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Total: 10647
Small molecule
Approved
Unknown
Unknown
Depressive Disorder, Major; Fatigue Syndrome, Chronic; Idiopathic Pulmonary Fibrosis; Kidney Diseases; Nasopharyngeal Carcinoma; Castleman Disease; Hearing Loss, Sensorineural; Leukemia; Leukemia, Lymphocytic, Chronic, B-Cell; Lymphoma; Colitis, Ulcerative; Cytomegalovirus Infections; Cytomegalovirus Retinitis; Infections; Virus Diseases
Unknown
Unknown
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Endometritis; Appendicitis; Pyelonephritis; Renal Insufficiency, Chronic; Tuberculosis; Tuberculosis, Pulmonary; Diabetic Foot; Gonorrhea; Infections; Osteomyelitis; Pneumonia; Urinary Tract Infections; Bacterial Infections
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
Unknown
Unknown
Hypotension, Orthostatic; Lecithin Cholesterol Acyltransferase Deficiency; Memory; Obesity; Subarachnoid Hemorrhage; Cocaine-Related Disorders; HIV Infections; Psychotic Disorders; Tobacco Use Disorder; Alzheimer Disease; Anxiety; Autistic Disorder; Dementia, Vascular; Depressive Disorder; Lewy Body Disease; Schizophrenia; Dementia
Unknown
Protein
Approved
OTHER
INTRAVENOUS; SUBCUTANEOUS
Acute Kidney Injury; Brain Diseases; Brain Injuries; Brain Ischemia; Dysgerminoma; Hematologic Neoplasms; Leukemia; Lymphoma; Breast Neoplasms; Kidney Diseases; Leukemia, Lymphocytic, Chronic, B-Cell; Lymphoma, Large B-Cell, Diffuse; Myelodysplastic Syndromes; Myocardial Infarction; Small Cell Lung Carcinoma; Anemia; Kidney Failure, Chronic; Neoplasms; Renal Insufficiency, Chronic
Erythropoietin receptor agonist
Small molecule
Approved
Unknown
Unknown
Aspergillosis; Wounds and Injuries; Candidemia; Candidiasis; Candidiasis, Invasive; Candidiasis, Oral; Infections; Mycoses
Unknown
Small molecule
Approved
Unknown
Unknown
Diabetes Mellitus; Fever; Glaucoma; Heart Failure; Mitral Valve Stenosis; Neoplasms; Pancreatic Neoplasms; Sleep Apnea Syndromes; Asthma; Hermanski-Pudlak Syndrome; Hernias, Diaphragmatic, Congenital; Hypoplastic Left Heart Syndrome; Liver Cirrhosis; Melanoma; Pulmonary Disease, Chronic Obstructive; Diabetes Mellitus, Type 2; Eisenmenger Complex; Heart Septal Defects, Atrial; Idiopathic Pulmonary Fibrosis; Optic Neuropathy, Ischemic; Persistent Fetal Circulation Syndrome; Ulcer; Familial Primary Pulmonary Hypertension; Heart Defects, Congenital; Hypertension; Hypertension, Pulmonary; Pulmonary Arterial Hypertension; Scleroderma, Systemic
Endothelin receptor, ET-A/ET-B antagonist
Small molecule
Approved
CANCER; DIABETES DRUGS & ENDOCRINOLOGY; MUSCULOSKELETAL; OTHER
INJECTION; INTRAVENOUS; IV (INFUSION)
Adenocarcinoma; Anemia, Sickle Cell; Chondrosarcoma; Menopause; Neuroblastoma; beta-Thalassemia; Bone Resorption; Carcinoma, Intraductal, Noninfiltrating; Complex Regional Pain Syndromes; Kidney Neoplasms; Leiomyosarcoma; Low Back Pain; Macular Degeneration; Mesothelioma; Nasopharyngeal Neoplasms; Osteosarcoma; Pancreatic Neoplasms; Primary Myelofibrosis; Progeria; Urogenital Neoplasms; Uterine Cervical Neoplasms; Arthritis, Rheumatoid; Bone Diseases, Metabolic; Bone Neoplasms; Breast Neoplasms; Carcinoma, Hepatocellular; Carcinoma, Non-Small-Cell Lung; Giant Cell Tumors; Lung Neoplasms; Lymphoma; Lymphoma, Non-Hodgkin; Neoplasms, Plasma Cell; Osteoarthritis, Hip; Osteogenesis Imperfecta; Osteonecrosis; Pain; Plasmacytoma; Sarcoma; Sarcoma, Ewing; Spinal Cord Injuries; Bone Diseases; Fractures, Bone; Hypercalcemia; Multiple Myeloma; Neoplasm Metastasis; Osteitis Deformans; Osteoporosis; Osteoporosis, Postmenopausal; Prostatic Neoplasms
Farnesyl diphosphate synthase inhibitor
Small molecule
Approved
IMMUNE SYSTEM; OTHER
ORAL
Urinary Tract Infections; Bronchitis, Chronic; Infections; Pharyngitis; Tonsillitis
Bacterial penicillin-binding protein inhibitor
Unknown
Approved
Unknown
Unknown
Pulmonary Embolism; Renal Insufficiency, Chronic; Respiratory Distress Syndrome; Stroke; Hypotension; Ischemic Stroke; Shock, Septic; Multiple Organ Failure; Sepsis; Thrombosis
Coagulation factor VIII inhibitor
Small molecule
Approved
Unknown
Unknown
Acquired Immunodeficiency Syndrome; Dysmenorrhea; HIV Infections; Lupus Erythematosus, Systemic; Pregnancy; Prostatic Hyperplasia
Progesterone receptor agonist
Oligosaccharide
Approved
Unknown
Unknown
Renal Insufficiency; Thromboembolism; Venous Thromboembolism; Angina, Unstable; Myocardial Infarction; Pulmonary Embolism; Venous Thrombosis
Antithrombin-III activator
Small molecule
Approved
OTHER; UROLOGY AND KIDNEY
ORAL
Aging; Amyotrophic Lateral Sclerosis; Bulbo-Spinal Atrophy, X-Linked; Prostatitis; Severe Acute Respiratory Syndrome; Alopecia; Hypogonadism; Prostatic Neoplasms, Castration-Resistant; Prostatic Hyperplasia; Prostatic Neoplasms
Steroid 5-alpha-reductase inhibitor
Small molecule
Approved
Unknown
Unknown
Pain; Migraine Disorders
Unknown
Small molecule
Approved
OTHER; RESPIRATORY
INHALATION
Lung Neoplasms; Tobacco Use Disorder; Asthma; Bronchial Spasm; Bronchitis, Chronic; Emphysema; Pulmonary Disease, Chronic Obstructive
Beta-2 adrenergic receptor agonist
Small molecule
Approved
Unknown
Unknown
Arthritis, Juvenile; Breast Neoplasms; Fatty Liver; Hepatitis B, Chronic; Hypertension, Pulmonary; Lymphoma; Neoplasms; Non-alcoholic Fatty Liver Disease; Asthma; Autistic Disorder; Child Development Disorders, Pervasive; Cystic Fibrosis; Dyspepsia; Eosinophilic Esophagitis; Neuralgia; Digestive System Diseases; Duodenal Ulcer; Esophageal Neoplasms; Esophagitis, Peptic; Gastritis; Gastroesophageal Reflux; Gastrointestinal Hemorrhage; Helicobacter Infections; Hemorrhage; Nausea; Osteoarthritis; Peptic Ulcer; Pre-Eclampsia; Stomach Ulcer; Ulcer
Unknown
Small molecule
Approved
IMMUNE SYSTEM; OTHER
ORAL
Hepatitis C; Hepatitis, Chronic; Insulin Resistance; Lymphoma; Parkinson Disease; Tuberculosis; Communicable Diseases; Hepatitis D; Lipodystrophy; Liver Cirrhosis, Biliary; Multiple Sclerosis; Acquired Immunodeficiency Syndrome; Severe Acute Respiratory Syndrome; Hepatitis B, Chronic; HIV Infections; Infections; Liver Diseases
Human immunodeficiency virus type 1 reverse transcriptase inhibitor
Small molecule
Approved
OTHER
INTRAVENOUS
Head and Neck Neoplasms; Ischemic Stroke; Lymphedema; Melanoma; Osteosarcoma; Breast Neoplasms; Carcinoma, Hepatocellular; Cholangiocarcinoma; Compartment Syndromes; Kidney Neoplasms; Myocardial Infarction; Renal Insufficiency, Chronic; Prostatic Neoplasms; Echocardiography
Diagnostic agent
Small molecule
Approved
Unknown
Unknown
HIV Infections; Metrorrhagia; Pregnancy
Progesterone receptor agonist
Small molecule
Approved
Unknown
Unknown
Migraine Disorders
Unknown
Small molecule
Approved
Unknown
Unknown
Hepatitis; Hepatitis B, Chronic; Hepatitis C, Chronic; Hepatitis D; Liver Cirrhosis, Biliary; HIV Infections; Severe Acute Respiratory Syndrome; Virus Diseases
Unknown
Small molecule
Approved
IMMUNE SYSTEM; OTHER; RESPIRATORY
ORAL
Lecithin Cholesterol Acyltransferase Deficiency; Carcinoma, Non-Small-Cell Lung; Common Cold; Conjunctivitis, Allergic; Dermatitis; Eczema; Multiple Sclerosis; Multiple Sclerosis, Chronic Progressive; Pruritus; Hypersensitivity; Rhinitis, Allergic, Perennial; Rhinitis, Allergic, Seasonal; Urticaria
Histamine H1 receptor antagonist
Small molecule
Approved
OTHER; PREGNANCY AND GYNECOLOGY
ORAL
Osteoarthritis, Knee; Pancreatitis; Pain; Pharyngitis; Arthritis, Rheumatoid; Dysmenorrhea; Osteoarthritis; Rheumatic Diseases
Cyclooxygenase-2 inhibitor
Small molecule
Approved
Unknown
Unknown
Acute Lung Injury; Carcinoma, Renal Cell; Carcinoma, Squamous Cell; Colorectal Neoplasms; Desmoplastic Small Round Cell Tumor; Fibrosarcoma; Head and Neck Neoplasms; Hematologic Neoplasms; Liver Cirrhosis; Lymphoma, Large-Cell, Anaplastic; Lymphoma, Non-Hodgkin; Pancreatic Neoplasms; Rhinitis, Allergic, Seasonal; Thymoma; Arthritis, Rheumatoid; Breast Neoplasms; Chordoma; Colonic Neoplasms; Desmoid Tumors; Fibroma; Glioblastoma; Hypereosinophilic Syndrome; Leukemia, Lymphoid; Leukemia, Myeloid, Acute; Lung Neoplasms; Malaria, Falciparum; Melanoma; Scleroderma, Systemic; Spinal Cord Injuries; Stomach Neoplasms; Thyroid Neoplasms; Tuberculosis; Gastrointestinal Stromal Tumors; Graft vs Host Disease; Hypertension, Pulmonary; Influenza, Human; Leukemia; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid; Neoplasms; Pneumonia; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Sarcoma; Severe Acute Respiratory Syndrome; Stroke
Unknown
Protein
Approved
CANCER
UNKNOWN
Brain Neoplasms; Coronary Disease; Glioma; Lymphoma, Follicular; Lymphoma, T-Cell, Cutaneous; Neuroblastoma; Osteosarcoma; Adenocarcinoma of Lung; Anemia, Aplastic; Breast Neoplasms, Male; Carcinoid Tumor; Carcinoma, Islet Cell; Carcinoma, Large Cell; Carcinoma, Renal Cell; Carcinoma, Squamous Cell; Colonic Neoplasms; Colorectal Neoplasms; Diabetes Mellitus, Type 1; Fallopian Tube Neoplasms; Head and Neck Neoplasms; Hematologic Neoplasms; Leukemia; Leukemia, Myeloid; Leukemia, Myeloid, Acute; Lymphoma, Mantle-Cell; Lymphoma, Non-Hodgkin; Lymphoma, T-Cell, Peripheral; Medulloblastoma; Melanoma; Myelodysplastic Syndromes; Nasopharyngeal Carcinoma; Neoplasms, Plasma Cell; Ovarian Neoplasms; Pancreatic Neoplasms; Peritoneal Neoplasms; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Prostatic Neoplasms; Rectal Neoplasms; Retinoblastoma; Small Cell Lung Carcinoma; Stomach Neoplasms; Testicular Neoplasms; Urethral Neoplasms; Urinary Bladder Neoplasms; Uterine Cervical Neoplasms; Wilms Tumor; Adrenal Cortex Neoplasms; Breast Neoplasms; Carcinoma, Non-Small-Cell Lung; Endometrial Neoplasms; Esophageal Neoplasms; Hodgkin Disease; Lung Neoplasms; Lymphoma; Lymphoma, Large B-Cell, Diffuse; Multiple Myeloma; Neoplasms, Germ Cell and Embryonal; Prostatic Neoplasms, Castration-Resistant; Sarcoma; Triple Negative Breast Neoplasms; Uterine Neoplasms; Infections; Neoplasms; Neutropenia
Granulocyte colony stimulating factor receptor agonist
Antibody
Approved
Unknown
Unknown
Mucopolysaccharidosis II; Mucopolysaccharidosis VI; Thyroid Neoplasms; Asthma; Bursitis; Choroidal Neovascularization; Colitis; Dupuytren Contracture; Glomerulosclerosis, Focal Segmental; Inflammation; Macular Degeneration; Netherton Syndrome; Osteoarthritis, Knee; Prostatic Hyperplasia; Sarcoidosis; Sciatica; Behcet Syndrome; Cystitis, Interstitial; Giant Cell Arteritis; Inflammatory Bowel Diseases; Osteoarthritis; Pyoderma; Severe Acute Respiratory Syndrome; Spondylarthropathies; Arthritis; Arthritis, Juvenile; Arthritis, Psoriatic; Arthritis, Rheumatoid; Colitis, Ulcerative; Crohn Disease; Hidradenitis Suppurativa; Immune System Diseases; Psoriasis; Spondylitis, Ankylosing; Uveitis
TNF-alpha inhibitor
Small molecule
Approved
Unknown
Unknown
Hyperpigmentation; Lentigo; Melanosis
Unknown
Small molecule
Approved
Unknown
Unknown
Amphetamine-Related Disorders; Cocaine-Related Disorders; Diabetes Mellitus, Type 1; Orthostatic Intolerance; Parkinson Disease; Tobacco Use Disorder; Alcoholism; Cognitive Dysfunction; Hypotension, Orthostatic; Marijuana Abuse; Opioid-Related Disorders; Phobia, Social; Sleep Apnea, Obstructive; Sleep Apnea Syndromes; Substance-Related Disorders; Syncope, Vasovagal; Tourette Syndrome; Autistic Disorder; Neoplasms; Schizophrenia; Attention Deficit Disorder with Hyperactivity
Unknown
Enzyme
Approved
CANCER
INTRAVENOUS
Burkitt Lymphoma; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Large-Cell, Anaplastic; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Tumor Lysis Syndrome; Gout; Hyperuricemia; Leukemia; Lymphoma
Uric acid oxidative enzyme
Small molecule
Approved
OTHER; PEDIATRICS
ORAL
Albinism; Alkaptonuria; Tyrosinemias
4-hydroxyphenylpyruvate dioxygenase inhibitor
Unknown
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
IMMUNE SYSTEM; OTHER; PEDIATRICS
ORAL
HIV Infections; Irritable Bowel Syndrome; Kidney Diseases; Liver Diseases; Bronchiolitis; Crohn Disease; Diabetes Mellitus, Type 2; Gastroenteritis; Hepatitis B, Chronic; Hepatitis C; Hepatitis C, Chronic; Malnutrition; Periodontitis; Sexually Transmitted Diseases; Tuberculosis; Arthritis, Rheumatoid; Brain Diseases; Clostridium Infections; Cryptosporidiosis; Dyspepsia; Enterocolitis, Pseudomembranous; Helicobacter Infections; Influenza, Human; Peritonitis; Respiratory Tract Diseases; Severe Acute Respiratory Syndrome; Amebiasis; Diarrhea
Pyruvate:ferredoxin oxidoreductase inhibitor
Small molecule
Approved
CARDIOVASCULAR; OTHER; RESPIRATORY
INHALATION; INTRAVENOUS; IV (INFUSION); SUBCUTANEOUS
Diabetes Mellitus, Type 1; Diabetic Foot; Raynaud Disease; Reperfusion Injury; Scleroderma, Systemic; Hernias, Diaphragmatic, Congenital; Ischemia; Peripheral Vascular Diseases; Persistent Fetal Circulation Syndrome; Pulmonary Disease, Chronic Obstructive; Respiratory Distress Syndrome; Familial Primary Pulmonary Hypertension; Idiopathic Pulmonary Fibrosis; Lung Diseases, Interstitial; Pulmonary Fibrosis; Hypertension, Pulmonary; Pulmonary Arterial Hypertension; Thrombosis
Prostanoid IP receptor agonist
Small molecule
Approved
IMMUNE SYSTEM; OTHER
INJECTION; INTRAVENOUS; IV (INFUSION); ORAL
Asthma; Graft vs Host Disease; Hematologic Neoplasms; HIV Infections; Keratitis; Leukemia, Lymphocytic, Chronic, B-Cell; Neoplasms; Neutropenia; Aspergillosis, Allergic Bronchopulmonary; Myelodysplastic Syndromes; Candidiasis, Invasive; Leishmaniasis; Leukemia; Leukemia, Myeloid, Acute; Neuroaspergillosis; Aspergillosis; Bacterial Infections and Mycoses; Candidemia; Candidiasis; Fusariosis; Infections; Mycoses
Cytochrome P450 51 inhibitor
Small molecule
Approved
CANCER
INTRAMUSCULAR
Carcinoma, Ductal; Carcinoma, Squamous Cell; Colorectal Neoplasms; Hereditary Breast and Ovarian Cancer Syndrome; Lymphoma; Lymphoma, Non-Hodgkin; Mesothelioma; Pancreatic Neoplasms; Small Cell Lung Carcinoma; Urinary Bladder Neoplasms; Carcinoma; Carcinoma, Intraductal, Noninfiltrating; Carcinoma, Non-Small-Cell Lung; Endometrial Neoplasms; Fibrous Dysplasia, Polyostotic; Genital Neoplasms, Female; Hypertension, Pulmonary; Lung Neoplasms; Lupus Erythematosus, Systemic; Ovarian Neoplasms; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Puberty, Precocious; Sarcoma, Endometrial Stromal; Carcinoma, Lobular; Neoplasm Metastasis; Breast Neoplasms; Neoplasms
Estrogen receptor alpha antagonist