Display Options:
Total: 10647
Small molecule
Approved
Unknown
Unknown
Cardiovascular Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Myasthenia Gravis; Glaucoma
Unknown
Small molecule
Approved
Unknown
Unknown
Glioma; Immunoblastic Lymphadenopathy; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Lymphoma, T-Cell, Peripheral; Precursor T-Cell Lymphoblastic Leukemia-Lymphoma; Leukemia, Biphenotypic, Acute; Lymphoma; Lymphoma, Mantle-Cell; Lymphoma, Non-Hodgkin; Multiple Sclerosis, Relapsing-Remitting; Myelodysplastic Syndromes; Leukemia; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Lymphoid; Leukemia, Myeloid, Acute; Leukemia, Promyelocytic, Acute; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Multiple Sclerosis; Multiple Sclerosis, Chronic Progressive; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Neoplasms
Unknown
Small molecule
Approved
OTHER
ORAL
Fibrosis; Glucose Intolerance; Huntington Disease; Liver Cirrhosis; Obesity; Severe Acute Respiratory Syndrome; Adenomatous Polyposis Coli; Arthritis, Rheumatoid; Chemical and Drug Induced Liver Injury; Cholangitis, Sclerosing; Cholestasis; Colorectal Neoplasms; Diabetes Mellitus; Heart Failure; Hepatitis D; Inflammation; Jaundice, Obstructive; Non-alcoholic Fatty Liver Disease; Parkinson Disease; Pregnancy; Cholelithiasis; Cholestasis, Intrahepatic; Diabetes, Gestational; Diabetes Mellitus, Type 2; Hepatitis C, Chronic; Liver Diseases; Liver Cirrhosis, Biliary
Bile acid receptor FXR agonist
Small molecule
Approved
OTHER
ORAL
Unknown
Norepinephrine transporter releasing agent
Small molecule
Approved
Unknown
Unknown
Brain Neoplasms; Cognitive Dysfunction; Colorectal Neoplasms; Diabetes Mellitus, Type 1; Dysthymic Disorder; Wounds and Injuries; Cocaine-Related Disorders; Epilepsy; Gastroesophageal Reflux; Hypertension, Pulmonary; Ischemic Stroke; Marijuana Abuse; Multiple Sclerosis, Chronic Progressive; Multiple System Atrophy; Obesity; Panic Disorder; Sciatica; Anxiety; Autistic Disorder; Bipolar Disorder; Cerebral Hemorrhage; Dementia; Depressive Disorder; Depressive Disorder, Major; Depressive Disorder, Treatment-Resistant; Enuresis; Fibromyalgia; Influenza, Human; Obsessive-Compulsive Disorder; Phobia, Social; Schizophrenia; Severe Acute Respiratory Syndrome; Stress Disorders, Post-Traumatic; Stroke; Tobacco Use Disorder
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Severe Combined Immunodeficiency; Castleman Disease; Infections; Leukemia-Lymphoma, Adult T-Cell; Liver Cirrhosis, Biliary; Lymphoma; Lymphoma, AIDS-Related; Paraparesis, Tropical Spastic; Sarcoma, Kaposi; Acquired Immunodeficiency Syndrome; AIDS Dementia Complex; AIDS-Related Complex; Diarrhea; Pneumonia, Pneumocystis; Pregnancy; Severe Acute Respiratory Syndrome; Tuberculosis; Autoimmune Diseases; HIV Infections; Virus Diseases
Human immunodeficiency virus type 1 reverse transcriptase inhibitor
Small molecule
Approved
Unknown
Unknown
Rectal Neoplasms; Cystitis; Infections; Otitis Externa; Pyelonephritis; Urinary Tract Infections
Bacterial DNA gyrase inhibitor
Small molecule
Approved
Unknown
Unknown
Reperfusion Injury; Heart Defects, Congenital; Hernias, Diaphragmatic, Congenital; Hypertension, Pulmonary; Muscle Cramp; Shock, Septic; Subarachnoid Hemorrhage; Vasospasm, Intracranial; Heart Failure; Cardiovascular Diseases
Unknown
Small molecule
Approved
OTHER; RESPIRATORY
ORAL
Osteomyelitis; Bronchitis, Chronic; Infections; Maxillary Sinusitis; Otitis Media; Pharyngitis; Sinusitis; Tonsillitis; Urinary Tract Infections
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Non-alcoholic Fatty Liver Disease
Unknown
Small molecule
Approved
Unknown
Unknown
Parkinson Disease; Carotid Stenosis; Atherosclerosis; Coronary Disease; Diabetes Mellitus, Type 2; Hypercholesterolemia; Hypertension; Prostatic Hyperplasia
Unknown
Small molecule
Approved
OTHER
VAGINAL
Vaginitis; Candidiasis, Vulvovaginal
Cytochrome P450 51 inhibitor
Small molecule
Approved
Unknown
Unknown
Depressive Disorder; Panic Disorder; Stress Disorders, Post-Traumatic; Bipolar Disorder; Depressive Disorder, Major; Obsessive-Compulsive Disorder
Serotonin transporter inhibitor
Small molecule
Approved
DERMATOLOGY; OTHER
TOPICAL
Bacterial Infections; Osteomyelitis; Sinusitis; Cystic Fibrosis; Hemangioma; Radiodermatitis; Epistaxis; Infections; Staphylococcal Infections; Telangiectasia, Hereditary Hemorrhagic; Impetigo; Nasal Obstruction
Isoleucyl-tRNA synthetase inhibitor
Small molecule
Approved
OTHER
ORAL
Unknown
Cyclooxygenase-2 inhibitor
Small molecule
Approved
CARDIOVASCULAR; OTHER
ORAL
Asthma; Inflammation; Leukemia, Myeloid, Acute; Metabolic Diseases; Porokeratosis; Stroke; Arthritis, Rheumatoid; Breast Neoplasms; Carotid Stenosis; Cerebrovascular Disorders; Cognitive Dysfunction; Fragile X Syndrome; HIV Infections; Intracranial Arteriosclerosis; Intracranial Arteriovenous Malformations; Learning Disabilities; Melanoma; Neurofibromatosis 1; Ovarian Neoplasms; Parkinson Disease; Prostatic Neoplasms, Castration-Resistant; Pulmonary Disease, Chronic Obstructive; Rett Syndrome; Xanthomatosis, Cerebrotendinous; Heart Diseases; Intermittent Claudication; Lipid Metabolism Disorders; Myocardial Ischemia; Peripheral Vascular Diseases; Atherosclerosis; Cardiovascular Diseases; Coronary Artery Disease; Coronary Disease; Hypercholesterolemia
HMG-CoA reductase inhibitor
Small molecule
Approved
Unknown
Unknown
Rheumatic Diseases
Cyclooxygenase inhibitor
Small molecule
Approved
OTHER
IMPLANTATION; INHALATION; NASAL; TOPICAL
Alopecia Areata; Hypersensitivity; Otitis Media with Effusion; Spinal Cord Injuries; Anemia, Sickle Cell; Dermatitis, Atopic; Eosinophilic Esophagitis; Pemphigoid, Bullous; Psoriasis; Radiodermatitis; Breast Neoplasms; Hypertrophy; Pulmonary Disease, Chronic Obstructive; Rhinitis, Allergic, Perennial; Severe Acute Respiratory Syndrome; Sinusitis; Sleep Apnea, Obstructive; Asthma; Lung Diseases, Obstructive; Nasal Obstruction; Nasal Polyps; Rhinitis, Allergic; Rhinitis, Allergic, Seasonal; Skin Diseases
Glucocorticoid receptor agonist
Small molecule
Approved
Unknown
Unknown
Bacterial Infections; Eye Infections
Unknown
Protein
Approved
OTHER
INJECTION
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
INJECTION
Cicatrix; Cardiomyopathy, Dilated; Hypertension
Angiotensin-converting enzyme inhibitor
Small molecule
Approved
OTHER
INJECTION
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Abortion, Incomplete; Infections; Clostridium Infections; Muscle Cramp; Non-alcoholic Fatty Liver Disease; Premature Birth; Abortion, Spontaneous; Leiomyoma; Menorrhagia; Myoma; Obesity; Pain; Postpartum Hemorrhage; Pre-Eclampsia; Pregnancy; Spondylitis, Ankylosing; Uterine Diseases; Duodenal Ulcer; Gastroesophageal Reflux; Hemorrhage; Osteoarthritis; Peptic Ulcer; Stomach Ulcer
Prostanoid EP3 receptor agonist
Small molecule
Approved
OTHER
ORAL
Chemical and Drug Induced Liver Injury; Cystinuria; Subarachnoid Hemorrhage
Reducing agent
Small molecule
Approved
Unknown
Unknown
Unknown
Bacterial dihydrofolate reductase inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Cardiovascular Diseases; Glaucoma
Unknown
Small molecule
Approved
Unknown
Unknown
Brain Neoplasms; Coronary Disease; Aortic Aneurysm, Thoracic; Stroke; Subarachnoid Hemorrhage; Hypertension; Muscle Cramp; Pre-Eclampsia; Cardiovascular Diseases
Unknown
Small molecule
Approved
OTHER
INJECTION
Esophageal and Gastric Varices
Calcium chelating agent
Small molecule
Approved
OTHER
INJECTION
Multiple Myeloma; Myelodysplastic Syndromes; Myeloproliferative Disorders; Neoplasm Metastasis; Neoplasms, Plasma Cell; Breast Neoplasms; Burkitt Lymphoma; Leukemia, Myeloid, Acute; Lymphoma, AIDS-Related; Lymphoma, B-Cell; Lymphoma, Large-Cell, Anaplastic; Lymphoma, Mantle-Cell; Nasopharyngeal Neoplasms; Pancreatic Neoplasms; Penile Neoplasms; Peritoneal Neoplasms; Rhabdomyosarcoma, Alveolar; Rhabdomyosarcoma, Embryonal; Urethral Neoplasms; Urinary Bladder Neoplasms; Uterine Neoplasms; Wilms Tumor; Carcinoma; Carcinoma, Non-Small-Cell Lung; Central Nervous System Neoplasms; Dermatofibrosarcoma; Endometrial Neoplasms; Fallopian Tube Neoplasms; Fibrosarcoma; Hemangiosarcoma; Histiocytoma; Hodgkin Disease; Kidney Neoplasms; Leiomyosarcoma; Leukemia; Leukemia, Biphenotypic, Acute; Liposarcoma; Lung Neoplasms; Lymphoma; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Non-Hodgkin; Lymphoma, T-Cell, Peripheral; Mediastinal Neoplasms; Neoplasms, Germ Cell and Embryonal; Neurilemmoma; Neuroblastoma; Osteosarcoma; Ovarian Neoplasms; Pheochromocytoma; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Precursor T-Cell Lymphoblastic Leukemia-Lymphoma; Retroviridae Infections; Rhabdomyosarcoma; Sarcoma; Sarcoma, Alveolar Soft Part; Sarcoma, Ewing; Sarcoma, Synovial; Small Cell Lung Carcinoma; Teratoma; Uterine Cervical Neoplasms; Neoplasms; Testicular Neoplasms
DNA inhibitor
Small molecule
Approved
CARDIOVASCULAR; OTHER
ORAL
Cerebrovascular Disorders; Intracranial Aneurysm; Schizophrenia; Cocaine-Related Disorders; Infertility; Muscle Cramp; Neuroma, Acoustic; Stroke; Poisoning; Subarachnoid Hemorrhage; Cardiovascular Diseases
Mineralocorticoid receptor antagonist
Small molecule
Approved
Unknown
Unknown
Onychomycosis; Tinea Pedis
Unknown