart Failure; Leukoplakia, Oral; Non-alcoholic Fatty Liver Disease; Pituitary ACTH Hypersecretion; Sarcoma; Atherosclerosis; Insulin Resistance; Diabetes Mellitus; Diabetes Mellitus, Type 2
Peroxisome proliferator-activated receptor gamma agonist
Small molecule
Approved
MUSCULOSKELETAL; OTHER; RHEUMATOLOGY
ORAL
Brain Neoplasms; Paraganglioma; Alzheimer Disease; Carcinoma, Non-Small-Cell Lung; Adenoma; Colorectal Neoplasms; Joint Diseases; Osteoarthritis; Osteoarthritis, Knee; Pain; Prostatic Neoplasms, Castration-Resistant; Stomach Neoplasms; Rheumatic Diseases
Cyclooxygenase-2 inhibitor
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER; UROLOGY AND KIDNEY
INJECTION; ORAL
Neoplasms; Prostatic Neoplasms, Castration-Resistant; Psoriasis; Hyperparathyroidism, Secondary; Parathyroid Diseases; Renal Insufficiency, Chronic
Vitamin D receptor agonist
Small molecule
Approved
Unknown
Unknown
Adenocarcinoma; Carcinoma, Non-Small-Cell Lung; Esophageal Neoplasms; Hodgkin Disease; Lymphoma, Follicular; Lymphoma, Non-Hodgkin; Neoplasms, Germ Cell and Embryonal; Ovarian Neoplasms; Pancreatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Sepsis; Small Cell Lung Carcinoma; Testicular Neoplasms; Thymoma; Breast Neoplasms; Carcinoma, Hepatocellular; Inflammatory Breast Neoplasms; Lymphoma, Large B-Cell, Diffuse; Lymphoma, T-Cell, Peripheral; Nasopharyngeal Carcinoma; Sarcoma; Stomach Neoplasms; Thrombosis; Triple Negative Breast Neoplasms; Urinary Bladder Neoplasms; Neoplasms
Unknown
Small molecule
Approved
OTHER
ORAL; TOPICAL
Carcinoma, Intraductal, Noninfiltrating; Multiple Myeloma; Pituitary ACTH Hypersecretion; Thyroid Neoplasms; Triple Negative Breast Neoplasms; Alopecia Areata; Alzheimer Disease; Breast Neoplasms; Leukemia; Leukemia, Myeloid, Acute; Lung Neoplasms; Myelodysplastic-Myeloproliferative Diseases; Myelodysplastic Syndromes; Parapsoriasis; Psoriasis; Sezary Syndrome; Carcinoma, Non-Small-Cell Lung; Cognitive Dysfunction; Lymphoma; Lymphoma, Large-Cell, Anaplastic; Mycosis Fungoides; Psychotic Disorders; Schizophrenia; Lymphoma, T-Cell; Lymphoma, T-Cell, Cutaneous; Neoplasms
Retinoid X receptor agonist
Small molecule
Approved
Unknown
Unknown
Anemia; Astrocytoma; Brain Neoplasms; Crohn Disease; Cystic Fibrosis; Diabetes Mellitus, Type 1; Gastroparesis; Glioblastoma; Granulomatous Disease, Chronic; Inflammation; Lupus Erythematosus, Systemic; Melanoma; Meningioma; Multiple Myeloma; Multiple Sclerosis; Multiple Sclerosis, Relapsing-Remitting; Neoplasms; Peripheral Arterial Disease; Prostatic Neoplasms; Pulmonary Alveolar Proteinosis; Adrenoleukodystrophy; Alcoholism; Alzheimer Disease; Amyotrophic Lateral Sclerosis; Asthma; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Cardiovascular Diseases; Cerebral Hemorrhage; Child Development Disorders, Pervasive; Cognitive Dysfunction; Depressive Disorder, Major; Glucose Intolerance; Hepatitis; Hepatitis C; Hepatitis C, Chronic; Hypertension, Pulmonary; Infections; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Leukoplakia, Oral; Liposarcoma; Liposarcoma, Myxoid; Lung Neoplasms; Obesity; Opioid-Related Disorders; Pancreatic Neoplasms; Parkinson Disease; Polycystic Kidney Diseases; Polycystic Ovary Syndrome; Prostatic Neoplasms, Castration-Resistant; Psoriasis; Renal Insufficiency, Chronic; Stroke; Thyroid Neoplasms; Arthritis, Rheumatoid; Atherosclerosis; Coronary Disease; Diabetes Mellitus, Type 2; Fatty Liver; Friedreich Ataxia; HIV-Associated Lipodystrophy Syndrome; HIV Infections; Hypercholesterolemia; Hypertension; Insulin Resistance; Liver Diseases; Metabolic Syndrome; Non-alcoholic Fatty Liver Disease; Diabetes Mellitus
Unknown
Small molecule
Approved
EYE; OTHER
OPHTHALMIC
Cataract; Osteomyelitis; Corneal Ulcer; Tuberculosis; Bacterial Infections; Conjunctivitis, Bacterial; Eye Infections; Infections
DNA gyrase inhibitor
Protein
Approved
Unknown
Unknown
Diabetes Mellitus; Diabetes Mellitus, Type 2
Insulin receptor agonist
Small molecule
Approved
Unknown
Unknown
Acne Vulgaris; Astrocytoma; Colonic Neoplasms; Colorectal Neoplasms; Crohn Disease; Dermatitis, Seborrheic; Glioma; Gliosarcoma; Oligodendroglioma; Sarcoma; Basal Cell Nevus Syndrome; Brain Neoplasms; Carcinoma, Basal Cell; Desmoid Tumors; Glioblastoma; Neurofibromatosis 1; Infections; Keratosis, Actinic; Paraganglioma; Neoplasms
Unknown
Small molecule
Approved
HEMATOLOGY
ORAL
Cerebellar Ataxia; Cognitive Dysfunction; HIV Infections; Myocardial Infarction; Amyotrophic Lateral Sclerosis; Friedreich Ataxia; Parkinson Disease; Stroke; Acute Kidney Injury; Hemochromatosis; Pantothenate Kinase-Associated Neurodegeneration; Anemia, Sickle Cell; beta-Thalassemia; Iron Overload; Thalassemia
Unknown
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Anxiety; Breast Neoplasms, Male; Carcinoma, Intraductal, Noninfiltrating; Diabetes Mellitus; Persian Gulf Syndrome; Pregnancy; Prostatic Neoplasms, Castration-Resistant; Tobacco Use Disorder; Adenomyosis; Alcoholism; Alzheimer Disease; Bipolar Disorder; Borderline Personality Disorder; Carcinoma, Non-Small-Cell Lung; Central Serous Chorioretinopathy; Cocaine-Related Disorders; Endometrial Neoplasms; Endometriosis; Fallopian Tube Neoplasms; Hepatitis C; HIV Infections; Ovarian Neoplasms; Peritoneal Neoplasms; Prostatic Neoplasms; Stress Disorders, Post-Traumatic; Abortion, Spontaneous; Breast Neoplasms; Depressive Disorder; Depressive Disorder, Major; Leiomyoma; Meningioma; Mental Disorders; Pituitary ACTH Hypersecretion; Cushing Syndrome
Glucocorticoid receptor antagonist
Small molecule
Approved
HEMATOLOGY; OTHER; UROLOGY AND KIDNEY
INTRAVENOUS
Hematologic Neoplasms; Hypertension, Pulmonary; Anemia; Anemia, Iron-Deficiency; Renal Insufficiency, Chronic
Supplement
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Oligosaccharide
Approved
Unknown
Unknown
Kidney Neoplasms; Ischemic Stroke; Thromboembolism; Carcinoma, Non-Small-Cell Lung; Thrombosis; Venous Thrombosis
Antithrombin-III activator
Protein
Approved
Unknown
Unknown
Polycystic Ovary Syndrome; Ovarian Hyperstimulation Syndrome; Anovulation; Hypogonadism; Infertility; Infertility, Female; Obesity; Primary Ovarian Insufficiency; Reproductive Techniques, Assisted
Luteinizing hormone/Choriogonadotropin receptor agonist
Antibody
Approved
CANCER
INJECTION; SINGLE-DOSE
Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Myelomonocytic, Juvenile; Leukemia, Promyelocytic, Acute; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Leukemia; Myelodysplastic Syndromes; Leukemia, Myeloid; Leukemia, Myeloid, Acute; Neoplasms
DNA disrupting agent
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
ORAL
Cocaine-Related Disorders; Hearing Loss, Noise-Induced; Tobacco Use Disorder; Essential Tremor; Hearing Loss; Obesity; Parkinson Disease; Alcoholism; Epilepsy, Complex Partial; Feeding and Eating Disorders; Migraine Disorders; Psychotic Disorders; Schizophrenia; Smoking Cessation; Weight Gain; Epilepsies, Partial; Epilepsy; Seizures
Sodium channel alpha subunit blocker
Small molecule
Approved
Unknown
Unknown
Acquired Immunodeficiency Syndrome; Brain Neoplasms; Carcinoma, Basal Cell; Carcinoma, Non-Small-Cell Lung; Central Nervous System Neoplasms; Colorectal Neoplasms; Glioblastoma; Gliosarcoma; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Melanoma; Polycythemia Vera; Primary Myelofibrosis; Thrombocythemia, Essential; Breast Neoplasms; Bronchiolitis Obliterans Syndrome; Carcinoma, Hepatocellular; Endometrial Neoplasms; Esophageal Neoplasms; Kidney Neoplasms; Leukemia, Lymphocytic, Chronic, B-Cell; Liver Neoplasms; Lung Neoplasms; Lupus Erythematosus, Systemic; Lymphoma; Multiple Myeloma; Neoplasms, Plasma Cell; Neuroblastoma; Pancreatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Small Cell Lung Carcinoma; Ureteral Neoplasms; Urethral Neoplasms; Urinary Bladder Neoplasms; Uterine Cervical Neoplasms; Leukemia; Leukemia, Myeloid, Acute; Myelodysplastic Syndromes; Leukemia, Promyelocytic, Acute; Neoplasms
Thioredoxin reductase 1 inhibitor
Small molecule
Approved
MUSCULOSKELETAL; OTHER
ORAL
Lupus Erythematosus, Systemic; Dysmenorrhea; Osteoarthritis, Knee; Pharyngitis; Pregnancy; Toothache; Low Back Pain; Migraine Disorders; Pain; Prostatic Neoplasms; Shoulder Pain; Spondylitis, Ankylosing; Tuberculosis; Arthritis, Juvenile; Arthritis, Rheumatoid; Osteoarthritis; Rheumatic Diseases
Cyclooxygenase-2 inhibitor
Protein
Approved
OTHER; PREGNANCY AND GYNECOLOGY
INJECTION
Arthritis, Rheumatoid; Endometriosis; Infertility; Ovarian Hyperstimulation Syndrome; Prostatic Hyperplasia
Unknown
Small molecule
Approved
OTHER
ORAL
Diabetes Mellitus; Diabetes Mellitus, Type 2
Sulfonylurea receptor 1, Kir6.2 blocker
Small molecule
Approved
Unknown
Unknown
Diabetes Mellitus; Infections; Pregnancy; Bipolar Disorder; Graves Disease; Congenital Hypothyroidism; Hypothyroidism; Lipid Metabolism Disorders
Unknown
Small molecule
Approved
IMMUNE SYSTEM
TOPICAL
Herpes Simplex; Virus Diseases
Envelope glycoprotein inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Protein
Approved
CARDIOVASCULAR; OTHER
INJECTION; INTRAVENOUS
Venous Thrombosis; Acute Disease; Aortic Valve Stenosis; Cardiovascular Diseases; Coronary Disease; Heart Diseases; Hematologic Diseases; Hemorrhage; Myocardial Infarction; Subarachnoid Hemorrhage; Acute Coronary Syndrome; Angina, Unstable; Syndrome; Thrombocytopenia; Thrombosis
Thrombin inhibitor
Small molecule
Approved
Unknown
Unknown
Renal Insufficiency; Pain; Periodontitis; Pulpitis
Unknown
Protein
Approved
Unknown
Unknown
HIV Infections; Lymphoma; Salivary Gland Neoplasms; Breast Neoplasms; Endometriosis; Infertility; Ovarian Hyperstimulation Syndrome; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Puberty, Precocious; Neoplasms
Unknown
Small molecule
Approved
Unknown
TOPICAL
Nausea; Communicable Diseases; Anemia; Arthritis, Psoriatic; Arthritis, Rheumatoid; Burns; Colitis, Ulcerative; Eczema; Infections; Prostatic Neoplasms; Psoriasis; Spondylitis, Ankylosing
Unknown
Small molecule
Approved
OTHER
INTRAVENOUS; ORAL
Burns; Cystic Fibrosis; Hematologic Neoplasms; Lung Diseases; Meningitis; Tuberculosis, Multidrug-Resistant; Abscess; Cellulitis; Gram-Positive Bacterial Infections; Optic Nerve Diseases; Pneumonia, Bacterial; Pneumonia, Pneumococcal; Skin Diseases; Staphylococcal Infections; Syphilis; Tuberculosis; Tuberculosis, Pulmonary; Bacteremia; Bacterial Infections; Infections; Osteomyelitis; Pneumonia
Bacterial 70S ribosome inhibitor
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
TRANSDERMAL
Amphetamine-Related Disorders; Central Nervous System Diseases; Cocaine-Related Disorders; Down Syndrome; Substance-Related Disorders; Anxiety; Brain Injuries; Cognitive Dysfunction; Delirium; Dementia, Vascular; Depressive Disorder; Neurobehavioral Manifestations; Schizophrenia; Supranuclear Palsy, Progressive; Alzheimer Disease; Dementia; Parkinson Disease
Cholinesterases; ACHE & BCHE inhibitor